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192

抑制剂 & 化合物

109

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Cat. No. Product Name Target Signaling Pathways
T4564 Ethacrynic acid

Edecrin,利尿酸,Etacrynic Acid,Hydromedin

Others; Calcium Channel; NF-κB; GST Membrane transporter/Ion channel; Metabolism; NF-κB; Others; oxidation-reduction
Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂,也是NF-κB 信号传导途径的有效抑制剂,并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道,从而导致气道平滑肌细胞松弛。它是利尿剂,具有抗炎特性,可减轻类维生素 A 诱导的小鼠耳部水肿。
T6044 Telotristat Etiprate

LX1606 (Hippurate),LX 1606 Hippurate,特罗司他马尿酸

Hydroxylase Metabolism
Telotristat Etiprate (LX 1606 Hippurate) 是一种色氨酸羟化酶抑制剂,可抑制血清素的产生。
T5039 Aminohippurate sodium

Sodium 4-aminohippurate Hydrate,Sodium p-aminohippurate,4-氨基马尿酸钠盐,p-Aminohippuric acid sodium salt

Others Others
Aminohippurate sodium (Sodium p-aminohippurate) 是能够利用肾血浆流量测量肾脏医学测试的诊断剂。
T19595 UDP-glucuronic acid trisodium

尿苷二磷酸葡萄糖醛酸三钠,UDP-​glucuronic acid trisodium,尿苷二磷酸葡糖醛酸

Others Others
UDP-glucuronic acid trisodium (UDP-​glucuronic acid trisodium) is an indispensable precursor for vital glycoconjugates in various biological domains. These glycoconjugates encompass mammalian glycosaminoglycans, plant cell wall polysaccharides, and bacterial capsule glycoglycerolipids.
T8365 Methenamine Hippurate

Antibacterial Microbiology/Virology
Methenamine hippurate 是一种口服活性尿液广谱抗菌剂。它对大多数常见的尿路病原体有效。
T13480 (S)-(-)-5-Fluorowillardiine

(S)-5-Fluorowillardiine,5-氟代尿嘧啶丙氨酸,(5S)-Fluorowillardiine

iGluR Membrane transporter/Ion channel; Neuroscience
(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) 是一种 AMPA 受体特异性激动剂。
T10824 cis-Urocanic acid

cis-UCA,(Z)-Imidazole-4-acrylic acid,(Z)-Urocanic acid,(E)-Urocanic acid,(Z)-3-(1H-Imidazol-5-yl)acrylic acid,顺式-尿刊酸

5-HT Receptor GPCR/G Protein; Neuroscience
cis-Urocanic acid ((E)-Urocanic acid) 是一种 5-HT2A 受体激动剂,cis-Urocanic acid 与 5-HT 受体结合的Kd 为 4.6 nM。cis-Urocanic acid 是一种免疫调节剂,通过与 5-HT2A 受体结合而诱导免疫抑制。
T22517 5,7-Dichlorokynurenic acid

5,7-二氯犬尿喹啉酸,5,7-dichlorokynurenic acid sodium,5,7-DCKA

NMDAR Neuroscience
5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) 是一种专门针对于NMDA 受体甘氨酸位点的竞争性拮抗剂(KB:65 nM)。它是犬尿酸的衍生物,可降低大鼠皮质细胞培养物中 NMDA 诱导的神经元损伤程度。
T19596 UDP-GlcNAc Disodium Salt

Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt

Others Others
UDP-GlcNAc Disodium Salt (UDP-α-D-N-Acetylglucosamine Disodium Salt) 是一种 O-GlcNAc 转移酶 (OGT) 的供体底物。
T15160 Dotinurad

(3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone

OAT Membrane transporter/Ion channel
Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) 是有效的尿酸盐重吸收选择性抑制剂,抑制尿酸盐转运蛋白 1的IC50为 37.2 nM,具有促尿酸排泄的作用。
T79854 Lingdolinurad

OAT Membrane transporter/Ion channel
Lingdolinurad 是一种靶向 hURAT1的尿酸转运蛋白抑制剂,可用于研究高尿酸血症或痛风。
T36125 Tienilic Acid

P450 Metabolism
Tienilic Acid 是一种具有一定肝毒性的排尿酸利尿剂
T8735 Sulbactum Sodium

5'-CDP,Cytidine-5′-diphosphate,胞苷-5'-二磷酸

Others Others
Sulbactum Sodium (5'-CDP) 由胞苷一磷酸 (CMP) 或尿苷一磷酸 (UMP) 通过磷酸基团的转移在尿苷酸激酶 (UMPK) 酶的催化下合成。
T61048 Puliginurad

YL-90148

OAT Membrane transporter/Ion channel
Puliginurad (YL-90148) 是一种具有有效性和选择性的尿酸盐转运蛋白 (URAT) 抑制剂,对尿酸的重吸收有抑制作用。Puliginurad 可用于预防和治疗高尿酸血症和痛风。
T32194 Irtemazole

R60844,R-60844,R 60844

Others Others
Irtemazole (R 60844) 是一种新型排尿酸物质,在治疗高尿酸血症和痛风方面很有价值。
T20545 Benzarone

Benzarona,Vasoc,苯扎隆,Venagil,Benzaronum

OAT Membrane transporter/Ion channel
Benzarone (Benzarona) 是人尿酸转运蛋白 1的有效抑制剂,IC50为 2.8 μM。它具有降低血清尿酸水平的作用。
T0601 Monobenzyl phthalate

邻苯二甲酸单苄酯,Phthalic Acid Monobenzyl Ester

Others; Endogenous Metabolite Metabolism; Others
Monobenzyl phthalate (Phthalic Acid Monobenzyl Ester) 是一种暴露于邻苯二甲酸盐(如,邻苯二甲酸二乙基己酯)后的尿代谢物 (urinary metabolite)。
T10632 Bucolome

Paramidin,5-Butyl-1-cyclohexylbarbituric acid,Paramidine,Bucolom,布可隆,Bucolomum

P450; Immunology/Inflammation related Immunology/Inflammation; Metabolism
Bucolome (Paramidine) 是一种 CYP2C9 抑制剂,具有排尿酸和抗炎活性。
T0457 Probenecid

Benemid,丙磺舒

HIV Protease; Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Probenecid (Benemid) 是一种苯甲酸衍生物,具有抗高尿酸特性。它也是一种选择性瞬时受体电位香草酸受体通道 2 激动剂,还可抑制pannexin 1通道。
T77517 URAT1 inhibitor 7

OAT Membrane transporter/Ion channel
URAT1 inhibitor 7 是一种新型高效的人尿酸转运蛋白 URAT1 抑制剂 (IC50:12 nM)。URAT1 inhibitor 7 对 CYP2C9 具有抑制作用,IC50为4.2 μM。URAT1 inhibitor 7 可用于研究高尿酸血症和痛风。
T0808 Diflunisal

Flovacil,二氟尼柳,Dolobid,MK-647,Fluniget,Dolobis

Epigenetic Reader Domain; COX Chromatin/Epigenetic; Immunology/Inflammation; Neuroscience
Diflunisal (Dolobid) 是一种水杨酸盐衍生物,是环氧合酶的抑制剂,具有非甾体抗炎和尿酸舒缓性能,可单独用作止痛剂和类风湿关节炎患者。
T1274 Benzbromarone

Desuric,Normurat,苯溴马隆,Urinorm

Apoptosis; P450; Xanthine Oxidase Apoptosis; Metabolism
Benzbromarone (Desuric) 是一种高效的,耐受性良好的非竞争性黄嘌呤氧化酶抑制剂,用作排尿酸剂,研究痛风。
T5987 Potassium oxonate

Oxonic Acid (potassium salt),氧嗪酸钾,Potassium otastat,Potassium azaorotate

Others Others
Potassium oxonate (Potassium azaorotate) 是用作尿酸酶抑制剂,都5-FU 磷酸化为5-fluorouridine-5'-monophosphate 具有抑制作用。
T21469 Cyclopenthiazide

Cyclomethiazide,Su-8341,SU 8341,环戊噻嗪

Others Others
Cyclopenthiazide (Cyclomethiazide) 是一种噻嗪类利尿剂,用于治疗高血压和心力衰竭。减少钙离子和尿酸的排泄,增加钠和钾离子的排泄。
T1896 Ro 61-8048

Hydroxylase Metabolism
Ro 61-8048 是一种选择性的、口服有效的犬尿氨酸 3-羟化酶抑制剂(IC50:37 nM)。它能够导致细胞喹啉酸浓度的显著增加。
T1672 Dimesna

地美司钠,BNP-7787

Others Others
Dimesna (BNP-7787) 是一种二硫代乙烷磺酸盐的合成衍生物,具有泌尿保护特性。
T60625 Tigulixostat

Tigulixostat 是吲哚基杂芳羧酸的新型衍生物。Tigulixostat 是一种非嘌呤选择性的黄嘌呤氧化酶抑制剂,可降低尿酸的生成。
T67822L Ulodesine

BCX4208

Endogenous Metabolite Metabolism
Ulodesine (BCX4208) 是一种嘌呤核苷磷酸化酶 (PNP) 抑制剂,对 PNP 有抑制作用,IC50 值为 2.293 nM/L。Ulodesine 可用于研究高尿酸血症。
T7542 Amino Tadalafil

氨基他达那非,氨基他达拉非

PDE Metabolism
Amino Tadalafil 是一种 Tadalafil 的类似物,是一种磷酸二酯酶 5 抑制剂,可用于多种疾病,如勃起功能障碍,肺动脉高压和下尿路功能障碍。
T72165 Xanthine oxidoreductase-IN-3

Xanthine Oxidase Metabolism
Xanthine oxidoreductase-IN-3 是一种具有口服活性的黄氨酸氧化还原酶 (XOR) 抑制剂(IC50 : 26.3 nM)。Xanthine oxidoreductase-IN-3 可用急性高尿酸血症的研究。
T72166 Xanthine oxidoreductase-IN-5

Xanthine Oxidase Metabolism
Xanthine oxidoreductase-IN-5 是一种具有口服活性的黄氨酸氧化还原酶 (XOR) 抑制剂(IC50 : 55 nM)。Xanthine oxidoreductase-IN-5 可用于急性高尿酸血症的研究。
T7704 KY-226

Phosphatase Metabolism
KY-226 是选择性的,口服活性的和变构蛋白酪氨酸磷酸酶 1B 抑制剂,IC50=0.25 μM,且不激活 PPARγ 。它可以保护神经元免受脑缺血损伤。它通过增强胰岛素和瘦素信号传导发挥抗糖尿病和抗肥胖作用。
T12499 PKR-IN-2

PKM Metabolism
PKR-IN-2 是丙酮酸激酶PKR 亚型的激活剂,可用于 PKR 功能相关疾病的研究,包括癌症、糖尿病、肥胖、自身免疫性疾病、良性前列腺增生等。
T7362 O-304

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
O-304 是 AMP 活化蛋白激酶 (AMPK) 的泛激活剂,可通过抑制 pAMPK 的去磷酸化来增加 AMPK 活性,可用于 2 型糖尿病和相关心血管并发症的研究。
T6288 Mozavaptan

莫扎伐坦,OPC31260l,OPC-31260

Vasopressin Receptor GPCR/G Protein
Mozavaptan (OPC-31260) 是 benzazepine 衍生物,是一种竞争性加压素受体拮抗剂,作用于 V1 和 V2 受体,IC50 分别为 1.2 μM 和 14 nM。它可在体内拮抗精氨酸加压素的抗利尿作用,可用于低钠血症、抗利尿激素不适当综合征和充血性心力衰竭的研究。
T15251 Etebenecid

乙磺舒,Urelim

Others Others
Etebenecid (Urelim) 是促尿酸排泄药,能够抑制青霉素自肾小管分泌。
T13257 Upamostat

PAI-1; Serine/threonin kinase; Serine Protease Cell Cycle/Checkpoint; Metabolism; Proteases/Proteasome
Upamostat 是一种丝氨酸蛋白酶抑制剂,也是一种具有口服活性的 WX-UK1 前药,是一种尿激酶型纤溶酶原激活剂 (uPA) 抑制剂。
T60561 Disulfamide

Carbonic Anhydrase Metabolism
Disulfamide 是一种具有口服活性的碳酸酐酶 (carbonic anhydrase) 抑制剂,其 IC50 值为 0.07 μM。Disulfamide 具有利尿作用,可通过抑制碳酸酐酶,阻止钠、碳酸氢盐在近曲小管中的重吸收,从而发挥作用。
T76684 Girentuximab

cG250,WX-G250,G250

Carbonic Anhydrase Metabolism
Girentuximab (G250) 是一种有效的抗碳酸酐酶 IX (CAIX)单克隆抗体,具有抗癌活性,可用于研究尿路上皮癌 PET (ZiPUP)。
T31976 Glymidine sodium

Others Others
Glymidine sodium 是口服有活性的抗糖尿病药物,也是肝脂肪分解的抑制剂。它通过抑制葡萄糖的形成,也对由于内源性脂质动员抑制而导致的丙酮酸氧化升高具有抑制作用。
T83974 OPC18750 HCl

PDE Metabolism
OPC18750 HCl 是一种潜在的磷酸二酯酶抑制剂,具有正肌力作用,可用于研究哮喘、癌症、糖尿病和精神疾病。
T4410 LM10

Others Others
LM10 是有效的色氨酸 2,3-双加氧酶的抑制剂。色氨酸 2,3-双加氧酶是一种无关的肝酶,它可通过犬尿氨酸途径降解色氨酸。它对研究癌症疾病具有潜在的研究价值。
T3658 Trifluridine/tipiracil hydrochloride mixture

Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Trifluridine/tipiracil hydrochloride mixture (TAS-102) 是一种新型口服组合药物,含有摩尔比为 2:1 的曲氟尿苷(TFT) 和盐酸替吡嘧啶 (TTP)。它主要通过抑制胸苷酸合酶 (TS) 和掺入 DNA 来显示抗肿瘤活性。
T6820 D-α-Hydroxyglutaric acid disodium

D-alpha-Hydroxyglutaric acid disodium salt,(R)-2-羟基戊二酸二钠盐,Disodium (R)-2-Hydroxyglutarate

ATPase; Others; Reactive Oxygen Species; Endogenous Metabolite; mTOR Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Others; PI3K/Akt/mTOR signaling
D-α-Hydroxyglutaric acid disodium (Disodium (R)-2-Hydroxyglutarate) 是神经代谢疾病 D-2-羟基戊二酸尿症中积累的主要代谢产物,可增加活性氧的产生。它是 α-酮戊二酸 (α-KG) 的弱竞争拮抗剂,可抑制多种α-KG 依赖性双加氧酶,Ki 为 10.87 mM。
T6376 Allopurinol Sodium

1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐,Allopurinol sodium salt,Sodium allopurinol

ROS Immunology/Inflammation
Allopurinol Sodium 是黄嘌呤氧化酶抑制剂,其IC50= 0.2~50 μM。它能够抗利什曼原虫,也可用于研究痛风以及高尿酸血症。
T4639 Azemiglitazone

MSDC 0602

Mitochondrial Metabolism; mTOR Metabolism; PI3K/Akt/mTOR signaling
Azemiglitazone (MSDC 0602) 是一种 PPARγ 保留的噻唑烷二酮类药物 (TZD),与能够线粒体丙酮酸载体 (MPC) 相互作用并抑制其活性,降低 pparγ 介导的副作用的风险,有用于 2 型糖尿病研究的潜能。
T0435 Sulfinpyrazone

(+/-)-Sulfinpyrazone,G-28315,苯磺保泰松,NSC 75925

COX Immunology/Inflammation; Neuroscience
Sulfinpyrazone (NSC-75925) 是一种口服有效的尿酸剂,具有抗血栓和血小板抑制作用。它可作用于慢性和间歇性痛风性关节炎。
T0922 Zoxazolamine

NSC 24995,Contrazole,氯苯恶唑胺,苯并恶唑胺

Others Others
Zoxazolamine (NSC-24995) 是排尿酸和肌肉松弛剂,被广泛用于药物测试,可作为啮齿动物细胞色素 P-450 活性变化的方便指标。
T2397 Topiroxostat

托匹司他,FYX-051

P450; ROS; Xanthine Oxidase Immunology/Inflammation; Metabolism
Topiroxostat (FYX-051) 是一种有效的口服黄嘌呤氧化还原酶 (XOR) 抑制剂,IC50=5.3 nM,Ki=5.7 nM。它还表现出弱的CYP3A4抑制活性 (18.6%)。它有用于高尿酸血症的研究潜力。
T24644 Piritrexim

BW 301U

DHFR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Piritrexim (BW 301U) 是一种可口服的脂溶性二氢叶酸还原酶抑制剂,具有肺毒性,用于研究尿路上皮癌和转移性乳腺癌。

化合物

Ethacrynic acid
Cat.No: T4564
Synonym: Edecrin,利尿酸,Etacrynic Acid,Hydromedin
Target: Others, Calcium Channel, NF-κB, GST
Telotristat Etiprate
Cat.No: T6044
Synonym: LX1606 (Hippurate),LX 1606 Hippurate,特罗司他马尿酸
Target: Hydroxylase
Aminohippurate sodium
Cat.No: T5039
Synonym: Sodium 4-aminohippurate Hydrate,Sodium p-aminohippurate,4-氨基马尿酸钠盐,p-Aminohippuric acid sodium salt
Target: Others
UDP-glucuronic acid trisodium
Cat.No: T19595
Synonym: 尿苷二磷酸葡萄糖醛酸三钠,UDP-​glucuronic acid trisodium,尿苷二磷酸葡糖醛酸
Target: Others
Methenamine Hippurate
Cat.No: T8365
Synonym:
Target: Antibacterial
(S)-(-)-5-Fluorowillardiine
Cat.No: T13480
Synonym: (S)-5-Fluorowillardiine,5-氟代尿嘧啶丙氨酸,(5S)-Fluorowillardiine
Target: iGluR
cis-Urocanic acid
Cat.No: T10824
Synonym: cis-UCA,(Z)-Imidazole-4-acrylic acid,(Z)-Urocanic acid,(E)-Urocanic acid,(Z)-3-(1H-Imidazol-5-yl)acrylic acid,顺式-尿刊酸
Target: 5-HT Receptor
5,7-Dichlorokynurenic acid
Cat.No: T22517
Synonym: 5,7-二氯犬尿喹啉酸,5,7-dichlorokynurenic acid sodium,5,7-DCKA
Target: NMDAR
UDP-GlcNAc Disodium Salt
Cat.No: T19596
Synonym: Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt
Target: Others
Dotinurad
Cat.No: T15160
Synonym: (3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone
Target: OAT
Lingdolinurad
Cat.No: T79854
Synonym:
Target: OAT
Tienilic Acid
Cat.No: T36125
Synonym:
Target: P450
Sulbactum Sodium
Cat.No: T8735
Synonym: 5'-CDP,Cytidine-5′-diphosphate,胞苷-5'-二磷酸
Target: Others
Puliginurad
Cat.No: T61048
Synonym: YL-90148
Target: OAT
Irtemazole
Cat.No: T32194
Synonym: R60844,R-60844,R 60844
Target: Others
Benzarone
Cat.No: T20545
Synonym: Benzarona,Vasoc,苯扎隆,Venagil,Benzaronum
Target: OAT
Monobenzyl phthalate
Cat.No: T0601
Synonym: 邻苯二甲酸单苄酯,Phthalic Acid Monobenzyl Ester
Target: Others, Endogenous Metabolite
Bucolome
Cat.No: T10632
Synonym: Paramidin,5-Butyl-1-cyclohexylbarbituric acid,Paramidine,Bucolom,布可隆,Bucolomum
Target: P450, Immunology/Inflammation related
Probenecid
Cat.No: T0457
Synonym: Benemid,丙磺舒
Target: HIV Protease, Antibacterial, TRP/TRPV Channel
URAT1 inhibitor 7
Cat.No: T77517
Synonym:
Target: OAT
Diflunisal
Cat.No: T0808
Synonym: Flovacil,二氟尼柳,Dolobid,MK-647,Fluniget,Dolobis
Target: Epigenetic Reader Domain, COX
Benzbromarone
Cat.No: T1274
Synonym: Desuric,Normurat,苯溴马隆,Urinorm
Target: Apoptosis, P450, Xanthine Oxidase
Potassium oxonate
Cat.No: T5987
Synonym: Oxonic Acid (potassium salt),氧嗪酸钾,Potassium otastat,Potassium azaorotate
Target: Others
Cyclopenthiazide
Cat.No: T21469
Synonym: Cyclomethiazide,Su-8341,SU 8341,环戊噻嗪
Target: Others
Ro 61-8048
Cat.No: T1896
Synonym:
Target: Hydroxylase
Dimesna
Cat.No: T1672
Synonym: 地美司钠,BNP-7787
Target: Others
Tigulixostat
Cat.No: T60625
Synonym:
Target:
Ulodesine
Cat.No: T67822L
Synonym: BCX4208
Target: Endogenous Metabolite
Amino Tadalafil
Cat.No: T7542
Synonym: 氨基他达那非,氨基他达拉非
Target: PDE
Xanthine oxidoreductase-IN-3
Cat.No: T72165
Synonym:
Target: Xanthine Oxidase
Xanthine oxidoreductase-IN-5
Cat.No: T72166
Synonym:
Target: Xanthine Oxidase
KY-226
Cat.No: T7704
Synonym:
Target: Phosphatase
PKR-IN-2
Cat.No: T12499
Synonym:
Target: PKM
O-304
Cat.No: T7362
Synonym:
Target: AMPK
Mozavaptan
Cat.No: T6288
Synonym: 莫扎伐坦,OPC31260l,OPC-31260
Target: Vasopressin Receptor
Etebenecid
Cat.No: T15251
Synonym: 乙磺舒,Urelim
Target: Others
Upamostat
Cat.No: T13257
Synonym:
Target: PAI-1, Serine/threonin kinase, Serine Protease
Disulfamide
Cat.No: T60561
Synonym:
Target: Carbonic Anhydrase
Girentuximab
Cat.No: T76684
Synonym: cG250,WX-G250,G250
Target: Carbonic Anhydrase
Glymidine sodium
Cat.No: T31976
Synonym:
Target: Others
OPC18750 HCl
Cat.No: T83974
Synonym:
Target: PDE
LM10
Cat.No: T4410
Synonym:
Target: Others
Trifluridine/tipiracil hydrochloride mixture
Cat.No: T3658
Synonym: Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
D-α-Hydroxyglutaric acid disodium
Cat.No: T6820
Synonym: D-alpha-Hydroxyglutaric acid disodium salt,(R)-2-羟基戊二酸二钠盐,Disodium (R)-2-Hydroxyglutarate
Target: ATPase, Others, Reactive Oxygen Species, Endogenous Metabolite, mTOR
Allopurinol Sodium
Cat.No: T6376
Synonym: 1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐,Allopurinol sodium salt,Sodium allopurinol
Target: ROS
Azemiglitazone
Cat.No: T4639
Synonym: MSDC 0602
Target: Mitochondrial Metabolism, mTOR
Sulfinpyrazone
Cat.No: T0435
Synonym: (+/-)-Sulfinpyrazone,G-28315,苯磺保泰松,NSC 75925
Target: COX
Zoxazolamine
Cat.No: T0922
Synonym: NSC 24995,Contrazole,氯苯恶唑胺,苯并恶唑胺
Target: Others
Topiroxostat
Cat.No: T2397
Synonym: 托匹司他,FYX-051
Target: P450, ROS, Xanthine Oxidase
Piritrexim
Cat.No: T24644
Synonym: BW 301U
Target: DHFR
Cat. No. Product Name Target Signaling Pathways
T0626 Uric Acid

尿酸,2,6,8-Trioxopurine,2,6,8-Trioxypurine,2,6,8-Trihydroxypurine,Lithic acid,Urate

Reactive Oxygen Species; Endogenous Metabolite; Phosphorylase Immunology/Inflammation; Metabolism; NF-κB
Uric Acid (Lithic acid) 是一种重要的抗氧化剂。Uric acid 能清除活性氧(ROS) ,如单线态氧和过氧亚硝酸盐,抑制脂质过氧化。Uric acid 有助于维持血压的稳定和抗氧化应激。
T3762 Hyaluronic acid

透明质酸,Hyaluronate,玻尿酸,hyaluronan

Others; Endogenous Metabolite Metabolism; Others
Hyaluronic acid (hyaluronan) 由玉米发酵得到,是由二糖的重复单元组成的生物聚合物,应用领域广泛。
T4815 Hippuric acid

尿酸,2-Benzamidoacetic acid,Benzoylglycine

Others; Endogenous Metabolite Metabolism; Others
Hippuric acid (2-Benzamidoacetic acid) 是一种正常的尿液成分,是苯酸和甘氨酸结合作用下产生的一种酰基甘氨酸,来自食物的芳香化合物的代谢。
T1436 4-Aminohippuric Acid

p-Aminohippuric acid,对氨基马尿酸

Amino Acids and Derivatives; Endogenous Metabolite Metabolism
4-Aminohippuric Acid 是诊断剂,能够用于肾脏检测,在肾血浆流量的测定中使用。
T3010 Xanthurenic Acid

8-Hydroxykynurenic acid,黄尿酸,4,8-Dihydroxyquinaldic acid,xanthurenate

Apoptosis; Endogenous Metabolite; GluR Apoptosis; Metabolism; Neuroscience
Xanthurenic Acid (8-Hydroxykynurenic acid) 是通过 3-羟基犬尿氨酸转氨而由色氨酸代谢产生的分子,可激活 mGlu2/3 代谢型谷氨酸受体。在下丘脑的感觉传输过程中,它被认为是Group II 代谢型谷氨酸受体的激动剂。
T10191L 7-Chlorokynurenic acid

7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA

GluR; NMDAR Neuroscience
7-Chlorokynurenic acid (7-chloro-4-hydroxy-2-carboxyquinoline) 是一种有效的选择性 NMDA 受体拮抗剂,对甘氨酸 B 激动剂位点的 IC50 为 0.56 μM。 7-Chlorokynurenic acid 抑制谷氨酸再摄取到突触小泡中,Ki 为 0.59 μM,并在神经轴输送后显示出镇痛作用。
T5221 Salicyluric acid

2-羟基马尿酸,N-Salicyloylglycine,N-(2-Hydroxybenzoyl)glycine,2-Hydroxy Hippuric Acid

Others; Endogenous Metabolite Metabolism; Others
Salicyluric acid (2-Hydroxy Hippuric Acid) 是内源性代谢产物的一种。
T5226 2-(2-Methylbenzamido)acetic acid

2-Methylhippuric acid,2-甲基马尿酸,O-Toluric acid,N-(O-Toluoyl)glycine

Others; Endogenous Metabolite Metabolism; Others
2-(2-Methylbenzamido)acetic acid (O-Toluric acid) 是一种能够在尿液中检测到的代谢物。
T41242 Uric acid sodium

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Uric acid sodium 是氧自由基 (oxygen radical) 的清除剂,是一种有效的、常见的抗氧化剂,有助于维持机体血压稳定和抗氧化应激。Uric acid sodium 能清除活性氧 (ROS),如单线态氧和过氧亚硝酸盐,对脂质过氧化有抑制作用,与痛风性关节病的发病机理和草酸钙结石的形成有关。
T4759 Urocanic acid

4-Imidazoleacrylic acid,尿刊酸

Others; Endogenous Metabolite Metabolism; Others
Urocanic acid (4-Imidazoleacrylic acid), synthesized in the epidermis, functions as a primary absorber of ultraviolet (UV) radiation in mammalian skin.
T13456 (S)-Willardiine

(-)-Willardiine,L-willardiine,Willardiine

iGluR Membrane transporter/Ion channel; Neuroscience
(S)-Willardiine (L-willardiine) 存在于金合欢和含羞草的种子中。 (S)-Willardiine 是一种 AMPA/红藻氨酸受体激动剂 (EC50 = 44.8 μM)。
T4928 L-Kynurenine

L-犬尿氨酸,(S)-Kynurenine

AhR; Aryl Hydrocarbon Receptor; Endogenous Metabolite Immunology/Inflammation; Metabolism
L-Kynurenine ((S)-Kynurenine) 是L-色氨酸的代谢物,是芳香烃受体激动剂,可抑制同种异体 T 细胞增殖并增加恶性 U87 神经胶质瘤细胞侵入胶原基质。
T19792 1,3,7-Trimethyluric acid

Others Others
1,3,7-Trimethyluric acid 是咖啡因的代谢产物。其与咖啡因的代谢比可以反映 CYP3A 活性的变化情况。
T8075 1,3-Dimethyluric acid

Endogenous Metabolite Metabolism
1,3-Dimethyluric acid 是尿路结石中的嘌呤成分之一,是一种人体茶碱代谢的产物。
TMA2440 Uridine 5'-monophosphate disodium salt

尿苷-5'-单磷酸二钠盐,Disodium UMP,尿苷酸二钠盐,Disodium uridine-5'-monophosphate,5'-UMP disodium salt,Disodium 5'-Uridylate

Others Others
Uridine 5'-monophosphate disodium salt (Disodium UMP) 是合成 RNA 的一种重要成分。
T3011 2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid

Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine,犬尿氨酸

Others; Endogenous Metabolite Metabolism; Others
2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid (3-Anthraniloylalanine) 是一种酮类和氨基酸衍生物,具有多种生物功能,包括血管舒张、免疫调节和神经调节活性。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 是烟酸的前体。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 的异常产生与神经系统疾病相关的认知缺陷和抑郁症状有关。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 在某些类型的癌细胞中过度表达,可能被用作评估癌症风险的生物标志物。
T7711 Uridine triphosphate

尿苷5'-三磷酸酯,UTP,Uridine 5'-triphosphate,三磷酸尿苷

Others; Endogenous Metabolite Metabolism; Others
Uridine triphosphate (Uridine 5'-triphosphate) 是一种核苷酸,调节胰腺内分泌和外分泌、增殖、通道、转运体和细胞内信号传导的功能。
T4718 Uridine 5'-monophosphate

Uridylic acid,尿苷5-单磷酸,UMP,Uridine phosphate,Uridine 5'-phosphoric acid,5'-Uridylic acid

Others; Endogenous Metabolite Metabolism; Others
Uridine 5'-monophosphate (Uridylic acid) 是一种单磷酸盐形式的尿嘧啶核苷酸,能够由从头途径或体内核苷酸和核酸的降解产物获得,是哺乳动物乳中的主要核苷酸类似物。
T4706 Uridine-5'-diphosphate disodium salt

UDP disodium salt,Uridine 5'-diphosphate disodium salt hyd,尿苷-5'-二磷酸二钠盐

DNA/RNA Synthesis; Endogenous Metabolite; P2Y Receptor Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience
Uridine-5'-diphosphate disodium salt (UDP disodium salt) 是一种选择性 P2Y6受体激动剂,EC50为300 nM,对人 P2Y6受体的 pEC50为6.52。它可刺激炎症介质的产生、吞噬作用和血管收缩,催化多种底物的葡糖醛酸糖化反应,用于核酸生物合成。
T10020 1-Methyluric acid

1-Methyl-2,6,8-trihydroxypurine,1-Methylurate

Endogenous Metabolite Metabolism
1-Methyluric acid (1-Methylurate) 作用于膀胱粘膜并增加胰岛素、甘油三酯、胆固醇和血糖的水平。
T8393 Uridine triphosphate trisodium salt

UTP, Trisodium Salt,Uridine 5'-triphosphate trisodium salt,尿苷-5'-三磷酸三钠盐,Uridine triphosphate (trisodium salt)

Others Others
Uridine triphosphate trisodium salt (UTP, Trisodium Salt) 是一种核苷酸,在正常和疾病状态,均能够调节胰腺内分泌和外分泌、通道、增殖、转运体和细胞内信号传导的功能。
T4735 2'-Deoxyuridine 5'-monophosphate disodium

2'-脱氧尿苷-5'-单磷酸二钠,2'-dUMP⋅2Na,2-脱氧尿嘧啶核苷-5'-单磷酸二钠盐,2'-Deoxyuridine 5'-monophosphate disodium salt

Others; Endogenous Metabolite Metabolism; Others
2'-Deoxyuridine 5'-monophosphate disodium (2'-dUMP⋅2Na) salt 能够被双底物酶胸苷酸合酶(TS) 还原甲基化为 dTMP (2'-deoxythymidine 5'-monophosphate)。其中 dTMP 是 DNA 合成所需的核苷酸。
T4743 Uridine 5′-diphosphoglucose disodium salt

二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal

Endogenous Metabolite; P2Y Receptor GPCR/G Protein; Metabolism; Neuroscience
Uridine 5′-diphosphoglucose disodium salt (UDP-Glucose sodium salt) 是一种内源性核苷酸糖,参与代谢中的糖基转移酶反应。它是 P2Y14 受体的激动剂,EC50为 0.35 μM。
TN6062 1,3,9-Trimethyluric acid

1,3,9-Trimethyluric acid exhibits in vitro cytotoxic activity against breast cancer (MCF-7), human neuroblastoma (SHSY5Y), human non-small cell lung cancer (A549) and human liver cancer (HEPG2) with IC50 value in the range of 1-3 uM. 1,3,9-Trimethyluric a
T4922 Uridine 5′-triphosphate tris salt

尿苷-5′-三磷酸酯 三羟甲基氨基甲烷盐,Uridine 5'-triphosphoric acid

Others; Endogenous Metabolite Metabolism; Others
Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) 是 P2Y 受体的激动剂,已用于研究细胞内 Ca2+ 的浓度,以及用于体外激酶测定的磷酸盐供体。
T4919 Ureidopropionic acid

Carbamoyl-b-alanine,3-酰脲丙酸,3-Ureidopropionic acid

Endogenous Metabolite Metabolism
Ureidopropionic acid (3-Ureidopropionic acid) 是尿嘧啶代谢的中间体。更具体地说,它是二氢尿嘧啶的分解产物,由二氢嘧啶酶产生。它通过β -脲丙酸酶进一步分解为β -丙氨酸。尿素丙酸本质上是β -丙氨酸的尿素衍生物。高水平的尿丙酸存在于β -尿丙酸酶(UP)缺乏的个体中。嘧啶代谢中的酶缺乏与抗肿瘤药物5-氟尿嘧啶的严重毒性风险有关。
T10815 Cinnamoylglycine

Endogenous Metabolite Metabolism
Cinnamoylglycine 是肉桂酸和的甘氨酸结合物,是人体尿液代谢物。它被用作的尿液标志物,能够作为在抗生素研究期之后定殖耐药性的标志物。
T5257 L-Homocitrulline

高瓜氨酸,Homo-L-citrulline,Homocitrulline

Others; Endogenous Metabolite Metabolism; Others
L-Homocitrulline (Homocitrulline) 是一种代谢物,可在尿素循环障碍患者的尿液中大量检测到。在某些情况下,由于尿素循环的鸟氨酸供应耗尽而导致的氨甲酰磷酸酯的积累可能是 L-Homocitrulline 和高精氨酸合成增强的原因。
TN1983 Neoisoastilbin

IL Receptor; TNF; NO Synthase Apoptosis; Immunology/Inflammation
Neoisoastilbin 具有抗炎、抗氧化、抗尿酸过多等生物特性。
T19340 Glutarylcarnitine

O-glutaroyl-L-carnitine

Endogenous Metabolite Metabolism
Glutarylcarnitine (O-glutaroyl-L-carnitine) 是大多数串联质谱新生儿筛查计划中监测的丙二酸尿症和谷草酸尿症 I 型的诊断代谢物。
T3012 Mangiferin

Alpizarin,Chinomin,芒果,Hedysarid

Apoptosis; Others; NF-κB; Nrf2 Apoptosis; Immunology/Inflammation; NF-κB; Others
Mangiferin (Hedysarid) 是一种Nrf2激活剂。它抑制NF-κB 亚基p65和p50的核移位,具有抗氧化、抗糖尿病、抗高尿酸血症、抗病毒、抗癌和抗炎活性。
T5550 2-Hydroxy-2-methylbutanoic acid

Others; Endogenous Metabolite Metabolism; Others
2-Hydroxy-2-methylbutanoic acid 是非正常的代谢物,与羟基戊二酸尿症以及枫糖尿病有关。
T7464 3,3-Dimethylglutaric acid

3,3-二甲基戊二酸,3,3-Dimethylpentanedioate

Others; Endogenous Metabolite Metabolism; Others
3,3-Dimethylglutaric acid (3,3-Dimethylpentanedioate) 是一种甲基支化脂肪酸,是一种人尿中偶见的内源性代谢物。
T8091 trans-4-Hydroxycyclohexanecarboxylic Acid

Others Others
trans-4-Hydroxycyclohexanecarboxylic acid 是一种合成环己烷酸的底物 (substrate)。它是肠道细菌代谢的副产物 (by-product),能够通过尿路排泄。
T4794 Glutaric acid

Endogenous Metabolite Metabolism
Glutaric acid 是一种 C5 二羧酸,是色氨酸和赖氨酸分解代谢途径中的中间体。Glutaric acid 影响周细胞的收缩性和迁移。Glutaric acid 是 I 型戊二酸尿症的生物指标。
TMA0958 Forsythoside F

连翘酯苷F,Arenarioside,三糖苯丙素苷

Xanthine Oxidase Metabolism
Forsythoside F (Arenarioside) 是一种黄嘌呤氧化酶 (xanthine oxidase) 抑制剂,具有抗高尿酸活性。
T4096 Quinolinic acid

喹啉酸,pyridine-2,3-dicarboxylic acid,QUIN

Endogenous Metabolite; NMDAR; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
Quinolinic acid (QUIN) 是一种内源性 N-甲基-D-天冬氨酸 (NMDA) 受体激动剂,由 L-色氨酸通过犬尿氨酸途径合成,具有调节 NMDA 神经元损伤和功能障碍的潜力。
T4816 6-Hydroxynicotinic acid

6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
6-Hydroxynicotinic acid (6-Hydroxypyridine-3-carboxylic acid) 用于核磁共振波谱或气相色谱-质谱法诊断尿路感染中的铜绿假单胞菌。在引起尿液感染的常见细菌中,只有铜绿假单胞菌从烟酸中产生6-羟基烟酸。
T13280 Valerylcarnitine

VALERYL-L-CARNITINE

Endogenous Metabolite Metabolism
Valerylcarnitine (VALERYL-L-CARNITINE) 是一种短链脂肪酸,可用于研究 2 型糖尿病。
T5984 Indole-3-carboxylic acid

3-Indoleformic acid,3-吲哚甲酸

Endogenous Metabolite Metabolism
Indole-3-carboxylic acid (3-Indoleformic acid) 是尿吲哚色氨酸代谢物,在肝病患者中浓度会升高。
T3732 Decanedioic acid

1,10-Decanedioic acid,皮脂酸,Sebacic acid,Sebacinsaure,1,8-Octanedicarboxylic acid

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Decanedioic acid (Sebacinsaure) 是普通尿酸,与肉毒碱-甲酰乙胺转运酶缺乏和中链酰辅酶缺乏症有关。
T4861 trans-Aconitic acid

ATPase; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
trans-Aconitic acid 是反式丙酮酸2-甲基转移酶的底物,存在于正常人尿液中,大量存在于 Reye 综合征和有机酸尿症。
T1362 Hypoxanthine

次黄嘌呤,6-羟基嘌呤,6-Hydroxypurine,Purin-6-ol,Sarcine,Sarkin

Others; Endogenous Metabolite Metabolism; Others
Hypoxanthine (Purin-6-ol),也被称为 purine-6-ol 或 Hyp,是一种天然存在的嘌呤衍生物,是腺苷代谢和核苷酸补救途径形成核酸的反应中间体。在正常情况下,Hypoxanthine 很容易转化为尿酸。Hypoxanthine 首先被氧化为黄嘌呤,黄嘌呤再被黄嘌呤氧化酶氧化为尿酸
T5298 4-hydroxy-3-methylbenzoic acid

4-羟基-3-甲基苯甲酸,4,3-Cresotic acid

Others; Endogenous Metabolite Metabolism; Others
4-hydroxy-3-methylbenzoic acid (4,3-Cresotic acid) 是一种来自健康人群的尿样中鉴定的正常有机酸。
T40426 Cytidine 5'-diphosphate trisodium salt

CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐

Others Others
Cytidine 5'-diphosphate trisodium salt (CDP) 可通过尿苷单磷酸激酶 (UMPK) 催化将磷酸基从 ATP 转移到胞苷一磷酸 (CMP) 生成用于合成 DNA 和 RNA 的胞苷三磷酸。
T5260 2-Methylpentanedioic acid

2-甲基戊二酸,2-Methylglutaric acid,alpha-Methylglutarate

Others; Endogenous Metabolite Metabolism; Others
2-Methylpentanedioic acid (alpha-Methylglutarate) 是一种琥珀酸的代谢产物,它通常存在于人体尿液、健康成人和儿童中。其中琥珀酸是一种柠檬酸循环中间体。
T13851 Pseudolaric Acid C2

Others Others
Pseudolaric Acid C2 是一种从 Pseudolarix kaempferi 二萜酸,是大鼠口服和静脉注射后血浆、尿液、胆汁和粪便中 Pseudolaric acid B 的特异性代谢产物。
T38427 dUTP trisodium

2'-Deoxyuridine-5'-triphosphate trisodium salt,Deoxyuridine triphosphate

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
dUTP trisodium (Deoxyuridine triphosphate) 是在 5'-位具有三磷酸基团的脱氧尿苷磷酸盐,可用于 PCR。
T21665 DL-α-Hydroxyglutaric acid disodium salt

disodium 2-hydroxypentanedioate,DL-Α-羟基戊二酸二钠

Others Others
DL-α-Hydroxyglutaric acid disodium salt (disodium 2-hydroxypentanedioate) 是一种 α-羟基酸,由 (R) -5-oxy-2-tetrahydrofuran 羧酸水解形成,在人类神经代谢疾病 D-α-羟基戊二酸尿症中过量产生。
T21977 p-Cresyl sulfate

Others Others
p-Cresyl Sulfate 是主要的尿毒症毒素,存在于慢性肾病患者的血液,来源于肝脏中酪氨酸和苯丙氨酸的代谢物。
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天然产物

Uric Acid
Cat.No: T0626
Synonym: 尿酸,2,6,8-Trioxopurine,2,6,8-Trioxypurine,2,6,8-Trihydroxypurine,Lithic acid,Urate
Target: Reactive Oxygen Species, Endogenous Metabolite, Phosphorylase
Hyaluronic acid
Cat.No: T3762
Synonym: 透明质酸,Hyaluronate,玻尿酸,hyaluronan
Target: Others, Endogenous Metabolite
Hippuric acid
Cat.No: T4815
Synonym: 尿酸,2-Benzamidoacetic acid,Benzoylglycine
Target: Others, Endogenous Metabolite
4-Aminohippuric Acid
Cat.No: T1436
Synonym: p-Aminohippuric acid,对氨基马尿酸
Target: Amino Acids and Derivatives, Endogenous Metabolite
Xanthurenic Acid
Cat.No: T3010
Synonym: 8-Hydroxykynurenic acid,黄尿酸,4,8-Dihydroxyquinaldic acid,xanthurenate
Target: Apoptosis, Endogenous Metabolite, GluR
7-Chlorokynurenic acid
Cat.No: T10191L
Synonym: 7-chloro-4-hydroxy-2-carboxyquinoline,7-氯犬尿酸,7-CKA
Target: GluR, NMDAR
Salicyluric acid
Cat.No: T5221
Synonym: 2-羟基马尿酸,N-Salicyloylglycine,N-(2-Hydroxybenzoyl)glycine,2-Hydroxy Hippuric Acid
Target: Others, Endogenous Metabolite
2-(2-Methylbenzamido)acetic acid
Cat.No: T5226
Synonym: 2-Methylhippuric acid,2-甲基马尿酸,O-Toluric acid,N-(O-Toluoyl)glycine
Target: Others, Endogenous Metabolite
Uric acid sodium
Cat.No: T41242
Synonym:
Target: Reactive Oxygen Species
Urocanic acid
Cat.No: T4759
Synonym: 4-Imidazoleacrylic acid,尿刊酸
Target: Others, Endogenous Metabolite
(S)-Willardiine
Cat.No: T13456
Synonym: (-)-Willardiine,L-willardiine,Willardiine
Target: iGluR
L-Kynurenine
Cat.No: T4928
Synonym: L-犬尿氨酸,(S)-Kynurenine
Target: AhR, Aryl Hydrocarbon Receptor, Endogenous Metabolite
1,3,7-Trimethyluric acid
Cat.No: T19792
Synonym:
Target: Others
1,3-Dimethyluric acid
Cat.No: T8075
Synonym:
Target: Endogenous Metabolite
Uridine 5'-monophosphate disodium salt
Cat.No: TMA2440
Synonym: 尿苷-5'-单磷酸二钠盐,Disodium UMP,尿苷酸二钠盐,Disodium uridine-5'-monophosphate,5'-UMP disodium salt,Disodium 5'-Uridylate
Target: Others
2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid
Cat.No: T3011
Synonym: Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine,犬尿氨酸
Target: Others, Endogenous Metabolite
Uridine triphosphate
Cat.No: T7711
Synonym: 尿苷5'-三磷酸酯,UTP,Uridine 5'-triphosphate,三磷酸尿苷
Target: Others, Endogenous Metabolite
Uridine 5'-monophosphate
Cat.No: T4718
Synonym: Uridylic acid,尿苷5-单磷酸,UMP,Uridine phosphate,Uridine 5'-phosphoric acid,5'-Uridylic acid
Target: Others, Endogenous Metabolite
Uridine-5'-diphosphate disodium salt
Cat.No: T4706
Synonym: UDP disodium salt,Uridine 5'-diphosphate disodium salt hyd,尿苷-5'-二磷酸二钠盐
Target: DNA/RNA Synthesis, Endogenous Metabolite, P2Y Receptor
1-Methyluric acid
Cat.No: T10020
Synonym: 1-Methyl-2,6,8-trihydroxypurine,1-Methylurate
Target: Endogenous Metabolite
Uridine triphosphate trisodium salt
Cat.No: T8393
Synonym: UTP, Trisodium Salt,Uridine 5'-triphosphate trisodium salt,尿苷-5'-三磷酸三钠盐,Uridine triphosphate (trisodium salt)
Target: Others
2'-Deoxyuridine 5'-monophosphate disodium
Cat.No: T4735
Synonym: 2'-脱氧尿苷-5'-单磷酸二钠,2'-dUMP⋅2Na,2-脱氧尿嘧啶核苷-5'-单磷酸二钠盐,2'-Deoxyuridine 5'-monophosphate disodium salt
Target: Others, Endogenous Metabolite
Uridine 5′-diphosphoglucose disodium salt
Cat.No: T4743
Synonym: 二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal
Target: Endogenous Metabolite, P2Y Receptor
1,3,9-Trimethyluric acid
Cat.No: TN6062
Synonym:
Target:
Uridine 5′-triphosphate tris salt
Cat.No: T4922
Synonym: 尿苷-5′-三磷酸酯 三羟甲基氨基甲烷盐,Uridine 5'-triphosphoric acid
Target: Others, Endogenous Metabolite
Ureidopropionic acid
Cat.No: T4919
Synonym: Carbamoyl-b-alanine,3-酰脲丙酸,3-Ureidopropionic acid
Target: Endogenous Metabolite
Cinnamoylglycine
Cat.No: T10815
Synonym:
Target: Endogenous Metabolite
L-Homocitrulline
Cat.No: T5257
Synonym: 高瓜氨酸,Homo-L-citrulline,Homocitrulline
Target: Others, Endogenous Metabolite
Neoisoastilbin
Cat.No: TN1983
Synonym:
Target: IL Receptor, TNF, NO Synthase
Glutarylcarnitine
Cat.No: T19340
Synonym: O-glutaroyl-L-carnitine
Target: Endogenous Metabolite
Mangiferin
Cat.No: T3012
Synonym: Alpizarin,Chinomin,芒果,Hedysarid
Target: Apoptosis, Others, NF-κB, Nrf2
2-Hydroxy-2-methylbutanoic acid
Cat.No: T5550
Synonym:
Target: Others, Endogenous Metabolite
3,3-Dimethylglutaric acid
Cat.No: T7464
Synonym: 3,3-二甲基戊二酸,3,3-Dimethylpentanedioate
Target: Others, Endogenous Metabolite
trans-4-Hydroxycyclohexanecarboxylic Acid
Cat.No: T8091
Synonym:
Target: Others
Glutaric acid
Cat.No: T4794
Synonym:
Target: Endogenous Metabolite
Forsythoside F
Cat.No: TMA0958
Synonym: 连翘酯苷F,Arenarioside,三糖苯丙素苷
Target: Xanthine Oxidase
Quinolinic acid
Cat.No: T4096
Synonym: 喹啉酸,pyridine-2,3-dicarboxylic acid,QUIN
Target: Endogenous Metabolite, NMDAR, iGluR
6-Hydroxynicotinic acid
Cat.No: T4816
Synonym: 6-Hydroxypyridine-3-carboxylic acid,6-羟基烟酸,2-Hydroxy-5-pyridinecarboxylic acid
Target: Others, Endogenous Metabolite
Valerylcarnitine
Cat.No: T13280
Synonym: VALERYL-L-CARNITINE
Target: Endogenous Metabolite
Indole-3-carboxylic acid
Cat.No: T5984
Synonym: 3-Indoleformic acid,3-吲哚甲酸
Target: Endogenous Metabolite
Decanedioic acid
Cat.No: T3732
Synonym: 1,10-Decanedioic acid,皮脂酸,Sebacic acid,Sebacinsaure,1,8-Octanedicarboxylic acid
Target: HIV Protease, Endogenous Metabolite
trans-Aconitic acid
Cat.No: T4861
Synonym:
Target: ATPase, Endogenous Metabolite
Hypoxanthine
Cat.No: T1362
Synonym: 次黄嘌呤,6-羟基嘌呤,6-Hydroxypurine,Purin-6-ol,Sarcine,Sarkin
Target: Others, Endogenous Metabolite
4-hydroxy-3-methylbenzoic acid
Cat.No: T5298
Synonym: 4-羟基-3-甲基苯甲酸,4,3-Cresotic acid
Target: Others, Endogenous Metabolite
Cytidine 5'-diphosphate trisodium salt
Cat.No: T40426
Synonym: CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐
Target: Others
2-Methylpentanedioic acid
Cat.No: T5260
Synonym: 2-甲基戊二酸,2-Methylglutaric acid,alpha-Methylglutarate
Target: Others, Endogenous Metabolite
Pseudolaric Acid C2
Cat.No: T13851
Synonym:
Target: Others
dUTP trisodium
Cat.No: T38427
Synonym: 2'-Deoxyuridine-5'-triphosphate trisodium salt,Deoxyuridine triphosphate
Target: DNA/RNA Synthesis
DL-α-Hydroxyglutaric acid disodium salt
Cat.No: T21665
Synonym: disodium 2-hydroxypentanedioate,DL-Α-羟基戊二酸二钠
Target: Others
p-Cresyl sulfate
Cat.No: T21977
Synonym:
Target: Others
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