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1638

抑制剂 & 化合物

284

天然产物

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Cat. No. Product Name Target Signaling Pathways
T80644 DNA polymerase-IN-1

Antiviral; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation
DNA polymerase-IN-1 作为DNA聚合酶抑制剂,展现出对肿瘤细胞的抗增殖活性,其半抑制浓度(IC50)为20.7 μM。DNA polymerase-IN-1 抑制 Taq DNA 聚合酶,IC 值低于 250μM。DNA polymerase-IN-1 通过RT-PCR检测在体外显示出抗逆转录病毒活性,可用于研究氧化损伤和结直肠癌。
T3103 L67

DNA Ligase Inhibitor

DNA; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
L67 (DNA Ligase Inhibitor) 是一种竞争性人类 DNA 连接酶抑制剂,抑制 DNA 连接酶 I 和 III,IC50为10μM。
T31554 DNA-Spermidine

DA-51,DA 51,DA51,DNA Spermidine

DNA-spermidine influences the activity of restricted endonuclease from several bacterial species.
T1904 SGI-1027

DNA Methyltransferase Inhibitor II,SGI1027

Apoptosis; DNA Methyltransferase Apoptosis; Chromatin/Epigenetic
SGI-1027 (DNA Methyltransferase Inhibitor II) 是一种 DNA 甲基转移酶(DNMT)抑制剂,对以 poly(dI-dC) 为底物的 DNMT3B,DNMT3A 和 DNMT1 的IC50值分别为 7.5 μM,8 μM 和 12.5 μM。
T2433 NU 7026

NU7026,DNA-PK Inhibitor II,LY293646

Apoptosis; ATM/ATR; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
NU 7026 (DNA-PK Inhibitor II) 是一种新型特异性的DNA-PK 抑制剂,IC50为 0.23 μM,也抑制PI3K,IC50为 13 μM。
T15146 DNA2 inhibitor C5

Others Others
DNA2 inhibitor C5 是竞争性特异性的DNA2 核酸酶活性抑制剂(IC50:20 μM)。它能够抑制DNA 依赖性 ATPase、 DNA2 的核酸酶、解旋酶和 DNA 结合活性。它可用于研究奥正癌症。
T27194 DNA Primase Inhibitor-13

DNA Primase Inhibitor-13 is a novel inhibitor of DNA primase.
T79922 Taq DNA polymerase

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Taq DNA 聚合酶是一种在PCR过程中广泛使用的耐热性酶,由Thermus aquaticus细菌产生,其功能是在高温下合成DNA链。
T63442 DNA Gyrase-IN-2

DNA Gyrase-IN-2 是细菌 DNA 促旋酶 B 抑制剂,能作用于大肠杆菌 DNA 促旋酶(IC50: 3.29-10.49 μM)和结核分枝杆菌 DNA 促旋酶(IC50: 4.41-5.61 μM),表现出抗菌和抗结核作用。
T60961 LANA-DNA-IN-1

LANA-DNA-IN-1 是 LANA-DNA 的有效抑制剂,对 LBS2、LBS1 和 LBS3 的 IC50值分别为 8 μM、9μM 和 8μM。 LANA-DNA-IN-1 对野生型 LANA 显示出 53 μM 的 IC50值。LANA-DNA-IN-1 可用于研究感染。
T74340 DNA crosslinker 4 dihydrochloride

DNA crosslinker 4 (dihydrochloride) 作为高效的DNA小沟结合剂,对NCI-H460、A2780和MCF-7癌细胞表现出显著抑制活性,适用于抗癌研究。
T74338 DNA crosslinker 2 dihydrochloride

DNA crosslinker 2 (dihydrochloride)为一种高效DNA小沟结合剂,其结合亲和力(ΔTm)达1.2°C。该化合物对NCI-H460、A2780及MCF-7癌细胞展示出抑制活性,适用于抗癌研究。
T63681 DNA Gyrase-IN-1

DNA Gyrase-IN-1 是有效的、选择性的 DNA 促旋酶抑制剂 (IC50: 2.6 μM)。DNA Gyrase-IN-1 能够较好的抑制结核分枝杆菌 (Mtb) 的活性 (MIC: 0.49 μM)。DNA Gyrase-IN-1 能够用于研究结核病。
T74337 DNA crosslinker 1 dihydrochloride

DNA crosslinker 1 (dihydrochloride)作为有效DNA小沟结合剂,具有1.1°C的结合亲和力(ΔTm),适用于抗癌研究。
T79308 DNA polymerase-IN-3

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DNA polymerase-IN-3 (Compd 5b) 为香豆素衍生物,对 Taq DNA聚合酶具有抑制活性,适用于增值性疾病研究。
T61828 DNA-PK-IN-8

DNA-PK-IN-8(化合物DK1)是一种高效、选择性且口服活性的DNA依赖蛋白激酶 (DNA-PK) 抑制剂,其IC50值为0.8 nM。与Doxorubicin联合应用时,该化合物能在多种癌细胞中展现出协同的抗增殖效应,并能显著地抑制HL-60肿瘤生长。
T81953 LANA-DNA-IN-2

LANA-DNA-IN-2 (Compound 20) 是抑制潜伏期相关核抗原 (LANA) 与 DNA 相互作用的化合物。它适用于研究卡波西肉瘤相关疱疹病毒 (KSHV) 感染。
T74848 DNA Gyrase-IN-6

Antibacterial agent 138 是细菌 DNA 促旋酶和拓扑异构酶 IV 的苯并噻唑抑制剂。Antibacterial agent 138 表现出良好的溶解度和血浆蛋白结合。Antibacterial agent 138 对革兰氏阳性和革兰氏阴性菌株具有抗菌活性。Antibacterial agent 138 是一种双重 GyrB 和 ParE 抑制剂。
T79240 DNA gyrase B-IN-2

DNA gyrase B-IN-2 (Compound E) 是一款基于2-aminobenzothiazole的DNA gyrase B抑制剂,针对ESKAPE病原体显示出强效活性。该化合物在低纳摩尔浓度下表现出优异的DNA gyrase B抑制能力(IC50< 10 nM),具备对多种ESKAPE病原体的广谱抗菌作用。对于大部分革兰氏阳性菌,最低抑菌浓度(MIC)低于0.03 μg/mL;针对革兰氏阴性病原体如E. coli, Acinetobacter baumannii, Pseudomonas aeruginosa和Klebsiella pneumoniae,MIC为4 - 16 μg/mL。此化合物适用于感染性疾病的研究应用。
T62191 DNA-PK-IN-5

DNA-PK-IN-5 是一种 DNA-PK 的有效抑制剂。DNA-PK-IN-5 能够抑制 DNA-PKcs 活性,明显降低肿瘤 DNA 修复,并诱导细胞凋亡。DNA-PK-IN-5 能够提高肿瘤组织对放疗的敏感性,克服耐药问题,提高对多种实体瘤和血液肿瘤的抑制效果。
T62034 DNA-PK-IN-7

DNA-PK-IN-7 是有效的 DNA-PK 抑制剂,IC50为 1 nM (WO2021104277A1, compound 5)。
T78712 DNA Gyrase-IN-8

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DNA Gyrase-IN-8是一种高效的DNA gyrase抑制剂,其IC50为8.45 µM,同时展现出了抗菌活性。
T63395 DNA Gyrase-IN-5

DNA Gyrase-IN-5 是 DNA gyrase 的有效抑制剂 (IC50: 0.10 μM),对野生型和耐药株均有抗细菌(antibacterial)作用。
T62895 DNA Gyrase-IN-4

DNA Gyrase-IN-4 (compound 8p) 是一种 DNA 促旋酶的有效抑制剂 (IC50: 0.13 μM)。DNA Gyrase-IN-4 对金黄色葡萄球菌 (MIC: 0.05 μg/ml)、单核增生李斯特菌 (MIC: 0.05 μg/ml)、沙门氏菌 (MIC: 0.05 μg/ml) 和大肠杆菌 (MIC: 8 μg/ml) 具有较好的抗菌作用。
T82536 DNA polymerase-IN-4

DNA polymerase-IN-4 (Compd 5c),香豆素衍生物,显示出抗逆转录病毒活性,IC50为134.22 μM。
T12019 Methylproamine

Others Others
Methylproamine 是一种与DNA 结合的辐射保护剂,可以修复辐射诱导的短暂活性氧。
T61857 DNA-PK-IN-4

DNA-PK-IN-4 (WO2021209055A1, compound 27), an imidazolinone derivative compound, is a highly effective inhibitor of DNA-PK, specifically targeting DNA-PKcs activity. By inhibiting DNA-PKcs, the compound significantly impairs tumor DNA repair mechanisms and triggers apoptosis in cells. With its potential application in cancer research, DNA-PK-IN-4 holds promise for further investigation [1].
T61533 DNA-PK-IN-9

DNA-PK-IN-9 (also known as compound YK6) is a highly potent inhibitor of DNA-dependent protein kinase (DNA-PK), displaying an IC50 value of 10.47 nM. DNA-PK-IN-9 holds significant potential in anticancer research [1].
T61370 DNA-PK-IN-6

DNA-PK-IN-6, a robust DNA-PK inhibitor, effectively hampers the activity of DNA-PKcs, thereby significantly impairing the DNA repair mechanism in tumors and instigating apoptosis in cells. Additionally, DNA-PK-IN-6 amplifies the responsiveness of tumor tissues to radiotherapy, overcomes the challenge of drug resistance, and augments its inhibitory impact on a diverse range of solid and hematological tumors[1].
T79165 DNA-PK-IN-10

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
DNA-PK-IN-10是一种DNA-PK抑制剂, 主要应用于乳腺癌与非小细胞肺癌的研究。
T78866 DNA Gyrase-IN-9

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DNA Gyrase-IN-9 (compound 4j) 是一款抗细菌剂,作用于 DNA gyrase。该化合物对抑制革兰氏阳性菌的最小抑菌浓度(MIC)范围为 0.5-2 μg/mL,最小杀菌浓度(MBC)为 2-8 μg/mL。在金黄色葡萄球菌中,DNA Gyrase-IN-9 的 DNA gyrase 抑制半数有效浓度(IC50)为 6.29 μg/mL。
T4517 L189

DNA; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
L189 是一种人类 DNA 连接酶抑制剂,抑制 hLigI/III/IV,IC50值分别为5、9 和 5 μM。
T61937 DNA Gyrase-IN-3

DNA Gyrase-IN-3 (Compound 28) 是细菌DNA 旋转酶 B (bacterial DNA gyrase B) 抑制剂。DNA Gyrase-IN-3抑制大肠杆菌DNA 旋转酶的 IC50为5.41-15.64 μM。DNA Gyrase-IN-3显示出抗结核和抗菌活性。
T61633 DNA-PK-IN-2

DNA-PK-IN-2 is a highly effective inhibitor of DNA-dependent protein kinase (DNA-PK), which is a complex enzyme composed of Ku70/Ku80 heterodimer and DNA-PK catalytic subunit (DNA-PKcs). With its potential applications in cancer research, DNA-PK-IN-2 demonstrates promise as a valuable tool for studying cancer diseases [1].
T62648 DNA-PK-IN-1

DNA-PK-IN-1 是一种 DNA-PK 的有效抑制剂。DNA 依赖性蛋白激酶 (DNA-PK) 是一种由 Ku70/Ku80 异二聚体和 DNA 依赖性蛋白激酶催化亚基 (DNA-PKcs) 组成的 DNA-PK 酶复合物。DNA-PK-IN-1 具有潜力进行癌症疾病的研究。
T61751 DNA-PK-IN-3

DNA-PK-IN-3 is a highly potent inhibitor of DNA-PK. This compound exerts a synergistic effect when combined with radiotherapy and chemotherapy, resulting in enhanced therapeutic outcomes and significant inhibition of tumor growth. Furthermore, DNA-PK-IN-3 demonstrates remarkable efficacy in reducing damage to normal cells, effectively minimizing adverse side effects. Due to these compelling properties, DNA-PK-IN-3 holds great potential for cancer research applications[1].
T74339 DNA crosslinker 3 dihydrochloride

DNA crosslinker 3 (dihydrochloride) (compound 1) 为一种与DNA结合的小沟结合剂,其结合亲和力(ΔTm)达1.4°C,常用于抗癌研究。
T79307 DNA polymerase-IN-2

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DNA polymerase-IN-2 (Compd 3c)为香豆素衍生物,对Taq DNA聚合酶具有抑制作用,IC50为48.25 μM,适用于增殖性疾病研究。
T8873 Bractoppin

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Bractoppin 是一种BRCA1 (t)BRCT domain 识别磷酸肽的选择性抑制剂,IC50为 74 nM。它优先抑制 BRCA1 -tBRCT 依赖的 DNA 损伤。它减少 BRCA1 对 DNA 断裂片段的招募,进而抑制损伤诱导的 G2 期阻滞和重组酶 RAD51 的组装。
T15080 DC-05

DNA Methyltransferase; Histone Methyltransferase Chromatin/Epigenetic
DC-05 是一种DNMT1的抑制剂,IC50和Kd 值分别为 10.3 和 1.09 μM。
T11469 GSK-3484862

DNA Methyltransferase Chromatin/Epigenetic
GSK-3484862 是 有效的 DNA 甲基转移酶 Dnmt1的非共价抑制剂。GSK-3484862 通过诱导 DNA 低甲基化起抗癌作用。GSK-3484862 介导小鼠胚胎干细胞的整体去甲基化。
T36757 DMT-dU-CE Phosphoramidite

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DMT-dU-CE Phosphoramidite 是一个核苷分子,通常用于合成 DNADNA 测序试验。
T63360 DNA topoisomerase II inhibitor 1

DNA topoisomerase II inhibitor 1 是 DNA 拓扑异构酶 II 的有效抑制剂,能够将细胞周期停滞在亚 G1 期,并诱导细胞凋亡 (apoptosis) ,具有抗增值作用。
T0164 Oxaliplatin

L-OHP,奥沙利铂

DNA Alkylator/Crosslinker; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Oxaliplatin (L-OHP) 是一种 DNA 烷化剂,一种 DNA 合成抑制剂。Oxaliplatin 会导致 DNA 交联损伤,阻止 DNA 复制和转录并导致细胞死亡。Oxaliplatin 可以诱导细胞自噬。
T64012 DNA gyrase B-IN-1

DNA gyrase B-IN-1 是 DNA gyrase B 的有效抑制剂,表现出良好的结合亲和力和稳定性。DNA gyrase B-IN-1 能够抑制 P. aeruginosa/i> DNA gyrase B (IC50: 2.2 μM)。
T78776 DNA gyrase B-IN-3

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DNA gyrase B-IN-3(Compound A),作为一种细菌DNA gyrase B抑制剂(IC50: <10 nM),针对革兰氏阳性菌株表现出抗菌活性。
T4339 YU238259

DNA-PK; Others DNA Damage/DNA Repair; Others; PI3K/Akt/mTOR signaling
YU238259 是一种新型的同源依赖性 DNA 修复 (HDR) 抑制剂,在基于细胞的 GFP 报告基因检测中不抑制非同源末端连接 (NHEJ),可研究癌症。
T62389 14α-Demethylase/DNA Gyrase-IN-2

14α-Demethylase/DNA Gyrase-IN-2 (Compound 6a) 是一种 14α-Demethylase/DNA Gyrase 的有效抑制剂,具有抗菌作用。
T15789 LTURM34

DNA-PK; PI3K; PI4K DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
LTURM34 是一种 DNA-PK 抑制剂,IC50 为 34 nM。它在广泛的肿瘤细胞系中显示出有效的抗增殖活性,对 DNA-PK 的选择性比 PI3K 高 170 倍。
T5198 Bobcat339

盐酸Bobcat339,Bobcat339 hydrochloride

DNA Methyltransferase Chromatin/Epigenetic
Bobcat339 是一种基于胞嘧啶的选择性TET 酶抑制剂,抑制TET1和TET2的IC50值分别为 33 和 73 μM。它可作为靶向 DNA 甲基化和基因转录新疗法的起点,用于表观遗传学领域研究。

化合物

DNA polymerase-IN-1
Cat.No: T80644
Synonym:
Target: Antiviral, DNA/RNA Synthesis
L67
Cat.No: T3103
Synonym: DNA Ligase Inhibitor
Target: DNA, DNA/RNA Synthesis
DNA-Spermidine
Cat.No: T31554
Synonym: DA-51,DA 51,DA51,DNA Spermidine
Target:
SGI-1027
Cat.No: T1904
Synonym: DNA Methyltransferase Inhibitor II,SGI1027
Target: Apoptosis, DNA Methyltransferase
NU 7026
Cat.No: T2433
Synonym: NU7026,DNA-PK Inhibitor II,LY293646
Target: Apoptosis, ATM/ATR, DNA-PK, PI3K
DNA2 inhibitor C5
Cat.No: T15146
Synonym:
Target: Others
DNA Primase Inhibitor-13
Cat.No: T27194
Synonym:
Target:
Taq DNA polymerase
Cat.No: T79922
Synonym:
Target: DNA/RNA Synthesis
DNA Gyrase-IN-2
Cat.No: T63442
Synonym:
Target:
LANA-DNA-IN-1
Cat.No: T60961
Synonym:
Target:
DNA crosslinker 4 dihydrochloride
Cat.No: T74340
Synonym:
Target:
DNA crosslinker 2 dihydrochloride
Cat.No: T74338
Synonym:
Target:
DNA Gyrase-IN-1
Cat.No: T63681
Synonym:
Target:
DNA crosslinker 1 dihydrochloride
Cat.No: T74337
Synonym:
Target:
DNA polymerase-IN-3
Cat.No: T79308
Synonym:
Target: DNA/RNA Synthesis
DNA-PK-IN-8
Cat.No: T61828
Synonym:
Target:
LANA-DNA-IN-2
Cat.No: T81953
Synonym:
Target:
DNA Gyrase-IN-6
Cat.No: T74848
Synonym:
Target:
DNA gyrase B-IN-2
Cat.No: T79240
Synonym:
Target:
DNA-PK-IN-5
Cat.No: T62191
Synonym:
Target:
DNA-PK-IN-7
Cat.No: T62034
Synonym:
Target:
DNA Gyrase-IN-8
Cat.No: T78712
Synonym:
Target: DNA/RNA Synthesis
DNA Gyrase-IN-5
Cat.No: T63395
Synonym:
Target:
DNA Gyrase-IN-4
Cat.No: T62895
Synonym:
Target:
DNA polymerase-IN-4
Cat.No: T82536
Synonym:
Target:
Methylproamine
Cat.No: T12019
Synonym:
Target: Others
DNA-PK-IN-4
Cat.No: T61857
Synonym:
Target:
DNA-PK-IN-9
Cat.No: T61533
Synonym:
Target:
DNA-PK-IN-6
Cat.No: T61370
Synonym:
Target:
DNA-PK-IN-10
Cat.No: T79165
Synonym:
Target: DNA-PK
DNA Gyrase-IN-9
Cat.No: T78866
Synonym:
Target: DNA/RNA Synthesis
L189
Cat.No: T4517
Synonym:
Target: DNA, DNA/RNA Synthesis
DNA Gyrase-IN-3
Cat.No: T61937
Synonym:
Target:
DNA-PK-IN-2
Cat.No: T61633
Synonym:
Target:
DNA-PK-IN-1
Cat.No: T62648
Synonym:
Target:
DNA-PK-IN-3
Cat.No: T61751
Synonym:
Target:
DNA crosslinker 3 dihydrochloride
Cat.No: T74339
Synonym:
Target:
DNA polymerase-IN-2
Cat.No: T79307
Synonym:
Target: DNA/RNA Synthesis
Bractoppin
Cat.No: T8873
Synonym:
Target: Others, DNA/RNA Synthesis
DC-05
Cat.No: T15080
Synonym:
Target: DNA Methyltransferase, Histone Methyltransferase
GSK-3484862
Cat.No: T11469
Synonym:
Target: DNA Methyltransferase
DMT-dU-CE Phosphoramidite
Cat.No: T36757
Synonym:
Target: DNA/RNA Synthesis
DNA topoisomerase II inhibitor 1
Cat.No: T63360
Synonym:
Target:
Oxaliplatin
Cat.No: T0164
Synonym: L-OHP,奥沙利铂
Target: DNA Alkylator/Crosslinker, DNA/RNA Synthesis, Autophagy
DNA gyrase B-IN-1
Cat.No: T64012
Synonym:
Target:
DNA gyrase B-IN-3
Cat.No: T78776
Synonym:
Target: DNA/RNA Synthesis
YU238259
Cat.No: T4339
Synonym:
Target: DNA-PK, Others
14α-Demethylase/DNA Gyrase-IN-2
Cat.No: T62389
Synonym:
Target:
LTURM34
Cat.No: T15789
Synonym:
Target: DNA-PK, PI3K, PI4K
Bobcat339
Cat.No: T5198
Synonym: 盐酸Bobcat339,Bobcat339 hydrochloride
Target: DNA Methyltransferase
Cat. No. Product Name Target Signaling Pathways
T13592 Calf thymus DNA

DNA from calf thymus, Thymonucleic acid

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Calf thymus DNA (DNA from calf thymus, Thymonucleic acid) 是一种从牛胸腺中提取出来的高质量双链模板DNA,可广泛应用于DNA 结合抗癌剂和调节DNA 结构和功能的DNA 结合剂的研究。
T21498 Phleomycin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Phleomycin 是在链霉菌中发现的,引起 DNA 切割的抗癌糖肽抗生素之一。 它类似于博来霉素,它结合并插入 DNA 以破坏双螺旋的完整性。
T1068 Dithranol

1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Dithranol (cignoline) 是蒽醌衍生物,可破坏线粒体功能和结构,用于治疗皮肤病。
T7520 Deoxycytidine triphosphate

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Deoxycytidine triphosphate 是一种核苷三磷酸,是合成 DNA 的原料,可用于实时荧光定量 PCR、cDNA 合成和 DNA 测序。
T37101 1-Hydroxyanthraquinone

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
1-Hydroxyanthraquinone 是口服有效的天然产物,来源于植物 Tabebuia avellanedae,显示出致癌活性。
T6S0139 Neobavaisoflavone

Apoptosis; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Neobavaisoflavone 是一种从Psoralea corylifolia 的种子中分离出来的类黄酮。它具有抗炎,抗癌和抗氧化的作用。它在中至高浓度下可抑制 DNA 聚合酶,也可抑制血小板聚集。
T13969 Xanthopterin (hydrate)

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Xanthopterin hydrate 是东方大黄蜂翅膀中黄色颗粒的主要成分,是一种非共轭的蝶啶天然产物,在 386/456 nm 处产生特征性的激发光。 它可抑制 RNA 合成,引起大鼠肾脏生长和肥大。
TN2132 Quinizarin

1,4-Dihydroxyanthraquinone,1,4-二羟基蒽醌

Others; DNA/RNA Synthesis; Antifungal Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Quinizarin (1,4-Dihydroxyanthraquinone) 是一种杀菌剂和杀虫剂,可抑制肿瘤细胞生长。
T40179 Sodium Camptothecin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Sodium Camptothecin 是一种植物生物碱,具有抗肿瘤活性。它是可逆 RNA 合成抑制剂,可以抑制腺病毒的复制。它能抑制 DNA 合成,并引起细胞内预形成的病毒 DNA 断裂。
TWP2911 Thymidine

beta-胸苷,5-Methyldeoxyuridine,Deoxyribothymidine,DThyd,NSC 21548,Thymidin

Others; DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Others
Thymidine (DThyd) 是一种细胞同步剂,是脱氧核糖核酸的特殊前体。它可在 DNA 复制前在 G1/S 边界阻滞细胞,是DNA 合成抑制因子。
T0064 Adenine

Vitamin B4,腺嘌呤,6-Aminopurine

DNA/RNA Synthesis; Endogenous Metabolite; AChR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Neuroscience
Adenine (6-Aminopurine) 是一种嘌呤衍生物,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T12651 Rabdosiin

(+)-Rabdosiin

Others Others
Rabdosiin ((+)-Rabdosiin) 是一种分离自 Rabdosia japonicaHara 中的咖啡酸四聚体,具有抗过敏、抗 HIV 和抑制 DNA 拓扑异构酶作用。
T2S1635 3-Isomangostin

MTH1 DNA Damage/DNA Repair
3-Isomangostin 可从莽吉柿壳中提取的一种天然产物,是一种乙酰胆碱酯酶选择性抑制剂,也是一种有效的人醛糖还原酶抑制剂,IC50 为 3.48 uM。它抑制 MutT 同源物 1 (MTH1),IC50 为 52 nM。它具有清除自由基、抗疟原虫和抗癌的活性。
T5270 5-Methylcytosine

Others; DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Others
5-Methylcytosine 是一种存在于真核 DNA 中的甲基化核苷酸碱基。它是由 DNA 甲基转移酶作用形成的表观遗传修饰。
T3606 γ-Oryzanol

谷维素,Gamma-Oryzanol,Oliver,γ-谷维素,Gammariza

DNA Methyltransferase Chromatin/Epigenetic
γ-Oryzanol (Gamma-Oryzanol) 是一种从米糠油中分离出来的营养提取物,是含有甾醇和阿魏酸的混合物,有助于破坏皮肤中的自由基。它有效抑制小鼠纹状体中的 DNA 甲基转移酶(DNMTs)。 它抑制DNMT1和DNMT3a,IC50分别为 3.2 和 22.3 μM。
T3717 Hinokitiol

4-Isopropyltropolone,桧木醇,β-thujaplicin,β-桧木醇

DNA Methyltransferase; Virus Protease; Estrogen/progestogen Receptor; Nrf2 Chromatin/Epigenetic; Endocrinology/Hormones; Immunology/Inflammation; Microbiology/Virology
Hinokitiol (4-Isopropyltropolone) 是从日本扁柏中分离到的一种挥发油成分,可抑制紫外线 B 诱导的角质形成细胞凋亡,可调节雌激素受体信号传导并抑制人乳腺癌细胞的增殖。它具有抗感染、抗氧化及抗肿瘤等活性。
TN1134 Euscaphic acid

Apoptosis; LDL; PI3K; DNA/RNA Synthesis; NO Synthase; Prostaglandin Receptor Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; PI3K/Akt/mTOR signaling
Euscaphic acid 是来源于枣的一种三萜,是DNA 聚合酶抑制剂,可诱导细胞凋亡。它抑制小牛 DNA 聚合酶 α 和大鼠 DNA 聚合酶 β 的IC50值分别为 61 和 108 μM。
T5901 3-Hydroxy-2-methylpyridine

Others Others
3-Hydroxy-2-methylpyridine 是分离自可可碱提取物,可用于合成嘧啶。
T7457 5-Methyl-2'-deoxycytidine

5-Methyldeoxycytidine,5-甲基-2'-脱氧胞苷,5MedCyd

DNA Methyltransferase; Endogenous Metabolite Chromatin/Epigenetic; Metabolism
5-Methyl-2'-deoxycytidine (5MedCyd) 是嘧啶核苷,当掺入到单链 DNA 中时,可以顺式作用以从头发出信号。
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
T6225 Adenine hydrochloride

Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hydrochloride (6-Aminopurine hydrochloride) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T35455 N-Nitrosodiethylamine

Diethylnitrosamine,NDEA

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
N-Nitrosodiethylamine (NDEA) 是致癌物质二烷基硝胺。它主要存在于水、烟草烟雾、腌制食品、油炸食品以及许多酒精饮料中。它与 DNA 修复/复制相关的核酶的变化相关。
TN3110 5-Geranoxy-7-methoxycoumarin

Anti-infection; Antibacterial; Antifungal Microbiology/Virology
5-Geranoxy-7-methoxycoumarin 是一种香豆素。它诱导细胞凋亡,具有抗癌、抗真菌和抗菌活性。
T1339 5-Azacytidine

阿托胞苷,Azacitidine,NSC 102816,Mylosar,Ladakamycin,5-氮杂胞苷,5-AzaC

Nucleoside Antimetabolite/Analog; DNA Methyltransferase; Antibacterial; Antibiotic; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology
5-Azacytidine (Ladakamycin) 是一种胞苷核苷类似物,一种 DNA 甲基化抑制剂,具有特异性。5-Azacytidine 通过降低 DNA 甲基化水平调节基因表达。5-Azacytidine 可以诱导细胞自噬,具有抗肿瘤活性。
TQ0184 Chebulinic acid

ATPase; Proton pump; DNA/RNA Synthesis; Antibacterial; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Stem Cells
Chebulinic acid 是从诃子果中提取的一种天然产物,结核分枝杆菌 DNA 促旋酶的有效抑制剂。它也能抑制 SMAD-3 phosphorylation 和 H+ K+-ATPase 的活性。
T6S0232 Eriodictyol

圣草酚,Huazhongilexone

Influenza Virus; DNA/RNA Synthesis; Nrf2; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology
Eriodictyol (Huazhongilexone) 是从中草药中得到的一种黄酮类天然产物,具有抗氧化、抗炎和抗糖尿病作用。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 18 nM。它可诱导Nrf2信号通路。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T1508 Decitabine

Dacogen,NSC 127716,地西他滨,Deoxycytidine,5-Aza-2'-deoxycytidine

Apoptosis; Nucleoside Antimetabolite/Analog; DNA Methyltransferase Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair
Decitabine (Deoxycytidine) 是脱氧胞苷类似物,一种 DNA 甲基转移酶抑制剂,具有口服活性。Decitabine 具有抗肿瘤活性和抗代谢活性。Decitabine 诱导细胞周期阻滞和凋亡。
T3332 Isosteviol

异甜菊醇,(-)-Isosteviol

IL Receptor; Potassium Channel; TNF; NF-κB; Reactive Oxygen Species; COX; Topoisomerase Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Isosteviol ((-)-Isosteviol) 是一种常见的天然甜味剂,属于四环二萜糖苷,是甜菊糖苷通过酸催化水解产生的。它抑制 DNA 聚合酶和 DNA 拓扑异构酶,具有抗菌、抗癌和抗结核作用。
T0974 Novobiocin Sodium

Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T1507 Streptozocin

STZ,Streptozotocin,链脲佐菌素,NSC-85998,链脲菌素,U 9889

DNA Alkylator/Crosslinker; DNA Alkylation; DNA/RNA Synthesis; Antibacterial; Antibiotic; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Streptozocin (NSC-85998) 是一种抗生素,可诱导 DNA 甲基化。Streptozocin 对产生胰岛素的胰岛 B 细胞具有毒性,常用于构建 1 型糖尿病的动物模型。该产品在溶液中不稳定,建议现配现用。
T6369 Adenine hemisulfate

硫酸腺嘌呤,Diadenine sulphate,Adenine sulfate,Adeninsulfat,1H-嘌呤-6-胺硫酸盐

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hemisulfate (Diadenine sulphate) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T16674 Pseudouridine

Endogenous Metabolite Metabolism
Pseudouridine 是非编码 RNA 中丰富的修饰核苷,通过稳定 RNA 结构增强核糖体 RNA 和的转移 RNA 功能。
T4593 ISOPIMPINELLIN

5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen

Antiviral; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology
Isopimpinellin (4,9-Dimethoxypsoralen) 是从 Pimpinella saxifrage 根部分离得到的一种天然产物,具有抗病毒和抗利什曼病活性。
TN1637 Eurycomalactone

Anti-infection; NF-κB Microbiology/Virology; NF-κB
Eurycomalactone 是一种NF-κB 抑制剂,IC50=0.5 μM,是一种天然产物。它可抑制蛋白合成,降低 cyclin D1 蛋白水平,但对 TNFα 诱导的 IκBα 降解或 IKKα/β 和 IκBα 的磷酸化水平没有作用。
TWS1977 Kamebakaurin

尾叶香茶菜丙素,Kamebakaurine

NF-κB NF-κB
Kamebakaurin (Kamebakaurine) 是一种提取自Isodon japonicus 中的天然产物,是一种NF-κB 的抑制剂,能够抑制 p50 的 DNA 结合活性。
T9715 Aplidine

SARS-CoV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Aplidine 是有效的eEF1A2(KD=80 nM) 靶向的抗癌药物。Aplidine 具有抗病毒活性,抑制SARS-CoV-2的 IC90为 0.88 nM。Aplidine 在多发性骨髓瘤,晚期癌症及 COVID-19 领域有研究的价值。
T2998 Dihydromyricetin

Ampelopsin,Ampeloptin,二氢杨梅素

Influenza Virus; GABA Receptor; DNA/RNA Synthesis; mTOR; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
Dihydromyricetin (Ampelopsin) 是一种来自 Ampelopsis Grossedentata 的天然抗氧化剂类黄酮,是二氢嘧啶酶抑制剂,IC50 为 48 μM。它通过抑制mTOR 信号从而激活自噬。它还是流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 22 μM。
T6995 Ochromycinone

STA 21,STA21,STA-21

Antibacterial; STAT JAK/STAT signaling; Microbiology/Virology; Stem Cells
Ochromycinone (STA 21) 是一种天然抗生素,也是一种 STAT3抑制剂。它可抑制 STAT3DNA 结合活性,STAT3二聚化。它具有抗癌和抗菌活性。
T13791 N2-methylguanine

6-羟基-2-氨甲基嘌呤

DNA/RNA Synthesis; Endogenous Metabolite; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
N2-methylguanine (N2-methylguanine) 是一种在人体体液中发现的内源性甲基化核苷,是一种修饰的核苷。
T7004 Tubercidin

结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine

Influenza Virus; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Tubercidin (Sparsomycin A) 是从Streptomyces tubercidicus 得到的抗生素,抑制粪链球菌生长的IC50值为 0.02 μM。它是腺苷磷酸化酶的弱抑制剂,并干扰腺苷和 AMP 的磷酸化。它有抗病毒作用。
T5368 Eicosapentaenoic Acid

Histone Demethylase; Others; Endogenous Metabolite Chromatin/Epigenetic; Metabolism; Others
Eicosapentaenoic Acid 是一种 ω-3 脂肪酸。
TN1097 β-Boswellic acid

Beta-boswellic acid,β-乳香酸

Lipoxygenase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
β-Boswellic acid (Beta-boswellic acid) 是从乳香的树胶脂中分离出来的一种天然产物。它是 5-脂氧合酶(5-LO) 产物形成的非还原型抑制剂,其直接与 5-LO 相互作用或阻断其易位。具有抗癌、抗肿瘤和抗高血脂活性。
T6116 Bleomycin Sulfate

Blenoxane,硫酸博来霉素,硫酸博莱霉素,NSC125066

DNA/RNA Synthesis; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Bleomycin Sulfate (Blenoxane) 是一种糖肽抗生素,一种 DNA 合成抑制剂。Bleomycin Sulfate 可以引起 DNA 链断裂而不引起 RNA 链断裂。Bleomycin Sulfate 具有抗肿瘤活性。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
T3343 5-methoxyflavone

5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
5-methoxyflavone (5-methoxy-2-phenylchromen-4-one) 是一种类黄酮,是DNA 聚合酶 β 的抑制剂和 β-淀粉样蛋白毒性的神经保护剂。它通过调控嗜离子 GABAA 受体,起到镇静中枢神经系统的作用。
T0909 Nalidixic acid

萘啶酸,NSC-82174

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Nalidixic acid (NSC-82174) 是一种喹诺酮类抗生素,对革兰氏阳性和革兰氏阴性细菌有效。它在较低浓度下有抑菌作用,而在较高浓度下有杀菌作用。它抑制 DNA 促旋酶和拓扑异构酶 IV 的亚基,并可逆地阻止易感细菌中的 DNA 复制。
T6758 Anisomycin

茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; JNK Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK; Microbiology/Virology
Anisomycin (NSC-76712) 是一种从各种链霉菌属中分离出来的抗生素。 它通过抑制肽基转移酶或 80S 核糖体系统来干扰蛋白质和 DNA 合成。
T40426 Cytidine 5'-diphosphate trisodium salt

CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐

Others Others
Cytidine 5'-diphosphate trisodium salt (CDP) 可通过尿苷单磷酸激酶 (UMPK) 催化将磷酸基从 ATP 转移到胞苷一磷酸 (CMP) 生成用于合成 DNA 和 RNA 的胞苷三磷酸。
T38427 dUTP trisodium

2'-Deoxyuridine-5'-triphosphate trisodium salt,Deoxyuridine triphosphate

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
dUTP trisodium (Deoxyuridine triphosphate) 是在 5'-位具有三磷酸基团的脱氧尿苷磷酸盐,可用于 PCR。
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天然产物

Calf thymus DNA
Cat.No: T13592
Synonym: DNA from calf thymus, Thymonucleic acid
Target: DNA/RNA Synthesis
Phleomycin
Cat.No: T21498
Synonym:
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Dithranol
Cat.No: T1068
Synonym: 1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin
Target: Others, DNA/RNA Synthesis
Deoxycytidine triphosphate
Cat.No: T7520
Synonym:
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, Endogenous Metabolite
1-Hydroxyanthraquinone
Cat.No: T37101
Synonym:
Target: DNA/RNA Synthesis
Neobavaisoflavone
Cat.No: T6S0139
Synonym:
Target: Apoptosis, DNA/RNA Synthesis
Xanthopterin (hydrate)
Cat.No: T13969
Synonym:
Target: Others, DNA/RNA Synthesis
Quinizarin
Cat.No: TN2132
Synonym: 1,4-Dihydroxyanthraquinone,1,4-二羟基蒽醌
Target: Others, DNA/RNA Synthesis, Antifungal
Sodium Camptothecin
Cat.No: T40179
Synonym:
Target: DNA/RNA Synthesis
Thymidine
Cat.No: TWP2911
Synonym: beta-胸苷,5-Methyldeoxyuridine,Deoxyribothymidine,DThyd,NSC 21548,Thymidin
Target: Others, DNA/RNA Synthesis, Endogenous Metabolite
Adenine
Cat.No: T0064
Synonym: Vitamin B4,腺嘌呤,6-Aminopurine
Target: DNA/RNA Synthesis, Endogenous Metabolite, AChR
Rabdosiin
Cat.No: T12651
Synonym: (+)-Rabdosiin
Target: Others
3-Isomangostin
Cat.No: T2S1635
Synonym:
Target: MTH1
5-Methylcytosine
Cat.No: T5270
Synonym:
Target: Others, DNA/RNA Synthesis, Endogenous Metabolite
γ-Oryzanol
Cat.No: T3606
Synonym: 谷维素,Gamma-Oryzanol,Oliver,γ-谷维素,Gammariza
Target: DNA Methyltransferase
Hinokitiol
Cat.No: T3717
Synonym: 4-Isopropyltropolone,桧木醇,β-thujaplicin,β-桧木醇
Target: DNA Methyltransferase, Virus Protease, Estrogen/progestogen Receptor, Nrf2
Euscaphic acid
Cat.No: TN1134
Synonym:
Target: Apoptosis, LDL, PI3K, DNA/RNA Synthesis, NO Synthase, Prostaglandin Receptor
3-Hydroxy-2-methylpyridine
Cat.No: T5901
Synonym:
Target: Others
5-Methyl-2'-deoxycytidine
Cat.No: T7457
Synonym: 5-Methyldeoxycytidine,5-甲基-2'-脱氧胞苷,5MedCyd
Target: DNA Methyltransferase, Endogenous Metabolite
Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Adenine hydrochloride
Cat.No: T6225
Synonym: Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride
Target: DNA/RNA Synthesis, Endogenous Metabolite
N-Nitrosodiethylamine
Cat.No: T35455
Synonym: Diethylnitrosamine,NDEA
Target: DNA/RNA Synthesis
5-Geranoxy-7-methoxycoumarin
Cat.No: TN3110
Synonym:
Target: Anti-infection, Antibacterial, Antifungal
5-Azacytidine
Cat.No: T1339
Synonym: 阿托胞苷,Azacitidine,NSC 102816,Mylosar,Ladakamycin,5-氮杂胞苷,5-AzaC
Target: Nucleoside Antimetabolite/Analog, DNA Methyltransferase, Antibacterial, Antibiotic, Autophagy
Chebulinic acid
Cat.No: TQ0184
Synonym:
Target: ATPase, Proton pump, DNA/RNA Synthesis, Antibacterial, TGF-beta/Smad
Eriodictyol
Cat.No: T6S0232
Synonym: 圣草酚,Huazhongilexone
Target: Influenza Virus, DNA/RNA Synthesis, Nrf2, Endogenous Metabolite
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Decitabine
Cat.No: T1508
Synonym: Dacogen,NSC 127716,地西他滨,Deoxycytidine,5-Aza-2'-deoxycytidine
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA Methyltransferase
Isosteviol
Cat.No: T3332
Synonym: 异甜菊醇,(-)-Isosteviol
Target: IL Receptor, Potassium Channel, TNF, NF-κB, Reactive Oxygen Species, COX, Topoisomerase
Novobiocin Sodium
Cat.No: T0974
Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin
Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy
Streptozocin
Cat.No: T1507
Synonym: STZ,Streptozotocin,链脲佐菌素,NSC-85998,链脲菌素,U 9889
Target: DNA Alkylator/Crosslinker, DNA Alkylation, DNA/RNA Synthesis, Antibacterial, Antibiotic, Autophagy
Adenine hemisulfate
Cat.No: T6369
Synonym: 硫酸腺嘌呤,Diadenine sulphate,Adenine sulfate,Adeninsulfat,1H-嘌呤-6-胺硫酸盐
Target: DNA/RNA Synthesis, Endogenous Metabolite
Pseudouridine
Cat.No: T16674
Synonym:
Target: Endogenous Metabolite
ISOPIMPINELLIN
Cat.No: T4593
Synonym: 5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen
Target: Antiviral, DNA/RNA Synthesis, Parasite
Eurycomalactone
Cat.No: TN1637
Synonym:
Target: Anti-infection, NF-κB
Kamebakaurin
Cat.No: TWS1977
Synonym: 尾叶香茶菜丙素,Kamebakaurine
Target: NF-κB
Aplidine
Cat.No: T9715
Synonym:
Target: SARS-CoV, DNA/RNA Synthesis
Dihydromyricetin
Cat.No: T2998
Synonym: Ampelopsin,Ampeloptin,二氢杨梅素
Target: Influenza Virus, GABA Receptor, DNA/RNA Synthesis, mTOR, Autophagy
Ochromycinone
Cat.No: T6995
Synonym: STA 21,STA21,STA-21
Target: Antibacterial, STAT
N2-methylguanine
Cat.No: T13791
Synonym: 6-羟基-2-氨甲基嘌呤
Target: DNA/RNA Synthesis, Endogenous Metabolite, Antibacterial
Tubercidin
Cat.No: T7004
Synonym: 结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine
Target: Influenza Virus, DNA/RNA Synthesis, Antibacterial, Antibiotic
Eicosapentaenoic Acid
Cat.No: T5368
Synonym:
Target: Histone Demethylase, Others, Endogenous Metabolite
β-Boswellic acid
Cat.No: TN1097
Synonym: Beta-boswellic acid,β-乳香酸
Target: Lipoxygenase, DNA/RNA Synthesis
Bleomycin Sulfate
Cat.No: T6116
Synonym: Blenoxane,硫酸博来霉素,硫酸博莱霉素,NSC125066
Target: DNA/RNA Synthesis, Antibiotic
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
5-methoxyflavone
Cat.No: T3343
Synonym: 5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮
Target: DNA/RNA Synthesis
Nalidixic acid
Cat.No: T0909
Synonym: 萘啶酸,NSC-82174
Target: Topoisomerase, Antibacterial, Antibiotic
Anisomycin
Cat.No: T6758
Synonym: 茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, JNK
Cytidine 5'-diphosphate trisodium salt
Cat.No: T40426
Synonym: CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐
Target: Others
dUTP trisodium
Cat.No: T38427
Synonym: 2'-Deoxyuridine-5'-triphosphate trisodium salt,Deoxyuridine triphosphate
Target: DNA/RNA Synthesis
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