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78

抑制剂 & 化合物

41

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Cat. No. Product Name Target Signaling Pathways
TP1327L OVA Peptide 257-264 2TFA (138831-86-4 free base)

OVA Peptide 257-264 2TFA 1262751-08-5(TFA-2TFA)

Others Others
OVA Peptide 257-264 2TFA (138831-86-4 free base) 是 OVA 的 I 类 (Kb) 限制性肽表位,OVA 是卵清蛋白的八聚体肽,由 I 类 MHC 分子 H-2Kb 呈递。
TP1591L OVA G4 peptide acetate(148274-82-2 free base)

SIIGFEKL acetate

Others Others
OVA G4 peptide acetate(148274-82-2 free base) (SIIGFEKL acetate) 是激动剂卵清蛋白 (OVA) 肽 (257-264) SIINFEKL 的变体。 OVA 肽是卵清蛋白的 I 类 (Kb) 限制性肽表位,由 I 类 MHC(主要组织相容性复合物)分子 H-2Kb(小鼠 MHC I 类基因)呈递。
T38665 OVA-E1 peptide TFA

OVA-E1 peptide TFA

p38 MAPK; JNK MAPK
OVA-E1 peptide TFA 在突变型和野生型胸腺细胞中都能同样地激活 p38 和 JNK 级联。
T39017 OVA-E1 peptide

OVA-E1 peptide

OVA-E1 peptide, a variant antagonist of SIINFEKL [OVA (257-264)], elicits comparable activation of the p38 and JNK cascades in both mutant and wild-type thymocytes.
T7619 OVA Peptide(257-264)

OVA Peptide 257-264,OVA Peptide 257-264 (2TFA)

Others Others
OVA Peptide(257-264) 是 OVA 的 I 类 (Kb)-限制性肽表位,其中OVA 是一种来自卵清蛋白的八聚体肽,由 I 类 MHC 分子 H-2Kb 所呈递。
T81589 OVA-A2 Peptide

SAINFEKL, OVA (257-264) Variant

OVA-A2 Peptide(SAINFEKL, OVA (257-264) Variant)是具备生物活性的A2肽(SAINFEKL)变体,具有抗原特性。
T40360 OVA (329-337)

OVA (329-337) is a 9-aa core epitope (329–337) located in the C-terminal end of the OVA peptide.
TP1612 OVA sequence (323-336)

OVA sequence 323-336

This peptide is a cognate helper T-lymphocyte peptide that is employed to enhance CTL epitope immunogencity
TP1327 OVA Peptide(257-264) TFA

OVA Peptide (257-264) TFA

OVA Peptide (257-264) TFA, an octameric peptide epitope from ovalbumin, is presented by the class I MHC molecule, H-2Kb, showcasing a class I (Kb)-restricted profile.
T39005 OVA (55-62)

OVA 55-62 is a truncated peptide derived from the ovalbumin (OVA) antigen, specifically designed to bind to the H2-Kb mouse major histocompatibility complex (MHC) class I molecule.
TP1591 OVA G4 peptide

G4 peptide (SIIGFEKL) is a variant of the agonist ovalbumin (OVA) peptide (257-264), SIINFEKL. OVA Peptide is a class I (Kb)-restricted peptide epitope of ovalbumin presented by the class I MHC (major histocompatibility complex) molecule, H-2Kb (class I genes of the mouse MHC).
TP1652 OVA G4 peptide TFA (148274-82-2 free base)

OVA G4 peptide TFA

OVA G4 peptide TFA is an TFA salt form of OVA G4 peptide. G4 peptide (SIIGFEKL) is a variant of the agonist ovalbumin (OVA) peptide (257-264), SIINFEKL. OVA Peptide is a class I (Kb)-restricted peptide epitope of ovalbumin presented by the class I MHC (major histocompatibility complex) molecule, H-2Kb (class I genes of the mouse MHC).
TP1339 OVA Peptide 323-339

OVA Peptide (323-339) represents a T and B cell epitope of Ovalbumin (Ova), which play an important role in the development and development of immediate hypersensitivity in BALB/c mice.
T81590 OVA peptide

OVA peptide,主要源于鸡蛋清,作为I类MHC(主要组织相容性复合体)分子H-2Kb(小鼠MHC的I类基因)所呈递的特定卵白蛋白Kb限制性表位。在过敏性研究领域,OVA peptide具有广泛应用。
T78000 OVA Peptide (323-339)

OVA Peptide (323-339) 是卵清蛋白(OVA)的T和B细胞表位,对BALB/c小鼠的瞬时超敏反应生成与发展至关重要。
T0227 Bromisoval

2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral

Others Others
Bromisoval (Isobromyl) 具有抗炎活性。
T28830 Sovaprevir

ACH 0141625,ACH0141625,ACH-0141625,ACH1625,ACH 1625,ACH-1625

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sovaprevir 是一种非结构性3(NS3)蛋白酶抑制剂,有抗病毒活性,用于治疗 HCV 感染。
T9088 Topovale

ARC111,ARC 111,ARC-111,Topoval

Topoisomerase DNA Damage/DNA Repair
Topovale (ARC111) 是一种有效的拓扑异构酶 I 抑制剂。Topovale 抑制缺氧介导的缺氧诱导因子 1alpha 的积累。 Topovale 对一组癌细胞表现出低 nM 细胞毒性。与 P388 细胞相比,在 CPT 抗性拓扑异构酶 I (TOP1) 缺陷的 P388/CPT45 细胞中,Topovale 细胞毒性和 Topovale 诱导的细胞凋亡减少了 > 100 倍。
T22276 Bis(maltolato)oxovanadium(IV)

双(麦芽醇)氧钒(IV),BMOV,Bis maltolato oxovanadium,Bis(maltolato)oxovanadium (IV),bis maltolato oxo vanadium,Bis(maltolato)oxovanadium (IV)

Phosphatase; Others Metabolism; Others
Bis(maltolato)oxovanadium(IV) (BMOV) 是一种有效的胰岛素增敏剂,也是一种有效的、竞争性的、可逆的、口服具有活性的光谱蛋白酪氨酸磷酸酶 (PTP) 抑制剂。它抑制HCPTPA,PTP1B,HPTPβ和SHP2的IC50分别为 126 nM,109 nM,26 nM 和 201 nM。
T1491 Atovaquone

Atavaquone,阿托伐醌

Others; P450; Dehydrogenase; Antibiotic; Parasite Metabolism; Microbiology/Virology; Others
Atovaquone (Atavaquone) 是具有口服活性的选择性寄生虫线粒体细胞色素bc1复合物的抑制剂。它抑制人类和P. falciparum 细胞色素bc1活性,IC50值分别为 460 nM 和 2.0 nM。它有抗疟作用,有潜力用于疟疾、弓形体病、肺孢子虫肺炎和巴贝斯虫病的相关研究。
T14494 Balovaptan

RG7314

Vasopressin Receptor GPCR/G Protein
Balovaptan (RG7314) 是一种高效和选择性的脑渗透性血管加压素 1a (hV1a) 受体拮抗剂,对人类 (hV1a) 和小鼠 (mV1a) 受体的 Ki 值分别为 1 和 39 nM,可用于自闭症的研究。
T76698 Rovalpituzumab

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Rovalpituzumab 是一种靶向 delta 样蛋白 3 (DLL3) 的人源化单克隆抗体。Rovalpituzumab 可用于合成抗体-活性分子偶联物 (ADC)。Rovalpituzumab 具有抗癌活性,可用于治疗小细胞肺癌 (SCLC)。
T16792 Rovazolac

ALX-101

Liver X Receptor Metabolism
Rovazolac (ALX-101) 是一种肝脏x受体 (LXR)调节剂,可用于研究免疫系统疾病和特应性皮炎。
T5600 Darovasertib

LXS196

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Darovasertib (LXS196) 是一种有效的、选择性的和具有口服活性的蛋白激酶C(PKC) 抑制剂,有用于葡萄膜黑素瘤的研究潜力,对 PKCα、PKCθ 和 GSK3β 的 IC50值分别为 1.9、0.4 和 3.1 μM。
T2189 Sodium orthovanadate

Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate

ATPase; Phosphatase Membrane transporter/Ion channel; Metabolism
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。
T34399 Rovatirelin

KPS-0373,S0373,S-0373,S 0373

AChE Neuroscience
Rovatirelin (S-0373) 是一种新合成的促甲状腺激素释放激素(TRH)类似物,通过乙酰胆碱和多巴胺神经传递改善胞嘧啶阿拉伯糖苷诱导的脊髓小脑变性大鼠模型的运动功能障碍。
T20456 5-Chlorovaleronitrile

AI3 20151,5-氯戊腈,AI3-20151,AI320151

Others Others
5-Chlorovaleronitrile (AI320151) 可用作定量结构毒性模型来预测水生毒性。
T31806 Flovagatran

TGN 255

Thrombin Proteases/Proteasome
Flovagatran (TGN 255) 是一种具有口服活性和有效性的凝血酶和肠外直接因子 II 抑制剂。Flovagatran 可用于研究静脉血栓栓塞。
T4538 palovarotene

Ro 3300074,R 667,帕罗伐汀

Retinoid Receptor; Autophagy Autophagy; Metabolism
Palovarotene (Ro 3300074) 是核视网膜酸受体γ 的激动剂。
T5638 novaluron

氟酰脲

Others Others
Novaluron 是具有杀虫剂作用的化学品,可用作昆虫生长调节剂的杀虫剂。
T11326 Frovatriptan succinate hydrate

Frovelan,夫罗曲坦琥珀酸盐水合物 ,Frova

5-HT Receptor GPCR/G Protein; Neuroscience
Frovatriptan succinate hydrate (Frova) 是一种有效、高亲和力、选择性和口服活性的 5-HT1B、HT1D 受体激动剂和中等有效的 5-HT7 受体激动剂,pKi 值分别为 8.6、8.4 和 6.7。它可有效治疗各种偏头痛,包括恶心、呕吐、畏光和畏声等相关症状。
T15273 Fedovapagon

VA483,A106483

Vasopressin Receptor GPCR/G Protein
Fedovapagon (VA106483) 是一种具有选择性和高效性的加压素 V2 受体 (V2R) 激动剂,可抑制斑马鱼节间血管的生长。Fedovapagon 可用于研究膀胱过度活动症、夜尿症和膀胱疼痛综合征。
T13231L Trovafloxacin mesylate

Others; DNA/RNA Synthesis; Topoisomerase; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Trovafloxacin是一种广谱氟喹诺酮类抗生素,可阻断 DNA 促旋酶 (DNA gyrase) 和拓扑异构酶 IV (topoisomerase IV) 的活性,也是一种有效的特异性 pannexin 1 通道抑制剂 (PANX1, IC50 = 4 μM)。
T39479 Rovanersen

WVE-120101,Rovanersen

Rovanersen (WVE-120101) is an antisense oligonucleotide that can be used for huntington’s disease research.
T76573 [8-L-arginine] deaminovasopressin

[8-L-arginine] deaminovasopressin (dAVP) 是一种抗利尿激素类似物。
T38347 Zelkovamycin

Zelkovamycin is a cyclic peptide antibiotic originally isolated from Streptomyces.1 It inhibits growth of X. oryzae, P. oryzae, S. aureus, and A. laidlawii in a concentration-dependent manner when used at concentrations ranging from 0.01 to 300 μg/ml.References1. Zhang, H., Tomoda, H., Tabata, N., et al. Zelkovamycin, a new cyclic peptide antibiotic from Streptomyces sp. K96-0670. I. Production, isolation and biological properties. J. Antibiot. (Tokyo) 52(1), 29-33 (1999). Zelkovamycin is a cycl...
T124998 Isovallesiachotamine

Isovallesiachotamine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124998。
T36098 Isovaleryl-L-carnitine (chloride)

Isovaleryl-L-carnitine is a naturally occurring acylcarnitine that is formed via metabolic conversion of L-leucine. It increases survival and decreases apoptosis in hepatocyte growth factor-deprived murine C2.8 hepatocytes when used at a concentration of 1 mM. Isovaleryl-L-carnitine inhibits amino acid deprivation-induced proteolysis and autophagy in isolated perfused rat liver when used at concentrations of 77 and 100 μM, respectively. Increased levels of isovaleryl carnitine are associated wit...
T71621 Eprovafen

Eprovafen is a lipooxygenase inhibitor.
T124476 Cannabigerovarinic acid

Cannabigerovarinic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124476。
T22695 Crovatin

Others Others
Crovatin is extracted from Croton laevigatus Vahl.
T13231 Trovafloxacin

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Trovafloxacin 是广谱喹诺酮类抗生素,对革兰氏阳性,革兰氏阴性和厌氧菌有活性。它可阻断 DNA 促旋酶 和拓扑异构酶 IV 的活性。它也是口服活性的 Pannexin 1通道选择性抑制剂,对 PANX1内向电流的 IC50为 4 μM。
T20790 Iprovalicarb

SZX 0722,Melody,SZX-0722,Fencaramid,SZX0722,Irprovalicarb

Iprovalicarb is a fungicide aimed at oomycetes.
T77136 Quisovalimab

Quisovalimab (AVTX-002; AEVI 002; SAR 252067) 是一种人源的抗LIGHT 单克隆抗体,LIGHT 是一种肿瘤坏死因子(TNF)相关细胞因子(TNFSF14),在急性呼吸窘迫综合征(ARDS)和细胞因子释放综合征(CRS)的 COVID-19 中发挥重要作用。Quisovalimab 可用于 COVID-19 急性呼吸窘迫综合征等研究。
T76921 Befovacimab

Befovacimab (BAY 1093884),一种全人源单克隆IgG2抗体,特异性结合于组织因子通路抑制剂(TFPI),适用于血友病A/B的研究。
TP2280 ovalbumin (324-338) [Gallus gallus]/[Coturnix coturnix]

Others Others
Ovalbumin is the main protein found in egg white, making up 60-65% of the total protein. Ovalbumin is an important protein in several different areas of research, including general studies of protein structure and properties. Ovalbumin is used for studies
T80602 Dovanvetmab

ZTS-00521505

Dovanvetmab (ZTS-00521505),一种IgG1-κ型抗体,专一性靶向Felcat IL31,由CHO(Chinese Hamster Ovary)细胞主要表达。
T33682 N-Isovalerylglutamic acid

N-Ivga

N-Isovalerylglutamic acid belongs to the class of organic compounds known as glutamic acid and derivatives.
T68380 Thiovardenafil

Thiovardenafil is the thiol analogue of the PDE 5 inhibitor Vardenafil.
T27336 Flovagatran sodium

TGN255,TGN-255,TGN 255

Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.

化合物

OVA Peptide 257-264 2TFA (138831-86-4 free base)
Cat.No: TP1327L
Synonym: OVA Peptide 257-264 2TFA 1262751-08-5(TFA-2TFA)
Target: Others
OVA G4 peptide acetate(148274-82-2 free base)
Cat.No: TP1591L
Synonym: SIIGFEKL acetate
Target: Others
OVA-E1 peptide TFA
Cat.No: T38665
Synonym: OVA-E1 peptide TFA
Target: p38 MAPK, JNK
OVA-E1 peptide
Cat.No: T39017
Synonym: OVA-E1 peptide
Target:
OVA Peptide(257-264)
Cat.No: T7619
Synonym: OVA Peptide 257-264,OVA Peptide 257-264 (2TFA)
Target: Others
OVA-A2 Peptide
Cat.No: T81589
Synonym: SAINFEKL, OVA (257-264) Variant
Target:
OVA (329-337)
Cat.No: T40360
Synonym:
Target:
OVA sequence (323-336)
Cat.No: TP1612
Synonym: OVA sequence 323-336
Target:
OVA Peptide(257-264) TFA
Cat.No: TP1327
Synonym: OVA Peptide (257-264) TFA
Target:
OVA (55-62)
Cat.No: T39005
Synonym:
Target:
OVA G4 peptide
Cat.No: TP1591
Synonym:
Target:
OVA G4 peptide TFA (148274-82-2 free base)
Cat.No: TP1652
Synonym: OVA G4 peptide TFA
Target:
OVA Peptide 323-339
Cat.No: TP1339
Synonym:
Target:
OVA peptide
Cat.No: T81590
Synonym:
Target:
OVA Peptide (323-339)
Cat.No: T78000
Synonym:
Target:
Bromisoval
Cat.No: T0227
Synonym: 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral
Target: Others
Sovaprevir
Cat.No: T28830
Synonym: ACH 0141625,ACH0141625,ACH-0141625,ACH1625,ACH 1625,ACH-1625
Target: HCV Protease
Topovale
Cat.No: T9088
Synonym: ARC111,ARC 111,ARC-111,Topoval
Target: Topoisomerase
Bis(maltolato)oxovanadium(IV)
Cat.No: T22276
Synonym: 双(麦芽醇)氧钒(IV),BMOV,Bis maltolato oxovanadium,Bis(maltolato)oxovanadium (IV),bis maltolato oxo vanadium,Bis(maltolato)oxovanadium (IV)
Target: Phosphatase, Others
Atovaquone
Cat.No: T1491
Synonym: Atavaquone,阿托伐醌
Target: Others, P450, Dehydrogenase, Antibiotic, Parasite
Balovaptan
Cat.No: T14494
Synonym: RG7314
Target: Vasopressin Receptor
Rovalpituzumab
Cat.No: T76698
Synonym:
Target: Gamma-secretase
Rovazolac
Cat.No: T16792
Synonym: ALX-101
Target: Liver X Receptor
Darovasertib
Cat.No: T5600
Synonym: LXS196
Target: PKC
Sodium orthovanadate
Cat.No: T2189
Synonym: Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate
Target: ATPase, Phosphatase
Rovatirelin
Cat.No: T34399
Synonym: KPS-0373,S0373,S-0373,S 0373
Target: AChE
5-Chlorovaleronitrile
Cat.No: T20456
Synonym: AI3 20151,5-氯戊腈,AI3-20151,AI320151
Target: Others
Flovagatran
Cat.No: T31806
Synonym: TGN 255
Target: Thrombin
palovarotene
Cat.No: T4538
Synonym: Ro 3300074,R 667,帕罗伐汀
Target: Retinoid Receptor, Autophagy
novaluron
Cat.No: T5638
Synonym: 氟酰脲
Target: Others
Frovatriptan succinate hydrate
Cat.No: T11326
Synonym: Frovelan,夫罗曲坦琥珀酸盐水合物 ,Frova
Target: 5-HT Receptor
Fedovapagon
Cat.No: T15273
Synonym: VA483,A106483
Target: Vasopressin Receptor
Trovafloxacin mesylate
Cat.No: T13231L
Synonym:
Target: Others, DNA/RNA Synthesis, Topoisomerase, Antibacterial
Rovanersen
Cat.No: T39479
Synonym: WVE-120101,Rovanersen
Target:
[8-L-arginine] deaminovasopressin
Cat.No: T76573
Synonym:
Target:
Zelkovamycin
Cat.No: T38347
Synonym:
Target:
Isovallesiachotamine
Cat.No: T124998
Synonym:
Target:
Isovaleryl-L-carnitine (chloride)
Cat.No: T36098
Synonym:
Target:
Eprovafen
Cat.No: T71621
Synonym:
Target:
Cannabigerovarinic acid
Cat.No: T124476
Synonym:
Target:
Crovatin
Cat.No: T22695
Synonym:
Target: Others
Trovafloxacin
Cat.No: T13231
Synonym:
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Iprovalicarb
Cat.No: T20790
Synonym: SZX 0722,Melody,SZX-0722,Fencaramid,SZX0722,Irprovalicarb
Target:
Quisovalimab
Cat.No: T77136
Synonym:
Target:
Befovacimab
Cat.No: T76921
Synonym:
Target:
ovalbumin (324-338) [Gallus gallus]/[Coturnix coturnix]
Cat.No: TP2280
Synonym:
Target: Others
Dovanvetmab
Cat.No: T80602
Synonym: ZTS-00521505
Target:
N-Isovalerylglutamic acid
Cat.No: T33682
Synonym: N-Ivga
Target:
Thiovardenafil
Cat.No: T68380
Synonym:
Target:
Flovagatran sodium
Cat.No: T27336
Synonym: TGN255,TGN-255,TGN 255
Target:
Cat. No. Product Name Target Signaling Pathways
T12500 Platycoside E

Platycodin E,桔梗苷E

Others Others
Platycoside E (Platycodin E) 是一种桔梗皂苷元型皂苷,从桔梗的根中分离获得,能够促进 ovalbumin 免疫小鼠中血清 OVA 特异性IgG2a 和IgG2b 抗体的产生。它具有溶血活性和佐剂潜力。
T0361 Isovaleramide

异戊酰胺,3-Methylbutanamide

Dehydrogenase Metabolism
Isovaleramide (3-Methylbutanamide) 是抗惊厥剂,能够调节中枢神经系统的活性。
T3S0507 Homovanillic acid

Homovaniuic acid,Vanilacetic acid,高香草酸,Vanillacetic acid

Others; Endogenous Metabolite Metabolism; Others
Homovanillic acid (Vanillacetic acid) 是一种多巴胺代谢物,它与乳糜泻、生长激素缺乏、芳香族氨基酸脱羧酶缺乏症以及脂联素还原酶缺乏症相关。
T5S2350 Beta-Acetoxyisovalerylshikonin

乙酰氧基异戊酰阿卡宁,Acetoxyisovalerylalkannin,β-乙酰氧基异戊酰阿卡宁

Others Others
Acetoxyisovalerylshikonin 是一种萘醌衍生物,提取自Arnebia euchroma 中。
T5609 Isovaleric acid

3-Methylbutyric acid,Isopentanoic acid,β-methylbutyric acid,异戊酸,3-Methylbutanoic acid,Delphinic acid

Others; Endogenous Metabolite Metabolism; Others
Isovaleric acid (Delphinic acid) 是天然脂肪酸,可能与人类新生儿死亡以及牙买加呕吐病有关。
TN6761 Menthyl isovalerate

Others Others
Menthyl isovalerate 是一种生物活性化学品。
T3740 Isovanillin

3-羟基-4-甲氧基苯甲醛,3-Hydroxy-p-anisaldehyde,3-Hydroxy-4-methoxybenzaldehyde,5-Formylguaiacol

Others Others
Isovanillin (5-Formylguaiacol) 是一种醛氧化酶抑制剂,具有解痉挛和止泻活性。
T26288 Clovamide

trans-Clovamide,N-trans-Caffeoy-L-dopa

Apoptosis; Influenza Virus; ROS; Antibacterial Apoptosis; Immunology/Inflammation; Microbiology/Virology
Clovamide (trans-Clovamide) 是一种天然存在的咖啡酰结合物,具有抗菌、抗炎、抗氧化和神经保护作用。它是一种极好的活性氧和氧自由基清除剂。
T0613 3-Hydroxyisovaleric acid

β-羟基异戊酸,Beta-Hydroxyisovaleric acid

Others; Endogenous Metabolite Metabolism; Others
3-Hydroxyisovaleric acid (Beta-Hydroxyisovaleric acid) 是尿液中排泄的内源性代谢产物 ,可作为生物素缺乏的早期和敏感指标。
T8264 3-Methyl-2-oxovaleric acid

Endogenous Metabolite Metabolism
3-Methyl-2-oxovaleric acid 是神经毒素,代谢毒素和酸性原,它是支链氨基酸不完整分解产生的异常代谢物。
T64744 Ovalbumins

Endogenous Metabolite Metabolism
Ovalbumins 是蛋清中的主要蛋白质。Ovalbumins 具有多种生物活性,如降压、抗菌、抗癌、抗氧化和免疫调节活性。Ovalbumins 是雌激素或孕酮处理的输卵管中合成的丰富的蛋白质。Ovalbumins 通常用作研究激素控制该组织中基因表达的标志物。
T5767 Isovanillic acid

3-羟基-4-甲氧基苯甲酸,3-Hydroxy-4-methoxybenzoic acid

Others Others
Isovanillic acid (3-Hydroxy-4-methoxybenzoic acid) 是一种酚醛酸化合物,从 S. frutescens 中分离得到,具有抗炎作用。
TN1742 Homovanillyl alcohol

高香草醇,4-羟基-3-甲氧基苯乙醇

TNF; Drug Metabolite Apoptosis; Metabolism
Homovanillyl alcohol 是羟基酪醇的生物代谢物。Hydroxytyrosol 是存在于原始橄榄油和葡萄酒中的酚类化合物。它能够保护红细胞免受氧化损伤,并对心血管具有保护作用。
T5245 N-Isovaleroylglycine

N-异戊酰氨基乙酸,Isovaleroylglycine,N-Isovalerylglycine

Others; Endogenous Metabolite Metabolism; Others
N-Isovaleroylglycine (Isovaleroylglycine) 是酰基甘氨酸,能够作为体重提高和肥胖的生物标记物。
T5089 5-Aminovaleric acid

Others; Endogenous Metabolite Metabolism; Others
5-Aminovaleric acid 被认为是 GABA 的亚甲基同系物,是GABA 的弱激动剂。它是赖氨酸降解产物。 它既能够内源性产生,也能够通过赖氨酸的细菌分解代谢产生。
T19384 Isovalerylcarnitine

Apoptosis; Cysteine Protease Apoptosis; Proteases/Proteasome
Isovalerylcarnitine (3-methylbutyrylcarnitine) 是 L-亮氨酸分解代谢和异戊酸的积累产生的小分子化合物,也是一种具有选择性和有效性的钙蛋白酶 (calpain) 激活剂,可促使细胞凋亡,与异戊酸血症有关,可作为异戊酸血症的标志。
TN7221 6-Bromovanillin

6-Bromovanillin 是一种生化试剂,可用于用于合成caridopa。Caridopa 一种芳香氨基酸脱羧酶抑制剂。
T1207 Lovastatin

MK-803,洛伐他汀,Mevinolin

Ferroptosis; HMG-CoA Reductase; Autophagy Apoptosis; Autophagy; Metabolism
Lovastatin (MK-803) 是一种 HMG-CoA 还原酶抑制剂,用于降低胆固醇。
TN2447 Isovalerylshikonin

Antibacterial Microbiology/Virology
Isovalerylshikonin 是太子参和紫草的天然产物。
T8163 Glucovanillin

葡萄糖香草醛,Vanillin 4-O-β-D-Glucoside,4-(β-D-葡萄糖氧基)-3-甲氧基苯甲醛

Others Others
Glucovanillin (Vanillin 4-O-β-D-Glucoside) 是提取于青荚中,通过细胞壁降解和葡萄糖酐水解的酶联合作用可转化为香草醛。
TN2002 Obovatol

BCL; Caspase; JAK Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Proteases/Proteasome; Stem Cells
Obovatol has antioxidant, neuroprotective, antiinflammatory, antithrombotic and antitumour effects, it is a potent NF-κB inhibitors for Alzheimer's disease treatment.
T13484 2-Oxovaleric acid

Others Others
2-Oxovaleric acid is a keto acid existed in human blood.
TN3646 Chlorovaltrate K

Others Others
Chlorovaltrate K shows moderate cytotoxicity against lung adenocarcinoma (A 549), metastatic prostate cancer (PC-3M), colon cancer (HCT-8) and hepatoma (Bel 7402) cell lines with IC50 values of 0.89-9.76 uM.
TN3844 Didrovaltrate

Calcium Channel Membrane transporter/Ion channel; Metabolism
Didrovaltrate shows cytotoxic against human cancer cell lines. Didrovaltrate blocks I(Ca-L) in a concentration-dependent manner and probably inhibits I(Ca-L) in its inactive state, which may contribute to its cardiovascular effect.
TN6164 2,4,6-Trihydroxyisovalerophenone

2',4',6'-Trihydroxyisovalerophenone

2,4,6-Trihydroxyisovalerophenone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6164,CAS号为 26103-97-9。
TN5738 Homovanillyl alcohol 4-O-glucoside

Homovanillyl alcohol 4-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5738,CAS号为 104380-15-6。
TN3855 Dihydroobovatin

Others Others
Dihydroobovatin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3855,CAS号为 104055-79-0。
TN6520 Methyl isovanillate

Methyl isovanillate is a natural product from Vitex agnus-castus.
TN3683 Clovanediol

Others Others
Clovanediol是一种天然产物,属于桃金娘科番石榴属,其产品编号为 TN3683,CAS号为 2649-64-1。Clovanediol可用作对照参考。
T0542 Isohomovanillic acid

3-羟基-4-甲氧基苯乙酸,Homoisovanillic acid

Others; Endogenous Metabolite Metabolism; Others
Isohomovanillic acid (Homoisovanillic acid) 是一种由乙酸乙酯在 pH 值为 2 的条件下从尿液中提取而来,在许多正常人尿中并不明显。
TN3504 β-Hydroxypropiovanillone

beta-Hydroxypropiovanillone

Others Others
beta-Hydroxypropiovanillone, an achiral compound, which is further degraded by lignin degradation. It shows tyrosinase inhibitory activities.
TN5533 Yukovanol

Yukovanol inhibits the proliferation of activated HSC-T6 cells in vitro.
T82024 Isovaleroyl oxokadsuranol

Isovaleroyl oxokadsuranol为从Kadsura longipedunculata中提取的一种木脂素化合物。
TN3303 8beta-(4-Hydroxytigloyloxy)ovatifolin

Others Others
8beta-(4-Hydroxytigloyloxy)ovatifolin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3303,CAS号为 554449-27-3。
TMA0750 De-O-methylacetovanillochromene

Others Others
De-O-methylacetovanillochromene 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TMA0750,CAS号为 67667-62-3。
T40618 cis-Clovamide

cis-Clovamide is a naturally occurring phenolic compound with noteworthy antioxidant, anti-inflammatory, and antiapoptotic properties.
TN5333 Clovanediol diacetate

Clovanediol diacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5333,CAS号为 2649-68-5。
TN1440 Beta-Hydroxyisovalerylshikonin

EGFR; Tyrosine Kinases; Prostaglandin Receptor; Src; AMPK; Fatty Acid Synthase Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; Metabolism; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Beta-hydroxyisovalerylshikonin 是分离自Lithospermium radix 的天然产物,具有抑制PTK 的作用, 对 EGFR 和 v-Src 受体作用的IC50分别为 0.7 μM 和 1 μM。它对多种肿瘤细胞系均有抑制作用,可以高效诱导 NCI-H522 和 DMS114 细胞的死亡。
TN6685 Homovanillic Acid Sulfate

Homovanillic acid sulfate is used as a reagent to detect oxidative enzymes, and is associated with dopamine levels in the brain.In psychiatry and neuroscience, brain and cerebrospinal fluid levels of homovanillic acid are measured as a marker of metabolic
TN2089 Platycodin D3

桔梗皂苷D3,桔梗皂苷 D3

HCV Protease; NF-κB Microbiology/Virology; NF-κB; Proteases/Proteasome
Platycodin D3 是桔梗中有抗HCV 活性的一种三萜皂苷类天然产物。
T4S2164 Narirutin

Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷

Others; Antibacterial Microbiology/Virology; Others
Narirutin (Naringenin-7-O-rutinoside) 是从Citrus unshiu 中分离的活性成分之一,具有抗氧化和抗炎活性。它是一种具有抗结核效力的shikimate 激酶抑制剂。

天然产物

Platycoside E
Cat.No: T12500
Synonym: Platycodin E,桔梗苷E
Target: Others
Isovaleramide
Cat.No: T0361
Synonym: 异戊酰胺,3-Methylbutanamide
Target: Dehydrogenase
Homovanillic acid
Cat.No: T3S0507
Synonym: Homovaniuic acid,Vanilacetic acid,高香草酸,Vanillacetic acid
Target: Others, Endogenous Metabolite
Beta-Acetoxyisovalerylshikonin
Cat.No: T5S2350
Synonym: 乙酰氧基异戊酰阿卡宁,Acetoxyisovalerylalkannin,β-乙酰氧基异戊酰阿卡宁
Target: Others
Isovaleric acid
Cat.No: T5609
Synonym: 3-Methylbutyric acid,Isopentanoic acid,β-methylbutyric acid,异戊酸,3-Methylbutanoic acid,Delphinic acid
Target: Others, Endogenous Metabolite
Menthyl isovalerate
Cat.No: TN6761
Synonym:
Target: Others
Isovanillin
Cat.No: T3740
Synonym: 3-羟基-4-甲氧基苯甲醛,3-Hydroxy-p-anisaldehyde,3-Hydroxy-4-methoxybenzaldehyde,5-Formylguaiacol
Target: Others
Clovamide
Cat.No: T26288
Synonym: trans-Clovamide,N-trans-Caffeoy-L-dopa
Target: Apoptosis, Influenza Virus, ROS, Antibacterial
3-Hydroxyisovaleric acid
Cat.No: T0613
Synonym: β-羟基异戊酸,Beta-Hydroxyisovaleric acid
Target: Others, Endogenous Metabolite
3-Methyl-2-oxovaleric acid
Cat.No: T8264
Synonym:
Target: Endogenous Metabolite
Ovalbumins
Cat.No: T64744
Synonym:
Target: Endogenous Metabolite
Isovanillic acid
Cat.No: T5767
Synonym: 3-羟基-4-甲氧基苯甲酸,3-Hydroxy-4-methoxybenzoic acid
Target: Others
Homovanillyl alcohol
Cat.No: TN1742
Synonym: 高香草醇,4-羟基-3-甲氧基苯乙醇
Target: TNF, Drug Metabolite
N-Isovaleroylglycine
Cat.No: T5245
Synonym: N-异戊酰氨基乙酸,Isovaleroylglycine,N-Isovalerylglycine
Target: Others, Endogenous Metabolite
5-Aminovaleric acid
Cat.No: T5089
Synonym:
Target: Others, Endogenous Metabolite
Isovalerylcarnitine
Cat.No: T19384
Synonym:
Target: Apoptosis, Cysteine Protease
6-Bromovanillin
Cat.No: TN7221
Synonym:
Target:
Lovastatin
Cat.No: T1207
Synonym: MK-803,洛伐他汀,Mevinolin
Target: Ferroptosis, HMG-CoA Reductase, Autophagy
Isovalerylshikonin
Cat.No: TN2447
Synonym:
Target: Antibacterial
Glucovanillin
Cat.No: T8163
Synonym: 葡萄糖香草醛,Vanillin 4-O-β-D-Glucoside,4-(β-D-葡萄糖氧基)-3-甲氧基苯甲醛
Target: Others
Obovatol
Cat.No: TN2002
Synonym:
Target: BCL, Caspase, JAK
2-Oxovaleric acid
Cat.No: T13484
Synonym:
Target: Others
Chlorovaltrate K
Cat.No: TN3646
Synonym:
Target: Others
Didrovaltrate
Cat.No: TN3844
Synonym:
Target: Calcium Channel
2,4,6-Trihydroxyisovalerophenone
Cat.No: TN6164
Synonym: 2',4',6'-Trihydroxyisovalerophenone
Target:
Homovanillyl alcohol 4-O-glucoside
Cat.No: TN5738
Synonym:
Target:
Dihydroobovatin
Cat.No: TN3855
Synonym:
Target: Others
Methyl isovanillate
Cat.No: TN6520
Synonym:
Target:
Clovanediol
Cat.No: TN3683
Synonym:
Target: Others
Isohomovanillic acid
Cat.No: T0542
Synonym: 3-羟基-4-甲氧基苯乙酸,Homoisovanillic acid
Target: Others, Endogenous Metabolite
β-Hydroxypropiovanillone
Cat.No: TN3504
Synonym: beta-Hydroxypropiovanillone
Target: Others
Yukovanol
Cat.No: TN5533
Synonym:
Target:
Isovaleroyl oxokadsuranol
Cat.No: T82024
Synonym:
Target:
8beta-(4-Hydroxytigloyloxy)ovatifolin
Cat.No: TN3303
Synonym:
Target: Others
De-O-methylacetovanillochromene
Cat.No: TMA0750
Synonym:
Target: Others
cis-Clovamide
Cat.No: T40618
Synonym:
Target:
Clovanediol diacetate
Cat.No: TN5333
Synonym:
Target:
Beta-Hydroxyisovalerylshikonin
Cat.No: TN1440
Synonym:
Target: EGFR, Tyrosine Kinases, Prostaglandin Receptor, Src, AMPK, Fatty Acid Synthase
Homovanillic Acid Sulfate
Cat.No: TN6685
Synonym:
Target:
Platycodin D3
Cat.No: TN2089
Synonym: 桔梗皂苷D3,桔梗皂苷 D3
Target: HCV Protease, NF-κB
Narirutin
Cat.No: T4S2164
Synonym: Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷
Target: Others, Antibacterial
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