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Search Results for " pparγ "

152

抑制剂 & 化合物

39

天然产物

1

TargetMol 试剂盒

5

重组蛋白

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Cat. No. Product Name Form Specificity Of Inhibition
CL0076 PPAR inhibitor/activator kit

PPAR inhibitor/activator kit

TargetMol 试剂盒

PPAR inhibitor/activator kit
Cat.No: CL0076
Cat. No. Product Name Target Signaling Pathways
T63561 PPARγ agonist 5

PPARγ agonist 5 是选择性的、有效的 PPARγ 激动剂,对癌症疾病表现出研究潜力。
T63514 PPARγ agonist 1

PPARγ agonist 1 是 PPARγ 的有效激动剂,能够高效的激活 hPPARγ ,并不引起完全激动,进而能够避免不良反应。PPARγ agonist 1 对代谢紊乱相关心血管疾病表现出研究潜力。
T61465 PPARγ agonist 3

PPARγ agonist 3, also known as Compound 18a, is a potent and selective agonist of PPARγ. This compound does not exhibit cytotoxicity towards both non-resistant and resistant cells. Notably, PPARγ agonist 3 demonstrates antitumor efficacy exclusively when co-administered with Imatinib [1].
T61731 PPARγ agonist 4

PPARγ agonist 4 (Compound 18b), a potent and selective PPARγ agonist, demonstrates antitumor efficacy only when used in conjunction with Imatinib. Notably, PPARγ agonist 4 does not exhibit cytotoxic effects on either non-resistant or resistant cells [1].
T61417 PPARγ agonist 7

PPARγ agonist 7 (Compound 3a) is a highly potent and selective agonist of the peroxisome proliferator-activated receptor gamma (PPARγ). It specifically stimulates adiponectin production in human bone marrow mesenchymal stem cells (hBM-MSCs), making it an innovative full agonist of PPARγ with an EC 50 value of 4.34 μM [1].
T79678 PPARγ-IN-2

PPAR DNA Damage/DNA Repair; Metabolism
PPARγ-IN-2 (Compound 5a) 是一款PPARγ抑制剂,可在3T3-L1前脂肪细胞中抑制TG积累,EC50值为0.106 μM。该化合物能够减轻HFC诱导的肥胖及相关代谢综合症状,同时降低脂肪组织内脂质的堆积。
T62581 PPARγ agonist 6

PPARγ agonist 6 (Compound 12) 是一种选择性 PPARγ 的有效激动剂。PPARγ agonist 6 具有潜力进行癌症疾病的研究。
T61743 PPARγ agonist 2

PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ. It exhibits significant potential for utilization in metabolic disease research [1].
T79182 PPARγ agonist 8

PPAR DNA Damage/DNA Repair; Metabolism
PPARγ agonist8,作为PPARγ的激动剂,能够诱导过氧化物酶体增殖反应元件(PPRE)-萤光素酶活性,其EC50值为0.2 μM。
T62554 PPARγ phosphorylation inhibitor 1

PPARγ phosphorylation inhibitor 1 (Compound 10) 是一种有效的 PPARγ结合剂 (IC50: 24 nM),具有抗糖尿病效果。PPARγ phosphorylation inhibitor 1 对 CDK5 介导的 PPARγ Ser273 磷酸化表现出抑制作用 (IC50: 160 nM),且几乎无 PPARγ 激动作用。
T75009 PPARγ/GR modulator 1

PPARγ/GR modulator 1 是一种口服活性的 PPARγ和糖皮质激素受体 (GR) 的双动激动剂,Ki 值分别为 3.3 和 33.6 μM。PPARγ/GR modulator 1 可用于研究代谢疾病,例如糖尿病。
T4353 SR-18292

SR 18292

Autophagy Autophagy; Metabolism
SR-18292 是一种 PPARγ 共激活因子-1α (PGC-1α) 抑制剂,可增加 PGC-1α 乙酰化,抑制糖异生基因表达并减少肝细胞中的葡萄糖生成。
T1802 ZLN005

Autophagy Autophagy; Metabolism
ZLN005 是一种有效的组织特异性 PGC-1α 转录激活剂。
T16695 Pyrintegrin

Integrin Cytoskeletal Signaling
Pyrintegrin 是一种 β1 整合素激动剂,也是 2,4-二取代的嘧啶,可促进胚胎干细胞存活。它可用作足细胞保护剂,能增强细胞-细胞外基质 (ECM) 粘附介导的整联蛋白信号传导,具有强大的成脂作用。
T21955 GQ-16

PPAR DNA Damage/DNA Repair; Metabolism
GQ-16 是 PPARγ 的部分激动剂,Ki 为 160 nM。 GQ-16 可减少脂肪生成作用并促进胰岛素敏化而不会增加体重。
T8763 PTGR2-IN-1

PTGR2-IN-22

Others Others
PTGR2-IN-1 是有效的 PTGR2抑制剂,IC50为 ~0.7 μM。它能够提高转染 PTGR2 的 HEK293T 细胞 15-keto-PGE2 依赖的 PPARγ 转录活性。
T6829 EPI-001

EPI001,EPI 001

Apoptosis; Androgen Receptor; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Metabolism
EPI-001 是一种选择性雄激素受体 (AR) 的抑制剂,靶向 AR 的反式激活单元 5,可抑制 AR 氨基末端结构域的反式激活,IC50值约为 6 μM。它也是一种选择性的PPARγ调节剂,对去势抵抗性前列腺癌具有活性。
T0214 Pioglitazone

U 72107,吡格列酮,匹格列酮

Ferroptosis; PPAR Apoptosis; DNA Damage/DNA Repair; Metabolism
Pioglitazone (U 72107) 是一种胰岛素增敏剂和噻唑烷二酮,适用于治疗 2 型糖尿病。它是一种选择性PPARγ激动剂,高亲和力结合到 PPARγ 配体结合域,作用于人和鼠 PPARγ的EC50分别为 0.93 和 0.99 μM。
T0334 Rosiglitazone

BRL49653,罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone (BRL49653) 是一种 PPARγ 激动剂、TRPC5 激活剂和 TRPM3 抑制剂,具有口服活性。Rosiglitazone 也是一种降糖剂,是噻唑烷二酮类胰岛素增敏剂。
T8780 AMG131

INT-131,AMG-131,CHS 131

PPAR DNA Damage/DNA Repair; Metabolism
AMG131 (CHS 131) 是一种新型非噻唑烷二酮(TZD) 选择性过氧化物酶体增殖物激活受体 (PPAR) γ 调节剂,可用于治疗 2 型糖尿病。
T6646 Rosiglitazone hydrochloride

盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone hydrochloride (BRL-49653 HCl) 是一种降血糖药物,通过与脂肪细胞中的 PPAR 受体结合来刺激胰岛素分泌。它对 PPARγ1、PPARγ2 和 PPARγ 的EC50值分别为 30 nM、100 nM 和 60 nM。它也是TRPC5的激活剂和TRPM3的抑制剂。
T62646 Pparδ agonist 5

Pparδ agonist 5 是一种选择性的、口服具有活力的 PPARδ 激动剂,其 EC50 为 0.335 μM,选择性好于 GW0742。Pparδ agonist 5 对体内骨密度和微结构的改善具有促进作用。
T78806 PPARδ agonist 9

PPAR DNA Damage/DNA Repair; Metabolism
PPARδ agonist9 (compound 21) 作为PPARδ激动剂,展现出EC50为3.6 nM的活性。在体内实验中,PPARδ agonist9能有效降低小鼠血清中MCP-1水平,并在LDLr-KO模型中显著抑制动脉粥样硬化的发展,其抑制率达50-60%。
T62968 PPARα/δ agonist 1

PPARα/δ agonist 1 是一种有效的 PPARα/PPARδ 双重激动剂,对 PPARα和 PPARδ 的 EC50 值分别为 7.0 nM 和 8.4 nM。PPARα/δ agonist 1 对 PPARγ 表现出很高的选择性 (EC50: 1316.1 nM)。PPARα/δ agonist 1 具有潜力进行非酒精性脂肪性肝炎的研究。
T62266 PPARα agonist 1

PPARα agonist 1 是一种完整的、有效的 PPARα激动剂。
T62277 PPARδ agonist 8

Pparδ agonist 8 是一种 Pparδ 的有效激动剂。其中过氧化物酶体增殖物激活受体 (PPAR) 属于核内受体转录因子超家族,在体内代谢稳态、炎症、细胞生长和分化的调节中具有关键作用。Pparδ agonist 8 具有潜力进行非酒精性脂肪肝 (NAFLD) 的研究。
T60535 PPARα/γ agonist 1

PPARα/γ agonist 1 是一种有效的双重 PPARα/γ部分激动剂,是用于研究血脂异常和糖尿病的有前途的化合物。PPARα/γ agonist 1 对 PPARα 和 PPARγ 的EC50值分别为 28 nM 和 69 nM。
T62205 Pparδ agonist 7

Pparδ agonist 7 是一种 Pparδ 的有效激动剂。其中过氧化物酶体增殖物激活受体 (PPAR) 属于核内受体转录因子超家族,在体内代谢稳态、炎症、细胞生长和分化的调节中发挥着关键作用。Pparδ agonist 7 对非酒精性脂肪肝 (NAFLD) 表现出研究潜力。
T2260 GW9662

2-氯-5-硝基-N-苯基苯酰胺,TIMTEC-BB SBB006523,GW 9662

PPAR DNA Damage/DNA Repair; Metabolism
GW9662 (TIMTEC-BB SBB006523) 是一种特异性 PPARγ 拮抗剂,IC50值为3.3 nM,在细胞中对 PPARγ 的功能选择性是 PPARα/δ 的 10 到 1000 倍。
T23389 SR1664

SR 1664

PPAR DNA Damage/DNA Repair; Metabolism
SR1664 是一种PPARγ拮抗剂,与结合PPARγ,可有效抑制 Cdk5 介导的PPARγ磷酸化,IC50为80 nM,Ki 为 28.67 nM。
T3170 Troglitazone

CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay,曲格列酮

Apoptosis; Ferroptosis; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism
Troglitazone (Romglizone) 是一种 PPARγ 激动剂,具有抗炎和抗肿瘤活性。
T16074 Mifobate

SR-202,米福贝特

PPAR DNA Damage/DNA Repair; Metabolism
Mifobate (SR-202) 是一种有效且特异性的 PPARγ拮抗剂,可选择性抑制噻唑烷二酮 (TZD) 诱导的 PPARγ 转录活性,IC50为140 μM,具有抗肥胖和抗糖尿病作用。
T67936 BAY-0069

PPAR DNA Damage/DNA Repair; Metabolism
BAY-0069 是一种 PPARγ 反向激活剂,具有有效性和选择性,对人 PPARγ 和鼠 PPARγ 具有抑制作用, IC50 分别为 6.3 nM 和 24 nM。BAY-0069 可用于研究癌症。
T6689 T0070907

PPAR DNA Damage/DNA Repair; Metabolism
T0070907 是一种有效且特异性的 PPARγ 抑制剂,Ki 值为1 nM,其选择性比 PPARα 和 PPARδ 高 800 倍以上。
T0214L Pioglitazone hydrochloride

U-72107E,AD 4833,U 72107A,Pioglitazone HCl,匹格列酮盐酸盐

Ferroptosis; PPAR Apoptosis; DNA Damage/DNA Repair; Metabolism
Pioglitazone hydrochloride (AD 4833) 是一种选择性PPARγ激动剂,高亲和力结合到 PPARγ 配体结合域。作用于人和鼠 PPARγ,EC50分别为 0.93 和 0.99 μM。它是一种口服活性噻唑烷二酮的盐酸盐,具有抗糖尿病特性和潜在的抗肿瘤活性。
T38715 MSDC-0602K

MSDC-0602K,Azemiglitazone potassium

PPAR DNA Damage/DNA Repair; Metabolism
MSDC-0602K (Azemiglitazone potassium) (Azemiglitazone potassium) is a PPARγ-sparing thiazolidinedione (Ps-TZD) compound that binds to PPARγ with an IC50 of 18.25 μM. It also modulates the mitochondrial pyruvate carrier (MPC). This compound, MSDC-0602K, has potential applications in researching fatty liver conditions, including dysfunctional lipid metabolism, inflammation, and insulin resistance. MSDC-0602K acts as an insulin sensitizer, improving insulinemia and fatty liver disease in mice both ...
TQ0120 CDDO-Im

RTA-403,CDDO-Imidazolide,TP-235

Others; Ferroptosis; Nrf2; PPAR Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Others
CDDO-Im (TP-235) 是一种 Nrf2和 PPAR 的激活剂,对 PPARα 和 PPARγ 的 Ki 分别为232 nM 和 344 nM。
T15453 GW7647

2-[[4-[2-[[环己基氨基)羰基](4-环己基丁基)氨基]乙基]苯基]硫基]-2-甲基丙酸

PPAR DNA Damage/DNA Repair; Metabolism
GW7647 是一种PPARα有效激动剂,对人 PPARα、PPARγ 和 PPARδ 的EC50值分别为 6、1.1 和 6.2 μM。
T67933 BAY-4931

PPAR DNA Damage/DNA Repair; Metabolism
BAY-4931 是一种有效的、共价的、选择性的 PPARγ反向激动剂,IC50为 0.17 nM。
T12834 Saroglitazar Magnesium

Others Others
Saroglitazar Magnesium 是一种新型过氧化物酶体增殖物激活受体(PPAR)激动剂,对PPARα (EC50 0.65pM)具有显著的激活活性以及对PPARγ(EC50 3 nM)有中等的激活活性。
T12835 Saroglitazar

Lipaglyn

PPAR DNA Damage/DNA Repair; Metabolism
Saroglitazar (Lipaglyn) 是 PPAR 的激动剂,对 PPARα 和 PPARγ 的 EC50 值为 0.65 pM 和 3 nM。
T17044 Tesaglitazar

PPAR DNA Damage/DNA Repair; Metabolism
Tesaglitazar 是一种有效且具有选择性的过氧化物 PPAR α / γ受体双重激动剂,对 PPARγ的亲和力比 PPARα更有效,对大鼠PPARα和人PPARα的EC50分别为13.4 μM 和3.6 μM,对大鼠PPARγ和人类 PPARγ的EC50都是0.2 μM。Tesaglitazar 诱导大鼠皮下组织间质间充质细胞DNA 合成和纤维肉瘤形成。
T8374 LJ570

PPAR DNA Damage/DNA Repair; Metabolism
LJ570 是一种 PPARα/γ 双激动剂,EC50 分别为 1.05 和 0.12 μM。
T14176 Aleglitazar

RO0728804,R1439

PPAR DNA Damage/DNA Repair; Metabolism
Aleglitazar (R1439) 是一种高效的 PPARα/γ 双重激动剂,对人 PPARα 和 PPARγ 作用的 IC50 分别为 38 nM 和 19 nM。Aleglitazar 可用于 II 型糖尿病的研究。
T7395 Lanifibranor

IVA337

PPAR DNA Damage/DNA Repair; Metabolism
Lanifibranor (IVA337) 是泛过氧化物酶体增殖物激活受体 (PPAR) 激动剂,对人类PPARα,PPARσ和PPARγ的EC50值分别为 1.5, 0.87 和 0.21 μM。
T19211 BM152054

Others Others
BM152054 是一种有效的 PPARγ配体,可以通过加强胰岛素作用来诱导外周组织对葡萄糖的利用。
T15581 Inolitazone

RS5444,Efatutazone,CS-7017,伊诺他酮

PPAR DNA Damage/DNA Repair; Metabolism
Inolitazone (RS5444) 是一种高亲和力PPARγ激动剂。在体外,Inotazone 显示生长抑制的IC50约为0.8 nM。
T26986 Cevoglitazar

LBM-642,LBM 642,LBM642

PPAR DNA Damage/DNA Repair; Metabolism
Cevoglitazar (LBM-642) 是一种 PPARɑ 激动剂和 PPARγ激动剂。Cevoglitazar 能有效减少肥胖小鼠和猴的食物摄入量和体重。
T15440 GSK376501A

PPAR DNA Damage/DNA Repair; Metabolism
GSK376501A 是一种具有选择性和有效性的的过氧化物酶体增殖物激活受体 γ (PPARγ) 调节剂,可用于研究 2 型糖尿病。
T19710 Ciglitazone

Ciglitazona,U 63287,ADD3878,ADD-3878,U-63287,ADD 3878

Apoptosis; p38 MAPK; PPAR Apoptosis; DNA Damage/DNA Repair; MAPK; Metabolism
Ciglitazone (ADD 3878) 是一种强效和选择性的PPARγ激动剂(EC50:3μM)和口服降糖药。Ciglitazone 抑制th17细胞的增殖和分化,降低胰岛素水平、血管内皮生长因子的产生和血压,诱导胃癌细胞的细胞周期停止。Ciglitazone 能诱导负鼠肾上皮细胞的凋亡,激活p38 MAPK 和凋亡诱导因子(AIF)的核转位。 Ciglitazone 在肥胖症和高血糖症的动物模型中表现出降血糖活性。

化合物

PPARγ agonist 5
Cat.No: T63561
Synonym:
Target:
PPARγ agonist 1
Cat.No: T63514
Synonym:
Target:
PPARγ agonist 3
Cat.No: T61465
Synonym:
Target:
PPARγ agonist 4
Cat.No: T61731
Synonym:
Target:
PPARγ agonist 7
Cat.No: T61417
Synonym:
Target:
PPARγ-IN-2
Cat.No: T79678
Synonym:
Target: PPAR
PPARγ agonist 6
Cat.No: T62581
Synonym:
Target:
PPARγ agonist 2
Cat.No: T61743
Synonym:
Target:
PPARγ agonist 8
Cat.No: T79182
Synonym:
Target: PPAR
PPARγ phosphorylation inhibitor 1
Cat.No: T62554
Synonym:
Target:
PPARγ/GR modulator 1
Cat.No: T75009
Synonym:
Target:
SR-18292
Cat.No: T4353
Synonym: SR 18292
Target: Autophagy
ZLN005
Cat.No: T1802
Synonym:
Target: Autophagy
Pyrintegrin
Cat.No: T16695
Synonym:
Target: Integrin
GQ-16
Cat.No: T21955
Synonym:
Target: PPAR
PTGR2-IN-1
Cat.No: T8763
Synonym: PTGR2-IN-22
Target: Others
EPI-001
Cat.No: T6829
Synonym: EPI001,EPI 001
Target: Apoptosis, Androgen Receptor, PPAR
Pioglitazone
Cat.No: T0214
Synonym: U 72107,吡格列酮,匹格列酮
Target: Ferroptosis, PPAR
Rosiglitazone
Cat.No: T0334
Synonym: BRL49653,罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
AMG131
Cat.No: T8780
Synonym: INT-131,AMG-131,CHS 131
Target: PPAR
Rosiglitazone hydrochloride
Cat.No: T6646
Synonym: 盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Pparδ agonist 5
Cat.No: T62646
Synonym:
Target:
PPARδ agonist 9
Cat.No: T78806
Synonym:
Target: PPAR
PPARα/δ agonist 1
Cat.No: T62968
Synonym:
Target:
PPARα agonist 1
Cat.No: T62266
Synonym:
Target:
PPARδ agonist 8
Cat.No: T62277
Synonym:
Target:
PPARα/γ agonist 1
Cat.No: T60535
Synonym:
Target:
Pparδ agonist 7
Cat.No: T62205
Synonym:
Target:
GW9662
Cat.No: T2260
Synonym: 2-氯-5-硝基-N-苯基苯酰胺,TIMTEC-BB SBB006523,GW 9662
Target: PPAR
SR1664
Cat.No: T23389
Synonym: SR 1664
Target: PPAR
Troglitazone
Cat.No: T3170
Synonym: CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay,曲格列酮
Target: Apoptosis, Ferroptosis, PPAR, Autophagy
Mifobate
Cat.No: T16074
Synonym: SR-202,米福贝特
Target: PPAR
BAY-0069
Cat.No: T67936
Synonym:
Target: PPAR
T0070907
Cat.No: T6689
Synonym:
Target: PPAR
Pioglitazone hydrochloride
Cat.No: T0214L
Synonym: U-72107E,AD 4833,U 72107A,Pioglitazone HCl,匹格列酮盐酸盐
Target: Ferroptosis, PPAR
MSDC-0602K
Cat.No: T38715
Synonym: MSDC-0602K,Azemiglitazone potassium
Target: PPAR
CDDO-Im
Cat.No: TQ0120
Synonym: RTA-403,CDDO-Imidazolide,TP-235
Target: Others, Ferroptosis, Nrf2, PPAR
GW7647
Cat.No: T15453
Synonym: 2-[[4-[2-[[环己基氨基)羰基](4-环己基丁基)氨基]乙基]苯基]硫基]-2-甲基丙酸
Target: PPAR
BAY-4931
Cat.No: T67933
Synonym:
Target: PPAR
Saroglitazar Magnesium
Cat.No: T12834
Synonym:
Target: Others
Saroglitazar
Cat.No: T12835
Synonym: Lipaglyn
Target: PPAR
Tesaglitazar
Cat.No: T17044
Synonym:
Target: PPAR
LJ570
Cat.No: T8374
Synonym:
Target: PPAR
Aleglitazar
Cat.No: T14176
Synonym: RO0728804,R1439
Target: PPAR
Lanifibranor
Cat.No: T7395
Synonym: IVA337
Target: PPAR
BM152054
Cat.No: T19211
Synonym:
Target: Others
Inolitazone
Cat.No: T15581
Synonym: RS5444,Efatutazone,CS-7017,伊诺他酮
Target: PPAR
Cevoglitazar
Cat.No: T26986
Synonym: LBM-642,LBM 642,LBM642
Target: PPAR
GSK376501A
Cat.No: T15440
Synonym:
Target: PPAR
Ciglitazone
Cat.No: T19710
Synonym: Ciglitazona,U 63287,ADD3878,ADD-3878,U-63287,ADD 3878
Target: Apoptosis, p38 MAPK, PPAR
Cat. No. Product Name Target Signaling Pathways
TN7060 Methyl oleanonate

PPAR DNA Damage/DNA Repair; Metabolism
Methyl oleanonate 是从柃木中分离得到的一种三萜类天然产物,是齐墩果酸衍生物,是一种PPARγ激动剂,具有抗癌作用。
T6917 Oleuropein

洋橄榄苦甙,橄榄苦苷

Apoptosis; Aromatase; ROS; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。
T5552 Methyl cinnamate

Tyrosinase; Antibacterial; AMPK Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Methyl cinnamate 是花椒的有效成分,也是一种天然香料。它是一种防止食品褐变的酪氨酸酶抑制剂,具有抗菌活性。它通过由 CaMKK2-AMPK 信号途径介导的机制具有抗脂活性。
T4S1173 Agrimol B

仙鹤草酚B,仙鹤草酚 B

Sirtuin; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物,可抑制脂肪形成,降低PPARγ的表达,诱导SIRT1易位和表达。
TN1475 Caulophyllogenin

Segetalic acid

IL Receptor; TNF; PPAR; Immunology/Inflammation related Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Caulophyllogenin 是一种部分 PPARγ 激动剂 (EC50 = 12.6 μM),来源于 Kalopanax pictus (五加科) 的茎皮。 Caulophyllogenin 抑制促炎细胞因子分泌,可用于预防和治疗炎症性疾病、2 型糖尿病、肥胖和代谢综合征的研究。
T3000 Magnolol

NSC 293099,厚朴酚,5,5'-Diallyl-2,2'-biphenyldiol

NF-κB; Retinoid Receptor; Antibacterial; PPAR; p53; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB
Magnolol (5,5'-Diallyl-2,2'-biphenyldiol) 是RXRα和PPARγ的激动剂,EC50值分别为 10.4 µM 和 17.7 µM。他是从厚朴的树皮中分离得到的一种木脂素。
T3917 Protopanaxatriol

20(R)-APPT,20(R)-Protopanaxatriol,原人参三醇,(20R)-Protopanaxatriol

PPAR DNA Damage/DNA Repair; Metabolism
Protopanaxatriol (20(R)-APPT) 是天然的人参皂苷的糖苷配基,包括 Re,Rf,Rg1,Rg2 和 Rh。
T5S0788 Oroxin A

木蝴蝶苷A,Baicalein 7-O-glucoside

PPAR DNA Damage/DNA Repair; Metabolism
Oroxin A (Baicalein 7-O-glucoside) 是从黄芩根中提取的一种天然产物,是PPARγ的部分激动剂,可激活 PPARγ 转录。它通过对接 PPARγ 的蛋白配体结合区域起到激活作用。它对 α-葡萄糖苷酶有抑制活性,具有抗氧化能力,可用于癌症研究。
TN5137 Tetramethylkaempferol

transporter; PPAR DNA Damage/DNA Repair; Metabolism
Tetramethylkaempferol 是一种 PPARγ 激动剂,它可以通过增加脂联素的水平来提高胰岛素敏感性,脂联素是一种与脂肪组织中胰岛素敏感性相关的重要脂肪细胞因子。 它可以浓度依赖性地增强甘油三酯的积累,甘油三酯是脂肪生成的标志物。
TN1990 Norathyriol

芒果苷元

Akt; DNA/RNA Synthesis; AMPK; PPAR Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Norathyriol 是来自芒果的芒果苷代谢物,具有抗氧化、抗癌、抗菌和抗炎活性。它以非竞争性方式抑制 α-葡萄糖苷酶,IC50为 3.12 μM。它还抑制PPARα、PPARβ和PPARγ,IC50分别为 92.8、102.4 和 153.5 µM。
T5764 Alliin

蒜氨酸,(S)-3-(Allylsulphinyl)-L-alanine

NF-κB; PPAR DNA Damage/DNA Repair; Metabolism; NF-κB
Alliin ((S)-3-(Allylsulphinyl)-L-alanine) 是一种从大蒜中提取的亚砜化合物,具有口服活性,表现出降血糖、抗氧化和抗炎特性。
TN1525 Convallatoxin

K-毒毛旋花子配质-3-L-鼠李糖甙,铃兰毒苷

NF-κB; P-gp; PPAR DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Convallatoxin 是从铃兰分离得到的一种强心苷。它是 P-糖蛋白底物,并识别 Val982 是参与其转运的重要氨基酸。它是配体诱导的 MOR 胞吞作用的增强剂,通过激活PPARγ和抑制NF-κB 改善结肠炎,具有抗炎和抗增殖特性。
T4S1545 Licarin B

(-)-Licarin B,Licarine B,(-)-利卡灵B

transporter; Antibacterial; PPAR DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Licarin B (Licarine B) 是来源于肉豆蔻种子的一种天然产物,是 NO 生成抑制剂,可通过激活 IRS-1/PI3K/AKT 通路中的PPARγ和GLUT4 改善胰岛素敏感性。
T0646 5-Aminosalicylic Acid

Mesalazine,5-ASA,5-氨基水杨酸,Mesalamine

NF-κB; Lipoxygenase; COX; Glutathione Peroxidase; Endogenous Metabolite; PAK; PPAR Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
5-Aminosalicylic Acid (5-ASA) 是一种特异性的PPARγ激动剂,还抑制 p21-激活激酶1(PAK1) 和NF-κB,具有抗炎活性。
TN1804 Isosilybin A

异水飞蓟素 A,异水飞蓟宾A,水飞蓟素 B2

Apoptosis; Tyrosinase; PPAR; ABC Apoptosis; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome
Isosilybin A 是从水飞蓟中分离出来的一种黄酮木脂素,可抑制癌细胞增殖并诱导 G1 期停滞和凋亡,通过靶向 Akt-NF-κB-雄激素受体轴激活前列腺癌细胞的凋亡机制,具有抗前列腺癌活性。
TN2232 Soyasaponin Ab

NOS; NF-κB; COX Immunology/Inflammation; Neuroscience; NF-κB
Soyasaponin Ab 是一种大豆皂苷。Soyasaponin Ab 在 3T3-L1 脂肪细胞中通过下调 PPARγ 产生抗肥胖的作用。
T37974 (S)-Coriolic acid

13(S)-HODE

Lipoxygenase; Mitochondrial Metabolism; PPAR DNA Damage/DNA Repair; Metabolism
(S)-Coriolic acid (13(S)-HODE) 是一种重要的细胞内信号剂,是亚油酸与植物和哺乳动物脂氧合酶反应生成的,在各种生物系统中参与细胞增殖和分化。(S)-Coriolic acid 在 1 μM 左右时,它能抑制肿瘤细胞与血管内皮的粘附,能下调 IRGpIIb/IIIa 受体的表达。(S)-Coriolic acid 是15-脂氧合酶 (15-LOX) 代谢产物,常作为内源性配体激活 PPARγ。(S)-Coriolic acid 诱导线粒体功能障碍 和气道上皮损伤。
T5S1550 Cinnamyl alcohol

肉桂醇,肉桂醇;beta-苯丙烯醇,Cinnamic Alcohol,Styryl Carbinol

PPAR DNA Damage/DNA Repair; Metabolism
Cinnamyl alcohol (Styryl Carbinol) 是从板栗花中分离得到的一种活性成分,抑制增加的 PPARγ表达,具有抗肥胖作用。
T7443 4'-Methoxychalcone

4'-甲氧基查耳酮,4'-甲氧基查尔酮

PARP; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
4'-Methoxychalcone 通过PPARγ活化调节脂肪细胞分化,并调节参与胰岛素敏感性的脂肪组织中各种脂肪因子的表达和分泌,具抗肿瘤和抗炎活性。
T3403 Glabridin

光甘草定,Q-100692,KB-289522,LS-176045

Reactive Oxygen Species; Tyrosinase; GABA Receptor; Antibacterial; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome
Glabridin (KB-289522) 能够结合并激活PPARγ,EC50值为 6115 nM,是一种从Glycyrrhiza glabra 中分到的异黄烷类天然产物。它具有抗炎、抗菌、抗肾炎、抗氧化、抗肿瘤、抗糖尿病、抗骨质疏松、保护神经、保护心血管、清除自由基等作用。
T22473 15-deoxy-Δ-12,14-Prostaglandin J2

Others Others
15-deoxy-Δ-12,14-Prostaglandin J2 is a PPARγ agonist.
T10327 Ankaflavin

PPAR DNA Damage/DNA Repair; Metabolism
Ankaflavin is isolated from Monascus-Fermented red rice and is a PPARγ agonist with anti-inflammatory activity. It shows the selective cytotoxic effect and induces cell death on cancer cells.
TWS0787 Oroxin A

木蝴蝶苷A,Baicalin-7-glucoside

PPAR; Glucosidase DNA Damage/DNA Repair; Metabolism
Oroxin A (Baicalin-7-glucoside) 是一种部分 PPARγ 激动剂,可在体外和体内激活 PPARγ 转录激活。 Oroxin A 还表现出对 α-葡萄糖苷酶的抑制活性和抗氧化能力。
T75690 Wistin

Wistin 可从 Caragana sinica 根部分离得到,是 PPARα和 PPARγ的激动剂。
T72961 Falcarindiol

法卡林二醇

Falcarindiol 是一种口服活性聚乙炔氧脂,能激活 PPARγ 并增加 ABCA1 表达,具有诱导细胞凋亡和自噬的功能。此外,Falcarindiol 还展现出抗炎、抗菌、抗癌和抗糖尿病等特性。
T3056 Bavachinin

补骨脂二氢黄酮加醚,补骨脂二氢黄酮甲醚,Bavachinin A,7-O-Methylbavachin

PPAR DNA Damage/DNA Repair; Metabolism
Bavachinin (Bavachinin A) 是一种具有抗炎症和抗血管生成作用的天然化合物。
TN4390 Kihadanin B

Akt; PPAR; FOXO1 Apoptosis; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Kihadanin B can repress the adipogenesis by decreasing lipid accumulation through the suppression of the Akt-FOXO1-PPARγ axis in 3T3-L1 adipocytes.
T81898 Lyciumamide A

DPP-IV-IN-5,一种从枸杞果实中分离得到的化合物,对过氧化物酶体增殖物激活受体(PPARγ)展示中等拮抗活性,其EC50值介于10.09至44.26 μM,同时对二肽基肽酶-4 (DPPIV)亦有抑制作用,IC50值为47.13 μM。
T10153 4-O-Methyl honokiol

Others Others
4-O-Methyl honokiol, a natural neolignan isolated from Magnolia officinalis, acts as a PPARγ agonist and inhibits NF-κB activity, used for cancer and inflammation research.
TN2535 1-Hydroxy-2-oxopomolic acid

transporter; PPAR; Fatty Acid Synthase DNA Damage/DNA Repair; Metabolism
1β-Hydroxy-2-oxopomolic acid inhibits adipocyte differentiation through downregulation of various adipocytokines by blocking PPARγ and C/EBPα expression.
T79949 Foenumoside B

PPAR DNA Damage/DNA Repair; Metabolism
Foenumoside B为从Lysimachia foenum-graecum中提取的三萜皂苷。该化合物通过激活AMPK信号传导和抑制PPARγ诱导的脂肪生成,调节脂质代谢向脂肪分解方向转变。因其调控作用,Foenumoside B常用于研究肥胖及相关代谢疾病。
TN5149 Tirotundin

NF-κB; COX; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Tirotundin is a PPARα/γ dual agonist, it exerts anti-diabetic effect through PPARγ pathway. It shows anti-inflammatory activity, it inhibits inhibit the activation of NF-kappa B, thereby, the synthesis of inflammatory mediators such as cytokines and chemo
TMA0127 Ficusin A

transporter; PPAR DNA Damage/DNA Repair; Metabolism
Ficusin has antioxidant, antilipidemic and antidiabetic effects, it can lower the levels of fasting blood glucose, plasma insulin, body weight gain in HFD-STZ induced diabetic rats, and can significantly enhance the PPARγ expression and improve the transl
TN2228 Soyasaponin Aa

大豆皂苷 AA,大豆皂苷Aa

PPAR DNA Damage/DNA Repair; Metabolism
Soyasaponin Aa and soyasaponin Ab dose-dependently markedly inhibit adipocyte differentiation and expression of various adipogenic marker genes, through the downregulation of the adipogenesis-related transcription factors PPARγ and C/EBPα± in 3T3-L1 adipo
TN5091 Tagitinin A

PPAR; Antifection DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Tagitinin A is a plant insecticidal compound, it has phytotoxic activity, it shows significant inhibition of wheat coleoptile growth, seed germination, and the growth of STS and weeds. Tagitinin A is also a PPARα/γ dual agonist , it exerts anti-diabetic e
T75611 Tibesaikosaponin V

Tibesaikosaponin V 是一种三萜双糖苷,可从北柴胡 (Bupleurum chinense DC) 的根的甲醇提取物中分离得到。Tibesaikosaponin V (TKV) 是一种三萜双糖苷,可从 Bupleurum chinense DC 根的甲醇提取物中分离得到。Tibesaikosaponin V 抑制脂质积累和甘油三酯含量的发生,对脂肪细胞没有细胞毒性。Tibesaikosaponin V 抑制核转录因子的 mRNA 表达,例如过氧化物酶体增殖物激活受体 γ (PPARγ) 和 CCAAT/增强子结合蛋白 α (C/EBPα)。Tibesaikosaponin V 抑制 3T3-L1 前脂肪细胞分化。Tibesaikosaponin V 可用于肥胖及其相关代谢紊乱的研究。
TN3366 Ailanthoidol

IL Receptor; NOS; COX; Prostaglandin Receptor; PPAR DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Ailanthoidol has anti-inflammatory activity, it inhibits inflammatory reactions by macrophages and protects mice from endotoxin shock. It also possesses potential as a chemopreventive agent against tumor promotion. Ailanthoidol has anti-adipogenic activit
TN5369 Dehydroleucodine

Dehydroleucodin

Dehydroleucodine has antidiarrheal, anti-inflammatory, anti-microbial, embryotoxicity, gastric cytoprotective, anti-cancer activities. Dehydroleucodine has an important inhibitory effect in cellular pathways regulating adipocyte differentiation by modulat
T83915 Norbixin hydrate

Norbixin是一种在B. orellana中发现的类胡萝卜素,具有多样的生物活性。在无细胞测试中,它与过氧化物酶体增殖物激活受体γ (PPARγ)结合(Ki = 1.15 µM)。在心脑血管代谢综合征大鼠模型中,Norbixin (47.7 mg/kg) 能够减轻高血糖、高胰岛素血症和胰岛素抗性,降低血清脂质水平及心脏中硫代巴比妥酸反应性物质(TBARS)和谷胱甘肽(GSH)的水平。在胆固醇诱导的动脉粥样硬化兔模型中,它降低氧化型LDL和主动脉蛋白氧化水平,并减少动脉粥样硬化面积。Norbixin(每天0.1和1 mg/kg)减少汞诱导的大鼠肝细胞和白细胞DNA损伤。此外,它还能预防与年龄相关的黄斑变性(AMD)Abca4-/- Rdh8-/-小鼠模型中的光感受器退化。

天然产物

Methyl oleanonate
Cat.No: TN7060
Synonym:
Target: PPAR
Oleuropein
Cat.No: T6917
Synonym: 洋橄榄苦甙,橄榄苦苷
Target: Apoptosis, Aromatase, ROS, PPAR
Methyl cinnamate
Cat.No: T5552
Synonym:
Target: Tyrosinase, Antibacterial, AMPK
Agrimol B
Cat.No: T4S1173
Synonym: 仙鹤草酚B,仙鹤草酚 B
Target: Sirtuin, PPAR
Caulophyllogenin
Cat.No: TN1475
Synonym: Segetalic acid
Target: IL Receptor, TNF, PPAR, Immunology/Inflammation related
Magnolol
Cat.No: T3000
Synonym: NSC 293099,厚朴酚,5,5'-Diallyl-2,2'-biphenyldiol
Target: NF-κB, Retinoid Receptor, Antibacterial, PPAR, p53, Autophagy
Protopanaxatriol
Cat.No: T3917
Synonym: 20(R)-APPT,20(R)-Protopanaxatriol,原人参三醇,(20R)-Protopanaxatriol
Target: PPAR
Oroxin A
Cat.No: T5S0788
Synonym: 木蝴蝶苷A,Baicalein 7-O-glucoside
Target: PPAR
Tetramethylkaempferol
Cat.No: TN5137
Synonym:
Target: transporter, PPAR
Norathyriol
Cat.No: TN1990
Synonym: 芒果苷元
Target: Akt, DNA/RNA Synthesis, AMPK, PPAR
Alliin
Cat.No: T5764
Synonym: 蒜氨酸,(S)-3-(Allylsulphinyl)-L-alanine
Target: NF-κB, PPAR
Convallatoxin
Cat.No: TN1525
Synonym: K-毒毛旋花子配质-3-L-鼠李糖甙,铃兰毒苷
Target: NF-κB, P-gp, PPAR
Licarin B
Cat.No: T4S1545
Synonym: (-)-Licarin B,Licarine B,(-)-利卡灵B
Target: transporter, Antibacterial, PPAR
5-Aminosalicylic Acid
Cat.No: T0646
Synonym: Mesalazine,5-ASA,5-氨基水杨酸,Mesalamine
Target: NF-κB, Lipoxygenase, COX, Glutathione Peroxidase, Endogenous Metabolite, PAK, PPAR
Isosilybin A
Cat.No: TN1804
Synonym: 异水飞蓟素 A,异水飞蓟宾A,水飞蓟素 B2
Target: Apoptosis, Tyrosinase, PPAR, ABC
Soyasaponin Ab
Cat.No: TN2232
Synonym:
Target: NOS, NF-κB, COX
(S)-Coriolic acid
Cat.No: T37974
Synonym: 13(S)-HODE
Target: Lipoxygenase, Mitochondrial Metabolism, PPAR
Cinnamyl alcohol
Cat.No: T5S1550
Synonym: 肉桂醇,肉桂醇;beta-苯丙烯醇,Cinnamic Alcohol,Styryl Carbinol
Target: PPAR
4'-Methoxychalcone
Cat.No: T7443
Synonym: 4'-甲氧基查耳酮,4'-甲氧基查尔酮
Target: PARP, PPAR
Glabridin
Cat.No: T3403
Synonym: 光甘草定,Q-100692,KB-289522,LS-176045
Target: Reactive Oxygen Species, Tyrosinase, GABA Receptor, Antibacterial, PPAR
15-deoxy-Δ-12,14-Prostaglandin J2
Cat.No: T22473
Synonym:
Target: Others
Ankaflavin
Cat.No: T10327
Synonym:
Target: PPAR
Oroxin A
Cat.No: TWS0787
Synonym: 木蝴蝶苷A,Baicalin-7-glucoside
Target: PPAR, Glucosidase
Wistin
Cat.No: T75690
Synonym:
Target:
Falcarindiol
Cat.No: T72961
Synonym: 法卡林二醇
Target:
Bavachinin
Cat.No: T3056
Synonym: 补骨脂二氢黄酮加醚,补骨脂二氢黄酮甲醚,Bavachinin A,7-O-Methylbavachin
Target: PPAR
Kihadanin B
Cat.No: TN4390
Synonym:
Target: Akt, PPAR, FOXO1
Lyciumamide A
Cat.No: T81898
Synonym:
Target:
4-O-Methyl honokiol
Cat.No: T10153
Synonym:
Target: Others
1-Hydroxy-2-oxopomolic acid
Cat.No: TN2535
Synonym:
Target: transporter, PPAR, Fatty Acid Synthase
Foenumoside B
Cat.No: T79949
Synonym:
Target: PPAR
Tirotundin
Cat.No: TN5149
Synonym:
Target: NF-κB, COX, PPAR
Ficusin A
Cat.No: TMA0127
Synonym:
Target: transporter, PPAR
Soyasaponin Aa
Cat.No: TN2228
Synonym: 大豆皂苷 AA,大豆皂苷Aa
Target: PPAR
Tagitinin A
Cat.No: TN5091
Synonym:
Target: PPAR, Antifection
Tibesaikosaponin V
Cat.No: T75611
Synonym:
Target:
Ailanthoidol
Cat.No: TN3366
Synonym:
Target: IL Receptor, NOS, COX, Prostaglandin Receptor, PPAR
Dehydroleucodine
Cat.No: TN5369
Synonym: Dehydroleucodin
Target:
Norbixin hydrate
Cat.No: T83915
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-02575 PPAR gamma/PPARG Protein, Human, Recombinant (His & GST)

CIMT1,PPARγ,GLM1,PPARgamma,PPARG1,PPARG2,NR1C3,pero...

Human Baculovirus Insect Cells
Peroxisome proliferator-activated receptor gamma (PPARG), a nuclear hormone receptor, plays a critical role in the lipid and glucose homeostasis, adipocyte differentiation, as well as intracellular insulin-signaling events. The peroxisome proliferator-activated receptor gamma (PPARgamma) regulates osteoblast and osteoclast differentiation, and is the molecular target of thiazolidinediones (TZDs), insulin sensitizers that enhance glucose utilization and adipocyte differentiation. Peroxisome proli...
TMPH-02827 PPAR gamma Protein, Mouse, Recombinant (His)

Mouse E. coli
PPAR gamma Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 63.3 kDa and the accession number is P37238.
TMPY-06830 PPAR alpha/PPARA Protein, Human, Recombinant (His)

NR1C1,PPARα,peroxisome proliferator-activated receptor α,PPA...

Human E. coli
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.36 kDa and the accession number is Q07869.
TMPH-03711 PPAR gamma Protein, Xenopus laevis, Recombinant (His)

Xenopus laevis E. coli
Receptor that binds peroxisome proliferators such as hypolipidemic drugs and fatty acids. Once activated by a ligand, the receptor binds to a promoter element in the gene for acyl-CoA oxidase and activates its transcription. It therefore controls the peroxisomal beta-oxidation pathway of fatty acids. Key regulator of adipocyte differentiation and glucose homeostasis. May play a role in the regulation of circadian rhythm.
TMPY-06837 PPAR alpha/PPARA Protein, Mouse, Recombinant (His)

PPARα,PPAR-alpha,peroxisome proliferator-activated receptor ...

Mouse E. coli
PPAR alpha/PPARA Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 31.49 kDa and the accession number is P23204.

重组蛋白

PPAR gamma/PPARG Protein, Human, Recombinant (His & GST)
Cat.No: TMPY-02575
Species: Human
Expression System: Baculovirus Insect Cells
PPAR gamma Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02827
Species: Mouse
Expression System: E. coli
PPAR alpha/PPARA Protein, Human, Recombinant (His)
Cat.No: TMPY-06830
Species: Human
Expression System: E. coli
PPAR gamma Protein, Xenopus laevis, Recombinant (His)
Cat.No: TMPH-03711
Species: Xenopus laevis
Expression System: E. coli
PPAR alpha/PPARA Protein, Mouse, Recombinant (His)
Cat.No: TMPY-06837
Species: Mouse
Expression System: E. coli
TargetMol Loading
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