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127

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T9982 PU23

MRP Immunology/Inflammation
PU 23 是一种多药抗性蛋白4(MRP4)的抑制剂。
T11888 LtaS-IN-1

Others; Antibacterial Microbiology/Virology; Others
LtaS-IN-1 是多药耐药粪肠球菌中脂磷壁酸合成的有效抑制剂,可改变细胞壁形态。 LtaS-IN-1 对抗肠球菌属 28 菌株,MIC 值从 0.5 μg/mL 到 64 μg/mL 不等。 LtaS-IN-1 抑制菌株 E1630 和 E1590,MIC 值为 0.5 μg/mL。
T1248 Sulfanitran

磺胺硝苯,乙酰磺胺对硝基苯

Antibacterial; Autophagy Autophagy; Microbiology/Virology
Sulfanitran 是一种用于家禽业的磺胺类抗生素。它也是一种多药耐药蛋白 2 (MRP2) 激动剂,可增加 MRP2 对雌二醇 17-β-D-葡糖醛酸的亲和力。
T8596 Ceefourin 1

MRP Immunology/Inflammation
Ceefourin 1 是一种具有高度选择性的多药抗性蛋白 4 (MRP4) 抑制剂。它能够抑制多种 MRP4 底物的转运,但对其他 ABC 转运蛋白无影响。它是苯并噻唑,常作为高危神经母细胞瘤的化学增敏剂。
T12341 P-gp inhibitor 1

Others; P-gp Membrane transporter/Ion channel; Neuroscience; Others
P-gp inhibitor 1 抑制逆转 P-糖蛋白介导的多药耐药性,EC50 为 57.9 nM(K562/A02 细胞)。
T1631 Sulbactam

CP45899,舒巴坦,舒巴坦酸

Antibacterial; Antibiotic Microbiology/Virology
Sulbactam (CP45899) 是一种竞争性、不可逆的 β-内酰胺酶抑制剂,抑制耐多药不动杆菌-鲍曼不动杆菌复合物。它具有抗菌活性。
T11071 Dofequidar fumarate

MS-209

P-gp Membrane transporter/Ion channel; Neuroscience
Dofequidar fumarate (MS-209) 是口服活性的喹啉化合物,通过抑制 ABCB1/P-gp 和 ABCC1/MDR 相关蛋白 1 来克服 MDR。
T4989 Fosfomycin Tromethamine

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T8426 Encequidar

HM30181,HM30181A

P-gp Membrane transporter/Ion channel; Neuroscience
Encequidar (HM30181A) 是一种选择性 P-糖蛋白抑制剂。
T6685 Sulbactam sodium

舒巴坦钠,CP-45899-2

Antibacterial; Antibiotic Microbiology/Virology
Sulbactam sodium (CP-45899-2) 是一种竞争性、不可逆的 β-内酰胺酶抑制剂。它具有抗菌活性,抑制耐多药不动杆菌-鲍曼不动杆菌复合物。
T16561 Polyoxyethylene stearate

POES,聚氧乙烯硬脂酸酯

Antibacterial; P-gp Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Polyoxyethylene stearate (POES) 是一种非离子乳化剂。
T10460 Batabulin

巴他布林,T138067

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Batabulin (T138067) 是一种抗肿瘤剂,可与 β-微管蛋白同种型的子集共价且选择性地结合,从而破坏微管聚合。它影响细胞形态并导致细胞周期停滞,最终诱导细胞凋亡。
T6287 Tariquidar

XR9576,他立喹达

P-gp Membrane transporter/Ion channel; Neuroscience
Tariquidar (XR9576) 是一种特异性有效的P-糖蛋白抑制剂,Kd 为 5.1 nM。
T0351 Risperidone

Risperidal,R 64 766,利培酮

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂,对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。
T4059 Selamectin

UK-124114,司拉克丁,塞拉菌素

Chloride channel; P-gp; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Selamectin (UK-124114) 是半合成的大环内酯,是一种驱虫剂,可增强线虫中谷氨酸和 GABA 门控氯离子通道的开放。它还是抗寄生虫剂,可激活神经元和咽肌中的谷氨酸门控氯离子通道,以预防恶丝虫,淋巴丝虫和线虫感染。它还是 P-糖蛋白底物和抑制剂,IC50为 120 nM。
T3131 Fosfomycin calcium

Phosphomycin calcium salt,Fosmicin,磷霉素钙

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T13383 Zamicastat

BIA 5-1058

BCRP; Hydroxylase; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Zamicastat (BIA 5-1058) 是多巴胺 β-羟化酶 (DBH) 抑制剂,可透过血脑屏障引起中枢和周边效应,具有降血压作用。它也是一种浓度依赖性的双重 P-gp 和 BCRP 抑制剂,IC50值分别为 73.8 和 17.0 μM。
T8389 Trifluoperazine

三氟拉嗪,trifluoroperazine

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine (trifluoroperazine) 是一种多巴胺 D2 受体抑制剂,可治疗精神分裂症。它是NUPR1抑制剂,具有抗癌活性。它是α1-adrenergic 受体拮抗剂,是流感病毒形态发生的可逆抑制剂。
T11578L Encequidar mesylate

HM30181 mesylate,HM30181A mesylate

P-gp Membrane transporter/Ion channel; Neuroscience
Encequidar mesylate (HM30181A mesylate) 是竞争性有效的 P-糖蛋白抑制剂。
T1634 Glibenclamide

格列本脲,Glyburide

Potassium Channel; Mitochondrial Metabolism; CFTR; P-gp; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
Glibenclamide (Glyburide) 是一种具有口服活性的 ATP 敏感的 K+通道抑制剂,可研究糖尿病和肥胖。它抑制 P-糖蛋白,可直接结合并阻断 KATP 的 SUR1亚基并抑制囊性纤维化跨膜传导调节蛋白。它通过诱导膜离子通透性干扰线粒体生物能,可诱导自噬。
T0100L Atazanavir

Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir (BMS-232632) 是一种高选择性的HIV-1蛋白酶抑制剂,可研究艾滋病毒感染。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 3.49 μM。它是CYP3A4的底物和抑制剂,也是P-糖蛋白的抑制剂和诱导剂。
T20656 Verapamil

NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil (CP-16533-1) 是一种钙通道阻滞剂,是一种口服有效的 P-gp 抑制剂。Verapamil 抑制 CYP3A4,可用于治疗高血压、心律失常和心绞痛的研究。
T16339 Norverapamil hydrochloride

(±)-Norverapamil hydrochloride,D591 hydrochloride,盐酸去甲维拉帕米

Calcium Channel; P-gp; Drug Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
Norverapamil hydrochloride (D591 hydrochloride) 是 Verapamil 的 N-去甲基代谢物,是 L 型钙通道阻滞剂和 P-糖蛋白 (P-gp) 功能抑制剂。
T1010 Verapamil hydrochloride

Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil hydrochloride (Verapamil HCl) 是一种钙通道阻滞剂,是一种可口服的 P 糖蛋白 (P-gp) 抑制剂,可抑制CYP3A4,用于高血压、心律不齐和心绞痛的研究。
T1222 Trifluoperazine dihydrochloride

Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine dihydrochloride (SKF5019) 是一种抗精神病药物,靶向中枢多巴胺受体。它是流感病毒形态发生的可逆抑制剂,是NUPR1抑制剂,具有抗癌活性。它是钙调蛋白抑制剂,还可抑制 P-糖蛋白,可研究精神分裂症。
T0100 Atazanavir sulfate

阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir sulfate (BMS-232632 sulfate) 是一种氮杂肽和 HIV 蛋白酶抑制剂,与其他抗 HIV 药物联合用于治疗 HIV 感染和艾滋病。它也是SARS-CoV 3CLpro 抑制剂,IC50为 3.49 μM。
T2657 Elacridar

GW0918,依克立达,GW120918,GF120918,GG918

BCRP; P-gp Membrane transporter/Ion channel; Neuroscience
Elacridar (GG918) 是一种有效的 P-糖蛋白和BCRP 的抑制剂。
T22330 Fenamic acid

N-苯基邻氨基苯甲酸,2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid

Chloride channel Membrane transporter/Ion channel
Fenamic acid (N-Phenylanthranilic acid) 是氯通道阻滞剂。
T6018 Zosuquidar trihydrochloride

唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride

P-gp Membrane transporter/Ion channel; Neuroscience
Zosuquidar trihydrochloride (LY-335979 trihydrochloride) 是一种P-糖蛋白抑制剂,Ki 值为 59 nM。
T10378 Artelinic acid

Others Others
Artelinic acid, a derivative of Artemisinin, is an antimalarial drug for the treatment of multidrug-resistant strains of Plasmodium falciparum.
T27954 LY-402913

LY 402913,LY402913

MRP Immunology/Inflammation
LY-402913 是一种选择性多药耐药蛋白 (MRP1) 抑制剂。
T9944 3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide

MRP Immunology/Inflammation
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide inhibits multidrug resistance protein (MRP1).
T3581 KS176

Potassium Channel; BCRP Membrane transporter/Ion channel
KS176是选择性高活性乳腺癌耐药蛋白多药转运通道抑制剂,在Pheo A 和Hoechst 检测中,IC50值分别为0.59和1.39 μM。
T60009 YS-370

P-gp Membrane transporter/Ion channel; Neuroscience
YS-370 是一种具有口服活性的 P-gp 抑制剂,对 CYP3A4 有中度抑制作用。 YS-370 有效逆转对紫杉醇和秋水仙碱的多药耐药性,与紫杉醇联合应用表现出更强的抗肿瘤活性。
T22269 Benzyldodecyldimethylammonium Chloride Dihydrate

Antibacterial Microbiology/Virology
Benzyldodecyldimethylammonium chloride dihydrate 可以用作杀虫试剂,可以靶向耐药性细菌,如耐甲氧西林金黄色葡萄球菌、耐多药铜绿假单胞菌等,且具有浓度依赖性。
T15409 GNF179

Parasite Microbiology/Virology
GNF179 是8,8-二甲基 IP 类似物。 它表现出对多药耐药菌株 W2 的效力,具有良好的体外代谢稳定性和体内口服生物相容性。
T5699 SSE15206

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
SSE15206 是一种克服多药耐药性的微管聚合抑制剂,其在 HCT116 细胞中的 GI50值为 197 nM。由于癌细胞中纺锤体形成不完整,导致 G2/M 停滞,有丝分裂异常。
T12343 Benzquinamide

BZQ,P2647,Benzoquinamide

Adrenergic Receptor GPCR/G Protein; Neuroscience
Benzquinamide (P2647) 是一种具有抗癌活性的止吐剂, 抑制p糖蛋白介导的药物外排,增强多重耐药细胞中抗癌药物的细胞毒性。Benzquinamide 对 α2A, α2B, 以及α2C 肾上腺素能受体(α2-AR)的 Ki值分别为 1,365, 691 和 545 nM。
T9830 GSK2556286

GSK286

Antibacterial Microbiology/Virology
GSK2556286 (GSK286) 是一种具有口服活性的结核分枝杆菌 (M. tuberculosis) 抑制剂。GSK2556286 对人巨噬细胞 (macrophages) 生长具有抑制作用,IC50值为 0.07 μM。GSK2556286对多重耐药 (MDR) 或广泛耐药 (XDR) 和药物敏感 (DS) 结核分枝杆菌均有效。
T64133L Laniquidar TFA

Laniquidar TFA(197509-46-9 Free base),R101933

P-gp Membrane transporter/Ion channel; Neuroscience
Laniquidar TFA (R101933) 是一种新型口服非竞争性P-糖蛋白(P-gp)抑制剂,IC50 值为 0.51 μM。Laniquidar的生物利用度有限,可用于调节多药耐药性转运体。Laniquidar可用于研究急性髓性白血病(AML)和骨髓增生异常综合征(MDS)。
T67727 MCT1-IN-3

Monocarboxylate transporter Membrane transporter/Ion channel
MCT1-IN-3是一种单羧酸转运蛋白1 (MCT1)抑制剂。溶质载体(SLC)单羧酸转运蛋白1 (MCT1);SLC16A1)是治疗癌症的一个有希望的靶点。MCT1-IN-3(化合物24)对MCT1转运抑制作用强,IC50值为81.0 nM。MCT1-IN-3对多药转运体ABCB1也有明显的抑制作用。
T3148 MK-571 sodium

L-660711 (sodium salt),L-660711 sodium salt,Verlukast sodium,L-660711,MK571,MK-571 sodium salt,Propanoic acid

Leukotriene Receptor; LTR GPCR/G Protein; Immunology/Inflammation
MK-571 sodium (L-660711 sodium salt) 是一种可口服的选择性白三烯 D4受体拮抗剂,在豚鼠和人肺膜的 Ki 分别为0.22 和 2.1 nM。
T35610 2,5-dimethyl Celecoxib

Apoptosis; Wnt/beta-catenin; Prostaglandin Receptor Apoptosis; Cytoskeletal Signaling; GPCR/G Protein; Immunology/Inflammation; Stem Cells
2,5-dimethyl Celecoxib 是塞来昔布衍生物和微粒体前列腺素 E 合酶 1 (mPGES-1) 的靶向抑制剂,mPGES-1 是炎症介质 PGE2 合成途径中的关键酶。
T24785 S-Fcme

S Fcme,SFcme

S-Fcme is an activator of multidrug resistance transporter that acts by stimulating the multidrug resistance transporter ATPase activity and competing for drug binding.
T33683 NITD-304

NITD304

NITD-304 is an anti-tuberculosis drug candidate for the treatment of multidrug-resistant tuberculosis (MDR-TB), showing effective activity against both MTB drug-sensitive and multidrug-resistant clinical isolates.
T23868 Ceefourin-2

Ceefourin2,Ceefourin 2

Ceefourin-2 is a highly selective multidrug resistance protein 4 inhibitor.
T26417 A 39355

A39355,A-39355

A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.
T70683 NA 382

NA 382 is a staurosporine derivative that inhibits multidrug resistance.
T28173 NIK-250

NIK250

NIK-250 is a P-glycoprotein inhibitor. NIK250 could reverse multidrug resistance in human glioma cells.
T26413 A 30312

A-30312,A30312

A 30312 is a fused indole, which overcomes multidrug resistance in P388/Adr cells in vitro. It potentiates the cytotoxicity of the antitumor drugs Adriamycin, vincristine and vinblastine in multidrug-resistant cells with no effect on drug-sensitive parent P388 cells.

化合物

PU23
Cat.No: T9982
Synonym:
Target: MRP
LtaS-IN-1
Cat.No: T11888
Synonym:
Target: Others, Antibacterial
Sulfanitran
Cat.No: T1248
Synonym: 磺胺硝苯,乙酰磺胺对硝基苯
Target: Antibacterial, Autophagy
Ceefourin 1
Cat.No: T8596
Synonym:
Target: MRP
P-gp inhibitor 1
Cat.No: T12341
Synonym:
Target: Others, P-gp
Sulbactam
Cat.No: T1631
Synonym: CP45899,舒巴坦,舒巴坦酸
Target: Antibacterial, Antibiotic
Dofequidar fumarate
Cat.No: T11071
Synonym: MS-209
Target: P-gp
Fosfomycin Tromethamine
Cat.No: T4989
Synonym:
Target: Antibacterial, Antibiotic
Encequidar
Cat.No: T8426
Synonym: HM30181,HM30181A
Target: P-gp
Sulbactam sodium
Cat.No: T6685
Synonym: 舒巴坦钠,CP-45899-2
Target: Antibacterial, Antibiotic
Polyoxyethylene stearate
Cat.No: T16561
Synonym: POES,聚氧乙烯硬脂酸酯
Target: Antibacterial, P-gp
Batabulin
Cat.No: T10460
Synonym: 巴他布林,T138067
Target: Apoptosis, Microtubule Associated
Tariquidar
Cat.No: T6287
Synonym: XR9576,他立喹达
Target: P-gp
Risperidone
Cat.No: T0351
Synonym: Risperidal,R 64 766,利培酮
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, P-gp
Selamectin
Cat.No: T4059
Synonym: UK-124114,司拉克丁,塞拉菌素
Target: Chloride channel, P-gp, Parasite
Fosfomycin calcium
Cat.No: T3131
Synonym: Phosphomycin calcium salt,Fosmicin,磷霉素钙
Target: Antibacterial, Antibiotic
Zamicastat
Cat.No: T13383
Synonym: BIA 5-1058
Target: BCRP, Hydroxylase, P-gp
Trifluoperazine
Cat.No: T8389
Synonym: 三氟拉嗪,trifluoroperazine
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
Encequidar mesylate
Cat.No: T11578L
Synonym: HM30181 mesylate,HM30181A mesylate
Target: P-gp
Glibenclamide
Cat.No: T1634
Synonym: 格列本脲,Glyburide
Target: Potassium Channel, Mitochondrial Metabolism, CFTR, P-gp, Autophagy
Atazanavir
Cat.No: T0100L
Synonym: Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632
Target: P450, SARS-CoV, HIV Protease, P-gp
Verapamil
Cat.No: T20656
Synonym: NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil
Target: P450, Calcium Channel, P-gp
Norverapamil hydrochloride
Cat.No: T16339
Synonym: (±)-Norverapamil hydrochloride,D591 hydrochloride,盐酸去甲维拉帕米
Target: Calcium Channel, P-gp, Drug Metabolite
Verapamil hydrochloride
Cat.No: T1010
Synonym: Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride
Target: P450, Calcium Channel, P-gp
Trifluoperazine dihydrochloride
Cat.No: T1222
Synonym: Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
Atazanavir sulfate
Cat.No: T0100
Synonym: 阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦
Target: P450, SARS-CoV, HIV Protease, P-gp
Elacridar
Cat.No: T2657
Synonym: GW0918,依克立达,GW120918,GF120918,GG918
Target: BCRP, P-gp
Fenamic acid
Cat.No: T22330
Synonym: N-苯基邻氨基苯甲酸,2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid
Target: Chloride channel
Zosuquidar trihydrochloride
Cat.No: T6018
Synonym: 唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride
Target: P-gp
Artelinic acid
Cat.No: T10378
Synonym:
Target: Others
LY-402913
Cat.No: T27954
Synonym: LY 402913,LY402913
Target: MRP
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide
Cat.No: T9944
Synonym:
Target: MRP
KS176
Cat.No: T3581
Synonym:
Target: Potassium Channel, BCRP
YS-370
Cat.No: T60009
Synonym:
Target: P-gp
Benzyldodecyldimethylammonium Chloride Dihydrate
Cat.No: T22269
Synonym:
Target: Antibacterial
GNF179
Cat.No: T15409
Synonym:
Target: Parasite
SSE15206
Cat.No: T5699
Synonym:
Target: Apoptosis, Microtubule Associated
Benzquinamide
Cat.No: T12343
Synonym: BZQ,P2647,Benzoquinamide
Target: Adrenergic Receptor
GSK2556286
Cat.No: T9830
Synonym: GSK286
Target: Antibacterial
Laniquidar TFA
Cat.No: T64133L
Synonym: Laniquidar TFA(197509-46-9 Free base),R101933
Target: P-gp
MCT1-IN-3
Cat.No: T67727
Synonym:
Target: Monocarboxylate transporter
MK-571 sodium
Cat.No: T3148
Synonym: L-660711 (sodium salt),L-660711 sodium salt,Verlukast sodium,L-660711,MK571,MK-571 sodium salt,Propanoic acid
Target: Leukotriene Receptor, LTR
2,5-dimethyl Celecoxib
Cat.No: T35610
Synonym:
Target: Apoptosis, Wnt/beta-catenin, Prostaglandin Receptor
S-Fcme
Cat.No: T24785
Synonym: S Fcme,SFcme
Target:
NITD-304
Cat.No: T33683
Synonym: NITD304
Target:
Ceefourin-2
Cat.No: T23868
Synonym: Ceefourin2,Ceefourin 2
Target:
A 39355
Cat.No: T26417
Synonym: A39355,A-39355
Target:
NA 382
Cat.No: T70683
Synonym:
Target:
NIK-250
Cat.No: T28173
Synonym: NIK250
Target:
A 30312
Cat.No: T26413
Synonym: A-30312,A30312
Target:
Cat. No. Product Name Target Signaling Pathways
TN1651 Furanodiene

Apoptosis; PARP; Reactive Oxygen Species; Caspase; CDK; P-gp Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Proteases/Proteasome
Furanodiene 是从姜黄中提取的一种萜类天然产物,可抑制外排转运蛋白Pgp 功能并降低 Pgp 蛋白水平。它通过抗血管生成和诱导ROS 产生,DNA 链断裂和细胞凋亡发挥抗癌作用。
T3S0012 coniferyl ferulate

P-gp; GST Membrane transporter/Ion channel; Neuroscience; oxidation-reduction
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。
T2S0223 Isosinensetin

异橙黄酮,6-Demethoxynobiletin

Antioxidant; HIV Protease; Antibacterial; P-gp Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; oxidation-reduction; Proteases/Proteasome
Isosinensetin (6-Demethoxynobiletin) 是从青皮中提取的一种甲氧基黄酮,具有抗氧化和抑制 HIV-1 蛋白酶的活性。
TN4761 Phellamurin

P-gp Membrane transporter/Ion channel; Neuroscience
Phellamurin 是一种来自黄檗叶的黄酮糖苷,可诱导细胞凋亡,具有抗肿瘤活性。它抑制肠道 P-糖蛋白,还抑制凤蝶的产卵。
T3002 Piperine

胡椒碱,1-Piperoylpiperidine,Bioperine

P450; Endogenous Metabolite; P-gp; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
Piperine (Bioperine) 是从胡椒中分离的一种生物碱,可以抑制P-糖蛋白和 CYP3A4 的活性,在HeLa 细胞中的IC50值为61.94±0.054 μg/mL。它已用于研究治疗多发性骨髓瘤和吞咽障碍的试验。
T2S0271 Voacamine

老刺木胺,Voacanginine

Cannabinoid Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Voacamine (Voacanginine) 是非洲马铃果中的一种吲哚生物碱,可抑制多药耐药肿瘤细胞中的 P-糖蛋白作用,具有强效的大麻素 CB1受体拮抗活性。
T1589 D-Cycloserine

RO-1-9213,D-环丝氨酸

Others; Antibacterial; Antibiotic; iGluR Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Others
D-Cycloserine (RO-1-9213) 是一种抗生素,靶向细菌细胞壁肽聚糖生物合成酶。它是一种NMDA 部分激动剂,可以改善认知功能,可研究耐多药结核病。
TJS1159 Chrysosplenetin

猫眼草黄素,Chrysosptertin B

P450; Ferroptosis; P-gp Apoptosis; Membrane transporter/Ion channel; Metabolism; Neuroscience
Chrysosplenetin 是青蒿和其他几种中草药中的一种多甲氧基化黄酮类天然产物,抑制 P-gp 活性并逆转由青蒿素诱导的上调的 P-gp 和 MDR1 水平。
T2S1200 Sinapine

Antioxidant; P-gp; AChE Membrane transporter/Ion channel; Neuroscience; oxidation-reduction
Sinapine 是萝卜中分离出来的一种生物碱,具有抗炎、抗氧化、抗肿瘤、抗血管生成和放射防护作用。它还是乙酰胆碱酯酶抑制剂,可用于研究阿尔茨海默症,共济失调,重症肌无力和帕金森氏病。
T3392 Sinapine thiocyanate

P-gp; AChE Membrane transporter/Ion channel; Neuroscience
Sinapine thiocyanate 是萝卜中分离出来的一种生物碱,具有抗炎、抗氧化、抗肿瘤、抗血管生成和放射防护作用。它还是乙酰胆碱酯酶抑制剂,可用于研究阿尔茨海默症,共济失调,重症肌无力和帕金森氏病。
T4034 Solamargine

Solamargin,δ-Solanigrine,澳洲茄边碱

Apoptosis; p38 MAPK; P-gp; STAT Apoptosis; JAK/STAT signaling; MAPK; Membrane transporter/Ion channel; Neuroscience; Stem Cells
Solamargine (δ-Solanigrine) 是一种来源于茄属植物的类固醇 Solasodine 的衍生物,诱导非选择性细胞毒性和 P-gp 抑制作用。它通过下调 MMP-2 和 MMP-9 的表达和活性来显著抑制 HepG2 细胞的迁移和侵袭,在多种癌症中均表现出抗癌活性。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
TN1757 Hypophyllanthin

叶下珠次素,(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂

Potassium Channel; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Hypophyllanthin 是珠子草中的一种木脂素,能直接抑制 P-gp 的活性,具有很强的抗炎活性。
T2799 (20S)-Protopanaxadiol

20-Epiprotopanaxadiol,20(S)-APPD,20 (S)-原人参二醇,原人参二醇

Apoptosis; Reactive Oxygen Species; P-gp Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) 是人参皂甙的代谢产物,是一种凋亡诱导剂,抑制Akt 活性并诱导多种肿瘤细胞凋亡。
TN1525 Convallatoxin

K-毒毛旋花子配质-3-L-鼠李糖甙,铃兰毒苷

NF-κB; P-gp; PPAR DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Convallatoxin 是从铃兰分离得到的一种强心苷。它是 P-糖蛋白底物,并识别 Val982 是参与其转运的重要氨基酸。它是配体诱导的 MOR 胞吞作用的增强剂,通过激活PPARγ和抑制NF-κB 改善结肠炎,具有抗炎和抗增殖特性。
TCS2336 Evodine

P-gp Membrane transporter/Ion channel; Neuroscience
Evodine 是吴茱萸中的主要柠檬苦素,是P-gp 有效抑制剂,可通过保留抗氧化剂防御系统,针对谷氨酸诱导的毒性具有保护作用。
T19768 γ-Tocotrienol

gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚

Others Others
γ-Tocotrienol (Plastochromanol) 是一种维生素 E 的活性形式。
T4085 Paris saponin VII

重楼皂苷 VII,Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII

Apoptosis; BCL; Others; PARP; p38 MAPK; Akt; Caspase; P-gp; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; MAPK; Membrane transporter/Ion channel; Neuroscience; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Paris saponin VII (Dioscini) 是从延龄草的根和根茎中分离的一种甾体皂苷。它减弱线粒体膜电位,增加凋亡相关蛋白的表达,并降低Bcl-2、caspase-9、caspase-3、PARP-1和p-Akt 的蛋白表达水平。它在 K562/ADR 细胞中诱导强烈的自噬,可研究白血病。
T5757 Loganetin

Antibacterial Microbiology/Virology
Loganetin 是无毒的天然产物,来源于Cornus officinalis Sieb. et Zucc.,可用于耐多药革兰氏阴性菌感染的研究。
T3S2019 Lathyrol

Others Others
Lathyrol 是一种具有抗癌功能的天然产物。
TN1342 8-Epidiosbulbin E acetate

8-表黄药子素E乙酸酯

Anti-infection; Antibacterial Microbiology/Virology
8-Epidiosbulbin E acetate 是从 Dioscorea bulbifera L.中发现的呋喃类化合物,对耐多药细菌具有广谱的质粒治疗活性。
T5A2455 Arenobufagin

沙蟾毒精,沙蟾毒经

Others Others
Arenobufagin 是一种蟾蜍甾烯,从蟾蜍毒液中提取得到,具有抗癌活性。
T6S1842 Tenacissoside G

Tenacissimoside A,通关藤苷G

Others Others
Tenacissoside G 是一种 C21 甾体,来自于Marsdenia tenacissima 茎部。它可逆转 P-糖蛋白过度表达的多药耐药癌细胞的多药耐药。
TN4221 Homoembelin

2,5-dihydroxy-3-nonyl-1,4-benzoquinone

Antibacterial Microbiology/Virology
Homoembelin (2,5-dihydroxy-3-nonyl-1,4-benzoquinone) 是来自 E. ribes 和 C. monocarpus 的色素,具有抗菌效果,可用于耐多药细菌感染的研究。
T6S0095 Genkwanin

7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether,芫花素

Virus Protease Microbiology/Virology
Genkwanin (Apigenin 7-methyl ether) 是一种O-甲基化黄酮,有抗炎活性,通过被动扩散和多药耐药蛋白介导的外排机制转运。
T2S1120 Ganoderenic acid B

P-gp Membrane transporter/Ion channel; Neuroscience
Ganoderenic acid B 是一种从Ganoderma lucidum 中提取的天然产物,可以通过抑制ABCB1的转运功能,增强化疗药物对ABCB1介导的耐多药癌细胞的细胞毒性来发挥作用。
T2S0265 Robinin

NSC 9222,刺槐素

TLR Immunology/Inflammation
Flavone glycoside from Robinia with antibacterial and diuretic properties; derived from kaempferol.The ability of robinin to reverse the multidrug resistance of the human colon cancer cell line Colo 320 expreβing MDR1/LRP was explored by monitoring their uptake of Rhodamine 123, but was shown to have minimal effect. Robinin (NSC-9222) was detected in lysates of the human breast cancer cell line MCF-7 using liquid chromatography-tandem maβ spectrometry.
TN2256 Taccalonolide B

根薯酮内酯B,根薯酮内酯 B

Microtubule Associated Cytoskeletal Signaling
Taccalonolide B 是从广西裂果薯中分离得到的一种微管稳定剂,具有抗肿瘤活性。它抑制 SK-OV-3 细胞的生长,IC50 为 208 nM,在体外对过表达 P-糖蛋白 (Pgp) 和多药耐药蛋白 (MRP7) 的细胞系有效。
T2S0410 Euphorbia factor L1

Euphorbiasteroid,大戟因子L1,大戟因子 L1

Apoptosis; P-gp Apoptosis; Membrane transporter/Ion channel; Neuroscience
Euphorbia factor L1 (Euphorbiasteroid) 可降低 Bcl-2,PI3K,AKT 和 mTOR 蛋白和 mRNA 水平,上调 caspase-9 and caspase-3 蛋白水平。它可诱导自噬,具有抗癌、抗脂肪生成、抗破骨细胞生成和多重耐药调节作用。
T4A2399 Cinobufotalin

华蟾毒它灵,华蟾素

IL Receptor; Akt; MRP; P-gp Cytoskeletal Signaling; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; PI3K/Akt/mTOR signaling
Cinobufotalin 是一种从蟾蜍的皮肤分泌物中提取的强心类固醇或丁二烯内酯。它已被用作强心药,利尿药和止血药,也是潜在的抗肺癌药物。
TN2254 Taccalonolide A

根薯酮内酯A,根薯酮内酯 A

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Taccalonolide A 是从水田七根茎中分离得到的一种类固醇,具有细胞毒性和抗疟活性。它在体外对过表达 p 糖蛋白、多药耐药蛋白 7 细胞系有抑制作用,抑制 SK-OV-3 细胞生长的 IC50值为 622 nM。它是微管稳定剂,能引起 G2-M 期滞留、Bcl-2 磷酸化,并引发细胞凋亡。
T4S1419 (±)-Praeruptorin A

Praeruptorin A,(±)-白花前胡甲素,白花前胡甲素,(-)-Praeruptorin A

p38 MAPK; Calcium Channel; Akt Cytoskeletal Signaling; MAPK; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
(±)-Praeruptorin A 是来自白花前胡的干燥根中的一种主要成分,用于研究伴有厚痰和呼吸困难的咳嗽,非天生性咳嗽和上呼吸道感染。它是顺式-内酯 (CKL) 的二酯化产物,可作为 Ca2+-反流阻滞剂,用于高血压的研究。
T13956 Uvarigrin

Others Others
Uvarigrin induces tumor multidrug resistance cell apoptosis and triggers Caspase-9 activation. Uvarigrin is isolated from the roots of Uvaria calamistrata.
T3S2016 Epoxylathyrol

Others Others
Epoxylathyrol derivatives have modulation of ABCB1-mediated multidrug resistance in human colon adenocarcinoma and mouse T-Lymphoma cells.
TMA0017 Sideroxylin

Antifection Microbiology/Virology
Sideroxylin can synergistically enhance the antimicrobial activity of the alkaloid berberine (also a constituent of H. canadensis) against Staphylococcus aureus by inhibition of the NorA multidrug resistance pump.
TN4962 Scholaricine

Others Others
Scholaricine reverses multidrug resistance in vincristine-resistant KB cells.
TN5114 Taxinine

P-gp Membrane transporter/Ion channel; Neuroscience
Taxinine and Taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells.
TN1522 Combretol

Antifection Microbiology/Virology
Combretol has leishmanicidal activity, it showed moderate activity (growth inhibition 87.3 and 73.0 %, respectively, at 50 μM) against a multidrug-resistant L. tropica line. Combretol also shows weakly active cytotoxic activity.
T23610 Acerinol

Acerinol is an active ingredient from traditional Chinese medicinal herbs. It could be used as a cancer multidrug resistance reversal agent. Acerinol can significantly stimulate the activity of ABCB1 ATPase without affecting the expression of ABCB1 on nei
T12518 Polymyxin B1

硫酸多粘 B1

Others Others
Polymyxin B1 is a potent antimicrobial lipopeptide first derived from Bacilus polymyxa. Polymyxin B1 has the potential for multidrug-resistant Gram-negative bacterial infections treatment.
TN3077 5,5'-Dimethoxylariciresinol 4-O-glucoside

5,5'-二甲氧基落叶松脂素4-O-葡萄糖苷

Others Others
5,5'-Dimethoxylariciresinol-4'-O-beta-D-glucoside is shown to effectively enhance chemosensitivity of resistant cells, which makes it may be a suitable candidate for potential multidrug resistance (MDR)-reversing agents.
TN5113 Taxinine B

Others Others
Taxinine and taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. Taxinine B shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arachidonic acid (AA).
TN1165 (Rac)-Myrislignan

1-(3,4-dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol,rac-myrislignan,ALPHA-[1-[2,6-二甲氧基-4-(2-丙烯-1-基)苯氧基]乙基]-4-羟

Others Others
1-(3,4-Dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol shows anti-staphylococcal activity against a total of five multidrug-resistant (MDR) and methicillin-resistant Staphylococcus aureus strains and the minimum inhibitory concentrations (MIC
T72735 Coleon-U-quinone

Coleon-U-quinone 是一种有效的P-gp 抑制剂。Coleon-U-quinone 能抑制癌细胞活力,能提高多药耐药肿瘤细胞对Doxorubicin 的敏感性。
T83055 Anti-inflammatory agent 57

Anti-inflammatory agent 57(Compound 13),一种天然产自Peucedanum praeruptorum根部的吡喃香豆素,既能逆转多药耐药性(MDR)又具备抗炎效果。
T79943 6-C-Methylquercetin-3,4'-dimethyl ether

Antibiotic Microbiology/Virology
6-C-Methylquercetin-3,4'-dimethyl etheris 是一种黄酮醇衍生物,提取自Bauhinia thonningii Schum叶。本化合物对多重耐药的革兰氏阴性细菌及耐甲氧西林金黄色葡萄球菌(MRSA)表现出抗菌活性。
T36815 Chevalone C

Chevalone C is a meroterpenoid fungal metabolite originally isolated from E. chevalieri. It is active against M. tuberculosis H37Ra (MIC = 6.3 μg/ml) and is cytotoxic to BC1 human breast cancer cells (IC50 = 8.7 μg/ml). Chevalone C inhibits the growth of multidrug-resistant isolates of E. coli, S. aureus, and E. faecium in a disc diffusion assay when used at a concentration of 15 μg/disc. It also induces cell death in HCT116 colorectal carcinoma cells.
T72737 Ganoderic acid R

Ganoderic acid R为一种高效的抗癌化合物,通过促进肿瘤细胞系的凋亡(apoptosis)机制来抑制其生长。它对多药耐药(MDR)肿瘤细胞系(KB-A-1/Dox)及敏感肿瘤细胞系(KB-A-1)展现出显著的细胞毒性效应。
T35754 Aszonapyrone A

Aszonapyrone A is a meroditerpene fungal metabolite that has been found in Neosartorya and has diverse biological activities.1,2,3 It inhibits the growth of MCF-7, NCI H460, and A375-C5 cancer cells (GI50s = 13.6, 11.6, and 10.2 μM, respectively).1 Aszonapyrone A is active against multidrug-resistant isolates of S. aureus, E. faecalis, and E. faecium (MICs = 8, 16, and 16 μg/ml, respectively) and inhibits S. aureus biofilm formation.2 It is also active against P. falciparum in vitro (IC50 = 1.34...
T15097 Deoxynivalenol

Vomitoxin,4-Deoxynivalenol

Deoxynivalenol (Vomitoxin) 是一种单端孢菌素家族镰刀菌属产生的霉菌毒素,常见于受到污染的食物和饲料中。Deoxynivalenol 通过紧密连接处的细胞旁路来穿过肠粘膜。Deoxynivalenol 转运不受P-糖蛋白 (PgP) 或多药耐药相关蛋白 (MRP) 抑制剂的影响。Deoxynivalenol 通常会导致人类和动物腹泻、呕吐和胃肠道炎症。
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天然产物

Furanodiene
Cat.No: TN1651
Synonym:
Target: Apoptosis, PARP, Reactive Oxygen Species, Caspase, CDK, P-gp
coniferyl ferulate
Cat.No: T3S0012
Synonym:
Target: P-gp, GST
Isosinensetin
Cat.No: T2S0223
Synonym: 异橙黄酮,6-Demethoxynobiletin
Target: Antioxidant, HIV Protease, Antibacterial, P-gp
Phellamurin
Cat.No: TN4761
Synonym:
Target: P-gp
Piperine
Cat.No: T3002
Synonym: 胡椒碱,1-Piperoylpiperidine,Bioperine
Target: P450, Endogenous Metabolite, P-gp, Autophagy
Voacamine
Cat.No: T2S0271
Synonym: 老刺木胺,Voacanginine
Target: Cannabinoid Receptor, P-gp
D-Cycloserine
Cat.No: T1589
Synonym: RO-1-9213,D-环丝氨酸
Target: Others, Antibacterial, Antibiotic, iGluR
Chrysosplenetin
Cat.No: TJS1159
Synonym: 猫眼草黄素,Chrysosptertin B
Target: P450, Ferroptosis, P-gp
Sinapine
Cat.No: T2S1200
Synonym:
Target: Antioxidant, P-gp, AChE
Sinapine thiocyanate
Cat.No: T3392
Synonym:
Target: P-gp, AChE
Solamargine
Cat.No: T4034
Synonym: Solamargin,δ-Solanigrine,澳洲茄边碱
Target: Apoptosis, p38 MAPK, P-gp, STAT
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Hypophyllanthin
Cat.No: TN1757
Synonym: 叶下珠次素,(7S,8S,9R)-9-(3,4-二甲氧基苯基)-6,7,8,9-四氢-4-甲氧基-7,8-双(甲氧基甲基)萘并[1,2-D]-1,3-二恶茂
Target: Potassium Channel, Calcium Channel, P-gp
(20S)-Protopanaxadiol
Cat.No: T2799
Synonym: 20-Epiprotopanaxadiol,20(S)-APPD,20 (S)-原人参二醇,原人参二醇
Target: Apoptosis, Reactive Oxygen Species, P-gp
Convallatoxin
Cat.No: TN1525
Synonym: K-毒毛旋花子配质-3-L-鼠李糖甙,铃兰毒苷
Target: NF-κB, P-gp, PPAR
Evodine
Cat.No: TCS2336
Synonym:
Target: P-gp
γ-Tocotrienol
Cat.No: T19768
Synonym: gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚
Target: Others
Paris saponin VII
Cat.No: T4085
Synonym: 重楼皂苷 VII,Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII
Target: Apoptosis, BCL, Others, PARP, p38 MAPK, Akt, Caspase, P-gp, Autophagy
Loganetin
Cat.No: T5757
Synonym:
Target: Antibacterial
Lathyrol
Cat.No: T3S2019
Synonym:
Target: Others
8-Epidiosbulbin E acetate
Cat.No: TN1342
Synonym: 8-表黄药子素E乙酸酯
Target: Anti-infection, Antibacterial
Arenobufagin
Cat.No: T5A2455
Synonym: 沙蟾毒精,沙蟾毒经
Target: Others
Tenacissoside G
Cat.No: T6S1842
Synonym: Tenacissimoside A,通关藤苷G
Target: Others
Homoembelin
Cat.No: TN4221
Synonym: 2,5-dihydroxy-3-nonyl-1,4-benzoquinone
Target: Antibacterial
Genkwanin
Cat.No: T6S0095
Synonym: 7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether,芫花素
Target: Virus Protease
Ganoderenic acid B
Cat.No: T2S1120
Synonym:
Target: P-gp
Robinin
Cat.No: T2S0265
Synonym: NSC 9222,刺槐素
Target: TLR
Taccalonolide B
Cat.No: TN2256
Synonym: 根薯酮内酯B,根薯酮内酯 B
Target: Microtubule Associated
Euphorbia factor L1
Cat.No: T2S0410
Synonym: Euphorbiasteroid,大戟因子L1,大戟因子 L1
Target: Apoptosis, P-gp
Cinobufotalin
Cat.No: T4A2399
Synonym: 华蟾毒它灵,华蟾素
Target: IL Receptor, Akt, MRP, P-gp
Taccalonolide A
Cat.No: TN2254
Synonym: 根薯酮内酯A,根薯酮内酯 A
Target: Apoptosis, Microtubule Associated
(±)-Praeruptorin A
Cat.No: T4S1419
Synonym: Praeruptorin A,(±)-白花前胡甲素,白花前胡甲素,(-)-Praeruptorin A
Target: p38 MAPK, Calcium Channel, Akt
Uvarigrin
Cat.No: T13956
Synonym:
Target: Others
Epoxylathyrol
Cat.No: T3S2016
Synonym:
Target: Others
Sideroxylin
Cat.No: TMA0017
Synonym:
Target: Antifection
Scholaricine
Cat.No: TN4962
Synonym:
Target: Others
Taxinine
Cat.No: TN5114
Synonym:
Target: P-gp
Combretol
Cat.No: TN1522
Synonym:
Target: Antifection
Acerinol
Cat.No: T23610
Synonym:
Target:
Polymyxin B1
Cat.No: T12518
Synonym: 硫酸多粘 B1
Target: Others
5,5'-Dimethoxylariciresinol 4-O-glucoside
Cat.No: TN3077
Synonym: 5,5'-二甲氧基落叶松脂素4-O-葡萄糖苷
Target: Others
Taxinine B
Cat.No: TN5113
Synonym:
Target: Others
(Rac)-Myrislignan
Cat.No: TN1165
Synonym: 1-(3,4-dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol,rac-myrislignan,ALPHA-[1-[2,6-二甲氧基-4-(2-丙烯-1-基)苯氧基]乙基]-4-羟
Target: Others
Coleon-U-quinone
Cat.No: T72735
Synonym:
Target:
Anti-inflammatory agent 57
Cat.No: T83055
Synonym:
Target:
6-C-Methylquercetin-3,4'-dimethyl ether
Cat.No: T79943
Synonym:
Target: Antibiotic
Chevalone C
Cat.No: T36815
Synonym:
Target:
Ganoderic acid R
Cat.No: T72737
Synonym:
Target:
Aszonapyrone A
Cat.No: T35754
Synonym:
Target:
Deoxynivalenol
Cat.No: T15097
Synonym: Vomitoxin,4-Deoxynivalenol
Target:
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