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1218

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T17870 cIAP1 ligand 1

E3 ligase Ligand 12

Others Others
cIAP1 ligand 1 (E3 ligase Ligand 12) 是基于 LCL161 衍生物的细胞凋亡蛋白配体,可募集 IAP 泛素连接酶以降解靶蛋白,可用于和雄激素受体配体偶联开发蛋白降解剂,可用于研究前列腺癌。
TP1484L α2β1 Integrin Ligand Peptide acetate

α2β1 Integrin Ligand Peptide acetate (134580-64-6)

Integrin Cytoskeletal Signaling
α2β1 Integrin Ligand Peptide acetate (α2β1 Integrin Ligand Peptide acetate (134580-64-6)) 是 α2β1 整合素受体的潜在拮抗剂。它与细胞膜上的 α2β1 整合素受体相互作用,介导细胞外信号进入细胞。
T13510 Sigma-LIGAND-1

Sigma receptor GPCR/G Protein
Sigma-LIGAND-1 是一种选择性 sigma 受体配体,在 DTG 和 PPP 位点的 IC50 分别为 16 nM,19 nM。Sigma-LIGAND-1 对多巴胺 D2 受体的 Ki 为 4000 nM。
T10053 5HT6-ligand-1

5-HT Receptor GPCR/G Protein; Neuroscience
5HT6-ligand-1 是一种具有口服活性的 5-HT6 受体配体 (Ki = 1.43 nM)。
T5835 PROTAC ERRα ligand 2

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
PROTAC ERRα ligand 2 是雌激素相关受体 α (ERRα)反向激动剂。它对 ERRα (IC50=5.67 nM) 的抑制作用比 XCT790 (IC50=61.3 nM) 高效约 11 倍。
T15191 PROTAC ERRα ligand 1

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
PROTAC ERRα ligand 1 是一种雌激素相关受体 α (ERRα) 拮抗剂,能够作用于 ERRα (IC50:0.04 μM)和 ERRγ (IC50:2.8 μM)。
TP1496L p5 Ligand for Dnak and DnaJ acetate

p5 Ligand for Dnak and DnaJ acetate(209518-24-1 free base)

HSP Cytoskeletal Signaling; Metabolism
p5 Ligand for Dnak and DnaJ acetate(209518-24-1 free base) 是一种九肽。它是 DnaK(大肠杆菌 Hsp70)和 DnaJ(大肠杆菌 Hsp40)的高亲和力配体。
T38476 Metallo β-lactamase ligand 1

Antibacterial Microbiology/Virology
Metallo β-lactamase ligand 1 是B 类β-内酰胺酶的抑制剂,具有抗菌活性。
T12551 PROTAC BRD4 ligand-1

Epigenetic Reader Domain; Ligands for Target Protein for PROTAC Chromatin/Epigenetic; PROTAC
PROTAC BRD4 ligand-1 是 PROTAC GNE-987 靶向 BRD4 蛋白的配体,也是一种 BET 的抑制剂。
T60015 TSPO ligand-2 

Carbonic acid

AUTACs PROTAC
TSPO ligand-2 (Carbonic acid) 是 AUTAC1 的配体,AUTAC1含有一个对氟苄基鸟嘌呤和一个烟曲霉醇部分。
T17879 E3 ligase Ligand 8

Others; Ligand for E3 Ligase Others; PROTAC
E3 ligase Ligand 8 是 E3 泛素连接酶配体。它能够利用 linker 与靶蛋白配体连接,形成 PROTAC 分子。PROTAC 可诱导促癌蛋白发生泛素化降解。
TP1704 Galanin Receptor Ligand M35 TFA

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Galanin Receptor Ligand M35 TFA(142846-71-7 free base) 是一种高亲和力配体和甘丙肽受体拮抗剂 (Kd=0.1 nM)。
T9809 E3 ligase Ligand 23

Ligand for E3 Ligase PROTAC
E3 ligase Ligand 23 是一种 cereblon 结合剂,可通过泛素蛋白酶体降解 Ikaros 或 Aiolos。
T9360 CRBN ligand-9

2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione

Ligand for E3 Ligase PROTAC
CRBN ligand-9 (2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione) 表现出对 CRBN 的抑制作用。
T13848 SMARCA-BD ligand 1 for Protac

Epigenetic Reader Domain Chromatin/Epigenetic
SMARCA-BD ligand 1 for Protac 能够与 BAF ATPase 亚基 SMARCA2 结合,可用于 PROTAC 技术,用于降解 SMARCA2。
T13890 SMARCA-BD ligand 1 for Protac dihydrochloride

Epigenetic Reader Domain Chromatin/Epigenetic
SMARCA-BD ligand 1 for Protac dihydrochloride 是一种能够与 BAF ATPase 亚基 SMARCA2 结合的化合物,基于 PROTAC 技术,使 SMARCA2 降解。
T7763 Thalidomide-4-OH

Cereblon ligand 2,E3 ligase Ligand 2

Ligand for E3 Ligase PROTAC
Thalidomide-4-OH (E3 ligase Ligand 2) 是一种基于 Thalidomide 的 Cereblon 配体,可用于募集 CRBN 蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。
T39997 PROTAC CDK9 ligand-1

PROTAC CDK9 ligand-1

PROTAC CDK9 ligand-1 is a CDK9 ligand that can be used in the synthesis of PROTACs.
T7752 (S,R,S)-AHPC-Me

VHL ligand 2,E3 ligase Ligand 1A

Ligand for E3 Ligase PROTAC
(S,R,S)-AHPC-Me (E3 ligase Ligand 1A) 是基于 (S,R,S)-AHPC 的的 VHL 配体,可用于募集 von Hippel-Lindau (VHL) 蛋白。它可有效降解去势抵抗性前列腺癌细胞中的 BET 蛋白,DC50<1 nM。它可用于合成 ARV-771。
T13671 (S,R,S)-AHPC-Me hydrochloride

VHL ligand 2 hydrochloride,E3 ligase Ligand 1

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-Me hydrochloride (VHL ligand 2 hydrochloride) is a chemical compound utilized in the synthesis of ARV-771, an exceptionally potent BET protein degrader. This compound selectively degrades BET protein in cells resistant to castration, exhibiting a remarkable DC50 <1 nM. Recognized as VHL ligand 2 hydrochloride, (S,R,S)-AHPC-Me hydrochloride serves as the VHL ligand derived from (S,R,S)-AHPC for the recruitment of von Hippel-Lindau (VHL) protein.
T39628 PROTAC BRD4 ligand-2

PROTAC BRD4 ligand-2

PROTAC BRD4 ligand-2 is a ligand for target BRD4 protein for PROTAC CFT-2718.
T7753 Thalidomide-O-COOH

Cereblon ligand 3,E3 ligase Ligand 3,TCE35031

Others; Ligand for E3 Ligase Others; PROTAC
Thalidomide-O-COOH (Cereblon ligand 3) 是一种基于 Thalidomide 的 Cereblon 配体,可用于募集 CRBN 蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。
T17869 cIAP1 ligand 2

E3 ligase Ligand 11

Others Others
cIAP1 ligand 2, a derivative of LCL161, is an IAP ligand that can be connected to the ABL ligand for protein via a linker, resulting in the formation of SNIPER.
T39629 BRD4 ligand-Linker Conjugate 1

BRD4 ligand-Linker Conjugate 1

BRD4 Ligand-Linker Conjugate 1 is a compound consisting of a ligand and a linker, specifically designed to bind to the target protein BRD4. This conjugate serves as a valuable tool for synthesizing PROTACs, molecules utilized for targeted protein degradation.
T17877 VH032-cyclopropane-F

VHL ligand 3,E3 ligase Ligand 19,Phenolic VH101

Others; Ligand for E3 Ligase Others; PROTAC
VH032-cyclopropane-F (Phenolic VH101) 是基于 VH032 的 VHL 配体。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子,如 PROTAC 1。PROTAC 1 是 SMARCA2 和 SMARCA4 的部分降解剂。
T17916 Pomalidomide-PEG4-C2-NH2

Cereblon Ligand-Linker Conjugates 8,E3 Ligase Ligand-Linker Conjugates 22

Others; Ligand for E3 Ligase Others; PROTAC
Pomalidomide-PEG4-C2-NH2 (E3 Ligase Ligand-Linker Conjugates 22) 是一种合成的 E3 连接酶配体- linker 偶联物,用于 PROTAC 技术中。
T73599 TSPO ligand-1

Autophagy Autophagy
TSPO ligand-1 对外周和中枢苯二氮卓受体有亲和力。TSPO ligand-1 是一种线粒体外膜跨膜结构域上与 AUTAC4 结合的蛋白,可诱导线粒体自噬 (autophagy) 促进胞内线粒体更新。TSPO ligand-1 参与胆固醇在胞内的转运,可作为脑损伤和神经变性的生物标志物。
T39609 cIAP1 Ligand-Linker Conjugates 16

cIAP1 Ligand-Linker Conjugates 16

cIAP1 Ligand-Linker Conjugates 16 refers to a specific type of ligase ligand-linker conjugate, possessing the ability to engage with E3 ligases, which finds application in the synthesis of PROTACs.
T17325 Pomalidomide-PEG4-C-COOH

Cereblon Ligand -Linker Conjugates 1,E3 Ligase Ligand-Linker Conjugates 1

Others; E3 Ligase Ligand-Linker Conjugate Others; PROTAC
Pomalidomide-PEG4-C-COOH (E3 Ligase Ligand-Linker Conjugates 1) 包含基于 Pomalidomide 的 cereblon 配体和 4 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T15189 Thalidomide-O-amido-C4-N3

E3 ligase Ligand-Linker Conjugates 18,Cereblon Ligand-Linker Conjugates 4

Others; Ligand for E3 Ligase Others; PROTAC
Thalidomide-O-amido-C4-N3 (Cereblon Ligand-Linker Conjugates 4) 是一种 E3 连接酶配体- linker 偶联物,包含基于 Thalidomide 的 cereblon 配体和 linker。
T17919 Thalidomide-O-amido-C6-NH2 TFA

E3 Ligase Ligand-Linker Conjugates 25 Trifluoroacetate,Cereblon Ligand-Linker Conjugates 11 TFA,E3 Ligase Ligand-Linker Conjugates 25 TFA

Others; Ligand for E3 Ligase Others; PROTAC
Thalidomide-O-amido-C6-NH2 TFA (Cereblon Ligand-Linker Conjugates 11 TFA) 包含基于 Thalidomide 的 cereblon 配体和 1 个 linker,是一种合成的 E3 连接酶配体-linker 偶联物。可用于 PROTAC 的合成分子。
T40142 Thalidomide-NH-CBP/p300 ligand 2

Thalidomide-NH-CBP/p300 ligand 2

Thalidomide-NH-CBP/p300 ligand 2 (P-007) is a PROTAC-based compound designed to degrade CBP and p300, acting as a functional antagonist (WO2020173440).
T7760 Thalidomide-O-amido-C3-NH2 TFA

Cereblon Ligand-Linker Conjugates 16 TFA,E3 Ligase Ligand-Linker Conjugates 52 TFA

E3 Ligase Ligand-Linker Conjugate; Ligand for E3 Ligase PROTAC
Thalidomide-O-amido-C3-NH2 TFA (Cereblon Ligand-Linker Conjugates 16 TFA) 包含基于 Thalidomide 的 cereblon 配体和 1 个 linker,是一种合成的 E3 连接酶配体-linker 偶联物,。
T7759 Thalidomide-O-amido-C4-NH2 TFA

E3 ligase Ligand-Linker Conjugates 19 TFA,Cereblon Ligand-Linker Conjugates 6 TFA

E3 Ligase Ligand-Linker Conjugate PROTAC
Thalidomide-O-amido-C4-NH2 TFA (E3 ligase Ligand-Linker Conjugates 19 TFA) 包含基于 Thalidomide 的 cereblon 配体和 1 个 linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T7758 Thalidomide-O-amido-PEG3-C2-NH2 TFA

E3 ligase Ligand-Linker Conjugates 14 TFA,Cereblon Ligand-Linker Conjugates 3 (TFA)

Others; E3 Ligase Ligand-Linker Conjugate; Ligand for E3 Ligase Others; PROTAC
Thalidomide-O-amido-PEG3-C2-NH2 TFA (Cereblon Ligand-Linker Conjugates 3 (TFA)) 包含基于 Thalidomide 的 cereblon 配体和 3 个单元的 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T17918 Thalidomide-O-amido-PEG2-C2-NH2 TFA

E3 Ligase Ligand-Linker Conjugates 24 TFA,Cereblon Ligand-Linker Conjugates 10 TFA

Others; E3 Ligase Ligand-Linker Conjugate Others; PROTAC
Thalidomide-O-amido-PEG2-C2-NH2 TFA (E3 Ligase Ligand-Linker Conjugates 24 TFA) 包含基于 Thalidomide 的 cereblon 配体和 2 个单元的 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T17922 (S,R,S)-AHPC-PEG3-NH2 hydrochloride

VHL Ligand-Linker Conjugates 1 hydrochloride,E3 ligase Ligand-Linker Conjugates 5,VH032-PEG3-NH2 hydrochloride,VHL Ligand-Linker Conjugates 1 HCl

Others; E3 Ligase Ligand-Linker Conjugate Others; PROTAC
(S,R,S)-AHPC-PEG3-NH2 hydrochloride (E3 ligase Ligand-Linker Conjugates 5) 是一种 E3 ligase ligand-linker conjugate,包含了 (S,R,S)-AHPC-based VHL ligand 和 3-unit PEG linker。
T82174 hRIO2 kinase ligand-1

Others Others
hRIO2 kinase ligand-1 是一种有效的 hRIO2 激酶的配体(Kd:520 nM)。
T17921 (S,R,S)-AHPC-PEG4-N3

VH032-PEG4-N3,VHL Ligand-Linker Conjugates 5,E3 ligase Ligand-Linker Conjugates 4

Others; PROTAC Linker Others; PROTAC
(S,R,S)-AHPC-PEG4-N3 (VHL Ligand-Linker Conjugates 5) is a synthesized conjugate that functions as a ligand-linker in E3 ligase-based systems. It is composed of the (S,R,S)-AHPC VHL ligand and a 4-unit PEG linker, both commonly employed in PROTAC technology.
T39440 CXCL12 ligand 1

CXCL12 ligand 1 is the first ligand of the sY12-binding pocket on chemokine CXCL12 .
T17920 (S,R,S)-AHPC-PEG1-N3

VHL Ligand-Linker Conjugates 9,VH032-PEG1-N3,E3 ligase Ligand-Linker Conjugates 3

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG1-N3 (E3 ligase Ligand-Linker Conjugates 3) 是 E3 连接酶配体和linker 连接得到的 偶联物,包含基于 (S,R,S)-AHPC 的 VHL 配体和 1 个单元 PEG linker。
T17909 (S,R,S)-AHPC-PEG3-N3

VHL Ligand-Linker Conjugates 8,VH032-PEG3-N3,E3 ligase Ligand-Linker Conjugates 12

Others; E3 Ligase Ligand-Linker Conjugate; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG3-N3 (VHL Ligand-Linker Conjugates 8) 包含基于 (S,R,S)-AHPC 的 VHL 配体和 3 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物。
T17889 cIAP1 Ligand-Linker Conjugates 14

E3 ligase Ligand-Linker Conjugates 36

Others Others
cIAP1 Ligand-Linker Conjugates 14 consist of an IAP ligand that targets the E3 ubiquitin ligase and a PROTAC linker. These conjugates, known as cIAP1 Ligand-Linker Conjugates 14, are used in the development of SNIPERs[1].
T17896 cIAP1 Ligand-Linker Conjugates 4

E3 ligase Ligand-Linker Conjugates 42

Others Others
cIAP1 Ligand-Linker Conjugates 4 is a chemical compound that comprises an IAP ligand specifically designed for the E3 ubiquitin ligase and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 4, has the potential to be utilized in the development of SNIPERs[1].
T17885 cIAP1 Ligand-Linker Conjugates 11

E3 ligase Ligand-Linker Conjugates 33

Others Others
cIAP1 Ligand-Linker Conjugates 11 is a chemical compound that combines an IAP ligand specifically designed for the E3 ubiquitin ligase with a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 11, is useful in the development of SNIPERs[1], allowing for the targeted degradation of proteins.
T17891 cIAP1 Ligand-Linker Conjugates 2

E3 ligase Ligand-Linker Conjugates 37

Others Others
cIAP1 Ligand-Linker Conjugates 2 is a chemical compound that combines an IAP ligand for the E3 ubiquitin ligase with a PROTAC linker. This compound is particularly useful in the design of SNIPERs [1].
T17893 cIAP1 Ligand-Linker Conjugates 5

E3 ligase Ligand-Linker Conjugates 39

Others Others
cIAP1 Ligand-Linker Conjugates 5 is a chemical compound consisting of an IAP ligand that targets the E3 ubiquitin ligase, and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 5, is specifically designed for the development of SNIPERs[1].
T18640 (S,R,S)-AHPC-C4-NH2 hydrochloride

VH032-C4-NH2 hydrochloride,E3 ligase Ligand-Linker Conjugates 28,VHL Ligand-Linker Conjugates 13

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-C4-NH2 hydrochloride (E3 ligase Ligand-Linker Conjugates 28) 是一种合成的 E3 连接酶配体- linker 偶联物,包含基于 (S,R,S)-AHPC 的 VHL 配体和 linker。
T17908 VHL Ligand-Linker Conjugates 15

E3 Ligase Ligand-Linker Conjugates 56

Others Others
VHL Ligand-Linker Conjugates 15 is a chemical compound that combines a VHL ligand, which targets the E3 ubiquitin ligase, with a PROTAC linker. It is specifically designed for the creation of PROTACs[1].
T15190L (S,R,S)-AHPC-PEG4-NH2

VHL Ligand-Linker Conjugates 4,E3 ligase Ligand-Linker Conjugates 7 Free Base,VH032-PEG4-NH2

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-PEG4-NH2 (VHL Ligand-Linker Conjugates 4) 是一种合成的 E3 连接酶配体-接头偶联物,包含基于 (S,R,S)-AHPC 的 VHL 配体和 4 单元 PEG 接头。

化合物

cIAP1 ligand 1
Cat.No: T17870
Synonym: E3 ligase Ligand 12
Target: Others
α2β1 Integrin Ligand Peptide acetate
Cat.No: TP1484L
Synonym: α2β1 Integrin Ligand Peptide acetate (134580-64-6)
Target: Integrin
Sigma-LIGAND-1
Cat.No: T13510
Synonym:
Target: Sigma receptor
5HT6-ligand-1
Cat.No: T10053
Synonym:
Target: 5-HT Receptor
PROTAC ERRα ligand 2
Cat.No: T5835
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
PROTAC ERRα ligand 1
Cat.No: T15191
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
p5 Ligand for Dnak and DnaJ acetate
Cat.No: TP1496L
Synonym: p5 Ligand for Dnak and DnaJ acetate(209518-24-1 free base)
Target: HSP
Metallo β-lactamase ligand 1
Cat.No: T38476
Synonym:
Target: Antibacterial
PROTAC BRD4 ligand-1
Cat.No: T12551
Synonym:
Target: Epigenetic Reader Domain, Ligands for Target Protein for PROTAC
TSPO ligand-2 
Cat.No: T60015
Synonym: Carbonic acid
Target: AUTACs
E3 ligase Ligand 8
Cat.No: T17879
Synonym:
Target: Others, Ligand for E3 Ligase
Galanin Receptor Ligand M35 TFA
Cat.No: TP1704
Synonym:
Target: Neuropeptide Y Receptor
E3 ligase Ligand 23
Cat.No: T9809
Synonym:
Target: Ligand for E3 Ligase
CRBN ligand-9
Cat.No: T9360
Synonym: 2-(2,6-dioxopiperidin-3-yl)-5-nitroisoindoline-1,3-dione
Target: Ligand for E3 Ligase
SMARCA-BD ligand 1 for Protac
Cat.No: T13848
Synonym:
Target: Epigenetic Reader Domain
SMARCA-BD ligand 1 for Protac dihydrochloride
Cat.No: T13890
Synonym:
Target: Epigenetic Reader Domain
Thalidomide-4-OH
Cat.No: T7763
Synonym: Cereblon ligand 2,E3 ligase Ligand 2
Target: Ligand for E3 Ligase
PROTAC CDK9 ligand-1
Cat.No: T39997
Synonym: PROTAC CDK9 ligand-1
Target:
(S,R,S)-AHPC-Me
Cat.No: T7752
Synonym: VHL ligand 2,E3 ligase Ligand 1A
Target: Ligand for E3 Ligase
(S,R,S)-AHPC-Me hydrochloride
Cat.No: T13671
Synonym: VHL ligand 2 hydrochloride,E3 ligase Ligand 1
Target: Others, Ligand for E3 Ligase
PROTAC BRD4 ligand-2
Cat.No: T39628
Synonym: PROTAC BRD4 ligand-2
Target:
Thalidomide-O-COOH
Cat.No: T7753
Synonym: Cereblon ligand 3,E3 ligase Ligand 3,TCE35031
Target: Others, Ligand for E3 Ligase
cIAP1 ligand 2
Cat.No: T17869
Synonym: E3 ligase Ligand 11
Target: Others
BRD4 ligand-Linker Conjugate 1
Cat.No: T39629
Synonym: BRD4 ligand-Linker Conjugate 1
Target:
VH032-cyclopropane-F
Cat.No: T17877
Synonym: VHL ligand 3,E3 ligase Ligand 19,Phenolic VH101
Target: Others, Ligand for E3 Ligase
Pomalidomide-PEG4-C2-NH2
Cat.No: T17916
Synonym: Cereblon Ligand-Linker Conjugates 8,E3 Ligase Ligand-Linker Conjugates 22
Target: Others, Ligand for E3 Ligase
TSPO ligand-1
Cat.No: T73599
Synonym:
Target: Autophagy
cIAP1 Ligand-Linker Conjugates 16
Cat.No: T39609
Synonym: cIAP1 Ligand-Linker Conjugates 16
Target:
Pomalidomide-PEG4-C-COOH
Cat.No: T17325
Synonym: Cereblon Ligand -Linker Conjugates 1,E3 Ligase Ligand-Linker Conjugates 1
Target: Others, E3 Ligase Ligand-Linker Conjugate
Thalidomide-O-amido-C4-N3
Cat.No: T15189
Synonym: E3 ligase Ligand-Linker Conjugates 18,Cereblon Ligand-Linker Conjugates 4
Target: Others, Ligand for E3 Ligase
Thalidomide-O-amido-C6-NH2 TFA
Cat.No: T17919
Synonym: E3 Ligase Ligand-Linker Conjugates 25 Trifluoroacetate,Cereblon Ligand-Linker Conjugates 11 TFA,E3 Ligase Ligand-Linker Conjugates 25 TFA
Target: Others, Ligand for E3 Ligase
Thalidomide-NH-CBP/p300 ligand 2
Cat.No: T40142
Synonym: Thalidomide-NH-CBP/p300 ligand 2
Target:
Thalidomide-O-amido-C3-NH2 TFA
Cat.No: T7760
Synonym: Cereblon Ligand-Linker Conjugates 16 TFA,E3 Ligase Ligand-Linker Conjugates 52 TFA
Target: E3 Ligase Ligand-Linker Conjugate, Ligand for E3 Ligase
Thalidomide-O-amido-C4-NH2 TFA
Cat.No: T7759
Synonym: E3 ligase Ligand-Linker Conjugates 19 TFA,Cereblon Ligand-Linker Conjugates 6 TFA
Target: E3 Ligase Ligand-Linker Conjugate
Thalidomide-O-amido-PEG3-C2-NH2 TFA
Cat.No: T7758
Synonym: E3 ligase Ligand-Linker Conjugates 14 TFA,Cereblon Ligand-Linker Conjugates 3 (TFA)
Target: Others, E3 Ligase Ligand-Linker Conjugate, Ligand for E3 Ligase
Thalidomide-O-amido-PEG2-C2-NH2 TFA
Cat.No: T17918
Synonym: E3 Ligase Ligand-Linker Conjugates 24 TFA,Cereblon Ligand-Linker Conjugates 10 TFA
Target: Others, E3 Ligase Ligand-Linker Conjugate
(S,R,S)-AHPC-PEG3-NH2 hydrochloride
Cat.No: T17922
Synonym: VHL Ligand-Linker Conjugates 1 hydrochloride,E3 ligase Ligand-Linker Conjugates 5,VH032-PEG3-NH2 hydrochloride,VHL Ligand-Linker Conjugates 1 HCl
Target: Others, E3 Ligase Ligand-Linker Conjugate
hRIO2 kinase ligand-1
Cat.No: T82174
Synonym:
Target: Others
(S,R,S)-AHPC-PEG4-N3
Cat.No: T17921
Synonym: VH032-PEG4-N3,VHL Ligand-Linker Conjugates 5,E3 ligase Ligand-Linker Conjugates 4
Target: Others, PROTAC Linker
CXCL12 ligand 1
Cat.No: T39440
Synonym:
Target:
(S,R,S)-AHPC-PEG1-N3
Cat.No: T17920
Synonym: VHL Ligand-Linker Conjugates 9,VH032-PEG1-N3,E3 ligase Ligand-Linker Conjugates 3
Target: Others, Ligand for E3 Ligase
(S,R,S)-AHPC-PEG3-N3
Cat.No: T17909
Synonym: VHL Ligand-Linker Conjugates 8,VH032-PEG3-N3,E3 ligase Ligand-Linker Conjugates 12
Target: Others, E3 Ligase Ligand-Linker Conjugate, Ligand for E3 Ligase
cIAP1 Ligand-Linker Conjugates 14
Cat.No: T17889
Synonym: E3 ligase Ligand-Linker Conjugates 36
Target: Others
cIAP1 Ligand-Linker Conjugates 4
Cat.No: T17896
Synonym: E3 ligase Ligand-Linker Conjugates 42
Target: Others
cIAP1 Ligand-Linker Conjugates 11
Cat.No: T17885
Synonym: E3 ligase Ligand-Linker Conjugates 33
Target: Others
cIAP1 Ligand-Linker Conjugates 2
Cat.No: T17891
Synonym: E3 ligase Ligand-Linker Conjugates 37
Target: Others
cIAP1 Ligand-Linker Conjugates 5
Cat.No: T17893
Synonym: E3 ligase Ligand-Linker Conjugates 39
Target: Others
(S,R,S)-AHPC-C4-NH2 hydrochloride
Cat.No: T18640
Synonym: VH032-C4-NH2 hydrochloride,E3 ligase Ligand-Linker Conjugates 28,VHL Ligand-Linker Conjugates 13
Target: Others, Ligand for E3 Ligase
VHL Ligand-Linker Conjugates 15
Cat.No: T17908
Synonym: E3 Ligase Ligand-Linker Conjugates 56
Target: Others
(S,R,S)-AHPC-PEG4-NH2
Cat.No: T15190L
Synonym: VHL Ligand-Linker Conjugates 4,E3 ligase Ligand-Linker Conjugates 7 Free Base,VH032-PEG4-NH2
Target: Others, Ligand for E3 Ligase
Cat. No. Product Name Target Signaling Pathways
T24729 Roseoflavin

Antibacterial Microbiology/Virology
Roseoflavin 是天然色素,起初分离自Streptomyces davawensis。Roseoflavin 是核黄素和黄素单核苷酸的抗代谢类似物,显示出抗菌活性。
TQ0176 (-)-Isocorypalmine

Tetrahydrocolumbamine,(-)-异延胡索单酚碱,(S)-Tetrahydrocolumbamine

Dopamine Receptor; Antifungal GPCR/G Protein; Microbiology/Virology; Neuroscience
(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine) 是一种多巴胺受体配体,从延胡索粗碱中分离得到。重组CYP719A21 对 (-)-Isocorypalmine 具有严格的底物特异性和高亲和力 (Km=4.63 μM)。
T8097 Methyl 3-aminopropanoate hydrochloride

β-Alanine methyl ester hydrochloride,3-氨基丙酸甲酯盐酸盐

Others Others
Methyl 3-aminopropanoate hydrochloride (β-Alanine methyl ester hydrochloride) 是由 Β-Alanine (I) 酯化得到。它可用于合成双齿吡啶酸配体。
T14063 7α,25-Dihydroxycholesterol

7α,25-OHC

EBI2/GPR183; Endogenous Metabolite GPCR/G Protein; Metabolism
7α,25-Dihydroxycholesterol 是一种孤儿 GPCR 受体EBI2 (GPR183)的内源性配体和有效选择性激动剂。它对激活 EBI2 有很强的作用 (EC50=140 pM;Kd=450 pM)。它能够作为一种趋化因子,指导 B 细胞、T 细胞和树突状细胞的迁移。
T4S0039 Baimaside

白麻苷,Quercetin-3-O-sophoroside,Quercetin 3-beta-D-sophoroside

Others Others
Baimaside (Quercetin-3-O-sophoroside) 是一种超氧阴离子的清除剂,分离自A. venetum 的花中。
TN1023 Miltirone

P450; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Miltirone 是存在于丹参中的一种天然产物,可作为中枢苯二氮受体部分激动剂,IC50值为 0.3 μM。
TP1232L Amylin, amide, rat acetate(124447-81-0,free base)

Amylin Receptor GPCR/G Protein
Amylin, amide, rat acetate(124447-81-0,free base) 是 AMY1 和 AMY3 受体以及 AMY2 受体的强效和高亲和力配体。
TN2077 (+/-)-Pinocembrin

NSC 43318,(±)-5,7-Dihydroxyflavanone

GPR; Others Endocrinology/Hormones; GPCR/G Protein; Others
(+/-)-Pinocembrin (NSC-43318) 是一种来自腋松的天然产物,它是一种 GPR120 配体,能促进 HaCaT 细胞系的伤口愈合。
T3806 kaempferide

Kaempferol 4'-O-methyl ether,山奈素,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Influenza Virus; Antibacterial; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology
kaempferide (4'-Methylkaempferol) 是一种存在于山柰中的O-甲基化黄酮醇,具有抗病毒活性。
T13815 Penicillic acid

Apoptosis; Caspase; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Proteases/Proteasome
Penicillic acid, a polyketide mycotoxin, synthesized by various species of Aspergillus and Penicillium, acts as an inhibitor of Fas ligand-induced apoptosis by impeding self-processing of caspase-8. Additionally, in vitro studies have shown that Penicillic acid displays cytotoxic properties in rat alveolar macrophages.
T8363 DL-Serine

PKM Metabolism
DL-Serine 是 D-丝氨酸和 L-丝氨酸的混合物,是一种基础代谢物。它具有抗病毒作用,能抑制烟草花叶病毒的增殖。
Fr12596 3-Acetylcoumarin

Others Others
3-Acetylcoumarin 作为室温下铜催化 CN 偶联反应的实用配体。它具有神经保护和杀螨特性。
T5026 Oxytocin

催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
Oxytocin (Oxytocin (Syntocinon)) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。
TJS1183 Cyclen

轮环藤宁,1,4,7,10-tetraazacyclododecane

Others Others
Cyclen (1,4,7,10-tetraazacyclododecane) 是一种氮杂冠醚的类似物,是制备有效的大环螯合物的中间体,是制备磁共振造影剂的前体物质。
TN3209 3′,4′,7-Trihydroxyflavone 

ATPase; Others; p38 MAPK; NF-κB MAPK; Membrane transporter/Ion channel; NF-κB; Others
3',4',7-Trihydroxyflavone 是分离自蚕豆荚的黄酮苷元化合物。
T5145 Oxytocin acetate

Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。
T3S0738 yangonin

Y100550,甲氧醉椒素

Cannabinoid Receptor; NF-κB; Autophagy Autophagy; GPCR/G Protein; NF-κB
Yangonin (Y100550) 是一种新型 CB1 受体配体,对人重组 CB1 受体具有亲和力。它可能是干预 NF-κB 依赖性病理状况的候选药物。
T36857 Estrone sulfate sodium

雌酮3-硫酸钠,Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate

Endogenous Metabolite Metabolism
Estrone sulfate sodium (17β-Estrone 3-sulfate) 是一种主要的循环血浆雌激素,无生物活性,通过类固醇硫酸酯酶(STS) 转化为生物活性雌激素雌酮。
T15705 Laminaran

β-1,3-Glucan

Laminaran 是一种从褐藻中分离出来的 β-1-3-葡聚糖,常作为 Dectin-1 的典型配体,具有抗癌、免疫调节和辐射防护作用。 Laminaran 可被葡糖酶催化。Laminaran 在体内外实验中显示出抗肿瘤活性,可用于预防和治疗癌症。
T7998 1,7-Diaminoheptane

Others Others
1,7-Diaminoheptane 是一种脂族胺家族的化合物。它可用于合成肽、拟肽和其他化合物,也被用作酶反应中的底物,金属配合物中的配体,以及有机合成中的试剂。
TN2143 3,7,4'-Trihydroxyflavone

Resokaempferol,5-Deoxykampferol

DNA DNA Damage/DNA Repair
3,7,4'-Trihydroxyflavone(5-Deoxykampferol) 是从黄檀心材中分离得到的一种具有 DNA 断链活性的黄酮类化合物,可抑制 NF-κB 配体 (RANKL) 受体激活剂诱导的 RAW 264.7 细胞和骨髓巨噬细胞中的破骨细胞分化、肌动蛋白环形成和骨吸收。
T4973 Paraxanthine

1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE

Endogenous Metabolite Metabolism
Paraxanthine (1,7-dimethylxanthine) 是一种 caffeine 的代谢物,能够刺激Ryanodine 受体通道来抑制多巴胺能细胞的死亡。
TL0005 3,5-O-Dicaffeoylquinic acid

Isochlorogenic Acid A,(-)-3,5-二咖啡酰奎宁酸,(-)-3,5-Dicaffeoyl quinic acid,3,5-Dicaffeoylquinic Acid

Others Others
3,5-O-Dicaffeoylquinic acid (Isochlorogenic Acid A) 能够改善由三甲基锡诱导的学习和记忆缺陷。
T0034 Cortisone acetate

醋酸可的松,Cortisone 21-acetate,NSC 49420

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Cortisone acetate (NSC-49420) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。它在高浓度下能够部分干预 Glucocorticoid 与Glucocorticoid-receptor 的结合。它具有免疫抑制和消炎的作用。
TN6694 5,6-Benzoflavone

β-Naphthoflavone,beta-NF

Antioxidant oxidation-reduction
5,6-Benzoflavone (β-Naphthoflavone) 是芳烃受体的外源配体,可破坏人肝癌 HepG2 细胞中的锌稳态。5,6-Benzoflavone (β-Naphthoflavone) 具有抗炎和抗氧化活性,抑制通过 AKT/Nrf-2/HO-1-NF-kappaB 信号转导轴,抑制 LPS 诱导的炎症,抑制TNF-α诱导的ICAM-1和VCAM-1表达,可用于研究神经退行性疾病。
T2915 Bardoxolone

RTA 401,齐墩果烷三萜化合物,CDDO

Others; Nrf2 Immunology/Inflammation; Others
Bardoxolone (CDDO) 是新型核调节因子激活剂。
T1168 Desonide

Tridesilon,地索奈德,Locapred,Prednacinolone

Glucocorticoid Receptor Endocrinology/Hormones
Desonide (Prednacinolone) 是一种非氟化皮质类固醇抗炎剂,能够作用于糖皮质激素受体。
T4S0498 Glaucocalyxin A

蓝萼甲素,Wangzaozin B,Leukamenin F

Apoptosis; Akt; Caspase; PI3K Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Glaucocalyxin A (Leukamenin F) 是来自日本黑纹病菌的一种对映型月桂基二萜,具有抗肿瘤作用。它通过调节PI3K/Akt 信号通路抑制 GLI1 的核易位,诱导骨肉瘤凋亡。
T37974 (S)-Coriolic acid

13(S)-HODE

Lipoxygenase; Mitochondrial Metabolism; PPAR DNA Damage/DNA Repair; Metabolism
(S)-Coriolic acid (13(S)-HODE) 是一种重要的细胞内信号剂,是亚油酸与植物和哺乳动物脂氧合酶反应生成的,在各种生物系统中参与细胞增殖和分化。(S)-Coriolic acid 在 1 μM 左右时,它能抑制肿瘤细胞与血管内皮的粘附,能下调 IRGpIIb/IIIa 受体的表达。(S)-Coriolic acid 是15-脂氧合酶 (15-LOX) 代谢产物,常作为内源性配体激活 PPARγ。(S)-Coriolic acid 诱导线粒体功能障碍 和气道上皮损伤。
T0798 Triamcinolone

Fluoxyprednisolone,曲安西龙,Aristocort,Rodinolone

Glucocorticoid Receptor; COX Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
Triamcinolone (Aristocort) 是一种皮质类固醇激素受体激动剂,也是一种合成的长效糖皮质激素,具有抗炎活性。
T14011 2-Arachidonoylglycerol

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
2-Arachidonoylglycerol 属于人内源性代谢物,是中枢神经系统中的一种内源性大麻素配体。
T4938 Potassium 1H-indol-3-yl sulfate

硫酸吲哚钾盐,Indoxyl sulfate potassium salt,Potassium 3-indoxyl sulfate

AhR; Endogenous Metabolite Immunology/Inflammation; Metabolism
Potassium 1H-indol-3-yl sulfate (Potassium 3-indoxyl sulfate) 是人芳烃受体(AhR)的激动剂。芳烃受体(AhR)最近被发现是免疫炎症条件的病理生理调节剂,Potassium 1H-indol-3-yl sulfate 已被证明是AhR的配体。Potassium 1H-indol-3-yl sulfate 也是膳食蛋白质中色氨酸的代谢物。色氨酸被肠道细菌代谢为吲哚,吲哚被吸收到血液中,然后在肝脏中进一步代谢为硫酸吲哚,通常通过尿液排出体外。在肾功能受损的慢性肾病患者中,Potassium 1H-indol-3-yl sulfate 可作为尿毒症毒素在血清中积累,诱导氧化应激并加速疾病进展。250 μM Potassium 1H-indol-3-yl sulfate 可诱导NF-Κb活化,促进大鼠近端小管细胞TGF-β1和Smad3的表达,与促纤维化活性相关。
T13735 Imidazoleacetic acid

Imidazolyl-4-acetic acid

Others Others
Imidazoleacetic acid, an endogenous ligand, stimulates imidazole receptors.
T38468 Glycodeoxycholic acid monohydrate

Glycodeoxycholic acid monohydrate is a nuclear receptor ligand.
T10821 Cirsiliol

Lipoxygenase Metabolism
Cirsiliol is a selective inhibitor of 5-lipoxygenase and a competitive low-affinity ligand of benzodiazepine receptors.
T16846 Sauristolactam

Saurolactam

Others Others
Sauristolactam inhibits the receptor activator of nuclear factor-κB ligand (RANKL)-induced osteoclastogenesis and has the potential to inhibit osteoclast differentiation. Sauristolactam, a natural aristolactam isolated from aerial portions of Saururus Chi
TN4628 Nelumol A

FXR Metabolism
Nelumol A, and nelumal A show a potency comparable to the endogenous ligand, they may as a valuable potential novel lead compound in the search for FXR agonists.
TN1484 Cheilanthifoline

NF-κB; Antifection Microbiology/Virology; NF-κB
Cheilanthifoline has anti-osteoclastogenic property, it gives significant inhibitions on receptor activator of nuclear factor-κB ligand-induced differentiation of mouse bone marrow-derived macrophages into multinucleated osteoclasts.
T75682 Cortisol sulfate

Cortisol sulfate (Cortisol 21-sulfate) 是皮质醇 的一种代谢物。Cortisol sulfate 是细胞内运皮质激素蛋白的一种特异性配体。
T82578 Desacetylxanthanol

Desacetylxanthanol (Compound 4),源自Xanthium strumarium的倍半萜类化合物,展现出抗肿瘤坏死因子相关凋亡诱导配体(TRAIL)活性。
T21577 Narasin (sodium salt)

Naracin sodium salt,naransin sodium,海南霉素,HainanMycin

NF-κB NF-κB
Narasin (sodium salt) (HainanMycin) 通过神经胶质瘤细胞中的 ER 应激诱导肿瘤坏死因子相关凋亡诱导配体 (TRAIL) 介导的细胞凋亡,并通过抑制 IκBα 的磷酸化来抑制 NF-κB 信号传导。
TN3537 Braylin

IL Receptor; TNF; NF-κB Apoptosis; Immunology/Inflammation; NF-κB
Braylin has anti-inflammatory, antinociceptive and immunomodulatory effects, which possibly act through the glucocorticoid receptor activation and by inhibition of the transcriptional activity of NF-κB. Braylin is also a phosphodiesterase-4 inhibitor, it could represent an ideal prototype of glucocorticoid receptor ligand, able to induce synergic immunomodulatory effects.
T21500 Sphingosine-1-phosphate

S1P

Endogenous Metabolite; S1P Receptor; LPL Receptor GPCR/G Protein; Metabolism
Sphingosine-1-phosphate (S1P) 是 S1P1-5 受体 (S1P1-5 receptors) 的激动剂和 GPR3、GPR6、GPR12 的配体。Sphingosine-1-phosphate 是细胞内的第二信使,动员 Ca2+ 作为 G 蛋白偶联受体的细胞外配体。Sphingosine-1-phosphate 是由鞘磷脂 (HY-113498) 或其他膜磷脂生成的重要脂质介质。
T82572 D-Glucosyl-β-1,1′-N-palmitoylsphingosine

C16 Glucosyl(β) Ceramide (d18:1/16:0)

D-Glucosyl-β-1,1′-N-palmitoylsphingosine (C16 Glucosyl(β) Ceramide (d18:1/16:0)) 是内源性Mincle配体,具免疫刺激活性。
TN4383 Kazinol U

IL Receptor; IκB/IKK; NOS; NF-κB Immunology/Inflammation; NF-κB
Kazinol U may have therapeutic value in delaying pancreatic β-cell destruction in type 1 diabetes by blocking the NF-κB pathway in pancreatic β-cells reduces cell damage. Kazinol U shows estrogenic activity with ligand-activity of estrogen receptor, transcriptional activity of estrogen -responsive element-reporter genes, it may have beneficial effects in the treatment of menopausal symptoms.
TN3539 Broussonin A

ERK; IL Receptor; IκB/IKK; NOS; NF-κB; Akt Cytoskeletal Signaling; Immunology/Inflammation; MAPK; NF-κB; PI3K/Akt/mTOR signaling
Broussonins A and B, new phytoalexins from diseased paper mulberry. Broussonin A shows estrogenic activity with ligand-binding activity of estrogen receptor, transcriptional activity of estrogen-responsive element-luciferase reporter genes. Broussonin A c
T36563 (E)-Guggulsterone

Bile acids are essential for solubilization and transport of dietary lipids, are the major products of cholesterol catabolism, and are physiological ligands for farnesoid X receptor (FXR), a nuclear receptor that regulates genes involved in lipid metabolism.1They are also inherently cytotoxic, as physiological imbalance contributes to increased oxidative stress.2,3Bile acid-controlled signaling pathways are promising novel targets to treat such metabolic diseases as obesity, type II diabetes, hy...

天然产物

Roseoflavin
Cat.No: T24729
Synonym:
Target: Antibacterial
(-)-Isocorypalmine
Cat.No: TQ0176
Synonym: Tetrahydrocolumbamine,(-)-异延胡索单酚碱,(S)-Tetrahydrocolumbamine
Target: Dopamine Receptor, Antifungal
Methyl 3-aminopropanoate hydrochloride
Cat.No: T8097
Synonym: β-Alanine methyl ester hydrochloride,3-氨基丙酸甲酯盐酸盐
Target: Others
7α,25-Dihydroxycholesterol
Cat.No: T14063
Synonym: 7α,25-OHC
Target: EBI2/GPR183, Endogenous Metabolite
Baimaside
Cat.No: T4S0039
Synonym: 白麻苷,Quercetin-3-O-sophoroside,Quercetin 3-beta-D-sophoroside
Target: Others
Miltirone
Cat.No: TN1023
Synonym:
Target: P450, GABA Receptor
Amylin, amide, rat acetate(124447-81-0,free base)
Cat.No: TP1232L
Synonym:
Target: Amylin Receptor
(+/-)-Pinocembrin
Cat.No: TN2077
Synonym: NSC 43318,(±)-5,7-Dihydroxyflavanone
Target: GPR, Others
kaempferide
Cat.No: T3806
Synonym: Kaempferol 4'-O-methyl ether,山奈素,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Influenza Virus, Antibacterial, Autophagy
Penicillic acid
Cat.No: T13815
Synonym:
Target: Apoptosis, Caspase, Antibacterial, Antibiotic
DL-Serine
Cat.No: T8363
Synonym:
Target: PKM
3-Acetylcoumarin
Cat.No: Fr12596
Synonym:
Target: Others
Oxytocin
Cat.No: T5026
Synonym: 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)
Target: Oxytocin Receptor
Cyclen
Cat.No: TJS1183
Synonym: 轮环藤宁,1,4,7,10-tetraazacyclododecane
Target: Others
3′,4′,7-Trihydroxyflavone 
Cat.No: TN3209
Synonym:
Target: ATPase, Others, p38 MAPK, NF-κB
Oxytocin acetate
Cat.No: T5145
Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素
Target: Oxytocin Receptor
yangonin
Cat.No: T3S0738
Synonym: Y100550,甲氧醉椒素
Target: Cannabinoid Receptor, NF-κB, Autophagy
Estrone sulfate sodium
Cat.No: T36857
Synonym: 雌酮3-硫酸钠,Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate
Target: Endogenous Metabolite
Laminaran
Cat.No: T15705
Synonym: β-1,3-Glucan
Target:
1,7-Diaminoheptane
Cat.No: T7998
Synonym:
Target: Others
3,7,4'-Trihydroxyflavone
Cat.No: TN2143
Synonym: Resokaempferol,5-Deoxykampferol
Target: DNA
Paraxanthine
Cat.No: T4973
Synonym: 1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE
Target: Endogenous Metabolite
3,5-O-Dicaffeoylquinic acid
Cat.No: TL0005
Synonym: Isochlorogenic Acid A,(-)-3,5-二咖啡酰奎宁酸,(-)-3,5-Dicaffeoyl quinic acid,3,5-Dicaffeoylquinic Acid
Target: Others
Cortisone acetate
Cat.No: T0034
Synonym: 醋酸可的松,Cortisone 21-acetate,NSC 49420
Target: Glucocorticoid Receptor, Endogenous Metabolite
5,6-Benzoflavone
Cat.No: TN6694
Synonym: β-Naphthoflavone,beta-NF
Target: Antioxidant
Bardoxolone
Cat.No: T2915
Synonym: RTA 401,齐墩果烷三萜化合物,CDDO
Target: Others, Nrf2
Desonide
Cat.No: T1168
Synonym: Tridesilon,地索奈德,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
Glaucocalyxin A
Cat.No: T4S0498
Synonym: 蓝萼甲素,Wangzaozin B,Leukamenin F
Target: Apoptosis, Akt, Caspase, PI3K
(S)-Coriolic acid
Cat.No: T37974
Synonym: 13(S)-HODE
Target: Lipoxygenase, Mitochondrial Metabolism, PPAR
Triamcinolone
Cat.No: T0798
Synonym: Fluoxyprednisolone,曲安西龙,Aristocort,Rodinolone
Target: Glucocorticoid Receptor, COX
2-Arachidonoylglycerol
Cat.No: T14011
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite
Potassium 1H-indol-3-yl sulfate
Cat.No: T4938
Synonym: 硫酸吲哚钾盐,Indoxyl sulfate potassium salt,Potassium 3-indoxyl sulfate
Target: AhR, Endogenous Metabolite
Imidazoleacetic acid
Cat.No: T13735
Synonym: Imidazolyl-4-acetic acid
Target: Others
Glycodeoxycholic acid monohydrate
Cat.No: T38468
Synonym:
Target:
Cirsiliol
Cat.No: T10821
Synonym:
Target: Lipoxygenase
Sauristolactam
Cat.No: T16846
Synonym: Saurolactam
Target: Others
Nelumol A
Cat.No: TN4628
Synonym:
Target: FXR
Cheilanthifoline
Cat.No: TN1484
Synonym:
Target: NF-κB, Antifection
Cortisol sulfate
Cat.No: T75682
Synonym:
Target:
Desacetylxanthanol
Cat.No: T82578
Synonym:
Target:
Narasin (sodium salt)
Cat.No: T21577
Synonym: Naracin sodium salt,naransin sodium,海南霉素,HainanMycin
Target: NF-κB
Braylin
Cat.No: TN3537
Synonym:
Target: IL Receptor, TNF, NF-κB
Sphingosine-1-phosphate
Cat.No: T21500
Synonym: S1P
Target: Endogenous Metabolite, S1P Receptor, LPL Receptor
D-Glucosyl-β-1,1′-N-palmitoylsphingosine
Cat.No: T82572
Synonym: C16 Glucosyl(β) Ceramide (d18:1/16:0)
Target:
Kazinol U
Cat.No: TN4383
Synonym:
Target: IL Receptor, IκB/IKK, NOS, NF-κB
Broussonin A
Cat.No: TN3539
Synonym:
Target: ERK, IL Receptor, IκB/IKK, NOS, NF-κB, Akt
(E)-Guggulsterone
Cat.No: T36563
Synonym:
Target:
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