289
44
6
17
Cat. No. | Product Name | ||
---|---|---|---|
L3400 | 临床期小分子药物库 | 3404 compounds | |
3404 个临床期化合物集合,可用于高通量筛选和高内涵筛选; | |||
L7860 | Mini片段亲电杂环化合物库 | 369 compounds | |
高溶解度共价杂环片段库中的 369 个化合物 | |||
L2120 | 抗癌临床化合物库 | 2545 compounds | |
2545 个具有抗癌活性小分子的独特集合,可用于高通量高内涵筛选。 | |||
L9300 | 大环化合物库 | 210 compounds | |
210 种活性已知的大环化合物,用于高通量、高内涵筛选; | |||
L3410 | 临床前化合物库 | 701 compounds | |
701 种临床前小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
L9610 | 环肽库 | 55 compounds | |
55 种环肽分子,可用于高通量和高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6411 |
Biapenem
CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627 |
Antibacterial; Antibiotic | Microbiology/Virology |
Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。 | |||
TQ0181 |
Resatorvid
CLI-095,TAK-242,瑞沙托维 |
TNF; TLR; Autophagy; Interleukin | Apoptosis; Autophagy; Immunology/Inflammation |
Resatorvid (TAK-242) 是一种 Toll 样受体 4 (TLR4) 的抑制剂,具有选择性。Resatorvid 直接与 Cys747 结合,阻止 TLR4 与 TIRAP 结合,从而阻止下游信号转导。Resatorvid 具有抗肿瘤活性、抗炎活性和神经保护作用。 | |||
TP1035L |
Cyclic somatostatin Acetate(38916-34-6(free base))
Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt) |
Others | Others |
Cyclic somatostatin Acetate(38916-34-6(free base)) (Somatostatin-14) 是一种环状十四肽,可调节许多内分泌和神经系统功能。 | |||
T6081 |
Milciclib
PHA-848125 |
Trk receptor; CDK; Autophagy | Autophagy; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors |
Milciclib (PHA-848125) 是一种 ATP 竞争性的 CDK 和原肌球蛋白受体激酶双重抑制剂,作用于 CDK2,IC50 为 45 nM。 | |||
T10898 |
Samuraciclib hydrochloride
ICEC0942 hydrochloride,CT7001 hydrochloride |
Apoptosis; CDK | Apoptosis; Cell Cycle/Checkpoint |
Samuraciclib hydrochloride (ICEC0942 hydrochloride) 是一种具有选择性,ATP 竞争性和口服活性的CDK7抑制剂,IC50为 41 nM。它以 GI50值为 0.2-0.3 µM 来抑制乳腺癌细胞系的生长,具有抗肿瘤作用。 | |||
T27636 |
Ispronicline
AZD-3480,RJR-1734,AZD 3480,TC 1734,AZD3480,TC-01734,TC-1734-112 |
AChR | Neuroscience |
Ispronicline (TC-1734) 是一种具有口服活性、选择性和有效性的 α4β2 nAChR 部分激动剂,具有抗抑郁、神经保护和持久的认知作用。Ispronicline 对 α4β2 nAChR 具有很高的亲和力,Ki= 11 nM。 | |||
T39403 |
Avotaciclib
BEY1107,Avotaciclib |
CDK | Cell Cycle/Checkpoint |
Avotaciclib (BEY1107) 是一种有效和具有口服活性的 cyclin dependent kinase 1 (CDK1) 抑制剂。Avotaciclib 可用于研究局部晚期或转移性胰腺癌。 | |||
T20864 |
7-Troc-paclitaxel
|
Others | Others |
7-Troc-paclitaxel 是紫杉醇的前体,紫杉醇具有抗肿瘤活性。 | |||
T40867 |
Simpinicline
OC-02 |
AChE | Neuroscience |
Simpinicline (OC-02)(OC-02)是一种高选择性烟碱乙酰胆碱受体(nAChR)激动剂,可激活三叉神经副交感神经通路,可用于治疗干眼症。 | |||
TP1573L |
CLIP 86-100 acetate(648881-58-7 free base)
|
Others | Others |
CLIP 86-100 acetate(648881-58-7 free base) 这是称为 CLIP 的 II 类相关不变链肽的氨基酸 86 至 100 片段。主要组织相容性复合物 II 类分子显示外源蛋白的肽片段,以触发免疫系统的防御反应。在将外源肽插入结合槽之前,去除一个占位肽 CLIP。这是通过分子 DM 实现的,它被证明可以增加 CLIP 肽与 II 类的解离速率。 | |||
TP1501L |
CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
|
MMP | Proteases/Proteasome |
CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base) 是基质金属蛋白酶 (MMP)-2 和 MMP-9 的抑制剂。它也被称为IV 型胶原酶或明胶酶。明胶酶是癌症治疗干预的潜在靶点,这些酶的抑制剂可以防止肿瘤进展。 | |||
T2138 |
Oxyphencyclimine Hydrochloride
盐酸奥克西利平,Spazamin,Daricon,Ulcociclinina |
AChR | Neuroscience |
Oxyphencyclimine Hydrochloride (Ulcociclinina) 是一种合成的叔胺和抗毒蕈碱剂,具有抗痉挛和抗分泌活性。 | |||
T11345L |
Lerociclib dihydrochloride
G1T38 dihydrochloride |
CDK | Cell Cycle/Checkpoint |
Lerociclib dihydrochloride (G1T38 dihydrochloride) 是一种有效的选择性CDK4/CDK6抑制剂,抑制CDK6/CyclinD3和CDK4/CyclinD1,IC50值分别为 2 nM 和 1 nM。 | |||
T1101 |
Minocycline hydrochloride
Minocycline HCl,盐酸米诺环素,美满霉素 |
HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic | Chromatin/Epigenetic; Metabolism; Microbiology/Virology |
Minocycline hydrochloride (Minocycline HCl) 是四环素抗生素,具有出色的吸收和组织渗透性,可用于多种细菌感染以及痤疮的治疗。米诺环素可导致在开始治疗后 1 至 3 个月内发生的急性肝炎样综合征或通常在长期治疗后具有自身免疫特征的更隐匿的慢性肝炎。 | |||
T0786 |
Clidinium bromide
克利溴铵,Ro 2-3773 |
AChR | Neuroscience |
Clidinium bromide (Ro 2-3773) 是季胺抗毒蕈碱剂,可通过减少胃酸和减慢肠道速度,缓解痉挛和腹部疼痛的症状。 | |||
T7193 |
Encenicline
EVP-6124 |
AChR | Neuroscience |
Encenicline (EVP-6124) 是一种新型α7神经元烟碱乙酰胆碱受体 (nAChRs)激动剂,用于治疗精神分裂症和阿尔茨海默病的认知障碍。 | |||
T2285 |
Encenicline hydrochloride
(R)-7-氯-N-(奎宁环-3-基)苯并[b]噻吩-2-甲酰胺盐酸盐,EVP-6124 (hydrochloride),EVP-6124 hydrochloride |
AChR | Neuroscience |
Encenicline hydrochloride (EVP-6124 hydrochloride) 是一种新型的α7神经元烟碱乙酰胆碱受体激动剂。 | |||
T15732 |
Ribociclib succinate
LEE011 琥珀酸盐,瑞博西尼琥珀酸盐,LEE011 succinate |
CDK | Cell Cycle/Checkpoint |
Ribociclib succinate (LEE011 succinate) 是一种高度特异性的CDK4/6抑制剂,IC50值分别为 10 nM 和 39 nM。它对细胞周期蛋白 B/CDK1 复合物的效力低 1000 倍。 | |||
TP1035 |
Cyclic somatostatin
SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14 |
Others | Others |
Cyclic somatostatin (SRIF-14) 是生长激素释放抑制因子,可用于研究胃十二指肠溃疡出血。 | |||
T16784 |
Roniciclib
BAY 1000394 |
CDK | Cell Cycle/Checkpoint |
Roniciclib (BAY 1000394) 是一种有效的泛 CDK 抑制剂和新型口服细胞毒剂,对 CDK1、CDK2、CDK3、CDK4、CDK7 和 CDK9 的 IC50值为 5-25 nM。 | |||
T77484 |
Atibuclimab
|
TNF | Apoptosis |
Atibuclimab 是一种靶向 CD14 的嵌合单克隆抗体,由小鼠可变区和人类 IgG4 Fc 区构成。Atibuclimab 可用于治疗肌萎缩侧索硬化症。Atibuclimab 可减少 LPS 诱导的病症,并对 LPS 诱导的促炎细胞因子释放有抑制作用,可延迟抗炎细胞因子可溶性 TNF 受体 I 型的释放, | |||
T60025 |
Eciruciclib
|
CDK | Cell Cycle/Checkpoint |
Eciruciclib 是一种具有抗肿瘤特性的 CDK 抑制剂。 | |||
T9636 |
Dalpiciclib
SHR-6390 |
CDK | Cell Cycle/Checkpoint |
Dalpiciclib (SHR-6390) 是一种高选择性、口服生物利用度和相当效力的 CDK4 和 CKD6 抑制剂,IC50 分别为 12.4 nM 和 9.9 nM。它通过抑制磷酸化 Rb 蛋白和诱导 G1 细胞周期阻滞在食管鳞状细胞癌中发挥有效的抗肿瘤活性。 | |||
T10096L |
Voruciclib
|
CDK | Cell Cycle/Checkpoint |
Voruciclib 是一种具有口服活性和选择性 CDK 抑制剂,Ki 为 0.626 nM-9.1 nM。它在多种弥漫性大 B 细胞淋巴瘤模型中抑制 MCL-1 的表达。它有效阻断 MCL-1 的转录调节子 CDK9。 | |||
T6450 |
Clinofibrate
克利贝特,S-8527,Lipoclin |
HMG-CoA Reductase; Autophagy | Autophagy; Metabolism |
Clinofibrate (Lipoclin) 是一种降脂剂,可抑制羟甲基戊二酰辅酶 A 还原酶。它用于控制血液中的高胆固醇和甘油三酯水平。 | |||
T21508 |
Anhydrotetracycline hydrochloride
|
Antibacterial; Antibiotic | Microbiology/Virology |
Anhydrotetracycline hydrochloride 是四环素的生物合成前体,是广谱的、有效的竞争性四环素破坏酶抑制剂。它是真核细胞中四环素控制的基因表达系统的效应子。 | |||
T3052 |
Sancycline
Bonomycin,Norcycline,Sancyclinum,山环素,6-Demethyl-6-deoxytetracycline |
Antibacterial | Microbiology/Virology |
Sancycline (Bonomycin) 是半合成四环素,通过可逆地结合 30S 核糖体亚基并通过阻断氨酰-tRNA 进入核糖体 A 位点来抑制蛋白质翻译。 | |||
T40652 |
Meclizine
Meclozine |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Meclizine (Meclozine) (Meclozine)具有抗组胺作用,可可逆地抑制组胺与H1受体的相互作用。Meclizine 是哌嗪类H1拮抗剂的一个成员。Meclizine 是一种有效的抗运动病剂。Meclizine 可通过血脑屏障。Meclizine 是小鼠组成型雄烷受体(CAR)的激动剂配体,也是人CAR 的反向激动剂。Meclizine 可用于polyQ 毒性疾病的研究,如亨廷顿病。 | |||
T38861L |
Tat-beclin 1 acetate
Tat-beclin 1 acetate(1423821-88-8 free base) |
HIV Protease; Autophagy | Autophagy; Microbiology/Virology; Proteases/Proteasome |
Tat-beclin 1 acetate 是一种有效的自噬诱导剂,并与自噬的负调节因子 GAPR-1 相互作用。 Tat-beclin 1 acetate 减少聚谷氨酰胺扩增蛋白聚集体的积累和几种病原体(包括 HIV-1)的复制。 | |||
T64318 |
Capecitabine-2',3'-cyclic Carbonate
|
Others | Others |
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。 | |||
T1110 |
Meclizine dihydrochloride
Meclozine dihydrochloride,NSC28728,Meclizine 2HCl,盐酸美克洛嗪 |
Apoptosis; Histamine Receptor | Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Meclizine dihydrochloride (NSC28728) 是一种组胺 H1 拮抗剂,用于治疗妊娠期间的晕动病、眩晕和恶心以及放射病。它是小鼠组成型雄甾烷受体激动剂,是人 CAR 的反向激动剂。它可透过血脑屏障,可用于多聚谷氨酰胺毒性障碍方面的研究。 | |||
T5189 |
Omadacycline
PTK 0796,Amadacycline |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。 | |||
T11227L1 |
Eravacycline HCl
Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl |
Antibiotic | Microbiology/Virology |
Eravacycline HCl (TP-434 HCl) 是一种具有广谱抗菌活性的强效抗生素。 | |||
T1569 |
Tigecycline
替加环素,GAR-936 |
ribosome; Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Tigecycline (GAR-936) 是甘氨酰环素抗生素,对 Acinetobacter baumannii(A. baumannii) 的 MIC50和 MIC90分别为 1 和 2 mg/L。它对 E. coli(MG1655 菌株) 的平均抑制浓度 (MIC) 约 125 ng/ mL。 | |||
T6199 |
Ribociclib
瑞博西尼,LEE011 |
VEGFR; CDK | Angiogenesis; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors |
Ribociclib (LEE011) 是一种口服有效的高特异性 CDK4/6 抑制剂,IC50值分别为 10 nM 和 39 nM。 | |||
T13044 |
Mevociclib
SY-1365 |
CDK | Cell Cycle/Checkpoint |
Mevociclib (SY-1365) 是一种高效选择性 CDK7抑制剂,Ki 值为 17.4 nM。它具有抗血液肿瘤和侵袭性实体肿瘤作用,有抗增殖和凋亡活性。 | |||
T12472 |
Pifithrin-α, p-Nitro, Cyclic
PFN-α |
p53 | Apoptosis |
Pifithrin-α, p-Nitro, Cyclic (PFN-α) 是 p53 的细胞渗透性和活性形式抑制剂。它对暴露于 Etoposide 的皮层神经元的保护作用比 Pifithrin-α 强一个数量级,ED50为30 nM。它也作为 p53 转录后的活性抑制剂。 | |||
T19870 |
Aceclidine
3-Acetoxyquinuclidine,1-azabicyclo[2.2.2]octan-3-yl acetate,NSC657843,3-quinuclidinyl acetate,NSC-657843,Glaucostat,NSC 657843,Quinuclidin-3-yl acetate |
AChR | Neuroscience |
Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) 是M3 mAChR 的调节剂,可用于有关通过降低眼内压治疗青光眼的研究。 | |||
T3207 |
Briciclib
ON 014185 |
CDK; PERK; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint |
Briciclib (ON 014185) 是一种 ON 013100 衍生物,是一种抑制 Y 细胞中 cyclin D1 积累的小分子。它可靶作用于eIF4E,有抑制实体瘤的潜力。 | |||
T4527 |
Seclidemstat
SP-2577 |
Histone Demethylase | Chromatin/Epigenetic |
Seclidemstat (SP-2577) 是非竞争性可逆KDM1A (LSD1)抑制剂,可用于尤文肉瘤的研究。它促进 SWI/SNF 复合物突变卵巢癌的抗肿瘤免疫,并抑制病毒产生、病毒 DNA 复制和晚期基因表达。 | |||
T3111 |
Abemaciclib methanesulfonate
abemaciclib mesylate,LY2835219,LY2835219 mesylate,LY2835219 (methanesulfonate) |
CDK | Cell Cycle/Checkpoint |
Abemaciclib methanesulfonate (LY2835219) 是一种选择性的CDK4/6抑制剂,能够抑制 CDK4/CDK6 的活性,IC50分别为 2 nM 和 10 nM。 | |||
T9694 |
Emraclidine
CVL-231 |
AChR | Neuroscience |
Emraclidine (CVL-231) 是一种毒蕈碱 M4 受体阳性变构调节剂,可用于神经系统疾病研究。 | |||
T24136 |
Heclin
|
E1/E2/E3 Enzyme | Ubiquitination |
Heclin 是一种 HECT E3 泛素连接酶抑制剂,通过抑制 Smurf2、Nedd4 和 WWP1 起作用,IC50 值分别为 6.8、6.3 和 6.9 μM。 | |||
T1912 |
Dinaciclib
SCH 727965,PS-095760 |
Apoptosis; CDK | Apoptosis; Cell Cycle/Checkpoint |
Dinaciclib (SCH 727965) 是一种 CDK 抑制剂,抑制 CDK1、CDK2、CDK5 和 CDK9 (IC50分=3/1/1/4 nM),具有选择性。Dinaciclib 具有潜在的抗肿瘤活性,可以抑制胸甘 (dThd) DNA 的整合。 | |||
T77191 |
Clivatuzumab
|
Others | Others |
Clivatuzumab为人源化抗粘液素单抗,可靶向大部分胰腺癌细胞表面高表达的MUC1表位,对多种肿瘤细胞均有较好的治疗效果。 | |||
T36983 |
Cyclic-di-GMP disodium
Cyclic diguanylate,5GP-5GP disodium,3',5'-Cyclic diguanylic acid,Cyclic di-GMP (sodium salt),cyclic diguanylate disodium,c-di-GMP,c-di-GMP disodium |
STING; Endogenous Metabolite | Immunology/Inflammation; Metabolism |
Cyclic-di-GMP disodium (5GP-5GP disodium) 是细菌的第二信使,也是一种 STING 激动剂,参与原核生物的多种过程,包括生物膜的形成、运动、和细胞周期的进展。Cyclic-di-GMP disodium 对癌细胞显示出抗增殖活性,可诱导 CD4 受体表达升高和细胞周期停滞。Cyclic-di-GMP disodium 可用于癌研究癌症。 | |||
TQ0053 |
Fadraciclib
CYC065 |
CDK | Cell Cycle/Checkpoint |
Fadraciclib (CYC065) 是一种口服有效的 ATP 竞争性的CDK2/CDK9激酶抑制剂,IC50分别为 5 和 26 nM。 | |||
T12367 |
Parsaclisib
INCB050465 |
PI3K | PI3K/Akt/mTOR signaling |
Parsaclisib (INCB050465) 是有效的、选择性的、具有口服活性的PI3Kδ抑制剂,其 IC50=1 nM。它相对于其他 PI3K I 类同工型的选择性约为 20000 倍。它可用于复发或难治性 B 细胞恶性肿瘤的研究。 | |||
T10464L |
Atuveciclib Racemate
BAY-1143572 Racemate,阿维西利 |
CDK | Cell Cycle/Checkpoint |
Atuveciclib Racemate (BAY-1143572 Racemate) 是 Atuveciclib 的外消旋混合物。 Atuveciclib 是口服有效的 P-TEFb/CDK9高选择性抑制剂,CDK9/CycT1的 IC50为13 nM。 | |||
T9702 |
Eclitasertib
|
RIP kinase | Apoptosis; NF-κB |
Eclitasertib 是一种受体相互作用蛋白激酶1抑制剂,IC50 <1 µΜ。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T30969 |
Clitocine
|
Apoptosis; BCL | Apoptosis |
Clitocine 是一种来从蘑菇中提取的一种腺苷类似物,是一种有效的转录通读剂,是一种无义突变的抑制剂,具有抗癌活性,可诱导携带 p53 无义突变等位基因的细胞产生 p53 蛋白。Clitocine 通过促进 Mcl-1 降解来增强 TRAIL 介导的人结肠癌细胞凋亡。 | |||
TCO2745 |
Cyclic AMP
Adenosine 3',5'-cyclophosphate,cAMP,腺苷环磷酸酯,环磷腺苷,Cyclic 3',5'-monophosphate adenosine,3',5'-AMP,Adenosine Cyclophosphate |
Others; Endogenous Metabolite | Metabolism; Others |
Cyclic AMP (cAMP)(Adenosine 3',5'-cyclophosphate) 是有丝分裂信使,可以促进 G1期到 S 期的细胞周期进程。 | |||
T1687L |
Doxycycline (hyclate)
Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate |
MMP; ribosome; Antibacterial; Antibiotic | Microbiology/Virology; Proteases/Proteasome |
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。 | |||
T6624 |
Oxytetracycline Dihydrate
土霉素二水合物,地霉素,Terramycin Dihydrate |
Others; Endogenous Metabolite; Antibacterial; Antibiotic; HSV | Metabolism; Microbiology/Virology; Others |
Oxytetracycline Dihydrate (Terramycin Dihydrate) 是一种四环素类抗生素,可抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,还具有抗 HSV-1的活性。 | |||
T5738 |
7-Epi 10-desacetyl paclitaxel
10-Deacetyl-7-epipaclitaxel,7-Epi-10-deacetyltaxol,7-表-10-去乙酰基云南紫杉宁A |
Others | Others |
7-Epi 10-desacetyl paclitaxel (10-Deacetyl-7-epipaclitaxel) 是紫杉醇衍生物,对 HeLa 细胞具有细胞毒性(IC50:85 μM)。 | |||
T8259 |
Doxycycline monohydrate
水合强力霉素,强力霉素一水物 |
MMP; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Proteases/Proteasome |
Doxycycline monohydrate 是一种四环素抗生素,是广谱金属蛋白酶抑制剂,具有抗菌活性。 | |||
T6447 |
Clindamycin
Clinimycin,Sobelin,Chlolincocin,克林霉素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Clindamycin (Sobelin) 从细菌核糖体中解离肽基-tRNA,破坏细菌蛋白质合成。 它是一种半合成广谱抗生素,由母体化合物林可霉素化学修饰而成。 | |||
T21430 |
Oxytetracycline Hydrochloride
Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin |
Antiviral; Endogenous Metabolite; Antibacterial; HSV | Immunology/Inflammation; Metabolism; Microbiology/Virology |
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。 | |||
TN1513 |
Clitorin
碟豆宁,碟豆素 |
PKC; Antifection | Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology |
Clitorin 是一种山奈酚糖苷,分离自 Acalypha indica 的花和叶,表现出抗氧化活性。 | |||
T0281 |
Meclocycline sulfosalicylate salt
磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream |
Antibacterial; Antibiotic | Microbiology/Virology |
Meclocycline sulfosalicylate salt (Mecloderm) 是一种具有广谱抗菌活性的四环素抗生素,可预防皮肤细菌感染。 | |||
T1304 |
Chlortetracycline hydrochloride
Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素 |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。 | |||
T0479 |
Cytisinicline
野靛碱,Baptitoxine,Cytisine,Baphitoxine,Sophorine,金雀花碱 |
AChR | Neuroscience |
Cytisinicline (Sophorine) 是从染料木中提取的一种生物碱,可用于帮助戒烟。它是 α4β2 烟碱乙酰胆碱能受体的部分激动剂,也是含 β4 受体和 α7 受体的偏完全性激动剂。 | |||
T0912 |
Tetracycline hydrochloride
NCI-c55561,盐酸四环素,Tetracycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。 | |||
T3875 |
CLINODISIDE A
|
Others | Others |
Clinodiside A 是来自中草药Clinopodium chinensis 中。 | |||
T1400 |
Demeclocycline hydrochloride
地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Demeclocycline hydrochloride (Declomycin) 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。 | |||
T1687 |
Doxycycline
Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素 |
MMP; ribosome; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Proteases/Proteasome |
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。 | |||
T3S0687 |
Ecliptasaponin D
|
Others | Others |
Ecliptasaponin D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T3S0687,CAS号为 206756-04-9。 | |||
T3S1916 |
Heteroclitin D
异型南五味子丁素,异南五味子丁素;异型南五味子丁素 |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Heteroclitin D 是异形南五味子中的一种木脂素,可抑制 L 型钙通道,具有抗脂质过氧化作用。 | |||
T5749 |
10-Deacetyl-7-xylosyl paclitaxel
10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,7-木糖甙-10-脱乙酰基紫杉醇,10-Deacetylpaclitaxel 7-Xyloside |
Others; Microtubule Associated | Cytoskeletal Signaling; Others |
10-Deacetyl-7-xylosyl paclitaxel (7-Xylosyl-10-deacetyltaxol) 是一种紫杉醇衍生物,具有改进的药理特性和更高的水溶性,用于治疗癌症。 | |||
TN1512 |
Clinopodiside A
|
Others | Others |
Clinopodiside A is a natural product from Clinopodium chinense. | |||
T0895 |
Oxytetracycline
土霉素,Terramycin |
ribosome; Endogenous Metabolite; Antibacterial; Antibiotic; HSV | Metabolism; Microbiology/Virology |
Oxytetracycline (Terramycin) 是一种四环素类抗生素。它强力抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,具有抗 HSV-1的活性。 | |||
T2S0690 |
Ecliptasaponin A
早莲苷 A,旱莲苷A,Echinocystic acid-3-o-glucoside |
Others | Others |
Ecliptasaponin A (Echinocystic acid-3-o-glucoside) 是一种墨旱莲 (Eclipta prostrate) 中分离得到的五环三萜皂苷。其中墨旱莲是一种具有多效作用的滋补草药,如抗炎、保肝、抗氧化和免疫调节。 | |||
T0518 |
Methacycline hydrochloride
Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Methacycline hydrochloride (Rondomycin) 是四环素抗生素,可抑制细菌蛋白质的合成。它是上皮-间质转化 (EMT) 抑制剂。它在体外可阻断 EMT,体内抑制纤维发生,不会直接影响 TGF-β1 Smad 信号传导。它是抗菌剂,有潜力研究肺纤维化。 | |||
T0912L |
Tetracycline
Deschlorobiomycin,Tetracyclinum,Tetracyclin,四环素 |
Others; ribosome; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Tetracycline (Tetracyclin) 是一种对多种革兰氏阳性和革兰氏阴性细菌有抑制活性的广谱抗生素。 | |||
TN7030 |
Heteroclitin G
|
Others | Others |
Heteroclitin G 被发现是 KIS 补血活性的潜在生物标志物,定量分析为进一步药理研究提供了研究基础。 | |||
T5065 |
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD
Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP |
PKA | Tyrosine Kinase/Adaptors |
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) 也称为 cGMP,是一种细胞调节剂,被描述为第二信使。它的水平随着各种激素的增加而增加,包括乙酰胆碱、胰岛素和催产素。 cGMP 激活蛋白激酶 G(PKG) 并调节离子通道电导,信号传导影响多种过程,包括平滑肌松弛和增殖、光转导和能量稳态。 | |||
T0968 |
Paclitaxel
Taxol,紫杉醇,NSC 125973 |
Apoptosis; Microtubule Associated; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling |
Paclitaxel (Taxol) 属于天然产物,是一种微管聚合物稳定剂。Paclitaxel 具有抗肿瘤活性;通过诱导有丝分裂停滞、细胞凋亡、细胞自噬等,导致细胞死亡。 | |||
T37687 | Cyclic ADP-ribose ammonium | ||
Cyclic ADP-ribose ammonium (cADPR ammonium) is a powerful calcium mobilization second messenger synthesized from NAD+ by an ADP-ribosyl cyclase. It primarily raises cytosolic calcium levels through Ryanodine receptor-mediated release from the endoplasmic reticulum, while also facilitating extracellular influx through the opening of TRPM2 channels [1][2][3]. | |||
TN3764 | Daphnicyclidin H | Others | Others |
Daphnicyclidin H is a natural product from Daphniphyllum humile and D.teijsmanni. | |||
TN3622 | Cephalocyclidin A | Others | Others |
Cephalocyclidin A是一种天然产物,属于三尖杉科三尖杉属,其产品编号为 TN3622,CAS号为 421583-14-4。Cephalocyclidin A可用作对照参考。 | |||
T75484 | Clionamine B | ||
Clionamine B, 一种海绵 Cliona celata 分离出来的刺激自噬的氨基类固醇,强烈刺激人乳腺癌 MCF-7 细胞的自噬。 | |||
TN4207 |
Heteroclitin B
|
Others | Others |
Heteroclitin B是一种天然产物,属于五味子科南五味子属,其产品编号为 TN4207,CAS号为 140461-47-8。Heteroclitin B可用作对照参考。 | |||
TN4208 |
Heteroclitin C
|
Others | Others |
Heteroclitin C is a natural product from Kadsura heteroclita. | |||
TN3765 | Daphnicyclidin I | Others | Others |
Daphnicyclidin I is a natural product from Daphniphyllum longeracemosum. | |||
T19253 |
Cyclic ADP-ribose
cADPR |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Cyclic ADP-ribose (cADPR) is an effective calcium mobilization second messenger, which is synthesized from NAD + by ADP-ribosyl cyclase. Cyclic ADP-ribose mainly increases cytosolic calcium through Ryanodine receptor-mediated endoplasmic reticulum release | |||
TN3763 | Daphnicyclidin D | Others | Others |
Daphnicyclidin D is a natural product from Daphniphyllum humile and D.teijsmanni. | |||
T64248 | Cyclic-di-GMP sodium | ||
Cyclic di-GMP sodium (c-di-GMP sodium) 是一种 STING 激活剂,也是一种无处不在的第二信使,具有调节生物膜的形成、运动和各种细菌的毒力的作用。 | |||
T72243 |
Cyclic-di-GMP diammonium
5GP-5GP diammonium,c-di-GMP diammonium ; cyclic diguanylate diammonium ; 5GP-5GP diammonium,c-di-GMP diammonium,cyclic diguanylate diammonium |
||
Cyclic di-GMP (c-di-GMP) diammonium 是一种STING 激活剂和无处不在的第二信使,调节生物膜的形成、运动和各种细菌的毒力。 | |||
T12712 |
Reutericyclin
Reutericycline |
Others | Others |
Reutericyclin is a unique tetramic acid, is an antibiotic produced by some strains of Lactobacillus reuteri. | |||
TN5863 | Dicliripariside A | ||
Dicliripariside A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5863,CAS号为 491613-65-1。 | |||
TN6058 | Daphnicyclidin F | ||
Daphnicyclidin F is a natural product from Daphniphyllum humile and D.teijsmanni. | |||
T79931 |
Mutanocyclin
|
||
Mutanocyclin 作为一种效能显著的抗真菌剂,能够抑制白色念珠菌 (C. albicans) 的丝状形成,并下调 HWP1、ECE1、FLO8、TEC1 基因的 mRNA 表达水平。此外,Mutanocyclin 在体外小鼠模型中亦能有效抑制酵母形态的发展。 | |||
T82209 |
Heteroclitin A
|
||
Heteroclitin A为一种可从五味子(Schisandra propinqua)茎部提取的木脂素。 | |||
T10909 |
Cyclic-di-GMP
c-di-GMP,cyclic diguanylate,5GP-5GP |
Others | Others |
Cyclic-di-GMP is a STING agonist and ubiquitous second messenger, which regulates the formation, motility and virulence of biofilms in various bacterial species. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01694 |
Clusterin Protein, Mouse, Recombinant (His)
SP-40,AI893575,Sgp-2,clusterin,Sugp-2,Cli,ApoJ,D14U... |
Mouse | HEK293 Cells |
Clusterin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.8 kDa and the accession number is Q06890. | |||
TMPY-01691 |
Clusterin Protein, Human, Recombinant (CLU34, His)
SGP-2,AAG4,KUB1,CLI,CLU2,TRPM2,APO-J,SP-40,CLU1,clu... |
Human | HEK293 Cells |
Clusterin Protein, Human, Recombinant (CLU34, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51.5 kDa and the accession number is P10909-2. | |||
TMPY-06908 |
Clusterin Protein, Human, Recombinant (sCLU, His)
KUB1,SP-40,TRPM-2,SGP2,CLI,TRPM2,APOJ,NA1/NA2,CLU1,... |
Human | HEK293 Cells |
Clusterin Protein, Human, Recombinant (sCLU, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 51.51 kDa and the accession number is NP_001822.3. | |||
TMPJ-00278 |
Clusterin Protein, Human, Recombinant (hFc & His)
CLU,NA1/NA2,TRPM-2,40,Apo-J,Clusterin,Complement Cytolysis I... |
Human | HEK293 Cells |
Clusterin Protein, Human, Recombinant (hFc & His) is expressed in HEK293 mammalian cells with C-Fc-6xHis tag. The predicted molecular weight is (33-45) and (60-85) KDa and the accession number is P10909. | |||
TMPJ-00279 |
Clusterin Protein, Human, Recombinant (His)
Clusterin,Ku70-Binding Protein 1,Apo-J,Testosterone-Represse... |
Human | HEK293 Cells |
Clusterin Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 28-40 KDa and the accession number is P10909. | |||
TMPY-02777 |
Cyclin E Protein, Human, Recombinant (His & GST)
cyclin E1,CCNE |
Human | Baculovirus Insect Cells |
Cyclin E Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 75 kDa and the accession number is P24864-1. | |||
TMPY-03535 |
Cyclin E Protein, Mouse, Recombinant (His & GST)
cyclin E1,AW538188,CycE1 |
Mouse | Baculovirus Insect Cells |
Cyclin E Protein, Mouse, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 74.8 kDa and the accession number is AAH62152.1. | |||
TMPH-01100 |
CLINT1 Protein, Human, Recombinant (His)
KIAA0171,Epsin-related protein,ENTH,CLINT1,Cli<... |
Human | E. coli |
Binds to membranes enriched in phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2). May have a role in transport via clathrin-coated vesicles from the trans-Golgi network to endosomes. Stimulates clathrin assembly. CLINT1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 72.3 kDa and the accession number is Q14677. | |||
TMPJ-00666 |
CLIC2 Protein, Human, Recombinant (His)
CLIC2,XAP121,Chloride Intracellular Channel Protein... |
Human | E. coli |
Chloride Intracellular Channel Protein 2 (CLIC2) is a critical component of all living cells; it regulatescellular traffic of Chloride ion and it can be inserted into membranes anf form chloride ion channels. Membrane insertion seems to be redox-regulated and may occur only under oxydizing conditions, channel activity depends on the pH. CLIC2 is involved in regulating membrane potential and organic solute transport. CLIC2 modulates the activity of RYR2 and inhibits Calcium influx. CLIC2 can be d... | |||
TMPJ-01363 |
CLIC5 Protein, Human, Recombinant (His)
Chloride Intracellular Channel Protein 5,CLIC5 |
Human | E. coli |
Chloride Intracellular Channel Protein 5 (CLIC5) is a single-pass membrane protein which belongs to the chloride channel CLIC family. It contains one GST C-terminal domain. Chloride intracellular channels are involved in chloride ion transport within various subcellular compartments. CLIC5 can insert into membranes and form selective ion channels regulated by actin that may transport chloride ions. It may play a role in the regulation of transepithelial ion absorption and secretion. CLIC5 specif... | |||
TMPY-04075 |
CLIC1 Protein, Human, Recombinant (His)
NCC27,G6,chloride intracellular channel 1 |
Human | E. coli |
Members of the CLIC family are largely soluble proteins that possess the intriguing property of spontaneous insertion into phospholipid bilayers to form integral membrane ion channels. Chloride intracellular channel 1 (CLIC1), a newly discovered member of the chloride channel protein family, has been implicated in multiple human cancers. CLIC1 is a Chloride Intracellular Ion Channel protein that exists either in a soluble state in the cytoplasm or as a membrane bound protein. CLIC1 acts as a put... | |||
TMPY-01550 |
Cyclin E Protein, Human, Recombinant (His)
cyclin E1,CCNE |
Human | Baculovirus Insect Cells |
Cyclin E Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 49.3 kDa and the accession number is P24864-1. | |||
TMPJ-00719 |
CLIC3 Protein, Human, Recombinant (His)
CLIC3,Chloride intracellular channel protein 3 |
Human | E. coli |
Chloride intracellular channel protein 3 (CLIC3) is encoded by the CLIC3 gene. CLIC3 is a single-pass membrane protein which belongs to the chloride channel CLIC family. It contains one GST C-terminal domain and one GST N-terminal domain. Chloride intracellular channel protein 3 high expressed in the placental, lung and heart, low expressed in skeletal muscle, kidney and pancreas. Chloride intracellular channel protein 3 can insert into membranes and forms chloride ion channels, may participate ... | |||
TMPY-01890 |
CLIC4 Protein, Human, Recombinant (His)
MTCLIC,chloride intracellular channel 4,p64H1,H1,hu... |
Human | E. coli |
Chloride intracellular channel protein 4, also known as Intracellular chloride ion channel protein p64H1 and CLIC4, is a member of the chloride channel CLIC family. It contains oneGST C-terminal domain. CLIC4 is a member of a family of intracellular chloride channels. It is regulated by p53, c-Myc, and tumor necrosis factor-alpha. CLIC4 is detected in epithelial cells from colon, esophagus and kidney (at protein level). CLIC4 has alternate cellular functions like a potential role in angio... | |||
TMPY-01401 |
Cyclin A1 Protein, Human, Recombinant (His)
cyclin A1,CT146 |
Human | Baculovirus Insect Cells |
Cyclin A1 is a member of the highly conserved cyclin family that is characterized by a dramatic periodicity in protein abundance, and belongs to the A-type cyclin subfamily. The mammalian A-type cyclin family consists of two members: cyclin A1 and cyclin A2. Different cyclins exhibit distinct expression. Cyclin A1 is expressed in mice exclusively in the germ cell lineage and high rate of cyclinA1 is found in human testis and certain myeloid leukaemia cells. Cyclin A1 is primarily function in the... | |||
TMPH-01004 |
Beclin-1 Protein, Human, Recombinant (His)
Protein GT197,GT197,Coiled-coil myosin-like BCL2-interacting... |
Human | E. coli |
Beclin-1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 57.9 kDa and the accession number is Q14457. | |||
TMPH-02538 |
Beclin-1 Protein, Mouse, Recombinant (His & SUMO)
Beclin-1,GT197,Coiled-coil myosin-like BCL2-interac... |
Mouse | E. coli |
Plays a central role in autophagy. Acts as core subunit of different PI3K complex forms that mediate formation of phosphatidylinositol 3-phosphate and are believed to play a role in multiple membrane trafficking pathways: PI3KC3-C1 is involved in initiation of autophagosomes and PI3KC3-C2 in maturation of autophagosomes and endocytosis. Involved in regulation of degradative endocytic trafficking and required for the abcission step in cytokinesis, probably in the context of PI3KC3-C2. Essential f... |