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845

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10775 c-Fms-IN-2

c-Fms Tyrosine Kinase/Adaptors
c-Fms-IN-2 是一种 c-FMS 激酶抑制剂 (IC50 = 24 nM)。
TNU0810 2′-C-Methyl-6-O-methylinosine

2′-C-Methyl-6-O-methylinosine

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
2′-C-Methyl-6-O-methylinosine (2′-C-Methyl-6-O-methylinosine) 是一种次黄嘌呤类似物,具有广泛的实物活性,可用于研究多种肿瘤疾病。
T7215 NM107

NM-107,2'-C-甲基胞嘧啶核苷,2'-C-Methylcytidine

HCV Protease Microbiology/Virology; Proteases/Proteasome
NM107 (2'-C-Methylcytidine) 是一种具有广谱抗病毒活性的核糖核苷,是丙型肝炎病毒 NS5B 聚合酶的核苷抑制剂,在野生型复制子细胞中的 EC50 为 1.85 μM。
T67743 4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-

Others Others
4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-是混合配体配位聚合物[Zn4(bdc)4(ppmh)2(H2O)]n 的配体。
T40005 Pomalidomide-C2-COOH

Others Others
Pomalidomide-C2-COOH 是一种合成的 E3 连接酶配体-接头偶联物,它结合了 PROTAC 技术中使用的基于 Pomalidomide 的 CRBN 配体和接头。
T40020 Pomalidomide-C2-acid

Others Others
Pomalidomide-C2-acid 是 PROTAC 的组成部分。
T8912 5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE

5-乙基-4,5,6,7-四氢-噻唑并[5,4-C]吡啶-2-胺

PLK Cell Cycle/Checkpoint
5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE 靶向 PLK1。
T7761 Pomalidomide-C2-NH2 hydrochloride

E3 Ligase Ligand-Linker Conjugate; Ligand for E3 Ligase PROTAC
Pomalidomide-C2-NH2 hydrochloride 包含基于 Pomalidomide 的 cereblon 配体和 1 个 linker,是合成的 E3 连接酶配体-linker 偶联物。
T4253 Skp2 Inhibitor C1

SKPin C1

Others; E1/E2/E3 Enzyme Others; Ubiquitination
Skp2 Inhibitor C1 (SKPin C1)(SKPin C1)是Skp2介导p27降解的特异性抑制剂。
T20889 AalphaC

2-Amino-alpha-carboline,Aalpha C,2-氨基-9H-吡啶[2,3-b]吲哚,Aalpha-C

Others Others
AalphaC (2-Amino-alpha-carboline) 是一种潜在的致癌物质。
T60531 2'-C-Methyladenosine

HCV Protease Microbiology/Virology; Proteases/Proteasome
2'-C-Methyladenosine 是丙型肝炎病毒(HCV)复制的抑制剂,分离自肾棒状杆菌。2'-C-Methyladenosine 抑制 HCV 复制子和 NS5B 催化的 RNA 合成,IC50值分别为 0.3 μM 和 1.9 μM。2'-C-Methyladenosine 还对Leishmania guyanensis (Lgy)和Leishmania braziliensis中的 LRV1有抑制作用。
T40518 C-Peptide 2, rat

C-Peptide 2, rat, a 31-amino-acid peptide, serves as a constituent in proinsulin. It possesses the ability to hinder glucose-triggered insulin secretion.
T16325 NITD008

7-Deaza-2'-C-acetylene-adenosine

Others Others
NITD008 (7-Deaza-2'-C-acetylene-adenosine) 是一种有效的和选择性的腺苷核苷抑制剂,是一种腺苷核苷类似物,具有广谱的抗病毒活性,抑制登革热病毒、动物杯状病毒和寨卡病毒。
T35653 2’-O,4’-C-Methyleneuridine

2'-O,4'-C-Methyleneuridine (Compound 15a) is a bicyclic nucleoside. [1]. Sharma VK, et al. Chemoenzymatic convergent synthesis of 2'-O,4'-C-methyleneribonucleosides. J Org Chem. 2014 Jul 3;79(13):6336-41.
T8871 C/EBPα inducer 1

4(3H)-Quinazolinone, 6-fluoro-2-[(1E)-2-(5-nitro-2-furanyl)ethenyl]-3-phenyl-

Others Others
C/EBPα inducer 1 (4(3H)-Quinazolinone, 6-fluoro-2-[(1E)-2-(5-nitro-2-furanyl)ethenyl]-3-phenyl-) 是一种C/EBPα和骨髓细胞分化的诱导剂。
T32826 LNA-Adenosine

LNA-A,LNA Adenosine,2'-O,4'-C-Methyleneadenosine

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
LNA-Adenosine (LNA-A) 是一种核苷类似物,可作为作为腺苷A3受体配体。
T37102 2'-O-Me-C(Bz) Phosphoramidite

2’-O-Me-C(Bz) Phosphoramidite is a modified phosphoramidite monomer, which can be used for the oligonucleotide synthesis.
TNU0442 2’-beta-C-Methyl inosine

2'-C-Methylinosine

Antiviral; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation
2’-beta-C-Methyl inosine (2'-C-Methylinosine) 是一种 HCV RNA聚合酶抑制剂,具有抗病毒活性,可用用于研究用于治疗丙型肝炎病毒感染。
T10654 c-Met-IN-2

c-Met/HGFR Tyrosine Kinase/Adaptors
c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.
TP1051L Protein Kinase C Peptide Substrate acetate

Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)

Others Others
Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) 以依赖于第二信使和特定衔接蛋白的方式靶向特定细胞间隔物,以响应激活 g 蛋白偶联受体、酪氨酸激酶受体或酪氨酸激酶偶联受体的细胞外信号。
T2117 PSI-6206

2'-deoxy-2'-fluoro-2'-C-methyluridine,RO 2433,GS-331007

HCV Protease Microbiology/Virology; Proteases/Proteasome
PSI-6206 (RO 2433) 是 PSI-6130 的脱氨衍生物,PSI-6206 是一种选择性 HCV RNA 聚合酶抑制剂,低效抑制HCV 复制,EC90为 >100 μM。PSI-6130 是一种有效的选择性 HCV NS5B 聚合酶抑制剂。
T5349 SCR-1481B1

麦他替尼胺丁三醇,c-Met inhibitor 2

VEGFR; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
SCR-1481B1 (c-Met inhibitor 2) 能够作用于依赖 Met 激活的癌症,对 VEGFR 具有抑制作用。
T22489 2'-MeCCPA

2-Chloro-N-cyclopentyl-2′-C-methyladenosine

HCV Protease; Adenosine Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome
2'-MeCCPA 是一种具有有效性和高选择性的 A1 腺苷受体 (A1AR) 激动剂,对 AR 的 K 值为 1.8 nM。2'-MeCCPA 抑制毛喉素刺激的腺苷酸环化酶活性,IC值为13.1 nM。2'-MeCCPA 具有镇痛活性,可用于研究 HCV 。
T40518L C-Peptide 2, rat acetate

C-Peptide 2, rat acetate (41594-08-5 Free base)

Others Others
C-Peptide 2, rat acetate 是一种可抑制葡萄糖诱导的胰岛素分泌胰岛素原组分,由31个氨基酸残基构成的多肽和醋酸盐组成。
T10650 c-Kit-IN-2

c-Kit Tyrosine Kinase/Adaptors
c-Kit-IN-2 is a c-KIT inhibitor (IC50: 82 nM), shows superior antiproliferative activities against all the three GIST cell lines, GIST430, GIST882, and GIST48 (GI50s: 1, 3, and 2 nM).
T9028 STING-IN-2

C-170

STING Immunology/Inflammation
STING-IN-2 (C-170) 是一种 STING 共价抑制剂,可抑制小鼠 STING (mmSTING) 和人类 STING (hsSTING),可用于自身炎症性疾病的研究。
T39503 Hepatitis Virus C NS3 Protease Inhibitor 2

Hepatitis Virus C NS3 Protease Inhibitor 2 is a peptide inhibitor derived from a product that targets the NS3 protease of the hepatitis C virus (HCV). Its inhibitory activity against the NS3 protease is characterized by a Ki value of 41 nM.
T41069 CHO-C-PEG2-C-CHO

CHO-C-PEG2-C-CHO

CHO-C-PEG2-C-CHO is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T0614 4-Amino-5-Chloro-2-Methoxybenzoic Acid

甲氧氯普胺杂质C,Metoclopramide EP Impurity C

Others Others
4-Amino-5-Chloro-2-Methoxybenzoic Acid (Metoclopramide EP Impurity C) 是一种Metoclopramide 代谢物。
T8005 Cardiogenol C hydrochloride

2-[[2-[(4-甲氧基苯基)氨基]-4-嘧啶基]氨基]乙醇盐酸盐,Cardiogenol C HCl,Cardiogenol C

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Cardiogenol C hydrochloride (Cardiogenol C) 是一种细胞渗透性嘧啶诱导剂,能够促使 ESCs 分化为心肌细胞。在有限的可塑性范围内,它可以对已经沿袭的祖细胞类型产生心肌生成效应,是一种心肌生成试剂,在动物模型中可以用作细胞移植研究中提高心脏修复的工具。
T29504 A(2)C

A2C,A 2C,A-2C

A(2)C is a biochemical.
T9013 Autogramin-2

tert-butyl 2-(4-isopropoxybenzamido)-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-carboxylate

Autophagy Autophagy
Autogramin-2 (tert-butyl 2-(4-isopropoxybenzamido)-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-carboxylate) 有效抑制由饥饿诱导的自噬,IC50为 0.27 μM。它也抑制 Rapamycin,通过抑制 mTORC1 诱导的自噬,IC50为 0.14 μM。
T13194 CSF1R-IN-2

c-Fms; c-Met/HGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
CSF1R-IN-2 是一种口服具有活力的、有效的 SRC,MET 和 c-FMS 抑制剂,它们的 IC50 值分别为 0.12 nM,0.14 nM 和 0.76 nM。
T19784 DBT

NSC701994,4,7-Bis(thiophen-2-yl)benzo[c][1,2,5]thiadiazole,NSC 701994,NSC-701994

Others Others
DBT (NSC-701994) 是一种远红/近红外荧光探针,用于肿瘤相关蛋白的特异性体外和体内成像。
T33467 MOMIPP

PI3K PI3K/Akt/mTOR signaling
MOMIPP 是一种 PIKfyve 抑制剂,是一种巨胞饮作用的诱导剂,可穿过血脑屏障 (BBB)。
T38237 2′-O-Methylcytidine

Nucleoside Antimetabolite/Analog; HCV Protease Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
2'-O-Methylcytidine 是 2'-代核苷,可抑制 HCV 复制。 它在体外抑制 NS5B 催化的 RNA 合成,其抑制方式是与底物核苷三磷酸竞争。
T21870 C-021

4-​Quinazolinamine, 2-​[1,​4'-​bipiperidin]​-​1'-​yl-​N-​cycloheptyl-​6,​7-​dimethoxy-

CCR Immunology/Inflammation; Microbiology/Virology
C 021 dihydrochloride 是一种 CC 趋化因子受体 4 (CCR4) 拮抗剂,抑制人和小鼠的功能趋化性,IC50分别为 140 和 39 nM。C-021 (4-​Quinazolinamine, 2-​[1,​4'-​bipiperidin]​-​1'-​yl-​N-​cycloheptyl-​6,​7-​dimethoxy-) 可有效阻止人 CCL22 衍生的 [35S]GTPγS 与受体结合,IC50为 18 nM。
T38279 C2-8

C2-8

C2-8 is an inhibitor of polyglutamine (polyQ) aggregation (IC50s = 25 and 0.05 μM for recombinant HDQ51 and in PC12 cells, respectively). It also inhibits polyQ aggregation in organotypic hippocampal slice cultures isolated from R6/2 transgenic mice and reduces neurodegeneration in a dose-dependent manner in a Drosophila model of Huntington's disease. C2-8 (100 and 200 mg/kg) reduces huntingtin aggregate size, reduces neuronal atrophy, and improves motor performance in a rotarod test in the R6/2...
T9939 JMJD6 inhibitor WL12

2H-1-Benzopyran-2-one, 3-(3H-imidazo[4,5-c]pyridin-2-yl)-6-methyl-,ZINC6733033

Others Others
JMJD6 inhibitor WL12 (ZINC6733033) 是一种JMJD6 抑制剂,能够抑制JMJD6依赖的癌细胞增殖,包括宫颈癌细胞和肝癌细胞,为研究JMJD6在癌症发展中的生物学功能提供了一个小分子探针。
T39392L C-Type Natriuretic Peptide (CNP) (1-22), human acetate

C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)

Others Others
C-Type Natriuretic Peptide (CNP) (1-22), human acetate 是一种利钠肽受体 B (NPR-B) 的激动剂,一种内皮衍生的松弛剂和生长抑制因子。 C-Type Natriuretic Peptide (CNP) (1-22), human acetate 抑制由组胺和 5-HT 或直接由毛喉素刺激的 cAMP 合成。
T40224 2',3'-cGAMP-C2-PPA

2',3'-cGAMP-C2-PPA

2',3'-cGAMP-C2-PPA (45) is a cyclic di-nucleotide that acts as a STING agonist (US20210015941A1). It is a drug-linker conjugate for antibody-drug conjugates (ADC) used in the targeted treatment of cancer.
T39582 2',3'-cGAMP-C2-SH

2',3'-cGAMP-C2-SH

2', 3'-cGAMP-C2-SH is a ADC cytotoxin.
T2242 Wnt-C59

4-(2-甲基-4-吡啶基)-N-[4-(3-吡啶基)苯基]苯乙酰胺,C59

Wnt/beta-catenin; Porcupine Cytoskeletal Signaling; Stem Cells
Wnt-C59 (C59) 是一种高效的、口服具有活力的PORCN 抑制剂(IC50:74 pM)。
T36671 C2 Phytoceramide (t18:0/2:0)

C2 Phytoceramide is a bioactive semisynthetic sphingolipid that inhibits formyl peptide-induced oxidant release (IC50 = 0.38 μM) in suspended polymorphonuclear cells. It increases COX-2 protein levels 15-fold through ERK signaling. It induces death of keratinocytes (20% viability) with an ED50 value of 30 μM, the same concentration at which 35% of cells in a TUNEL assay are apoptotic. C2 Phytoceramide also has antiproliferative effects in CHO cells, with greater than 80% cytotoxicity achieved at...
T39597 diABZI-C2-NH2

diABZI-C2-NH2

DiABZI-C2-NH2, a STING agonist with a primary amine functionality, is an active analogue.
T50001 Tinoridine

ethyl 2-amino-6-benzyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate,替诺立定

P450 Metabolism
Tinoridine 通过抑制环氧合酶-2COX-2)的产生来发挥作用,具有抗炎、抗过敏和抗凝血等活性。
T36230 C2 Ceramide (d14:1/2:0)

C2 Ceramide (d14:1/2:0)

C2 Ceramide (d14:1/2:0) is a bioactive sphingolipid. Dietary administration of C2 ceramide (d14:1/2:0) (100 μM) induces lipotoxic cardiomyopathy via increasing diastolic and systolic diameter as well as reducing fractional shortening and the number of normal cardiac contractile events in Drosophila.
T40726 Azide-C2-Azide

Azide-C2-Azide

Azide-C2-Azide is a cleavable linker vital in ADC synthesis. Azide-C2-Azide joins cytotoxic drugs to antibodies, enabling precise delivery to cells or proteins. The cleavable nature ensures controlled drug release, optimizing ADC effectiveness.
T38011 C2 Adamantanyl Globotriaosylceramide (d18:1/2:0)

C2 Adamantanyl globotriaosylceramide (AdaGb3) is a bioactive sphingolipid and water-soluble form of globotriaosylceramide that contains an adamantanyl group in place of the fatty acyl chain. It inhibits Vero toxin binding to globotriaosylceramide in an ELISA assay when used at a concentration of 10 μM. AdaGb3 decreases cell surface expression of P-glycoprotein (P-gp) and reduces efflux of rhodamine 123 in MDCK cells. It also increases apical-to-basal transport of vinblastine in human intestinal ...
T37440 C2 Adamantanyl Galactosylceramide (d18:1/2:0)

C2 Adamantanyl Galactosylceramide (d18:1/2:0) (AdaGalCer) is a bioactive sphingolipid. It reduces globotriaosylceramide 3 synthesis from exogenous lactosylceramide in microsomes. AdaGalCer stimulates recombinant glucocerebrosidase activity in a pH-dependent manner. It activates glucocerebrosidase to decrease glucosylceramide accumulation in fibroblasts and lymphoblasts isolated from patients with Gaucher and Fabry disease, respectively.

化合物

c-Fms-IN-2
Cat.No: T10775
Synonym:
Target: c-Fms
2′-C-Methyl-6-O-methylinosine
Cat.No: TNU0810
Synonym: 2′-C-Methyl-6-O-methylinosine
Target: Nucleoside Antimetabolite/Analog
NM107
Cat.No: T7215
Synonym: NM-107,2'-C-甲基胞嘧啶核苷,2'-C-Methylcytidine
Target: HCV Protease
4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-
Cat.No: T67743
Synonym:
Target: Others
Pomalidomide-C2-COOH
Cat.No: T40005
Synonym:
Target: Others
Pomalidomide-C2-acid
Cat.No: T40020
Synonym:
Target: Others
5-ETHYL-4,5,6,7-TETRAHYDRO-THIAZOLO[5,4-C]PYRIDIN-2-YLAMINE
Cat.No: T8912
Synonym: 5-乙基-4,5,6,7-四氢-噻唑并[5,4-C]吡啶-2-胺
Target: PLK
Pomalidomide-C2-NH2 hydrochloride
Cat.No: T7761
Synonym:
Target: E3 Ligase Ligand-Linker Conjugate, Ligand for E3 Ligase
Skp2 Inhibitor C1
Cat.No: T4253
Synonym: SKPin C1
Target: Others, E1/E2/E3 Enzyme
AalphaC
Cat.No: T20889
Synonym: 2-Amino-alpha-carboline,Aalpha C,2-氨基-9H-吡啶[2,3-b]吲哚,Aalpha-C
Target: Others
2'-C-Methyladenosine
Cat.No: T60531
Synonym:
Target: HCV Protease
C-Peptide 2, rat
Cat.No: T40518
Synonym:
Target:
NITD008
Cat.No: T16325
Synonym: 7-Deaza-2'-C-acetylene-adenosine
Target: Others
2’-O,4’-C-Methyleneuridine
Cat.No: T35653
Synonym:
Target:
C/EBPα inducer 1
Cat.No: T8871
Synonym: 4(3H)-Quinazolinone, 6-fluoro-2-[(1E)-2-(5-nitro-2-furanyl)ethenyl]-3-phenyl-
Target: Others
LNA-Adenosine
Cat.No: T32826
Synonym: LNA-A,LNA Adenosine,2'-O,4'-C-Methyleneadenosine
Target: Nucleoside Antimetabolite/Analog
2'-O-Me-C(Bz) Phosphoramidite
Cat.No: T37102
Synonym:
Target:
2’-beta-C-Methyl inosine
Cat.No: TNU0442
Synonym: 2'-C-Methylinosine
Target: Antiviral, DNA/RNA Synthesis
c-Met-IN-2
Cat.No: T10654
Synonym:
Target: c-Met/HGFR
Protein Kinase C Peptide Substrate acetate
Cat.No: TP1051L
Synonym: Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)
Target: Others
PSI-6206
Cat.No: T2117
Synonym: 2'-deoxy-2'-fluoro-2'-C-methyluridine,RO 2433,GS-331007
Target: HCV Protease
SCR-1481B1
Cat.No: T5349
Synonym: 麦他替尼胺丁三醇,c-Met inhibitor 2
Target: VEGFR, c-Met/HGFR
2'-MeCCPA
Cat.No: T22489
Synonym: 2-Chloro-N-cyclopentyl-2′-C-methyladenosine
Target: HCV Protease, Adenosine Receptor
C-Peptide 2, rat acetate
Cat.No: T40518L
Synonym: C-Peptide 2, rat acetate (41594-08-5 Free base)
Target: Others
c-Kit-IN-2
Cat.No: T10650
Synonym:
Target: c-Kit
STING-IN-2
Cat.No: T9028
Synonym: C-170
Target: STING
Hepatitis Virus C NS3 Protease Inhibitor 2
Cat.No: T39503
Synonym:
Target:
CHO-C-PEG2-C-CHO
Cat.No: T41069
Synonym: CHO-C-PEG2-C-CHO
Target:
4-Amino-5-Chloro-2-Methoxybenzoic Acid
Cat.No: T0614
Synonym: 甲氧氯普胺杂质C,Metoclopramide EP Impurity C
Target: Others
Cardiogenol C hydrochloride
Cat.No: T8005
Synonym: 2-[[2-[(4-甲氧基苯基)氨基]-4-嘧啶基]氨基]乙醇盐酸盐,Cardiogenol C HCl,Cardiogenol C
Target: Wnt/beta-catenin
A(2)C
Cat.No: T29504
Synonym: A2C,A 2C,A-2C
Target:
Autogramin-2
Cat.No: T9013
Synonym: tert-butyl 2-(4-isopropoxybenzamido)-6,7-dihydrothiazolo[5,4-c]pyridine-5(4H)-carboxylate
Target: Autophagy
CSF1R-IN-2
Cat.No: T13194
Synonym:
Target: c-Fms, c-Met/HGFR, Src
DBT
Cat.No: T19784
Synonym: NSC701994,4,7-Bis(thiophen-2-yl)benzo[c][1,2,5]thiadiazole,NSC 701994,NSC-701994
Target: Others
MOMIPP
Cat.No: T33467
Synonym:
Target: PI3K
2′-O-Methylcytidine
Cat.No: T38237
Synonym:
Target: Nucleoside Antimetabolite/Analog, HCV Protease
C-021
Cat.No: T21870
Synonym: 4-​Quinazolinamine, 2-​[1,​4'-​bipiperidin]​-​1'-​yl-​N-​cycloheptyl-​6,​7-​dimethoxy-
Target: CCR
C2-8
Cat.No: T38279
Synonym: C2-8
Target:
JMJD6 inhibitor WL12
Cat.No: T9939
Synonym: 2H-1-Benzopyran-2-one, 3-(3H-imidazo[4,5-c]pyridin-2-yl)-6-methyl-,ZINC6733033
Target: Others
C-Type Natriuretic Peptide (CNP) (1-22), human acetate
Cat.No: T39392L
Synonym: C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)
Target: Others
2',3'-cGAMP-C2-PPA
Cat.No: T40224
Synonym: 2',3'-cGAMP-C2-PPA
Target:
2',3'-cGAMP-C2-SH
Cat.No: T39582
Synonym: 2',3'-cGAMP-C2-SH
Target:
Wnt-C59
Cat.No: T2242
Synonym: 4-(2-甲基-4-吡啶基)-N-[4-(3-吡啶基)苯基]苯乙酰胺,C59
Target: Wnt/beta-catenin, Porcupine
C2 Phytoceramide (t18:0/2:0)
Cat.No: T36671
Synonym:
Target:
diABZI-C2-NH2
Cat.No: T39597
Synonym: diABZI-C2-NH2
Target:
Tinoridine
Cat.No: T50001
Synonym: ethyl 2-amino-6-benzyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate,替诺立定
Target: P450
C2 Ceramide (d14:1/2:0)
Cat.No: T36230
Synonym: C2 Ceramide (d14:1/2:0)
Target:
Azide-C2-Azide
Cat.No: T40726
Synonym: Azide-C2-Azide
Target:
C2 Adamantanyl Globotriaosylceramide (d18:1/2:0)
Cat.No: T38011
Synonym:
Target:
C2 Adamantanyl Galactosylceramide (d18:1/2:0)
Cat.No: T37440
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1661 Ganoderic acid C2

灵芝酸 C2

Reductase; Histamine Receptor; Immunology/Inflammation related Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Ganoderic acid C2 是分离自灵芝的一种三萜化合物, 具有潜在的抗肿瘤生物活性,以及抗组胺、抗衰老和细胞毒性作用。它对rat lens aldose reductase 具有很高的抑制活性,IC50为 3.8 µM。
T13851 Pseudolaric Acid C2

Others Others
Pseudolaric Acid C2 是一种从 Pseudolarix kaempferi 二萜酸,是大鼠口服和静脉注射后血浆、尿液、胆汁和粪便中 Pseudolaric acid B 的特异性代谢产物。
TN2373 (E/Z)-Ginkgolic acid C17:2

Ginkgolic Acid C17:2

Dehydrogenase Metabolism
(E/Z)-Ginkgolic acid C17:2 (Ginkgolic Acid C17:2) 是一种可从银杏中提取的天然产物,可靶向人二氢乳清酸脱氢酶 (DHODH).
T7607 PSI-6130

R 1656,2'-去氧-2'-氟-2'-C-甲基胞苷

HCV Protease Microbiology/Virology; Proteases/Proteasome
PSI-6130 (R 1656) 是高效选择性 HCV NS5B 聚合酶抑制剂,抑制 HCV 复制,IC50值为 0.6 μM。
TN2379 2-C-Methyl-D-erythritol

Others Others
2-C-Methyl-D-erythritol is a natural product from the fruit of Carum ajowan
TN2782 2''-O-Acetylsprengerinin C

Others Others
2''-O-Acetylsprengerinin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2782CAS号为 1220707-33-4。
TN1949 Moracin C

桑辛素 C,5-(6-羟基-2-苯并呋喃基)-2-(3-甲基-2-丁烯基)-1,3-苯二醇

ROS; NO Synthase Immunology/Inflammation
Moracin C 是一种发现于Morus mesozygia、Morus alba var. multicaulis 中的天然化合物,是一种抗炎剂。Moracin C 可抑制细胞中的一氧化氮(NO)释放和LPS 激活的活性氧(ROS)。
TN7180 2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-

4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C

Others Others
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- (Meridianin C)是一种海洋来源的天然产物,存在于Aplidium meridianum。
TN6772 Malabaricone C

Others Others
Malabaricone C 是天然的鞘磷脂合成酶抑制剂,对 SMS 1 和 SMS 2 的IC50分别为 3 和 1.5 μM。
T3671 Vitexin-2"-O-rhamnoside

牡荆素鼠李糖苷,牡荆素-2-O-鼠李糖苷,2''-O-Rhamnosylvitexin,Vitexin-2-O-rhaMnoside,Vitexin-2''-O-rhamnoside,Apigenin-8-C-glucoside

Others Others
Vitexin-2"-O-rhamnoside (Apigenin-8-C-glucoside) 是一种黄酮苷类化合物,存在于Cratagus pinnatifidaBge 中,对 H2O2介导的氧化应激损伤具有保护作用,可用于研究心血管系统疾病。
TN2499 2'-O-Methylbroussonin C

1-(4-Hydroxy-2-methoxyphenyl)-3-(4-hydroxy-3-prenylphenyl)propane

Others Others
2'-O-Methylbroussonin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2499,CAS号为 376362-03-7。
T22644 C2 Ceramide

Ceramide

Others Others
A potent modulator of cell proliferation and differentiation.
T3919 Ginsenoside Rb2

Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2

GPR; Others; Influenza Virus; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Others
Ginsenoside Rb2 (Ginsenoside C) 是人参提取物中的一种主要生物活性成分,具有抗病毒活性,可上调 GPR120 基因表达。
TN1195 17-Hydroxy sprengerinin C

17-羟基麦冬皂苷C

BCL; Others; Caspase Apoptosis; Others; Proteases/Proteasome
17-Hydroxy sprengerinin C 是从黄精的根茎中分离得到的一种糖苷化合物,具有更强的抗癌活性。17-Hydroxy sprengerinin C 降低 Blc-2 和 pro-caspase3 的表达并增加 Bax 的产生。
TN3301 8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C

Others Others
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3301,CAS号为 93395-31-4。
TQ0054 Purpureaside C

Others Others
Purpureaside C 是一种酚类糖苷类,具有显着的促炎、免疫调节和抗菌作用。
TN2750 2-C-Methyl-D-erythrono-1,4-lactone

Others Others
(-)-2-C-Methyl-D-erythrono-1,4-lactone is inactive alone, but elicits oviposition behavior when mixes with other fractions.
T11848 Licorice glycoside C2

甘草苷 C2

Others Others
Licorice glycoside C2 is a oleanane-type triterpene oligoglycoside isolated from Glycyrrhiza uralensis.
T3810 Saikosaponin B2

柴胡皂苷 B2,柴胡皂甙 B2

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。
T2873 Ginsenoside Rg2

Chikusetsusaponin I,Panaxoside Rg2,人参皂苷Rg2,Prosapogenin C2,(20S)Ginsenoside Rg2,人参皂苷 Rg2

Beta Amyloid; GSK-3; NF-κB Neuroscience; NF-κB; PI3K/Akt/mTOR signaling; Stem Cells
Ginsenoside Rg2 (Chikusetsusaponin I) 是一种人参的主要活性成分。它能够降低Aβ1-42积聚,抑制脂多糖介导的VCAM-1和ICAM-1表达的增加。
TN7108 Urolithin C

Apoptosis; Calcium Channel; Reactive Oxygen Species; IGF-1R; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Tyrosine Kinase/Adaptors
Urolithin C 属于多酚类,是鞣花酸的肠道微生物代谢产物,具有胰岛素分泌的葡萄糖依赖性激活活性。Urolithin C 是 L 型 Ca2+通道开放剂,可增强 Ca2+的流入。它通过线粒体介导的途径诱导细胞凋亡,并刺激活性氧的形成。
TN6785 Dihydrocatalpol

(2S,3R,4S,5S,6R)-2-[[(1aS,1bS,2S,5aR,6S,6aS)-6-hydroxy-1a-(hydroxymethyl)-2,4,5,5a,6,6a-hexahydro-1bH-oxireno[5,6]cyclopenta[1,3-c]pyran-2-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol

Others Others
Dihydrocatalpol ((2S,3R,4S,5S,6R)-2-[[(1aS,1bS,2S,5aR,6S,6aS)-6-hydroxy-1a-(hydroxymethyl)-2,4,5,5a,6,6a-hexahydro-1bH-oxireno[5,6]cyclopenta[1,3-c]pyran-2-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol) 是一种从地黄中提取的天然产物。
TN6837 Syringopicroside

2-(4-hydroxyphenyl)ethyl (1S,4aS,7R)-7-methyl-6-oxo-1-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-1H,4aH,5H,6H,7H,7aH-cyclopenta[c]pyran-4-carboxylate

Others Others
Syringopicroside (2-(4-hydroxyphenyl)ethyl (1S,4aS,7R)-7-methyl-6-oxo-1-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-1H,4aH,5H,6H,7H,7aH-cyclopenta[c]pyran-4-carboxylate) 是一种来自 Syringa oblata Lindl (S. oblata) 的具有抗菌活性的天然药物。
T6S0052 Chelerythrine

Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine (Broussonpapyrine) 是一种天然生物碱,为有效、选择性的 Ca2+/磷脂依赖性PKC 拮抗剂,IC50值为 0.7 μM。它具有抗肿瘤、抗糖尿病、抗炎的活性。它抑制BclXL-Bak BH3肽结合,IC50为 1.5 μM,并从 BclXL 取代了 Bax。它诱导细胞凋亡和自噬。
T13108 Pamufetinib

H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115

VEGFR; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
Pamufetinib (TAS-115) 是VEGFR 和c-Met/HGFR 抑制剂,能够抑制 rVEGFR2 (IC50:30 nM)和 rMET (IC50:32 nM)的活性。
T3419 Chelerythrine chloride

白屈菜红碱,盐酸白屈菜红碱

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine chloride 是一种可渗透细胞的蛋白激酶 C 抑制剂,对磷酸盐受体具有竞争性,而对 ATP 是非竞争性的。它诱导细胞凋亡和自噬。
T7792 Hispidin

6-[(1E)-2-(3,4-二羟基苯基)乙烯基]-4-羟基-2H-吡喃-2-酮

Endogenous Metabolite; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
Hispidin 是来自裂蹄木层孔菌的酚类天然产物,是一种 PKC 抑制剂,具有很强的抗氧化、抗癌、抗糖尿病和抗痴呆作用。
T8301 Amaranth

Acid Red 27,酸性红 27

Others Others
Amaranth (Acid Red 27) 是一种阴离子染料, 可应用到天然和合成纤维、皮革、纸张及苯酚-甲醛树脂。它是一种暗红色至紫色的偶氮染料,可用作食品染料和化妆品。
T2185 L-Ascorbic acid 2-phosphate trisodium

L-抗坏血酸-2-磷酸三钠盐(维生素C),L-Ascorbic acid 2-phosphate trisodium salt,Sodium L-ascorbyl-2-phosphate,Sodium ascorbyl phosphate,2-Phospho-L-ascorbic acid trisodium salt,Sodium ascorbyl monophosphate,L-抗坏血酸-2-磷酸三钠盐

Reactive Oxygen Species; c-Met/HGFR; Endogenous Metabolite Immunology/Inflammation; Metabolism; NF-κB; Tyrosine Kinase/Adaptors
L-Ascorbic acid 2-phosphate trisodium (Sodium ascorbyl phosphate) 是长效的维生素 C 衍生物,能够刺激胶原蛋白的表达和形成。Sodium L-ascorbyl-2-phosphate 提高成骨细胞分化过程中 hASC 中的碱性磷酸酶活性和 runx2A 的表达,因此,能够促进人脂肪干细胞的成骨分化。
T6S1529 Cynarin

Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花

Antioxidant; Antiviral; Influenza Virus; Reactive Oxygen Species Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Cynarin (1,5-Dicaffeoylquinic acid) 是一种抗窒息剂,具有抗氧化、抗组胺和抗病毒等多种生物活性。
TN5525 Orientin 2''-O-rhamnoside

2''-O-Rhamnosylorientin,Luteolin 8-C-neohesperidoside

Orientin 2''-O-rhamnoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5525,CAS号为 81398-30-3。
TN5698 8-Glucosyl-5,7-dihydroxy-2-isopropylchromone

5,7-Dihydroxy-2-isopropylchromone 8-C-glucoside

8-Glucosyl-5,7-dihydroxy-2-isopropylchromone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5698,CAS号为 188785-44-6。
T83150 Ajugasterone C 2-acetate

Ajugasterone C 2-acetate,一种可从Cyanotis arachnoidea分离得到的蜕皮类固醇。
T82799 C-2′-Decoumaroylaloeresin G

C-2′-Decoumaroylaloeresin G (化合物8)为一种色酮糖苷,源自芦荟属植物。
TN3265 Yuehgesin C

8-(3-Ethoxy-2-hydroxy-3-methylbutyl)-7-methoxycoumarin

Others Others
Yuehgesin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3265,CAS号为 125072-68-6。
T2764 (S)-10-Hydroxycamptothecin

10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。
T5736 1,3-Dicaffeoylquinic acid

CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid

Reactive Oxygen Species; Akt; PI3K Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
1,3-Dicaffeoylquinic acid (CYNARIN) 是一种咖啡酰奎宁酸衍生物,具有抗氧化、自由基清除作用。
T4069 Fatsiaside C

2)-alpha-L-arabinopyranoside'>Oleanolic acid-3-O-beta-D-glucopyranosyl (1->2)-alpha-L-arabinopyranoside

Others Others
Fatsiaside C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T4069,CAS号为 60213-69-6。
T81397 Procyanidin C2

Procyanidine C2

Procyanidin C2,源自Fagopyrum dibotrys (D. Don) Hara,为酚苷类化合物。
T79941 Antimycin A2c

Apoptosis Apoptosis
Anticanceragent 141(compound AE)是一种针对HPV感染宫颈癌具有抑制作用的抗霉素生物碱。该化合物能够抑制宫颈癌HeLa细胞的增殖并导致细胞周期在S期停滞。Anticanceragent 141破坏线粒体功能,诱导caspase依赖性细胞凋亡,并激活ROS介导的泛素依赖性蛋白酶体系统,进而引起E6/E7癌蛋白的降解。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
T7060 Amantadine

1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine

Others Others
Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
T81363 Pseudolaric acid C2-O-β-D-glucoside

Pseudolaric acid C2-O-β-D-glucoside, 一种天然产物,来源于Pseudolarix kaempferi,并通过分离提取得到。
TN1201 25(S)-Ruscogenin-1-O-α-L-rhamnopyranosyl (1→2)-β-D-xylopyranoside

25(S)-鲁斯可皂苷元-1-O-Α-L-吡喃鼠李糖基-(1→2)-Β-D-吡喃木糖苷,山麦冬皂苷C,(1beta,3beta,25S)-3-Hydroxyspirost-5-en-1-yl 2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-xylopyranoside

Others Others
(1beta,3beta,25S)-3-Hydroxyspirost-5-en-1-yl 2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-xylopyranoside is a natural product
TN1321 6'-​O-​Cinnamoyl harpagide

6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷

Others Others
6'-O-Cinnamoylharpagide has anti-inflammatory activity.
TN1488 Chrysin 6-C-glucoside 8-C-arabinoside

Others Others
Chrysin 6-C-glucoside 8-C-arabinoside 是α±-葡萄糖苷酶抑制剂,α±-葡萄糖苷酶抑制剂广泛用于2型糖尿病的治疗。
TN1487 Chrysin 6-C-arabinoside 8-C-glucoside

Others Others
Chrysin 6-C-arabinoside 8-C-glucoside 是α±-葡萄糖苷酶抑制剂,α±-葡萄糖苷酶抑制剂广泛用于2型糖尿病的治疗。
T1192 Protoporphyrin IX

PPIX,原卟啉,原卟啉IX

Others; Endogenous Metabolite Metabolism; Others
Protoporphyrin IX (PPIX) 是一种四吡咯,是血红素、细胞色素 c 和叶绿素的代谢前体。
TN1977 Neochamaejasmine B

新狼毒素B

Antifection Microbiology/Virology
Neochamaejasmin B 是一种提取自Stellera chamaejasme L.的双黄酮化合物。它在 C-2/C-3 和 C-2″/C-3″ 位置具有顺反几何结构。
T2S1158 4,5-Dicaffeoylquinic acid

3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C

Others; HBV; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。
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天然产物

Ganoderic acid C2
Cat.No: TN1661
Synonym: 灵芝酸 C2
Target: Reductase, Histamine Receptor, Immunology/Inflammation related
Pseudolaric Acid C2
Cat.No: T13851
Synonym:
Target: Others
(E/Z)-Ginkgolic acid C17:2
Cat.No: TN2373
Synonym: Ginkgolic Acid C17:2
Target: Dehydrogenase
PSI-6130
Cat.No: T7607
Synonym: R 1656,2'-去氧-2'-氟-2'-C-甲基胞苷
Target: HCV Protease
2-C-Methyl-D-erythritol
Cat.No: TN2379
Synonym:
Target: Others
2''-O-Acetylsprengerinin C
Cat.No: TN2782
Synonym:
Target: Others
Moracin C
Cat.No: TN1949
Synonym: 桑辛素 C,5-(6-羟基-2-苯并呋喃基)-2-(3-甲基-2-丁烯基)-1,3-苯二醇
Target: ROS, NO Synthase
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-
Cat.No: TN7180
Synonym: 4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C
Target: Others
Malabaricone C
Cat.No: TN6772
Synonym:
Target: Others
Vitexin-2"-O-rhamnoside
Cat.No: T3671
Synonym: 牡荆素鼠李糖苷,牡荆素-2-O-鼠李糖苷,2''-O-Rhamnosylvitexin,Vitexin-2-O-rhaMnoside,Vitexin-2''-O-rhamnoside,Apigenin-8-C-glucoside
Target: Others
2'-O-Methylbroussonin C
Cat.No: TN2499
Synonym: 1-(4-Hydroxy-2-methoxyphenyl)-3-(4-hydroxy-3-prenylphenyl)propane
Target: Others
C2 Ceramide
Cat.No: T22644
Synonym: Ceramide
Target: Others
Ginsenoside Rb2
Cat.No: T3919
Synonym: Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2
Target: GPR, Others, Influenza Virus, Endogenous Metabolite
17-Hydroxy sprengerinin C
Cat.No: TN1195
Synonym: 17-羟基麦冬皂苷C
Target: BCL, Others, Caspase
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C
Cat.No: TN3301
Synonym:
Target: Others
Purpureaside C
Cat.No: TQ0054
Synonym:
Target: Others
2-C-Methyl-D-erythrono-1,4-lactone
Cat.No: TN2750
Synonym:
Target: Others
Licorice glycoside C2
Cat.No: T11848
Synonym: 甘草苷 C2
Target: Others
Saikosaponin B2
Cat.No: T3810
Synonym: 柴胡皂苷 B2,柴胡皂甙 B2
Target: Others, HCV Protease
Ginsenoside Rg2
Cat.No: T2873
Synonym: Chikusetsusaponin I,Panaxoside Rg2,人参皂苷Rg2,Prosapogenin C2,(20S)Ginsenoside Rg2,人参皂苷 Rg2
Target: Beta Amyloid, GSK-3, NF-κB
Urolithin C
Cat.No: TN7108
Synonym:
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, IGF-1R, Endogenous Metabolite
Dihydrocatalpol
Cat.No: TN6785
Synonym: (2S,3R,4S,5S,6R)-2-[[(1aS,1bS,2S,5aR,6S,6aS)-6-hydroxy-1a-(hydroxymethyl)-2,4,5,5a,6,6a-hexahydro-1bH-oxireno[5,6]cyclopenta[1,3-c]pyran-2-yl]oxy]-6-(hydroxymethyl)oxane-3,4,5-triol
Target: Others
Syringopicroside
Cat.No: TN6837
Synonym: 2-(4-hydroxyphenyl)ethyl (1S,4aS,7R)-7-methyl-6-oxo-1-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-1H,4aH,5H,6H,7H,7aH-cyclopenta[c]pyran-4-carboxylate
Target: Others
Chelerythrine
Cat.No: T6S0052
Synonym: Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine
Target: Apoptosis, BCL, PKC, Autophagy
Pamufetinib
Cat.No: T13108
Synonym: H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115
Target: VEGFR, c-Met/HGFR
Chelerythrine chloride
Cat.No: T3419
Synonym: 白屈菜红碱,盐酸白屈菜红碱
Target: Apoptosis, BCL, PKC, Autophagy
Hispidin
Cat.No: T7792
Synonym: 6-[(1E)-2-(3,4-二羟基苯基)乙烯基]-4-羟基-2H-吡喃-2-酮
Target: Endogenous Metabolite, PKC
Amaranth
Cat.No: T8301
Synonym: Acid Red 27,酸性红 27
Target: Others
L-Ascorbic acid 2-phosphate trisodium
Cat.No: T2185
Synonym: L-抗坏血酸-2-磷酸三钠盐(维生素C),L-Ascorbic acid 2-phosphate trisodium salt,Sodium L-ascorbyl-2-phosphate,Sodium ascorbyl phosphate,2-Phospho-L-ascorbic acid trisodium salt,Sodium ascorbyl monophosphate,L-抗坏血酸-2-磷酸三钠盐
Target: Reactive Oxygen Species, c-Met/HGFR, Endogenous Metabolite
Cynarin
Cat.No: T6S1529
Synonym: Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花
Target: Antioxidant, Antiviral, Influenza Virus, Reactive Oxygen Species
Orientin 2''-O-rhamnoside
Cat.No: TN5525
Synonym: 2''-O-Rhamnosylorientin,Luteolin 8-C-neohesperidoside
Target:
8-Glucosyl-5,7-dihydroxy-2-isopropylchromone
Cat.No: TN5698
Synonym: 5,7-Dihydroxy-2-isopropylchromone 8-C-glucoside
Target:
Ajugasterone C 2-acetate
Cat.No: T83150
Synonym:
Target:
C-2′-Decoumaroylaloeresin G
Cat.No: T82799
Synonym:
Target:
Yuehgesin C
Cat.No: TN3265
Synonym: 8-(3-Ethoxy-2-hydroxy-3-methylbutyl)-7-methoxycoumarin
Target: Others
(S)-10-Hydroxycamptothecin
Cat.No: T2764
Synonym: 10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT
Target: Apoptosis, Topoisomerase
1,3-Dicaffeoylquinic acid
Cat.No: T5736
Synonym: CYNARIN,1,3-二咖啡酰奎宁酸,Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1S,​3R,​4R,​5R)​-,1,3-O-Dicaffeoylquinic acid,1,5-Dicaffeoylquinic acid
Target: Reactive Oxygen Species, Akt, PI3K
Fatsiaside C
Cat.No: T4069
Synonym: 2)-alpha-L-arabinopyranoside'>Oleanolic acid-3-O-beta-D-glucopyranosyl (1->2)-alpha-L-arabinopyranoside
Target: Others
Procyanidin C2
Cat.No: T81397
Synonym: Procyanidine C2
Target:
Antimycin A2c
Cat.No: T79941
Synonym:
Target: Apoptosis
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
Amantadine
Cat.No: T7060
Synonym: 1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine
Target: Others
Pseudolaric acid C2-O-β-D-glucoside
Cat.No: T81363
Synonym:
Target:
25(S)-Ruscogenin-1-O-α-L-rhamnopyranosyl (1→2)-β-D-xylopyranoside
Cat.No: TN1201
Synonym: 25(S)-鲁斯可皂苷元-1-O-Α-L-吡喃鼠李糖基-(1→2)-Β-D-吡喃木糖苷,山麦冬皂苷C,(1beta,3beta,25S)-3-Hydroxyspirost-5-en-1-yl 2-O-(6-deoxy-alpha-L-mannopyranosyl)-beta-D-xylopyranoside
Target: Others
6'-​O-​Cinnamoyl harpagide
Cat.No: TN1321
Synonym: 6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷
Target: Others
Chrysin 6-C-glucoside 8-C-arabinoside
Cat.No: TN1488
Synonym:
Target: Others
Chrysin 6-C-arabinoside 8-C-glucoside
Cat.No: TN1487
Synonym:
Target: Others
Protoporphyrin IX
Cat.No: T1192
Synonym: PPIX,原卟啉,原卟啉IX
Target: Others, Endogenous Metabolite
Neochamaejasmine B
Cat.No: TN1977
Synonym: 新狼毒素B
Target: Antifection
4,5-Dicaffeoylquinic acid
Cat.No: T2S1158
Synonym: 3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C
Target: Others, HBV, Endogenous Metabolite
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