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Search Results for " antiallergic "

36

抑制剂 & 化合物

24

天然产物

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Cat. No. Product Name Target Signaling Pathways
T63825 Antiallergic agent-1

Antiallergic agent-1 是 Src 家族激酶抑制剂,是一种新的有价值的先导化合物,具有作为抗过敏剂的潜力。
T3979 Emedastine

LY188695,依美斯汀,Emadine

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Emedastine (LY188695) 是一种可口服的,选择性和高亲和力的组胺 H1受体拮抗剂,Ki 值为 1.3 nM。它是苯并咪唑衍生物,可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T6426 Buclizine dihydrochloride

盐酸安其敏,Longifene,Buclina,Buclizine HCl,UCB-4445

5-HT Receptor; AChR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Buclizine dihydrochloride (Buclina) 是可口服的一种哌嗪组胺 H1 受体拮抗剂,主要具有止吐和抗眩晕活性。
T2335 Ebastine

Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ebastine (Kestine) 是一种可口服的组胺 H1 受体拮抗剂,用于过敏性鼻炎的症状和慢性特发性荨麻疹的研究。
T6488 Epinastine hydrochloride

Alesion,Epinastine HCl,WAL-801CL HCl,依匹斯汀盐酸盐,Elestat

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Epinastine hydrochloride (WAL-801CL HCl) 是抗组胺剂和肥大细胞稳定剂,是一种可口服的选择性组胺 H1 受体拮抗剂,可抑制 IL-8 释放,具有抗过敏作用。
T67953 Elbanizine

Others Others
Elbanizine 显示出抗过敏、抗哮喘、抗组胺和解痉的活性。
T4566 Lodoxamide

Lodoxamidum,洛草氨酸

GPR; Histamine Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Lodoxamide (Lodoxamidum) 是一种抗过敏药物,作为肥大细胞稳定剂,对治疗哮喘和过敏性结膜炎有效。
T1425 Pemirolast potassium

BMY 26517,TWT-8152,吡嘧司特钾

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pemirolast potassium (TWT-8152) 是 H1组胺受体拮抗剂和肥大细胞稳定剂,是一种具有抗过敏特性的嘧啶酮衍生物。
T14326 AS-35

Others Others
AS-35 is an orally effective, potent and selective antagonist of leukotrienes, antagonizes LTC4-, LTD4 and LTE4-induced contractions of the ileum. With IC50 values of 8 nM, 4 nM and 3 nM, respectively. It has antiallergic activities.
T68128 Picumast

Picumast 是一种具有抗过敏活性,可被用于治疗哮喘,可能用于治疗治疗过敏性气道疾病。
T2270 Trans-Tranilast

Tranilast trans-,反式-曲尼司特,反-曲尼司特

RAAS Endocrinology/Hormones
Trans-Tranilast 是抗过敏剂,可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T2690 Tranilast

曲尼司特,MK 341,SB 252218

RAAS; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
Tranilast (SB 252218) 是一种抗过敏药物,可抑制炎症细胞释放脂质介质和细胞因子,抑制前列腺素 D2 (PGD2)产生,IC50为 0.1 mM。它拮抗血管紧张素 II 并抑制其在血管平滑肌细胞中的生物学作用,具有抗炎和免疫调节作用。
T67959 Pirodomast

Thrombin; Serine Protease Proteases/Proteasome
Pirodomast 是血栓素 A(TXA2)合成酶抑制剂。Pirodomast 能抑制白三烯(LT)D4、C4、E4 的形成和血栓素 B2(TXB2)的活性,但对组胺、甲氧胆碱、血清素、LTC4 或血小板活化因子诱导的豚鼠支气管痉挛的拮抗作用较弱或无效。Pirodomast 在体外对豚鼠气管只有微弱的松弛活性。Pirodomast 是一种潜在的抗过敏化合物,在体外可抑制胰蛋白酶的蛋白水解活性,在体内可阻止抗原诱发过敏绵羊的即时和晚期哮喘反应,抑制抗原诱导的过敏绵羊对组胺和卡巴胆碱的气道高反应性。
T9084 Cetirizine Impurity B dihydrochloride

De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride,西替利嗪杂质B二盐酸盐,西替利嗪杂质04

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) 是 Cetirizine dihydrochloride 的杂质。Cetirizine 是一种抗组胺剂,是口服有活力的、特异性 H1受体拮抗剂。它能够抑制过敏反应期间嗜酸性粒细胞趋化,可以标记抗过敏特性。
T1278 Astemizole

Laridal,Histaminos,Paralergin,阿司咪唑

Potassium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。
T1666 Fludrocortisone acetate

9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate

Glucocorticoid Receptor; Autophagy Autophagy; Endocrinology/Hormones
Fludrocortisone acetate (9α-Fludrocortisone acetate) 是一种合成的盐皮质激素,可减少尿液中钠丢失量,也用于增加血压,有用于阿狄森氏病的研究潜力。
T19839 Oxatomide

Oxatomida

P2X Receptor; Calcium Channel; 5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Oxatomide (Oxatomida) 是一种有效且具有口服活性的双重 H1 组胺受体 和 P2X7 受体双重拮抗剂,具有抗组胺和抗过敏活性。Oxatomide 可用于阻断人 P2X7 受体中 ATP 诱导的电流 ,IC50 为 0.95 μM。Oxatomide 对 ATP 诱导的 Ca2+ 内流具有抑制作用,IC50 值为 0.43 μM。Oxatomide 对 5-羟色胺具有抑制作用。Oxatomide可用于治疗免疫系统疾病和研究超敏反应。
T23679 AHR-13268D

AHR 13268D,AHR13268D

AHR-13268D is a new agent of antiallergic/antihistaminic.
T25648 LC 6

LC-6,LC6

LC 6 is an orally active antiallergic agent.
T25413 Fenethazine

RP 3015,Lisergan,Phenetazine,RP-3015,Ethysene

Fenethazine is an effective antihistamine used as an antiallergic drug.
T25547 Isospaglumate sodium

Isospaglumate trisodium,Sodium isospaglumate

Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.
T68927 AY 25674

AY 25674 is a drug with antiallergic properties which has been shown to inhibit passive anaphylaxis in rat.
T15666 KP136

AL136

Others Others
KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).
T71540 CI 959

CI 959 is a novel antiallergic compound which is a potent inhibitor of receptor-mediated histamine release from human basophils. It inhibits thromboxanes.
T31191 Dagapamil hydrochloride

Dagapamil hydrochloride 是一种钙通道阻滞剂。Dagapamil hydrochloride 在动物模型中具有降压、抗心律失常、心脏保护、抗过敏和抑制血小板聚集的作用。
T13144 Thiazinamium chloride

Multergan chloride

Others Others
Thiazinamium chloride possesses potent anticholinergic and antiallergic activity and inhibits synthesis of TxB2(IC50 value of 0.2 µM).
T26523 Abroquinone A

Abroquinone A, a natural isoflavanquinone, has been shown to block cytosolic phospholipase A(2) and 5-lipoxygenase activation in neutrophils, it may have pharmaceutical potential as an antiallergic agent.
T40430 Cetirizine Impurity D

Cetirizine Impurity D is an impurity of Cetirizine. Cetirizine is a second-generation antihistamine that acts as a specific, orally active, and long-acting antagonist of the histamine H1-receptor. Cetirizine exhibits antiallergic properties and inhibits eosinophil chemotaxis in response to allergies.
T83201 Acetyl heptapeptide-4

Acetyl heptapeptide-4,一种抗过敏(antiallergic)生物活性肽,已报道作为化妆品成分使用。
T62421 Buclizine

Buclizine 是一种口服具有活力的抗组胺、抗过敏化合物。Buclizine 也是一种大鼠的强致畸剂,表现出抗肿瘤作用。
T31191L Dagapamil

Dagapamilum

Dagapamil 是一种钙通道阻滞剂。Dagapamil 在动物模型中具有降压、抗心律失常、心脏保护、抗过敏和抑制血小板聚集的作用。
T63394 MrgprX2 antagonist-6

MrgprX2 antagonist-6 是一种高效抗过敏剂,对肥大细胞脱颗粒具有抑制作用。
T60289 Pemirolast

Pemirolast 是一种具有口服活性的抗过敏剂。Pemirolast 通过抑制感觉神经肽的释放来减轻紫杉醇超敏反应,可用于对支气管哮喘和结膜炎的研究。
T60366 Epinastine

Epinastine (WAL801) 是一种抗组胺剂和肥大细胞稳定剂。Epinastine 是一种有效的,选择性的,口服活性的组胺 H1 受体 (histamine H1 receptor) 拮抗剂。Epinastine 还抑制人嗜酸性粒细胞释放 IL-8 并具有抗过敏作用。
T70904 Tylogenin

Tylogenin, a steroidal aglycone generated by acid hydrolysis from two seasonal glycosides occurring in Tylophora sylvatica, inhibits IgE-induced basophil mediator release for allergic reactions. In the rabbit basophil-dependent serotonin release (BDSR) assay system, the inhibitory activity of tylogenin was significantly greater than that of its parent glycosides, tylophoroside and acetyltylophoroside, and that of dexamethasone. The activity of tylogenin was found to increase with the incubation ...
T73665 Bufrolin

Bufrolin,作为Cromoglycate(组胺释放抑制剂)的类似物,是一种高效的GPR35激动剂,能够促进β-arrestin-2与人GPR35a或大鼠GPR35之间的相互作用。此外,Bufrolin亦可作为抗过敏性肥大细胞稳定剂,有效抑制内化肽诱导的抗炎反应,并且在内化肽连接药剂的药物递送研究中,被作为抗炎剂使用。

化合物

Antiallergic agent-1
Cat.No: T63825
Synonym:
Target:
Emedastine
Cat.No: T3979
Synonym: LY188695,依美斯汀,Emadine
Target: Histamine Receptor
Buclizine dihydrochloride
Cat.No: T6426
Synonym: 盐酸安其敏,Longifene,Buclina,Buclizine HCl,UCB-4445
Target: 5-HT Receptor, AChR, Histamine Receptor
Ebastine
Cat.No: T2335
Synonym: Ebastel,依巴斯汀,LAS-W 090,Ebastin,Kestine,RP64305
Target: Histamine Receptor
Epinastine hydrochloride
Cat.No: T6488
Synonym: Alesion,Epinastine HCl,WAL-801CL HCl,依匹斯汀盐酸盐,Elestat
Target: 5-HT Receptor, Histamine Receptor
Elbanizine
Cat.No: T67953
Synonym:
Target: Others
Lodoxamide
Cat.No: T4566
Synonym: Lodoxamidum,洛草氨酸
Target: GPR, Histamine Receptor
Pemirolast potassium
Cat.No: T1425
Synonym: BMY 26517,TWT-8152,吡嘧司特钾
Target: Histamine Receptor
AS-35
Cat.No: T14326
Synonym:
Target: Others
Picumast
Cat.No: T68128
Synonym:
Target:
Trans-Tranilast
Cat.No: T2270
Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特
Target: RAAS
Tranilast
Cat.No: T2690
Synonym: 曲尼司特,MK 341,SB 252218
Target: RAAS, Prostaglandin Receptor
Pirodomast
Cat.No: T67959
Synonym:
Target: Thrombin, Serine Protease
Cetirizine Impurity B dihydrochloride
Cat.No: T9084
Synonym: De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride,西替利嗪杂质B二盐酸盐,西替利嗪杂质04
Target: Histamine Receptor
Astemizole
Cat.No: T1278
Synonym: Laridal,Histaminos,Paralergin,阿司咪唑
Target: Potassium Channel, Histamine Receptor
Fludrocortisone acetate
Cat.No: T1666
Synonym: 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate
Target: Glucocorticoid Receptor, Autophagy
Oxatomide
Cat.No: T19839
Synonym: Oxatomida
Target: P2X Receptor, Calcium Channel, 5-HT Receptor, Histamine Receptor
AHR-13268D
Cat.No: T23679
Synonym: AHR 13268D,AHR13268D
Target:
LC 6
Cat.No: T25648
Synonym: LC-6,LC6
Target:
Fenethazine
Cat.No: T25413
Synonym: RP 3015,Lisergan,Phenetazine,RP-3015,Ethysene
Target:
Isospaglumate sodium
Cat.No: T25547
Synonym: Isospaglumate trisodium,Sodium isospaglumate
Target:
AY 25674
Cat.No: T68927
Synonym:
Target:
KP136
Cat.No: T15666
Synonym: AL136
Target: Others
CI 959
Cat.No: T71540
Synonym:
Target:
Dagapamil hydrochloride
Cat.No: T31191
Synonym:
Target:
Thiazinamium chloride
Cat.No: T13144
Synonym: Multergan chloride
Target: Others
Abroquinone A
Cat.No: T26523
Synonym:
Target:
Cetirizine Impurity D
Cat.No: T40430
Synonym:
Target:
Acetyl heptapeptide-4
Cat.No: T83201
Synonym:
Target:
Buclizine
Cat.No: T62421
Synonym:
Target:
Dagapamil
Cat.No: T31191L
Synonym: Dagapamilum
Target:
MrgprX2 antagonist-6
Cat.No: T63394
Synonym:
Target:
Pemirolast
Cat.No: T60289
Synonym:
Target:
Epinastine
Cat.No: T60366
Synonym:
Target:
Tylogenin
Cat.No: T70904
Synonym:
Target:
Bufrolin
Cat.No: T73665
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3254 PHYTOL

植醇,trans-Phytol,(E)-Phytol

Antibacterial; PPAR; Parasite DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
PHYTOL (trans-Phytol) 是一种从叶绿素中提取的二萜醇,广泛应用于食品添加剂和医药领域,具有很好的抗血吸虫特性。它具有抗伤害、抗氧化、抗炎、抗过敏等作用。它对结核分枝杆菌和金黄色葡萄球菌具有抗菌活性。
TN1712 Gossypin

NF-κB; S6 Kinase MAPK; NF-κB; PI3K/Akt/mTOR signaling
Gossypin 是一种从Hibiscus vitifolius 中分离得到的黄酮,能够抑制NF-κB 和 NF-κB 的调节基因表达。在小鼠原代骨髓细胞和 RAW264.7 细胞中,它也可抑制 RANKL 诱导的破骨细胞形成。它具有抗氧化、抗炎、抗癌、抗衰老、抗糖尿病和保护肝脏的活性。
T3776 Rhapontigenin

丹叶大黄素,Protigenin

P450; Antibacterial; Antifungal Metabolism; Microbiology/Virology
Rhapontigenin (Protigenin) 是一种基于机制的选择性细胞色素 P450 1A1 (IC50: 400 nM) 灭活剂。它是一种芳烃羟化酶,可激活作为致癌物质的多环芳烃。它是白藜芦醇的天然类似物,具有抗癌,抗氧化剂,抗真菌和抗菌活性。
T5S2360 Corydaline

Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline

P450; Virus Protease; Opioid Receptor; AChE Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Corydaline (Corydalin) 是从 Corydalis yanhusuo 提取的一种异喹啉生物碱,是一种新型促动力植物药的主要活性成分之一。它促进胃排空和小肠转运,促进胃的调节,具有抗乙酰胆碱酯酶、抗过敏和镇痛活性。
T1035 Hesperidin

橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷

Apoptosis; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Hesperidin (Cirantin) 是一种广泛存在于柑橘类水果中黄烷酮糖苷,具有减少炎症介质并发挥重要的抗氧化作用,还有抗肿瘤和抗过敏活性。
TWO2771 2-Adamantanol

2-金刚烷醇,Adamantan-2-Ol,2-Hydroxyadamantane

Others Others
2-Adamantanol (2-Hydroxyadamantane) 用于合成抗过敏药物Mizolastine。
T3S2027 Rubusoside

Others Others
Rubusoside 是天然的增溶剂及甜味剂,具有良好的抗血管新生和抗过敏药的特性。
T2891 Ammonium glycyrrhizinate

Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,甘草酸单胺,Monoammonium glycyrrhizinate hydrate,Glycyrram

Others Others
Ammonium glycyrrhizinate (Glycyrram) 具有抗炎、抗胃溃疡、抗过敏、抗肝炎等药理功能。
TN1136 Procyanidin A1

原花青素 A1,Proanthocyanidin A1,原花色素A1

LDL; Calcium Channel; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism
Procyanidin A1 (Proanthocyanidin A1) 是一种原花青素二聚体,具有抗过敏作用,可抑制蛋白激酶 C 激活下游脱粒或 RBL-213 细胞内部储存的 Ca2+流入。
T1027 Luteolin

木犀草素,Luteolol,Flacitran,Digitoflavone,Luteoline

Apoptosis; Nrf2; Endogenous Metabolite; PDE; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism
Luteolin (Luteolol) 属于黄酮类天然产物,是一种 Nrf2 抑制剂、PDE 抑制剂。Luteolin 具有多种生物活性,包括抗肿瘤、抗氧化、抗炎、抗菌、抗病毒、抗过敏和促凝血等。
TN2429 Capsiate

Antioxidant; TRP/TRPV Channel Membrane transporter/Ion channel; oxidation-reduction
Capsiate 是一种具有口服活性的 TRPV1 激动剂,是非刺激性辣椒素类似物,可作为抗过敏剂,具有抗炎、抗氧、降糖和抑制血管生成活性。
T0795 Rutin

Quercetin 3-O-rutinoside,芦丁,Rutoside

Beta Amyloid; Prostaglandin Receptor; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rutin (Quercetin 3-O-rutinoside) 是槐果实中的一种黄酮类天然产物,具有抗炎、降糖、抗氧化、神经保护、肾脏保护、肝脏保护和降低Aβ低聚物活性等多种生物活性。它能穿过血脑屏障,通过抑制细胞凋亡、线粒体功能紊乱和氧化应激抑制万古霉素诱导的肾小管细胞凋亡。
T3S0195 Nootkatone

诺卡酮,努特卡酮,诺卡酮

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Nootkatone 是一种神经保护剂,来自于Alpiniae OxyphyllaeFructus ,具有抗氧化和抗炎活性。它能够改善脂多糖诱导的阿尔茨海默氏病小鼠模型的认知障碍。
T2S2173 (E)-Naringenin chalcone

Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮

Others Others
Naringenin chalcone (Isosalipurpol) 是一种黄酮醇生物合成的中间体,在查耳酮异构酶的作用下,自发代谢成柚皮素。它具有抗炎和抗过敏活性。
TMA0955 Thunberginol C

Antifection Microbiology/Virology
Thunberginol C exhibits antimicrobial activity against oral bacteria. It shows antiallergic activity in the in vitro bioassay using the Schults-Dale reaction in sensitized guinea pig bronchial muscle.
T82563 Dichotomine H

Dichotomine H,一种从银柴胡 (Stellaria dichotoma L.) 提取的 p-咔啉生物碱,具有显著的抗过敏活性。
TN2155 Rhodiocyanoside A

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP IgE and inhibits the PCA reaction in rats.
T82250 Gymconopin C

Gymconopin C 在小鼠耳部被动皮肤过敏模型中显示出抗过敏活性。
TMA0627 Taxiresinol

TNF Apoptosis
Taxiresinol shows anticancer, antinociceptive, and antiallergic activities, it shows inhibitory activity on induced histamine release from the human basophilic cell line, KU812. Taxiresinol can protect the hepatocytes from apoptosis via an inhibition of TNF- alpha production by activated macrophages and a direct inhibition of apoptosis induced by TNF- alpha in D-GalN/LPS-treated mice.
TN1009 Epimagnolin B

NF-κB; NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; NF-κB
Epimagnolin B 是一种双环氧木质素,分离自木兰中。它能够抑制 LPS 激活的小胶质细胞中 NO 的产生。它具有抗过敏以及抗炎作用。
TN3614 Cearoin

檀木

ERK; BCL; PARP; IκB/IKK; TNF; NF-κB; ROS; Caspase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; MAPK; NF-κB; Proteases/Proteasome
Cearoin has anti-inflammatory, and antiallergic activities, it can markedly inhibit inflammatory responses including LPS-induced NO production by suppressing the expression of iNOS mRNA and LPS-induced mRNA expression of TNFα and CCL2. Cearoin induces aut
TN5164 trans-Hinokiresinol

IL Receptor; TNF; NOS; LTR Apoptosis; Immunology/Inflammation
Hinokiresinol is a novel inhibitor of LTB4 binding to the human neutrophils, it has antiallergic effect, it inhibits IgE-induced mouse passive cutaneous anaphylaxis reaction. Hinokiresinol (trans-hinokiresinol) and nyasol (cis-hinokiresinol) are estrogen
T82248 Gymnoside I

Gymnoside I(化合物1)是糖苷氧基苄基2-异丁基苹果酸,其在小鼠被动皮肤过敏反应(PCA)实验中展现出抗过敏效能。该化合物有望在哮喘、神经衰弱和慢性肝炎治疗研究中应用。
T8291 2-Carene

Others Others
2-Carene 是一种天然存在的双环单萜,存在于许多精油中,如松树、雪松和柏树。它被发现具有抗炎、抗真菌和抗菌活性,以及抗氧化、抗肿瘤和抗过敏活性,还有神经保护、心脏保护和肝脏保护作用。

天然产物

PHYTOL
Cat.No: T3254
Synonym: 植醇,trans-Phytol,(E)-Phytol
Target: Antibacterial, PPAR, Parasite
Gossypin
Cat.No: TN1712
Synonym:
Target: NF-κB, S6 Kinase
Rhapontigenin
Cat.No: T3776
Synonym: 丹叶大黄素,Protigenin
Target: P450, Antibacterial, Antifungal
Corydaline
Cat.No: T5S2360
Synonym: Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline
Target: P450, Virus Protease, Opioid Receptor, AChE
Hesperidin
Cat.No: T1035
Synonym: 橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷
Target: Apoptosis, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
2-Adamantanol
Cat.No: TWO2771
Synonym: 2-金刚烷醇,Adamantan-2-Ol,2-Hydroxyadamantane
Target: Others
Rubusoside
Cat.No: T3S2027
Synonym:
Target: Others
Ammonium glycyrrhizinate
Cat.No: T2891
Synonym: Glycamil,Monoammonium glycyrrhizinate,Ammonium Glycyrrhizate,甘草酸单胺,Monoammonium glycyrrhizinate hydrate,Glycyrram
Target: Others
Procyanidin A1
Cat.No: TN1136
Synonym: 原花青素 A1,Proanthocyanidin A1,原花色素A1
Target: LDL, Calcium Channel, PKC
Luteolin
Cat.No: T1027
Synonym: 木犀草素,Luteolol,Flacitran,Digitoflavone,Luteoline
Target: Apoptosis, Nrf2, Endogenous Metabolite, PDE, Autophagy
Capsiate
Cat.No: TN2429
Synonym:
Target: Antioxidant, TRP/TRPV Channel
Rutin
Cat.No: T0795
Synonym: Quercetin 3-O-rutinoside,芦丁,Rutoside
Target: Beta Amyloid, Prostaglandin Receptor, Autophagy
Nootkatone
Cat.No: T3S0195
Synonym: 诺卡酮,努特卡酮,诺卡酮
Target: AMPK
(E)-Naringenin chalcone
Cat.No: T2S2173
Synonym: Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮
Target: Others
Thunberginol C
Cat.No: TMA0955
Synonym:
Target: Antifection
Dichotomine H
Cat.No: T82563
Synonym:
Target:
Rhodiocyanoside A
Cat.No: TN2155
Synonym:
Target: Histamine Receptor
Gymconopin C
Cat.No: T82250
Synonym:
Target:
Taxiresinol
Cat.No: TMA0627
Synonym:
Target: TNF
Epimagnolin B
Cat.No: TN1009
Synonym:
Target: NF-κB, NO Synthase, Prostaglandin Receptor
Cearoin
Cat.No: TN3614
Synonym: 檀木
Target: ERK, BCL, PARP, IκB/IKK, TNF, NF-κB, ROS, Caspase
trans-Hinokiresinol
Cat.No: TN5164
Synonym:
Target: IL Receptor, TNF, NOS, LTR
Gymnoside I
Cat.No: T82248
Synonym:
Target:
2-Carene
Cat.No: T8291
Synonym:
Target: Others
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