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230

抑制剂 & 化合物

52

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Cat. No. Product Name Target Signaling Pathways
T9882 RUVBL1/2 ATPase-IN-1

Others Others
RUVBL1/2 ATPase-IN-1 是一种有效的 RUVBL1/2 ATPase 抑制剂,IC50 值分别为 6.0 和 7.7 μM。 RUVBL1/2 ATPase-IN-1 可用于癌症疾病的研究。
T83967 ATPase-IN-3

ATPase Membrane transporter/Ion channel
ATPase-IN-3 是一种 ATP 酶 (ATPase) 抑制剂,可用于研究与代谢相关的疾病。
T61553 ATPase-IN-2

ATPase-IN-2 is a compound that acts as an inhibitor of ATPase, with an IC50 value of 0.9 μM. It also inhibits the glycohydrolase activity of C. difficile toxin B (TcdB) with an AC50 value of 30.91 μM. ATPase-IN-2 is commonly utilized in ATP-related research [1].
T0712 Suloctidil

ATPase; Platelet aggregation Membrane transporter/Ion channel; Others
Suloctidil 是一种外周血管扩张剂,作用于大鼠脑突触, 影响Na+/ K+ ATP 酶活性和膜流动性,可治疗痴呆和血栓形成病症。
T6443 Chloroprocaine hydrochloride

盐酸氯普鲁卡因,Chloroprocaine HCl

ATPase; Others Membrane transporter/Ion channel; Others
Chloroprocaine hydrochloride (Chloroprocaine HCl) 是一种 Na/K-ATPase 活性抑制剂,IC50为 13 mM,可阻断外周神经。
T20626 Esomeprazole

Proton pump; Cysteine Protease Membrane transporter/Ion channel; Proteases/Proteasome
Esomeprazole 是奥美拉唑(omeprazole) 的S-异构体,抑制溶酶体半胱氨酸蛋白酶legumain,防止癌症转移。它是一种质子泵抑制剂(PPI)。
T0490 Chlorpropamide

Diabinese,氯磺丙脲

ATPase; ABC Membrane transporter/Ion channel
Chlorpropamide (Diabinese) 是口服降糖剂,可用于研究非胰岛素依赖型糖尿病。
T9008 NPD8733

Others Others
NPD8733 是癌细胞增强的成纤维细胞迁移抑制剂。它是与多种细胞活动 (AAA+) 蛋白家族相关的 ATP 酶的成员,能够与含 valosin 的蛋白 (VCP)/p97特异性结合,对癌症疾病具有潜在的研究价值。
T2176 2,3-Butanedione 2-Monoxime

Diacetyl monoxime,2,3-Butanedione-2-monoxime

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
2,3-Butanedione 2-Monoxime (Diacetyl monoxime) 是一种肌球蛋白 ATP 酶(myosin ATPase) 抑制剂。它诱导肌质网 Ca2+释放,能够有效抑制骨骼肌和心肌收缩。
T9230 KM 91104

ATPase Membrane transporter/Ion channel
KM 91104 是一种细胞通透性 V-ATPase 抑制剂,选择性作用于 V-ATPase 的 a3-b2 亚单位。
T3293 Apoptozole

Apoptosis Activator VII

Apoptosis; HSP Apoptosis; Cytoskeletal Signaling; Metabolism
Apoptozole (Apoptosis Activator VII) 是一种Hsc70和Hsp70的 ATPase 结构域抑制剂,可诱导凋亡,Kd 值分别为 0.21 和 0.14 μM。
T6796 CB-5083

CB5083,CB 5083

p97 Ubiquitination
CB-5083 是一种有效的、选择性的、可口服的 p97 AAA ATPase 抑制剂,IC50为 11 nM。
T9168 NSC 617145

NSC617145,NSC-617145

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
NSC 617145 (NSC617145) 是一种 WRN 解旋酶抑制剂,IC50值为 230 nM。它以浓度依赖性方式抑制 WRN 解旋酶的 ATP 酶,并诱导双链断裂和染色体异常。
T36816 S-trityl-L-Cysteine

STLC

Kinesin Cytoskeletal Signaling
S-Trityl-L-cysteine 是别构驱动蛋白Eg5的选择性抑制剂。rityl-L-cysteine 抑制基础 ATPase 活性的IC50为 1 μM,抑制微管激活的 ATPase 活性的IC50为 140 nM。S-Trityl-L-cysteine 显示出抗肿瘤活性。
T6700 Tenatoprazole

泰妥拉唑,TU-199

Proton pump Membrane transporter/Ion channel
Tenatoprazole (TU-199) 是一种口服有效的,基于咪唑吡啶的质子泵抑制剂。它抑制猪胃H+/K+-ATP 酶活性,IC50为6.2 μM。它阻断泛素与 ESCRT-1 因子 Tsg101 的相互作用,抑制几种包膜病毒的产生,包括 EBV。
T6953 Prilocaine

Citanest,丙胺卡因,Propitocaine,NSC 40027

ATPase; Sodium Channel Membrane transporter/Ion channel
Prilocaine (NSC-40027) 是一种氨基酰胺类局部麻醉剂,作用于神经元膜上的钠通道并限制癫痫发作的扩散。它是Na/K-ATPase 抑制剂,具有神经毒性作用。
T2686L Esomeprazole Sodium

埃索美拉唑钠,(S)-Omeprazole sodium

ATPase; Proton pump Membrane transporter/Ion channel
Esomeprazole Sodium ((S)-Omeprazole sodium) 是一种口服有效的活性质子泵抑制剂。Esomeprazole sodium 通过抑制胃壁细胞中的 H+, K+-ATPase 来降低酸分泌,在胃食管反流疾病中有研究价值。Esomeprazole 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T2621 Rostafuroxin

PST 2238

ATPase; RSV Membrane transporter/Ion channel; Microbiology/Virology
Rostafuroxin (PST 2238) 是洋地黄毒苷衍生物,是一种口服有效的 Na+,K+-ATPase 抑制剂,具有抗高血压和抗 RSV 活性,用于研究治疗原发性高血压的试验。
T0796 Prilocaine hydrochloride

Prilocaine HCl,Propitocaine hydrochloride,Xylonest,盐酸丙胺卡因

ATPase; Sodium Channel Membrane transporter/Ion channel
Prilocaine hydrochloride (Prilocaine HCl) 是一种氨基酰胺类局部麻醉剂,作用于神经元膜上的钠通道并限制癫痫发作的扩散。它是Na/K-ATPase 抑制剂,具有神经毒性作用。
T1734 Rabeprazole Sulfide

雷贝拉唑相关物质E,Rabeprazole Related Compound E

Proton pump; Antibacterial Membrane transporter/Ion channel; Microbiology/Virology
Rabeprazole Sulfide (Rabeprazole Related Compound E) 是 Rabeprazole 的活性代谢产物。Rabeprazole 是一种质子泵抑制剂类的抗溃疡药物,有效抑制幽门螺旋杆菌的活性,可通过与胃壁细胞中的(H+/K+)-ATPase 相互作用来抑制胃酸分泌,可研究各种消化系统疾病。
T10616 BRM/BRG1 ATP Inhibitor-1

Epigenetic Reader Domain Chromatin/Epigenetic
BRM/BRG1 ATP Inhibitor-1 是变构双 Brahma 同源物 (BRM)/SWI/SNF 相关的基质相关肌动蛋白依赖性调节剂,染色质亚家族 A 成员 2 和 BRG1/SMARCA4 ATP 酶活性抑制剂,IC50值低于 0.005 μM。
T7144 BTS

N-Tosylbenzylamine,N-苄基-对甲苯磺酸胺,N-Benzyl-p-toluenesulfonamide

ATPase; Myosin Cytoskeletal Signaling; Membrane transporter/Ion channel
BTS (N-Tosylbenzylamine) 是一种选择性骨骼肌肌球蛋白 II 亚片段 1 (S1) ATPase 活性抑制剂,可特异性抑制骨骼肌快速纤维的收缩。它对肌动蛋白和 Ca2+刺激的肌球蛋白 S1 ATPase 的 IC50值约为 5 µM。
T2686 Esomeprazole Magnesium

(S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium

ATPase; Proton pump Membrane transporter/Ion channel
Esomeprazole Magnesium (NEXIUM) 是一种口服有效的 H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病中具有研究价值。Esomeprazole magnesium 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T6928 Pantoprazole

SKF96022,泮托拉唑,BY1023

Apoptosis; Proton pump; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel
Pantoprazole (BY1023) 是一种质子泵抑制剂,用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。
T8386 Esomeprazole Magnesium trihydrate

埃索美拉唑镁三水合物,埃索美拉唑镁(三水),(S)-Omeprazole magnesium trihydrate

Proton pump Membrane transporter/Ion channel
Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) 是一种口服有效的H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病的研究中具有价值。它是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T1651 Rabeprazole sodium

Dexrabeprazole Sodium,LY307640 sodium,Habeprazole Sodium,雷贝拉唑钠,Rebeprazole sodium,Aciphex Sodium

Apoptosis; Proton pump Apoptosis; Membrane transporter/Ion channel
Rabeprazole sodium (Habeprazole Sodium) 是一种质子泵抑制剂,不可逆地抑制胃 H+/K+-ATPase,可研究胃溃疡和胃食管反流。它诱导细胞凋亡,也抑制尿苷核苷核糖水解酶 ,IC50为 0.3 μM。
T0161 Pantoprazole Sodium Hydrate

SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)

Apoptosis; Potassium Channel; Proton pump; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel
Pantoprazole Sodium Hydrate (BY1023 (sodium hydrate)) 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑,是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T6929 Pantoprazole sodium

Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc

Apoptosis; Others; Proton pump; HIF; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others
Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T27812 Leminoprazole

ATPase Membrane transporter/Ion channel
Leminoprazole 是一种可口服的 H+,K(+)-ATPase 抑制剂,可保护胃黏膜细胞免受各种细胞损伤,可用于治疗胃溃疡。
T7540 2,5-Di-tert-butylhydroquinone

BHQ,2,5-二特丁基对苯二酚

Calcium Channel; Lipoxygenase; COX Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
2,5-Di-tert-butylhydroquinone (BHQ) 是一种有效和选择性的内质网 Ca2+-ATPase 抑制剂,可调节5-LO 以及COX-2活性,IC50分别为 1.8 和 14.1 μM。
T22280 BRITE-338733

BRITE338733

ATPase; Antibacterial Membrane transporter/Ion channel; Microbiology/Virology
BRITE-338733 是一种新型ATPase 抑制剂,抑制 RecA 在细菌中的表达,IC50 值为 4.7 µM,用于治疗细菌感染。
T2404 Vonoprazan fumarate

富马酸沃诺拉赞,TAK-438

ATPase Membrane transporter/Ion channel
Vonoprazan fumarate (TAK-438) 是一种新型 P-CAB(钾竞争性酸阻滞剂),可可逆地抑制 H+/K+、ATP 酶。
T7134 Mavacamten

MYK-461,SAR439152

Myosin Cytoskeletal Signaling
Mavacamten (MYK-461) 是一种可口服的心肌肌球蛋白 ATP 酶抑制剂,在牛心脏和人心脏中的IC50值分别为 490和711 nM。
T21254 Vonoprazan Fumarate

TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞

Proton pump Membrane transporter/Ion channel
Vonoprazan Fumarate (TAK438) 是质子泵的有效抑制剂,是口服有效的高效钾竞争性酸阻断剂,具有抗分泌活性。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50为 19 nM。它被开发用于研究酸相关疾病,如消化性溃疡和胃食管反流病。
T17030 Tegoprazan

ATPase; Proton pump Membrane transporter/Ion channel
Tegoprazan 是一种口服有效的、高选择性胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,能够控制胃酸分泌和运动,在体外检测的对猪、犬、人的 H+/K+-ATP 酶的 IC50为0.29-0.52 μM。
T9553 8-[(2,6-dimethylbenzyl)amino]-2,3-dimethylimidazo[1,2-a]pyridine-6-carboxylic acid

Others Others
8-[(2,6-dimethylbenzyl)amino]-2,3-dimethylimidazo[1,2-a]pyridine-6-car 是一种 H+/K+ ATPase 抑制剂,IC50=0.38μM。
T2189 Sodium orthovanadate

Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate

ATPase; Phosphatase Membrane transporter/Ion channel; Metabolism
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。
T16865 SCH28080

ATPase; Proton pump Membrane transporter/Ion channel
SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂,具有抗溃疡活性、抗分泌和细胞保护活性。
T12503 (+)-Blebbistatin

Others Others
(+)-Blebbistatin 是 (–)-Blebbistatin 的非活性对映异构体。 (–)-Blebbistatin 是一种选择性肌球蛋白 II ATPase 抑制剂。
T7373 CDN1163

Calcium Channel Membrane transporter/Ion channel; Metabolism
CDN1163 是肌膜/内质网 Ca2+-ATPase (SERCA)的变构激活剂,可改善 Ca2+稳态,可减轻糖尿病和代谢紊乱。
T60032 BRM/BRG1 ATP Inhibitor-2

Epigenetic Reader Domain Chromatin/Epigenetic
BRM/BRG1 ATP Inhibitor-2 是 BRG1/BRM ATPase 的抑制剂,可用于治疗 BAF 相关疾病的研究。
T17313 (+)-SJ733

SJ000557733

ATPase; Parasite Membrane transporter/Ion channel; Microbiology/Virology
(+)-SJ733 (SJ000557733) 是一种有效的 Na+-ATPase PfATP4 抑制剂,具有抗疟活性,可用于研究疟疾。
T67763 PK095

ATPase Membrane transporter/Ion channel
PK095是一个基于胍的F1F0-ATPase 抑制剂家族。
T2039 GSK-923295

Apoptosis; Kinesin Apoptosis; Cytoskeletal Signaling
GSK923295 是一种特异性的变构着丝粒相关蛋白-E 驱动蛋白 ATPase 活性抑制剂,作用于人类和犬类此酶,Ki 分别为 3.2±0.2 nM 和 1.6±0.1 nM。
T13848 SMARCA-BD ligand 1 for Protac

Epigenetic Reader Domain Chromatin/Epigenetic
SMARCA-BD ligand 1 for Protac 能够与 BAF ATPase 亚基 SMARCA2 结合,可用于 PROTAC 技术,用于降解 SMARCA2。
T28136 NC-1300-B

NC1300B,NC 1300 B

ATPase Membrane transporter/Ion channel
NC-1300-B 抑制 H(+)-K(+)-ATP 酶,可用于研究胃溃疡。
T14965 Ciliobrevin D

ATPase; Hedgehog/Smoothened GPCR/G Protein; Membrane transporter/Ion channel; Stem Cells
Ciliobrevin D 是细胞渗透性,可逆和特异性的 AAA + ATPase 运动细胞质动力蛋白抑制剂。它在体外抑制依赖于动力蛋白的微管滑动和 ATPase 活性。它抑制Hedgehog 信号和初级纤毛形成。
T20436 DHQ

2,3-dihydroxy-quinoxalin,2,3-二羟基喹喔啉

ATPase Membrane transporter/Ion channel
DHQ (2,3-dihydroxy-quinoxalin) 是单纯疱疹病毒胸苷激酶的 ATPase 活性诱导剂。
T10435 Linaprazan

利那拉生,AZD0865

Potassium Channel Membrane transporter/Ion channel
Linaprazan (AZD0865) 通过K+竞争抑制胃中的H+,K+ -ATPase. (IC 50: 1.0 ± 0.2 μM)。Linaprazan 对酸有很强的抑制作用。
T27303 Farglitazar

GI-262570,GI 262570,GI262570

Farglitazar is a PPAR-γ agonist. GI262570 stimulates the ENaC and Na,K-ATPase system resulting in the increasing of water and sodium reabsorption in distal nephron.

化合物

RUVBL1/2 ATPase-IN-1
Cat.No: T9882
Synonym:
Target: Others
ATPase-IN-3
Cat.No: T83967
Synonym:
Target: ATPase
ATPase-IN-2
Cat.No: T61553
Synonym:
Target:
Suloctidil
Cat.No: T0712
Synonym:
Target: ATPase, Platelet aggregation
Chloroprocaine hydrochloride
Cat.No: T6443
Synonym: 盐酸氯普鲁卡因,Chloroprocaine HCl
Target: ATPase, Others
Esomeprazole
Cat.No: T20626
Synonym:
Target: Proton pump, Cysteine Protease
Chlorpropamide
Cat.No: T0490
Synonym: Diabinese,氯磺丙脲
Target: ATPase, ABC
NPD8733
Cat.No: T9008
Synonym:
Target: Others
2,3-Butanedione 2-Monoxime
Cat.No: T2176
Synonym: Diacetyl monoxime,2,3-Butanedione-2-monoxime
Target: Akt
KM 91104
Cat.No: T9230
Synonym:
Target: ATPase
Apoptozole
Cat.No: T3293
Synonym: Apoptosis Activator VII
Target: Apoptosis, HSP
CB-5083
Cat.No: T6796
Synonym: CB5083,CB 5083
Target: p97
NSC 617145
Cat.No: T9168
Synonym: NSC617145,NSC-617145
Target: DNA/RNA Synthesis
S-trityl-L-Cysteine
Cat.No: T36816
Synonym: STLC
Target: Kinesin
Tenatoprazole
Cat.No: T6700
Synonym: 泰妥拉唑,TU-199
Target: Proton pump
Prilocaine
Cat.No: T6953
Synonym: Citanest,丙胺卡因,Propitocaine,NSC 40027
Target: ATPase, Sodium Channel
Esomeprazole Sodium
Cat.No: T2686L
Synonym: 埃索美拉唑钠,(S)-Omeprazole sodium
Target: ATPase, Proton pump
Rostafuroxin
Cat.No: T2621
Synonym: PST 2238
Target: ATPase, RSV
Prilocaine hydrochloride
Cat.No: T0796
Synonym: Prilocaine HCl,Propitocaine hydrochloride,Xylonest,盐酸丙胺卡因
Target: ATPase, Sodium Channel
Rabeprazole Sulfide
Cat.No: T1734
Synonym: 雷贝拉唑相关物质E,Rabeprazole Related Compound E
Target: Proton pump, Antibacterial
BRM/BRG1 ATP Inhibitor-1
Cat.No: T10616
Synonym:
Target: Epigenetic Reader Domain
BTS
Cat.No: T7144
Synonym: N-Tosylbenzylamine,N-苄基-对甲苯磺酸胺,N-Benzyl-p-toluenesulfonamide
Target: ATPase, Myosin
Esomeprazole Magnesium
Cat.No: T2686
Synonym: (S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium
Target: ATPase, Proton pump
Pantoprazole
Cat.No: T6928
Synonym: SKF96022,泮托拉唑,BY1023
Target: Apoptosis, Proton pump, Autophagy
Esomeprazole Magnesium trihydrate
Cat.No: T8386
Synonym: 埃索美拉唑镁三水合物,埃索美拉唑镁(三水),(S)-Omeprazole magnesium trihydrate
Target: Proton pump
Rabeprazole sodium
Cat.No: T1651
Synonym: Dexrabeprazole Sodium,LY307640 sodium,Habeprazole Sodium,雷贝拉唑钠,Rebeprazole sodium,Aciphex Sodium
Target: Apoptosis, Proton pump
Pantoprazole Sodium Hydrate
Cat.No: T0161
Synonym: SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate)
Target: Apoptosis, Potassium Channel, Proton pump, Autophagy
Pantoprazole sodium
Cat.No: T6929
Synonym: Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc
Target: Apoptosis, Others, Proton pump, HIF, Autophagy
Leminoprazole
Cat.No: T27812
Synonym:
Target: ATPase
2,5-Di-tert-butylhydroquinone
Cat.No: T7540
Synonym: BHQ,2,5-二特丁基对苯二酚
Target: Calcium Channel, Lipoxygenase, COX
BRITE-338733
Cat.No: T22280
Synonym: BRITE338733
Target: ATPase, Antibacterial
Vonoprazan fumarate
Cat.No: T2404
Synonym: 富马酸沃诺拉赞,TAK-438
Target: ATPase
Mavacamten
Cat.No: T7134
Synonym: MYK-461,SAR439152
Target: Myosin
Vonoprazan Fumarate
Cat.No: T21254
Synonym: TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞
Target: Proton pump
Tegoprazan
Cat.No: T17030
Synonym:
Target: ATPase, Proton pump
8-[(2,6-dimethylbenzyl)amino]-2,3-dimethylimidazo[1,2-a]pyridine-6-carboxylic acid
Cat.No: T9553
Synonym:
Target: Others
Sodium orthovanadate
Cat.No: T2189
Synonym: Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate
Target: ATPase, Phosphatase
SCH28080
Cat.No: T16865
Synonym:
Target: ATPase, Proton pump
(+)-Blebbistatin
Cat.No: T12503
Synonym:
Target: Others
CDN1163
Cat.No: T7373
Synonym:
Target: Calcium Channel
BRM/BRG1 ATP Inhibitor-2
Cat.No: T60032
Synonym:
Target: Epigenetic Reader Domain
(+)-SJ733
Cat.No: T17313
Synonym: SJ000557733
Target: ATPase, Parasite
PK095
Cat.No: T67763
Synonym:
Target: ATPase
GSK-923295
Cat.No: T2039
Synonym:
Target: Apoptosis, Kinesin
SMARCA-BD ligand 1 for Protac
Cat.No: T13848
Synonym:
Target: Epigenetic Reader Domain
NC-1300-B
Cat.No: T28136
Synonym: NC1300B,NC 1300 B
Target: ATPase
Ciliobrevin D
Cat.No: T14965
Synonym:
Target: ATPase, Hedgehog/Smoothened
DHQ
Cat.No: T20436
Synonym: 2,3-dihydroxy-quinoxalin,2,3-二羟基喹喔啉
Target: ATPase
Linaprazan
Cat.No: T10435
Synonym: 利那拉生,AZD0865
Target: Potassium Channel
Farglitazar
Cat.No: T27303
Synonym: GI-262570,GI 262570,GI262570
Target:
Cat. No. Product Name Target Signaling Pathways
T1719 Bufalin

ATPase Membrane transporter/Ion channel
Bufalin 是蟾酥中的一种成分,是Na+/K+-ATPase 抑制剂,具有抗肿瘤活性,可与其基 α1、α2 和 α3 结合,Kd 值分别为 42.5、45 和 40 nM。
TJP2872 Acevaltrate

Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate

ATPase; Others Membrane transporter/Ion channel; Others
Acevaltrate (Acevaltratum) 对人小细胞肺癌细胞系 GLC(4) 和人结肠直肠癌细胞系 COLO 320 具有高细胞毒性,IC50 值为 1-6 uM。它抑制大鼠肾和脑半球中 Na+/K+-ATP 酶活性,IC50分别为 22.8 和 42.3 μM。
T5S0890 Oleandrin

Neriostene,Folinerin,Foliandrin,欧夹竹桃苷

Apoptosis; ATPase; Potassium Channel; Sodium Channel Apoptosis; Membrane transporter/Ion channel
Oleandrin (Folinerin) 是夹竹桃属中的一种类固醇,可抑制Na+/K+-ATPase 活性,IC50为 620 nM。
T0295 Digitoxin

Digitoxoside,洋地黄毒苷,Unidigin,洋地黄毒甙,Digitoxinum,洋地黄

ATPase; Others Membrane transporter/Ion channel; Others
Digitoxin (Digitoxinum) 是Na+/K+-ATPase 有效抑制剂, EC50 值为0.78 μM。
TN5073 Strophanthidin

毒毛旋花子甙元,Strophanthidine,葡萄球菌素

ATPase; Calcium Channel Membrane transporter/Ion channel; Metabolism
Strophanthidin (Strophanthidine) 是黄花夹竹桃中的一种类固醇,可增加舒张期和收缩期胞内 Ca2+浓度。它在 0.1 和 1 nmol/L 增加Na+/K+-ATPase 活性,1到100 μ mol/L 抑制Na+/K+-ATPase 活性,10 和 100 nmol/L 对Na+/K+-ATPase 活性无影响。
T2922 Phlorizin

Floridzin,根皮甙,根皮苷,NSC 2833,Phloridzin

ATPase; SGLT GPCR/G Protein; Membrane transporter/Ion channel
Phlorizin (Phloridzin) 是非选择性的SGLT 抑制剂,也是Na+/K+-ATPase 抑制剂,对于hSGLT1和hSGLT2的Ki 值分别为 300 和 39 nM。
T8183 Deslanoside

洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C

ATPase; Drug Metabolite Membrane transporter/Ion channel; Metabolism
Deslanoside (Desacetyllanatoside C) 是一种快速作用的强心苷,可抑制Na-K-ATPase 膜泵,导致细胞内钠和钙浓度增加。它用于研究充血性心力衰竭和因折返机制引起的室上性心律失常,并在研究慢性心房颤动时控制心室率。
T2O2668 Oleic acid

Elaidoic acid,9Z-Octadecenoic acid,Oleate,9-Octadecenoic Acid,Glycon Wo,9-cis-Octadecenoic acid,油酸

Apoptosis; ATPase; Others; Endogenous Metabolite Apoptosis; Membrane transporter/Ion channel; Metabolism; Others
Oleic acid (Glycon Wo) 属于天然产物,是一种常见的饱和脂肪酸,在存在于多种动物、植物的脂肪和油脂中。Palmitic acid 是一种 Na+/K+ATP 酶激活剂。
T6368 Abscisic Acid

Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)

Others; Proton pump; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Abscisic Acid (Dormin) 是具有口服活性的植物激素,存在于蔬菜和水果中,也是内源性的哺乳动物激素。它是生长抑制剂,可以调节植物生长发育。他抑制质子泵,并导致 Ca2+依赖性的质膜去极化。它是 LANCL2 的天然配体,属于胰岛素敏感化合物,在糖尿病前期,2 型糖尿病和代谢综合征的研究中具有价值。
T2822 Ginsenoside Rb1

Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III

ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。
T6062 Brefeldin A

BFA,布雷非德菌素 A,Ascotoxin,Cyanein,Decumbin

ATPase; Mitophagy; Antibiotic; Autophagy; HSV; CRISPR/Cas9 Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Brefeldin A (Cyanein) 属于大环内酯类抗生素,是一种 ATPase 抑制剂 (IC50=0.2 μM)。Brefeldin A 可以诱导肿瘤细胞分化和凋亡,也具有抑制自噬的活性。
TN1860 Licoflavone B

甘草黄酮 B,甘草黄酮B

ATPase; Anti-infection; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Licoflavone B 是从甘草中得到的一种类黄酮,抑制曼氏血吸虫 ATPase 和 ADPase 的活性,IC50值分别为 23.78 µM 和 31.50 µM。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T3432 Cinobufagin

华蟾蜍精,华蟾酥毒基,Cinobufagine

Apoptosis; ATPase; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel
Cinobufagin (Cinobufagine) 是一种具有抗肿瘤功效的天然产物。
T15027 Cyclopiazonic acid

环匹阿尼酸,环二氮酸

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cyclopiazonic acid 是一种神经毒性次级代谢产物 (SM),源于A. flavus,是一种纳摩尔内质网钙 ATP 酶抑制剂 (Ca2+ATPase; SERCA),是植物细胞死亡的有效诱导剂。
TQ0184 Chebulinic acid

ATPase; Proton pump; DNA/RNA Synthesis; Antibacterial; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Stem Cells
Chebulinic acid 是从诃子果中提取的一种天然产物,结核分枝杆菌 DNA 促旋酶的有效抑制剂。它也能抑制 SMAD-3 phosphorylation 和 H+ K+-ATPase 的活性。
T6323 Oligomycin A

MCH 32,寡霉素A

ATPase; Antibiotic; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Oligomycin A (MCH 32) 是从链霉菌属中得到的一种线粒体F0F1-ATPase 抑制剂,抑制氧化磷酸化和线粒体偶联膜上发生的所有 ATP 依赖性过程。
T6740 Bafilomycin A1

巴佛洛霉素A1,巴佛洛霉素 A1

Apoptosis; Proton pump; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology
Bafilomycin A1 属于大环内酯类抗生素,是一种 V-ATPase (IC50=0.44 nM),具有特异性和可逆性。Bafilomycin A1 是自噬晚期阶段抑制剂,阻断自噬体与溶酶体的融合。Bafilomycin A1 也诱导凋亡。
T3926 Echinatin

刺甘草查尔酮,Retrochalcone

Free radical scavengers oxidation-reduction
Echinatin (Retrochalcone) 是分离自中草药甘草中,具有保肝和抗炎活性。在大鼠中,它可以被快速吸收和消除,并广泛分布,绝对生物利用度约为 6.81%。
T36390 Sodium oleate

Oleic acid sodium salt,Sodium oleate,cis-9-Octadecenoic acid sodium salt

ATPase Membrane transporter/Ion channel
Sodium oleate (cis-9-Octadecenoic acid sodium salt) (Oleic acid sodium) 是人脂肪细胞和其他组织中最常见的单不饱和脂肪酸钠盐。Sodium oleate 是一种 Na+/K+ ATP 酶激活剂。
T0974 Novobiocin Sodium

Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T3868 Agnuside

牡荆油,穗花牡荆苷,chasteberry oil

COX; Prostaglandin Receptor; P-gp GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Agnuside (chasteberry oil) 是从黄荆中分离得到的一种天然产物,可下调炎性介质PGE2和LTB4,减少细胞因子的表达,具有抗关节炎活性。
T4897 Inosine-5'-triphosphate trisodium salt

ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt

Others; Endogenous Metabolite Metabolism; Others
Inosine-5'-triphosphate trisodium salt (ITP) 是三磷酸核苷,能够作为 ATPases 和 GTPases 的底物。
TQ0302 Thapsigargin

毒胡萝卜素

Apoptosis; SARS-CoV; Calcium Channel Apoptosis; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Thapsigargin 属于天然产物,是一种肌/内质网 Ca2+ ATP 酶 (SERCA) 的抑制剂,也是一种内质网应激诱导剂。Thapsigargin 通过阻断细胞将钙泵入肌浆和内质网的能力来提高胞浆钙浓度。
T5079 Adenosine 5'-diphosphate sodium salt

腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt

Others; Endogenous Metabolite Metabolism; Others
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
T4973 Paraxanthine

1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE

Endogenous Metabolite Metabolism
Paraxanthine (1,7-dimethylxanthine) 是一种 caffeine 的代谢物,能够刺激Ryanodine 受体通道来抑制多巴胺能细胞的死亡。
T6S1049 Wilforine

ATPase Membrane transporter/Ion channel
Wilforine 是一倍半萜吡啶化合物,T. wilfordii 植物中的重要生物活性化合物,可有效治疗特发性肺纤维化。它具有抗炎和杀虫活性。
T5075 Phytic acid potassium

植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt

Others; Endogenous Metabolite Metabolism; Others
Phytic acid potassium (Inositol polyphosphate dipotassium salt) 是内源性代谢产物的一种。
T7190 Actein

Apoptosis; Akt; JNK; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Actein 是从升麻的根茎中分离的一种三萜糖苷,通过促进ROS/JNK 活化和钝化人膀胱癌中的AKT 途径来抑制细胞增殖,诱导自噬和凋亡。
T5S1982 Periplocin

Periplocoside,杠柳毒苷

Apoptosis; Others Apoptosis; Others
Periplocin (Periplocoside) 是从黑龙骨中分离出的一种强心类固醇。它可促进肿瘤细胞凋亡并抑制肿瘤生长。它通过激活 Na/K-ATPase 介导的 Src/ERK 和 PI3K/Akt 途径,具有促进伤口愈合的潜力。
T13618 Citreoviridin

Others Others
Citreoviridin, a toxin from Penicillium citreoviride NRRL 2579, inhibits brain synaptosomal Na+/K+-ATPase whereas, in microsomes, both Na+/K+-ATPase and Mg2+-ATPase activities are significantly stimulated in a dose-dependent manner.
T38609 Mycalolide B

Mycalolide-B is a marine sponge-derived compound that functions as a selective inhibitor of actomyosin ATPase. It effectively hinders ATP-induced contraction and Mg2+-ATPase activity in the absence of Ca2+.
T14995 Concanamycin A

X 4357B,刀豆素A,Antibiotic X 4357B,Concanamycin

Others Others
Concanamycin A is a macrolide antibiotic. It also is a specific inhibitor of vacuolar-type H+-ATPase (V-ATPase).
TN6631 Chamigrenol

Chamigrenol is a promising candidate for the development of potent Na+/K+ ATPase inhibitors and antimicrobial agents. It inhibited the activities of Na+/K+-ATPase, with the IC50 value of 15.9 ± 0.54 μg/mL.
T25211 CC 1014

CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885

CC 1014 is a polypeptide antibiotic isolated from Penicillium lilacinum that inhibits phosphorylation of ADP, Mg ATPase.
TN5141 Thevetin B

ATPase; Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Thevetin B 是一种强心苷,是Na+-, K+-依赖性腺苷三磷酸酶 (Na+,K+-ATPase) 的抑制剂,来自 Thevetia peruviana。
TN4697 Odoroside H

ATPase; Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Odoroside H has anticancer activities, the cytotoxic effects are induced by the inhibition of the plasma membrane bound Na(+)/K(+)-ATPase.
TN3914 Echinatine

ATPase; IL Receptor; TNF Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel
Echinatin exerts a protective effect against ischemia/reperfusion (I/R)-induced myocardial injury on hearts, this effect may be attributed to the antioxidant and anti-inflammatory activities of this compound. Echinatin can inhibit DNP-ATPase activity whil
T10455 Bafilomycin B1

巴佛洛霉素 B1

Others Others
Bafilomycin B1, a macrolide antibiotic isolated from Streptomyces sp, acts as an inhibitor of K+-dependent ATPase of E. coli. It also inhibits Gram-positive bacteria and fungi.
T14293 Annonacin

Others Others
Annonacin is an Acetogenin and promotes cytotoxicity via a pathway inhibiting the mitochondrial complex and it is the active agent found in Graviola leaf extract to act as an inhibitor of sodium/potassium (NKA) and sarcoplasmic reticulum (SERCA) ATPase pu
TN2306 Wilfordine

ATPase; Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Wilfordine is an insecticidally active alkaloid, Na+-K+-ATPase may be an acting target of wilfordine against some larvae of insect.
T16719 Radicicol

根赤壳菌素,Monorden

HSP Cytoskeletal Signaling; Metabolism
Radicicol is an antifungal antibiotic, impairs mitochondrial replication by targeting P. falciparum topoisomerase VIB. Radicicol is an inhibitor of Hsp90 (IC50: 1 μM). Radicicol binds to the ATPase domain of Hsp90 and prevents maturation of Hsp90 clients,
TN5060 Stauntosaponin A

ATPase; Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Stauntosaponin A and stauntosaponin B show moderate inhibitory activities against Na+/K+-ATPase with IC50 values of 21 and 29 uM, respectively.
T23610 Acerinol

Acerinol is an active ingredient from traditional Chinese medicinal herbs. It could be used as a cancer multidrug resistance reversal agent. Acerinol can significantly stimulate the activity of ABCB1 ATPase without affecting the expression of ABCB1 on nei
TN3075 5,2',6'-Trihydroxy-6,7,8-trimethoxyflavone

ATPase Membrane transporter/Ion channel
5,2',6'-Trihydroxy-6,7,8-trimethoxyflavone (ED 50 =4.5 ug/ml ) shows cytotoxicity against L1210 cell and has inhibiting effects on ATPase from the cell.
T35605 Apoptolidin

Apoptolidin is an apoptosis inducer originally isolated from Nocardiopsis bacteria. It inhibits the mitochondrial F1FO ATPase (Ki = 4-5 μM). Apoptolidin selectively kills transformed glial cells without significantly affecting untransformed cells. It also has antibiotic and antifungal actions.
T27977 Manzamine A

Keramamine A

Manzamine A is a GSK-3 inhibitor and vacuolar ATPase uncoupler found in marine sponges. It inhibits autophagy and tumor growth in cancer models, suppresses foam cell formation in macrophages, prevents growth of gram negative and gram positive bacteria, an
T38069 Aquastatin A

Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC50= 3.2 μM) andS. aureusfatty acid synthesis (IC50= 3.5 μM).2Aquastatin A also inhibits the Na+/K+-ATPase and H+/K+-ATPase (IC50s = 7.1 and 6.2 μM, respectively), as well as protein tyrosine phosphatase 1B (PTP1B; IC50= 0.19 μM).1,3 1.Hamano, K., Kinoshita-Okami, M., Minagawa, K....
T72645 Norbatzelladine L

Norbatzelladine L 是一种 Pdr5p 转运蛋白催化活性和功能活性的抑制剂。Norbatzelladine L 抑制 Pdr5p ATPase 活性,IC50值为 3.8 µM。Norbatzelladine L 具有抗真菌 (antifungal)、抗寄生虫 (antiparasitic)、抗病毒 (antiviral)、抗细菌 (antibacterial) 和抗肿瘤活性。
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天然产物

Bufalin
Cat.No: T1719
Synonym:
Target: ATPase
Acevaltrate
Cat.No: TJP2872
Synonym: Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate
Target: ATPase, Others
Oleandrin
Cat.No: T5S0890
Synonym: Neriostene,Folinerin,Foliandrin,欧夹竹桃苷
Target: Apoptosis, ATPase, Potassium Channel, Sodium Channel
Digitoxin
Cat.No: T0295
Synonym: Digitoxoside,洋地黄毒苷,Unidigin,洋地黄毒甙,Digitoxinum,洋地黄
Target: ATPase, Others
Strophanthidin
Cat.No: TN5073
Synonym: 毒毛旋花子甙元,Strophanthidine,葡萄球菌素
Target: ATPase, Calcium Channel
Phlorizin
Cat.No: T2922
Synonym: Floridzin,根皮甙,根皮苷,NSC 2833,Phloridzin
Target: ATPase, SGLT
Deslanoside
Cat.No: T8183
Synonym: 洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C
Target: ATPase, Drug Metabolite
Oleic acid
Cat.No: T2O2668
Synonym: Elaidoic acid,9Z-Octadecenoic acid,Oleate,9-Octadecenoic Acid,Glycon Wo,9-cis-Octadecenoic acid,油酸
Target: Apoptosis, ATPase, Others, Endogenous Metabolite
Abscisic Acid
Cat.No: T6368
Synonym: Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)
Target: Others, Proton pump, Endogenous Metabolite
Ginsenoside Rb1
Cat.No: T2822
Synonym: Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
Brefeldin A
Cat.No: T6062
Synonym: BFA,布雷非德菌素 A,Ascotoxin,Cyanein,Decumbin
Target: ATPase, Mitophagy, Antibiotic, Autophagy, HSV, CRISPR/Cas9
Licoflavone B
Cat.No: TN1860
Synonym: 甘草黄酮 B,甘草黄酮B
Target: ATPase, Anti-infection, Parasite
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
Cinobufagin
Cat.No: T3432
Synonym: 华蟾蜍精,华蟾酥毒基,Cinobufagine
Target: Apoptosis, ATPase, Autophagy
Cyclopiazonic acid
Cat.No: T15027
Synonym: 环匹阿尼酸,环二氮酸
Target: Calcium Channel
Chebulinic acid
Cat.No: TQ0184
Synonym:
Target: ATPase, Proton pump, DNA/RNA Synthesis, Antibacterial, TGF-beta/Smad
Oligomycin A
Cat.No: T6323
Synonym: MCH 32,寡霉素A
Target: ATPase, Antibiotic, Antifungal
Bafilomycin A1
Cat.No: T6740
Synonym: 巴佛洛霉素A1,巴佛洛霉素 A1
Target: Apoptosis, Proton pump, Antibacterial, Antibiotic, Autophagy
Echinatin
Cat.No: T3926
Synonym: 刺甘草查尔酮,Retrochalcone
Target: Free radical scavengers
Sodium oleate
Cat.No: T36390
Synonym: Oleic acid sodium salt,Sodium oleate,cis-9-Octadecenoic acid sodium salt
Target: ATPase
Novobiocin Sodium
Cat.No: T0974
Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin
Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy
Agnuside
Cat.No: T3868
Synonym: 牡荆油,穗花牡荆苷,chasteberry oil
Target: COX, Prostaglandin Receptor, P-gp
Inosine-5'-triphosphate trisodium salt
Cat.No: T4897
Synonym: ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt
Target: Others, Endogenous Metabolite
Thapsigargin
Cat.No: TQ0302
Synonym: 毒胡萝卜素
Target: Apoptosis, SARS-CoV, Calcium Channel
Adenosine 5'-diphosphate sodium salt
Cat.No: T5079
Synonym: 腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt
Target: Others, Endogenous Metabolite
Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
Paraxanthine
Cat.No: T4973
Synonym: 1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE
Target: Endogenous Metabolite
Wilforine
Cat.No: T6S1049
Synonym:
Target: ATPase
Phytic acid potassium
Cat.No: T5075
Synonym: 植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt
Target: Others, Endogenous Metabolite
Actein
Cat.No: T7190
Synonym:
Target: Apoptosis, Akt, JNK, Autophagy
Periplocin
Cat.No: T5S1982
Synonym: Periplocoside,杠柳毒苷
Target: Apoptosis, Others
Citreoviridin
Cat.No: T13618
Synonym:
Target: Others
Mycalolide B
Cat.No: T38609
Synonym:
Target:
Concanamycin A
Cat.No: T14995
Synonym: X 4357B,刀豆素A,Antibiotic X 4357B,Concanamycin
Target: Others
Chamigrenol
Cat.No: TN6631
Synonym:
Target:
CC 1014
Cat.No: T25211
Synonym: CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885
Target:
Thevetin B
Cat.No: TN5141
Synonym:
Target: ATPase, Potassium Channel, Sodium Channel
Odoroside H
Cat.No: TN4697
Synonym:
Target: ATPase, Potassium Channel, Sodium Channel
Echinatine
Cat.No: TN3914
Synonym:
Target: ATPase, IL Receptor, TNF
Bafilomycin B1
Cat.No: T10455
Synonym: 巴佛洛霉素 B1
Target: Others
Annonacin
Cat.No: T14293
Synonym:
Target: Others
Wilfordine
Cat.No: TN2306
Synonym:
Target: ATPase, Potassium Channel, Sodium Channel
Radicicol
Cat.No: T16719
Synonym: 根赤壳菌素,Monorden
Target: HSP
Stauntosaponin A
Cat.No: TN5060
Synonym:
Target: ATPase, Potassium Channel, Sodium Channel
Acerinol
Cat.No: T23610
Synonym:
Target:
5,2',6'-Trihydroxy-6,7,8-trimethoxyflavone
Cat.No: TN3075
Synonym:
Target: ATPase
Apoptolidin
Cat.No: T35605
Synonym:
Target:
Manzamine A
Cat.No: T27977
Synonym: Keramamine A
Target:
Aquastatin A
Cat.No: T38069
Synonym:
Target:
Norbatzelladine L
Cat.No: T72645
Synonym:
Target:
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