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抑制剂 & 化合物

129

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Cat. No. Product Name Target Signaling Pathways
T60063 Fluorogen binding modulator-1

Fluorogen binding modulator-1

Others Others
Fluorogen binding modulator-1 (Fluorogen binding modulator-1)是一种氟-氟激活蛋白结合对的非荧光抑制剂。
T67737 gp120-α4β7 binding inhibitor 11

HIV Protease Microbiology/Virology; Proteases/Proteasome
gp120-α4β7 binding inhibitor 11是一种抗HIV 药物。gp120-α4β7 binding inhibitor 11干扰HIV 相关糖蛋白gp12G 与整合素α4β7的结合(IC50=1.64nM)。
TP1736L Fibrinogen-Binding Peptide 137235-80-4(fb-acetate)

Others Others
Fibrinogen-Binding Peptide 137235-80-4(fb-acetate) 是纤维蛋白原受体上玻连蛋白结合位点的推定肽模拟物。它结合纤维蛋白原并抑制血小板与纤维蛋白原的粘附和血小板聚集,还抑制血小板与玻连蛋白的粘附
T40361 Integrin Binding Peptide

Integrin Binding Peptide, derived from fibronectin, holds the potential as an essential component for preparing PEG hydrogels.
T18595 Dasatinib carbaldehyde

PROTAC ABL binding moiety 4,BMS-354825 carbaldehyde

Others; Ligands for Target Protein for PROTAC Others; PROTAC
Dasatinib carbaldehyde (PROTAC ABL binding moiety 4) 基于 ABL 抑制剂达沙替尼,通过接头与 IAP 配体结合,形成 SNIPER [1]。
TP2360 A2-Binding peptide

A2-Binding peptide has involved in the assembly of MHC Class I molecules.
TP1120 Interphotoreceptor Retinoid Binding Protein Fragment (IRBP)

IRBP,Interphotoreceptor Retinoid Binding Protein Fragment IRBP

Interphotoreceptor Retinoid Binding Protein Fragment (IRBP) is a 20-residue peptide, which is a major pathogenic epitope. It exists in the first homologous repeat of interstitial visual pigment Binding Protein peptide (IRBP 161-180) and can induce post-uv
TP1736 Fibrinogen-Binding Peptide

Fibrinogen-Binding Peptide (designed by anticomplementarity hypothesis) is a presumptive peptide mimic of the vitronectin binding site on the fibrinogen receptor. Fibrinogen, a soluble plasma protein, is a cofactor in platelet activation. It is converted
T13915L PROTAC BRD9-binding moiety 1 hydrochloride

PROTAC BRD9-binding moiety 1 hydrochloride (2097512-23-5 free base)

Others Others
PROTAC BRD9-binding moiety 1 hydrochloride binds to BRD9, and used for inhibiting BRD9 activity, based on PROTAC.
TP1710 Calmodulin Binding Peptide 1

Calmodulin Binding Peptide 1, a potent CaM-binding peptide with picomolar (pM) affinity, originates from smooth muscle myosin light-chain kinase (MLCK peptide). It effectively blocks inositol trisphosphate (IP3)-induced calcium (Ca2+) release [1].
TP1120L IRBP acetate(211426-18-5 free base)

Interphotoreceptor Retinoid Binding Protein Fragment IRBP

Others Others
IRBP acetate(211426-18-5 free base) (Interphotoreceptor Retinoid Binding Protein Fragment IRBP) 是一种含有 20 个残基的肽,是一种主要的致病表位。它存在于间质视觉色素结合蛋白肽(IRBP 161-180)的第一个同源重复序列中,可诱导葡萄膜炎后(EAU)。
TP1778 Fibrinogen Binding Inhibitor Peptide

Fibrinogen Binding Inhibitor Peptide, a synthetic dodecapeptide, represents the specific platelet receptor recognition site of the human fibrinogen g-chain (residues 400-411).
T13841 PROTAC Her3-binding moiety 1

Others Others
PROTAC Her3-binding moiety 1 is a Her3 Ligand for PROTAC.
T13915 PROTAC BRD9-binding moiety 1

Epigenetic Reader Domain Chromatin/Epigenetic
PROTAC BRD9-binding moiety 1 that binds to BRD9, and used for inhibiting BRD9 activity, based on PROTAC.
T18599 PROTAC BRD4-binding moiety 1

Others Others
PROTAC BRD4-binding moiety 1 is a BRD4 ligand that binds to the cereblon ligand through a linker, enabling the formation of a PROTAC complex. This complex efficiently degrades BRD4[1].
T12557 PROTAC BET-binding moiety 1

Others Others
PROTAC BET-binding moiety 1 is a key intermediate in the synthesis of high affinity BET inhibitors
T12558 PROTAC BET-binding moiety 2

Others Others
PROTAC BET-binding moiety 2 is an BET bromodomain inhibitor.
TP1153L Fibronectin Adhesion-promoting Peptide acetate

Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate

Others Others
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate)(125720-21-0 free base) 是在纤连蛋白的羧基末端肝素结合结构域中发现的肝素结合氨基酸序列之一。
TP2254 GTP-Binding Protein Fragment, G alpha

Others Others
Using specific antisera raised against synthetic peptides, we find that three distinct GTP-binding protein alpha subunits remain bound to the plasma membrane even after activation with nonhydrolyzable GTP analog. Trypsin cleaves each alpha subunit at a si
TP1119 Interphotoreceptor retinoid-binding protein(668-687)

IRBP(668-687)

Interphotoreceptor retinoid-binding protein(668-687)is an amino acid residue of human retinoid-binding protein(IRBP) 668-687, which can induce uveitis.
T76542 ErbB-2-binding peptide

ErbB-2-binding peptide (HER2-binding peptide)为具结合肿瘤功能的肽类,其在癌症研究中显示出应用潜力。
TP2302 vitamin D binding protein precursor (353-363) [Homo sapiens]

Others Others
Human vitamin D-binding protein (hDBP) is an abundant, multifunctional, and highly polymorphic serum glycoprotein synthesized by the liver1.
T82151 Hyaluronan-binding peptide, biotin labeled

Hyaluronan-binding peptide, biotin labeled 是通过 C 端 GGGSK 残基生物素化的透明质酸结合肽,能够干预 HA 与 CD44 受体的作用,并阻碍 T 细胞增殖。 HA 在细胞外基质和细胞表面广泛表达,参与多种生物过程,包括受精、胚胎发育、伤口修复、血管新生、炎症反应和肿瘤转移。
T76527 Hepatitis B Virus Receptor Binding Fragment

Hepatitis B Virus Receptor Binding Fragment(hepatitis B peptide 4980)为一合成肽类似物,特异性结合Hep G2细胞。基于病毒中和粘附阻断理念,此Fragment可望激发保护性抗体生成,展现作为免疫原的巨大潜力。
TP2299 tumor protein p53 binding protein fragment [Homo sapiens]/[Mus musculus]

Others Others
Tumor protein p53 binding protein (53BP1) has been identified in a yeast two-hybrid screen as a protein that interacts with the central DNA–binding domain of p532. Similar to breast cancer susceptibility gene 13, 4 (BRCA1; 53BP1 enhances p53-dependent tra
T74256 PROTAC BRD9-binding moiety 5

PROTACBRD9-binding moiety 5 是一种选择性 BRD9结合剂,IC50为 4.20 μM,可用于合成 PROTACs。PROTACBRD9-binding moiety 5 对癌细胞具有抗增殖活性。
TP2190 vitamin D binding protein precrusor (208-218) [Homo sapiens]/[Oryctolagus cuniculus]

Others Others
Vitamin D-binding protein is a multifunctional, highly expressed, polymorphic serum protein. These range from the transport of vitamin D metabolites to possible roles in the immune system and host defense. The molecular weight range, the time course of ap
TP1153 Fibronectin Adhesion-promoting Peptide

Heparin Binding Peptide

Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin.
T80233 p53 CBS

p53 Consensus binding sequence

p53 CBS(p53共有DNA结合位点)是一种具备生物活性的肽类化合物。
T82059 Interphotoreceptor retinoid-binding protein(668-687) TFA

IRBP(668-687) TFA

Interphotoreceptor retinoid-binding protein(668-687) TFA 为光受体视黄醇结合蛋白的668至687氨基酸片段,具有诱发葡萄膜炎的能力。
T80992 Thrombospondin (TSP-1)-derived CD36 binding motif

Thrombospondin (TSP-1)-derived CD36 binding motif 是一种源自基质结合糖蛋白TSP-1的生物活性肽,具备与CD36相互作用的关键结合基序。该肽通过二硫键形成环状结构,与癌症转移、肿瘤粘附和新血管形成等过程相关。研究表明,它能竞争性抑制血小板聚集和肿瘤转移。
T83742 SBP1 TFA

Spike Binding Peptide 1

Spike binding peptide 1 (SBP1) 为对应于血管紧张素转换酶2 (ACE2) 的第21至43位氨基酸的肽。已将脂质纳米粒子 (LNPs) 包裹的抗病毒化合物奥司他韦磷酸盐与SBP1结合并通过体外研究评估其控制释放奥司他韦磷酸盐的长期潜力。SBP1 (2%) 固定于交联的羟基丙烯酸酯和乙基黄原酸乙酯网络,提高了对严重急性呼吸系统冠状病毒2(SARS-CoV-2)刺突糖蛋白,亦称表面糖蛋白,的网络捕获效率。
T18612 Bestatin-amido-Me

PROTAC IAP binding moiety 1

Others Others
Bestatin-amido-Me, a derivative of Bestatin, acts as an IAP ligand and interacts with ABL inhibitor through a linker to produce SNIPER[1].
T18641 SirReal1-O-propargyl

PROTAC Sirt2-binding moiety 1

Others Others
SirReal1-O-propargyl is a selective and highly potent Sirtuin 2 (Sirt2) inhibitor, with an IC50 of 2.4 μM. SirReal1-O-propargyl, the SirReal1-based moiety, binds to the cereblon ligand via a linker to form PROTAC to degrade Sirt2[1].
T76566 Fsh receptor-binding inhibitor fragment(bi-10)

FSHreceptor-binding inhibitor fragment(bi-10) 是一种有效的 FSH 拮抗剂。FSHreceptor-binding inhibitor fragment(bi-10) 阻断 FSH 与 FSHR 的结合,并在受体水平上改变 FSH 的作用。FSHreceptor-binding inhibitor fragment(bi-10) 导致小鼠排卵抑制和卵泡闭锁。FSHreceptor-binding inhibitor fragment(bi-10) 通过下调卵巢中 FSHR 和 ERβ的过度表达来抑制卵巢癌发生。
T83756 S1H TFA

Site 1-binding Helix

S1H是一种人造肽类模拟物,模仿人类生长激素的第36至51个氨基酸,且为生长激素受体的拮抗剂。在溶液中呈现α-螺旋结构,并在100和200纳摩尔(nM)的浓度下,能降低SK-MEL-28和MALME-3M黑色素瘤细胞系以及IM-9 B细胞淋巴细胞中,由人类生长激素及泌乳素诱导的STAT5磷酸化。
TP1152 Fibronectin Adhesion-promoting Peptide TFA

Heparin Binding Peptide TFA

Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin. It promotes assembly of mesenchymal stem cell (MSC) spheroids into lar
T19172 A-1210477-piperazinyl

PROTAC Mcl1-binding moiety 1

Others Others
A-1210477-piperazinyl is a compound that specifically targets and binds to the protein myeloid cell leukemia 1 (MCL1). This compound is utilized in PROTAC technology, which harnesses the ability to selectively degrade target proteins.
T18601 Desmethyl-QCA276

PROTAC BRD4-binding moiety 4

Others Others
Desmethyl-QCA276, the QCA276-based moiety, binds to cereblon ligand via a linker to form PROTAC to degrade BET. QCA276 is a BET inhibitor with an IC50 of 10 nM, and with a Ki of 2.3 nM[1].
T13914 SLF-amido-C2-COOH

PROTAC FKBP12-binding moiety 1

Others Others
SLF-amido-C2-COOH is a synthetic ligand for FKBP (SLF), and can be used in the synthesis of PROTACs.
T18613 MV-1-NH-Me

PROTAC IAP binding moiety 2

Others Others
MV-1-NH-Me, an MV-1-derived IAP ligand, connects to an ABL inhibitor through a linker, resulting in the formation of SNIPER[1].
T18594 HG-7-85-01-Decyclopropane

PROTAC ABL binding moiety 3

Others Others
Decyclopropane, also known as HG-7-85-01, is a chemical compound with ABL inhibitor properties. It binds to the IAP ligand through a linker, resulting in the formation of SNIPER [1].
T81356 PTBP1-RNA-binding inhibitor P6 TFA

PTBP1 α3-helix derived peptide P6 TFA

PTBP1-RNA-binding inhibitor P6 (PTBP1 α3-helix derived peptide P6) TFA 为剪接因子PTBP1的特定钉合肽抑制剂,用于抑制PTBP1调控的RNA选择性剪接事件。该抑制剂通过与PTBP1的RNA识别基序相结合,从而发挥其作用。
T18593 GNF5-amido-Me

PROTAC ABL binding moiety 2

Others Others
GNF5-amido-Me, the moiety based on GNF5 (ABL inhibitor),binds through a linker to the IAP ligand forming SNIPER[1].
T18611 AP1867-2-(carboxymethoxy)

PROTAC FKBP12-binding moiety 2

Others Others
AP1867-2-(carboxymethoxy), a moiety based on the synthetic FKBP12F36V-directed ligand AP1867, connects to the CRBN ligand through a linker to generate dTAG molecules[1].
T83729 Tat-CIRP TFA

Tat-Cold-inducible RNA Binding Protein

Tat-CIRP是一种肽类抑制剂,用于抑制髓样分化2蛋白(MD-2,亦称淋巴细胞抗原96 [LY96])与寒冷诱导的RNA结合蛋白(CIRP)之间的蛋白-蛋白相互作用。它通过与MD-2结合,干扰MD-2与CIRP之间的相互作用,这一作用在共免疫沉淀实验中得到证实。在体内实验中,Tat-CIRP (10及20 mg/kg) 能够减少由中脑动脉闭塞(MCAO)引发的小鼠脑梗死体积。同样,在通过血栓引发脑梗死的恒河猴模型中,Tat-CIRP同样能减少脑梗死体积,并缩短患中风一侧手臂抓取并放下食物的时间。
T37473 SBFI AM

Sodium-binding Benzofuran Isophthalate Acetoxymethyl ester

SBFI AM is a membrane-permeant, fluorescent Na+ indicator dye. It is selective for Na+ over K+ with Kd values of 20 and 120 mM for these ions, respectively. [1]Increasing concentration of Na+ increases the ratio of excitation efficiency at 330-345 nm to that at 370-390 nm with emission collected at 450-550 nm. [1] Therefore, ratio fluorometry and imaging can be performed with the same wavelengths. SBF AM is suitable for single intracellular dye injection and is typically used for high-resolutio...
T15585 IRBP(668-687) (TFA)

Interphotoreceptor retinoid-binding protein(668-687) TFA

Others Others
Interphotoreceptor retinoid-binding protein TFA is the amino acid residue 668 to 687 of human interphotoreceptor retinoid-binding protein (IRBP). It also induces uveitis.
T14298 Rimiducid

Apoptosis; Others; Fatty Acid Synthase Apoptosis; Metabolism; Others
Rimiducid 是一种可渗透脂质的他克莫司类似物,是一种二聚剂,通过交联 FKBP 结构域起作用。它将 Caspase 9 自杀开关二聚化并迅速诱导细胞凋亡。
T83193 Acetyl-Heme-Binding Protein 1 (1-21) (human)

Acetyl-Heme-Binding Protein 1 (1-21) (human)为一种由Acetyl-Heme-Binding Protein 1前21个氨基酸组成的短肽。该肽具有与血红素结合的能力,参与血红素代谢及血红蛋白释放过程。

化合物

Fluorogen binding modulator-1
Cat.No: T60063
Synonym: Fluorogen binding modulator-1
Target: Others
gp120-α4β7 binding inhibitor 11
Cat.No: T67737
Synonym:
Target: HIV Protease
Fibrinogen-Binding Peptide 137235-80-4(fb-acetate)
Cat.No: TP1736L
Synonym:
Target: Others
Integrin Binding Peptide
Cat.No: T40361
Synonym:
Target:
Dasatinib carbaldehyde
Cat.No: T18595
Synonym: PROTAC ABL binding moiety 4,BMS-354825 carbaldehyde
Target: Others, Ligands for Target Protein for PROTAC
A2-Binding peptide
Cat.No: TP2360
Synonym:
Target:
Interphotoreceptor Retinoid Binding Protein Fragment (IRBP)
Cat.No: TP1120
Synonym: IRBP,Interphotoreceptor Retinoid Binding Protein Fragment IRBP
Target:
Fibrinogen-Binding Peptide
Cat.No: TP1736
Synonym:
Target:
PROTAC BRD9-binding moiety 1 hydrochloride
Cat.No: T13915L
Synonym: PROTAC BRD9-binding moiety 1 hydrochloride (2097512-23-5 free base)
Target: Others
Calmodulin Binding Peptide 1
Cat.No: TP1710
Synonym:
Target:
IRBP acetate(211426-18-5 free base)
Cat.No: TP1120L
Synonym: Interphotoreceptor Retinoid Binding Protein Fragment IRBP
Target: Others
Fibrinogen Binding Inhibitor Peptide
Cat.No: TP1778
Synonym:
Target:
PROTAC Her3-binding moiety 1
Cat.No: T13841
Synonym:
Target: Others
PROTAC BRD9-binding moiety 1
Cat.No: T13915
Synonym:
Target: Epigenetic Reader Domain
PROTAC BRD4-binding moiety 1
Cat.No: T18599
Synonym:
Target: Others
PROTAC BET-binding moiety 1
Cat.No: T12557
Synonym:
Target: Others
PROTAC BET-binding moiety 2
Cat.No: T12558
Synonym:
Target: Others
Fibronectin Adhesion-promoting Peptide acetate
Cat.No: TP1153L
Synonym: Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate
Target: Others
GTP-Binding Protein Fragment, G alpha
Cat.No: TP2254
Synonym:
Target: Others
Interphotoreceptor retinoid-binding protein(668-687)
Cat.No: TP1119
Synonym: IRBP(668-687)
Target:
ErbB-2-binding peptide
Cat.No: T76542
Synonym:
Target:
vitamin D binding protein precursor (353-363) [Homo sapiens]
Cat.No: TP2302
Synonym:
Target: Others
Hyaluronan-binding peptide, biotin labeled
Cat.No: T82151
Synonym:
Target:
Hepatitis B Virus Receptor Binding Fragment
Cat.No: T76527
Synonym:
Target:
tumor protein p53 binding protein fragment [Homo sapiens]/[Mus musculus]
Cat.No: TP2299
Synonym:
Target: Others
PROTAC BRD9-binding moiety 5
Cat.No: T74256
Synonym:
Target:
vitamin D binding protein precrusor (208-218) [Homo sapiens]/[Oryctolagus cuniculus]
Cat.No: TP2190
Synonym:
Target: Others
Fibronectin Adhesion-promoting Peptide
Cat.No: TP1153
Synonym: Heparin Binding Peptide
Target:
p53 CBS
Cat.No: T80233
Synonym: p53 Consensus binding sequence
Target:
Interphotoreceptor retinoid-binding protein(668-687) TFA
Cat.No: T82059
Synonym: IRBP(668-687) TFA
Target:
Thrombospondin (TSP-1)-derived CD36 binding motif
Cat.No: T80992
Synonym:
Target:
SBP1 TFA
Cat.No: T83742
Synonym: Spike Binding Peptide 1
Target:
Bestatin-amido-Me
Cat.No: T18612
Synonym: PROTAC IAP binding moiety 1
Target: Others
SirReal1-O-propargyl
Cat.No: T18641
Synonym: PROTAC Sirt2-binding moiety 1
Target: Others
Fsh receptor-binding inhibitor fragment(bi-10)
Cat.No: T76566
Synonym:
Target:
S1H TFA
Cat.No: T83756
Synonym: Site 1-binding Helix
Target:
Fibronectin Adhesion-promoting Peptide TFA
Cat.No: TP1152
Synonym: Heparin Binding Peptide TFA
Target:
A-1210477-piperazinyl
Cat.No: T19172
Synonym: PROTAC Mcl1-binding moiety 1
Target: Others
Desmethyl-QCA276
Cat.No: T18601
Synonym: PROTAC BRD4-binding moiety 4
Target: Others
SLF-amido-C2-COOH
Cat.No: T13914
Synonym: PROTAC FKBP12-binding moiety 1
Target: Others
MV-1-NH-Me
Cat.No: T18613
Synonym: PROTAC IAP binding moiety 2
Target: Others
HG-7-85-01-Decyclopropane
Cat.No: T18594
Synonym: PROTAC ABL binding moiety 3
Target: Others
PTBP1-RNA-binding inhibitor P6 TFA
Cat.No: T81356
Synonym: PTBP1 α3-helix derived peptide P6 TFA
Target:
GNF5-amido-Me
Cat.No: T18593
Synonym: PROTAC ABL binding moiety 2
Target: Others
AP1867-2-(carboxymethoxy)
Cat.No: T18611
Synonym: PROTAC FKBP12-binding moiety 2
Target: Others
Tat-CIRP TFA
Cat.No: T83729
Synonym: Tat-Cold-inducible RNA Binding Protein
Target:
SBFI AM
Cat.No: T37473
Synonym: Sodium-binding Benzofuran Isophthalate Acetoxymethyl ester
Target:
IRBP(668-687) (TFA)
Cat.No: T15585
Synonym: Interphotoreceptor retinoid-binding protein(668-687) TFA
Target: Others
Rimiducid
Cat.No: T14298
Synonym:
Target: Apoptosis, Others, Fatty Acid Synthase
Acetyl-Heme-Binding Protein 1 (1-21) (human)
Cat.No: T83193
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TWS1977 Kamebakaurin

尾叶香茶菜丙素,Kamebakaurine

NF-κB NF-κB
Kamebakaurin (Kamebakaurine) 是一种提取自Isodon japonicus 中的天然产物,是一种NF-κB 的抑制剂,能够抑制 p50 的 DNA 结合活性。
T6995 Ochromycinone

STA 21,STA21,STA-21

Antibacterial; STAT JAK/STAT signaling; Microbiology/Virology; Stem Cells
Ochromycinone (STA 21) 是一种天然抗生素,也是一种 STAT3抑制剂。它可抑制 STAT3DNA 结合活性,STAT3二聚化。它具有抗癌和抗菌活性。
T2144 Tacrolimus

他克莫司,Fujimycin,FK506,FR900506

Phosphatase; Others; Antibacterial; Antibiotic; mTOR; Autophagy Autophagy; Metabolism; Microbiology/Virology; Others; PI3K/Akt/mTOR signaling
Tacrolimus (Fujimycin) 可与 FKBP12 结合形成高亲和力复合物 (Ki: 0.2 nM),抑制钙/钙调蛋白依赖性蛋白磷酸酶的活性。
T6569 Mimosine

Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine

Others Others
Mimosine (Leucenol) 是一种酪氨酸类似物,具有抗癌和抗炎等活性。它可通过其强大的铁结合活性作为抗氧化剂,是一种 Fe(III) 螯合剂。它作用于人类白血病细胞,通过金属离子螯合、线粒体激活和诱导活性氧产生来诱导细胞凋亡。
T2481 Ascomycin

FK520,Immunomycin,子囊霉素,FR-900520

Phosphatase; Others; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology; Others
Ascomycin (Immunomycin) 是 Tacrolimus 的乙基类似物,具有免疫抑制特性。它也是一种大环聚酮类抗生素,具有抗疟疾、抗真菌和抗痉挛等多种生物活性。它可防止移植排斥,并具有用于各种皮肤病研究的潜力。
T1537 Rapamycin

Sirolimus,AY 22989,雷帕霉素,NSC-2260804

Others; Endogenous Metabolite; Antibiotic; mTOR; Autophagy; Antifungal Autophagy; Metabolism; Microbiology/Virology; Others; PI3K/Akt/mTOR signaling
Rapamycin (AY 22989) 属于大环内酯类天然产物,是一种 mTOR 抑制剂,具有特异性(HEK293 细胞:IC50=0.1 nM)。Rapamycin 具有免疫抑制活性,并能诱导自噬。
T20879 Tacrolimus monohydrate

FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506

Phosphatase; Others; Antibacterial; Antibiotic; Autophagy Autophagy; Metabolism; Microbiology/Virology; Others
Tacrolimus monohydrate (LCP-Tacro) 是大环内酯类化合物,它与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶,从而抑制 T 淋巴细胞信号转导和 IL-2 转录。具有强免疫抑制特性。
TN1653 Fustin

ERK; Beta Amyloid; AChR MAPK; Neuroscience
Fustin 是植物漆树 (Rhus verniciflua Stokes) 的植物性黄烷醇成分。 Fustin 对 6-羟基多巴胺诱导的神经元细胞死亡具有保护作用。
T5S0273 Hypaphorine

Lenticin,Glyyunnanenine,Tryptophan Betaine,刺桐碱

Others Others
Hypaphorine (Lenticin) 是一种提取自 Pisolithus tinctorius 中的吲哚类生物碱,对啮齿动物具有有神经学影响降糖活性。
T21351 Maytansine

NSC-153858,NSC153858,Maitansina,NSC 153858,Maitansine,美坦新

Microtubule Associated; Antibiotic Cytoskeletal Signaling; Microbiology/Virology
Maytansine (NSC-153858) 是从变叶美登木中分离的一种高效微管靶向天然产物,可诱导有丝分裂阻滞并在亚纳摩尔浓度杀死肿瘤细胞。
TN6722 Terminolic acid

2α,6β,23-trihydroxyl oleanolic acid

Antibacterial Microbiology/Virology
Terminolic acid (2α,6β,23-trihydroxyl oleanolic acid) 是一种从 Combretum racemosum 中分离得到的五环三萜糖苷,可通过与 IL-1β 和 IL-6 的受体活性位点结合抑制促炎细胞因子,并通过与 IL-4 受体结合位点结合增强抗炎细胞因子。它还表现出适度的抗菌活性。
T7097 Cytochalasin B

Phomin,细胞松弛素 B,细胞松弛素B

Arp2/3 Complex Cytoskeletal Signaling
Cytochalasin B is a mycotoxin binding to the barbed end of actin filaments. It can disrupt the formation of actin polymers (Kd: 1.4-2.2 nM for F-actin).
T4839 Ac-Ala-OH

N-Acetylalanine,N-Acetyl-L-alanine,N-乙酰-L-丙氨酸

Others; Endogenous Metabolite Metabolism; Others
Ac-Ala-OH (N-Acetyl-L-alanine) 是鸟嘌呤核苷酸结合蛋白G(I)/G(S)/G(O) γ -2亚基、髓鞘碱性蛋白、GTP-结合核蛋白 Ran、原肌球蛋白 α - 4链、HIV-1 Rev 结合蛋白2、Xaa-Pro 二肽酶、胸腺酶 β -10、肌动蛋白样蛋白3、丙氨酸转氨酶、丝氨酸/苏氨酸蛋白磷酸酶PP1 - β催化亚基、10 kda 热休克蛋白(线粒体)、钙调蛋白和 β -1-syntrophin 的底物。
T13592 Calf thymus DNA

DNA from calf thymus, Thymonucleic acid

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Calf thymus DNA (DNA from calf thymus, Thymonucleic acid) 是一种从牛胸腺中提取出来的高质量双链模板DNA,可广泛应用于DNA 结合抗癌剂和调节DNA 结构和功能的DNA 结合剂的研究。
TN1202 (-)-α-Pinene

左旋-α-蒎烯,左旋-alpha-蒎烯,(1S)-(-)-Alpha-Pinene

Virus Protease; GABA Receptor; Endogenous Metabolite; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) 是一种单萜类化合物,通过延长 GABAergic 突触传递、作为 GABAA-BZD 受体的部分调节剂并直接与 GABAA 受体的 BZD 结合位点结合来增强 NREMS 的数量而不影响 NREMS 的强度。
T0912L Tetracycline

Deschlorobiomycin,Tetracyclinum,Tetracyclin,四环素

Others; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Others
Tetracycline (Tetracyclin) 是一种对多种革兰氏阳性和革兰氏阴性细菌有抑制活性的广谱抗生素。
T30086 Anthragallol

Anthragallic acid,1,2,3-Trihydroxyanthraquinone

Others Others
Anthragallol(1,2,3-Trihydroxyanthraquinone) 通过与 DNA 结合而显示出细胞毒性。Anthragallol 可作为分析试剂,可用于生产棕色酸洗色料。
T16552 Pleuromutilin

Mutilin 14-glycolate,Drosophilin B,截短侧耳素

Antibacterial; Antibiotic Microbiology/Virology
Pleuromutilin (Drosophilin B) 通过与细菌的 50S 核糖体亚基结合来抑制细菌蛋白质的合成。
T1653 Liothyronine

Tresitope,O-(4-Hydroxy-3-iodophenyl)-3,5-diiodo-L-tyrosine,碘噻罗宁,Triiodothyronine,三碘甲状腺原氨酸,L-3,3',5-Triiodothyronine,3,3',5-Triiodo-L-thyronine,Lyothyronine

Thyroid hormone receptor(THR); Endogenous Metabolite Endocrinology/Hormones; Metabolism
Liothyronine (Tresitope) 是一种有效的甲状腺激素,能够激活 β1 甲状腺激素受体 (TRβ1)。
T5855 Edrophonium chloride

AChE Neuroscience
Edrophonium chloride 是一种乙酰胆碱酯酶抑制剂,可通过特异性结合其催化位点来防止神经递质乙酰胆碱的分解。
T3806 kaempferide

Kaempferol 4'-O-methyl ether,山奈素,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Influenza Virus; Antibacterial; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology
kaempferide (4'-Methylkaempferol) 是一种存在于山柰中的O-甲基化黄酮醇,具有抗病毒活性。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
T5081 Adenine monohydrochloride hemihydrate

腺嘌呤盐酸盐,Adenine hydrochloride hydrate,6-Aminopurine hydrochloride hydrate

Endogenous Metabolite; Adenosine Receptor GPCR/G Protein; Metabolism; Neuroscience
Adenine monohydrochloride hemihydrate 是内源性代谢产物的一种。
TJS1183 Cyclen

轮环藤宁,1,4,7,10-tetraazacyclododecane

Others Others
Cyclen (1,4,7,10-tetraazacyclododecane) 是一种氮杂冠醚的类似物,是制备有效的大环螯合物的中间体,是制备磁共振造影剂的前体物质。
TN6779 Clausine E

Others Others
Clausine E 是脂肪量和肥胖相关蛋白 (FTO) 脱甲基酶活性的抑制剂。 Clausine E 与 FTO 的结合是由正熵和负焓变化驱动的。
T2219 Puromycin dihydrochloride

CL13900 dihydrochloride,Puromycin 2HCl,嘌呤霉素二盐酸盐水合物,嘌呤霉素二盐酸盐

ribosome; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Puromycin dihydrochloride (CL13900 dihydrochloride) 属于肉桂酰胺腺苷抗生素,是一种蛋白质合成的抑制剂。Puromycin dihydrochloride 通过与 RNA 结合来抑制蛋白质合成,具有抗肿瘤和抗锥虫活性。
T13502 3-Oxo-5β-cholanoic acid

3-氧代-5β-胆烷酸,Dehydrolithocholic acid

ROR Metabolism
3-Oxo-5β-cholanoic acid (Dehydrolithocholic acid) 是胆汁酸的一种代谢产物。3-Oxo-5β-cholanoic acid 直接与关键转录因子RORγt(Kd=1.13 μM) 结合抑制TH17细胞分化。
TN2165 Rubrofusarin gentiobioside

Rubrofusarin-6-O-beta-D-gentiobioside,红链霉素-龙胆二糖苷,芸苔红素龙胆苷

ERK; NF-κB; TGF-beta/Smad MAPK; NF-κB; Stem Cells
Rubrofusarin gentiobioside (Rubrofusarin-6-O-beta-D-gentiobioside) 一种分离自决明子的、具有清除自由基作用的化合物。
T3810 Saikosaponin B2

柴胡皂苷 B2,柴胡皂甙 B2

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。
TN2030 P-Hydroxyphenethyl trans-ferulate

反式-阿魏酸对羟基苯乙酯

5-HT Receptor GPCR/G Protein; Neuroscience
p-Hydroxyphenethyl trans-ferulate 具有抗高血糖 (酵母α-葡萄糖苷酶,IC5019.24 ± 1.73 µmol L-1),抗氧化,抗炎活性,也具有抗癌特性和血清素能特性。
T3829 Ginsenoside F3

人参皂苷F3

Others; IFNAR; Interleukin Immunology/Inflammation; Others
Ginsenoside F3 是一种皂苷,提取自Panax ginseng 叶片。它能够调节1 型 (IL-2, IFN-γ) 及 2 型细胞因子(IL-4 and IL-10) 的产生和表达,有免疫增强的作用。
TN2269 Tetramethylcurcumin

Apoptosis; STAT Apoptosis; JAK/STAT signaling; Stem Cells
Tetramethylcurcumin 是一种新型姜黄素类似物,是一种有效的 STAT3 磷酸化、DNA 结合活性和体外反式激活抑制剂。它具有抗炎和抗癌作用。
T21430 Oxytetracycline Hydrochloride

Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin

Antiviral; Endogenous Metabolite; Antibacterial; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。
T65128 Tartaric acid disodium dihydrate

Disodium L-(+)-Tartrate Dihydrate

Phosphatase; Endogenous Metabolite Metabolism
Tartaric acid disodium dihydrate (Disodium L-(+)-Tartrate Dihydrate) 常用来制作分子生物学和细胞培养中的缓冲液,。Tartaric acid disodium dihydrate 是酸性磷酸酶抑制剂, 可增加秋水仙碱结合 tubulin1的概率。
T7054 N-Benzoyl-(2R,3S)-3-phenylisoserine

N-苯甲酰基-(2R,3S)-3-苯基异丝氨酸,taxol side chain

Antiviral Immunology/Inflammation
N-Benzoyl-(2R,3S)-3-phenylisoserine (taxol side chain) 是一种制备用于研究结合位点位置的强效抗癌药物紫杉醇的中间体。 它显示出细胞毒性、抗病毒和免疫调节活性。
TN1325 (2S)-6-Prenylnaringenin

(2S)-6-异戊烯基柚皮素,6-异戊二烯基柚皮素,6-Prenylnaringenin,6-PN

GABA Receptor Membrane transporter/Ion channel; Neuroscience
(2S)-6-Prenylnaringenin (6-Prenylnaringenin) 是强效植物雌激素 8-prenylnaringenin 的异构体,是前脑中最有效的化合物,在 α+β 结合位点上起GABAA 正变构调节剂的作用。
T6389 Anacardic Acid

漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid

Others; Epigenetic Reader Domain; Histone Acetyltransferase; Antibacterial Chromatin/Epigenetic; Microbiology/Virology; Others
Anacardic Acid (6-pentadecylsalicylic Acid) 是从腰果壳中提取液中分离到的酸类物质,是一种组蛋白乙酰转移酶抑制剂,对 p300 和 PCAF 的 IC50值分别为 ∼8.5 μM 和 ∼5 μM。
T4717 25-Hydroxycholesterol

25-羟基胆固醇,25-羟基胆甾醇

Others; Endogenous Metabolite; HMG-CoA Reductase Metabolism; Others
25-Hydroxycholesterol 是胆固醇的代谢产物,由巨噬细胞响应 Toll 样受体激活而分泌。它有效抑制 B 细胞产生 IgA,EC50约为 65 nM。
T2S0633 Raspberry ketone

Oxyphenalon,Rasketone,Aloenin,4-(4-Hydroxyphenyl)-2-butanone,p-Hydroxybenzyl acetone,Frambinone,覆盆子酮

PPAR DNA Damage/DNA Repair; Metabolism
Raspberry ketone (p-Hydroxybenzyl acetone) 是覆盆子中主要的芳香族天然产物,主要用作化妆品的香料和食品增味剂,也可作 PPAR-α激动剂。
TN7235 4-methoxylonchocarpin

TNF; NF-κB Apoptosis; NF-κB
4-methoxylonchocarpin 是从Abrus precatorius 的根中分离出来的以一种有效的抗炎化合物。4-methoxylonchocarpin 通过抑制LPS 与巨噬细胞的TLR4结合来抑制NF-κB 激活TNF 表达,抑制TNBS 引起的小鼠结肠炎。
T20939 Bimatoprost acid

17-phenyl trinor PGF2α,17-phenyl trinor Prostaglandin F2α

GPR Endocrinology/Hormones; GPCR/G Protein
Bimatoprost acid (17-phenyl trinor PGF2α) 是一种代谢稳定的 PGF2α 类似物,对 FP 受体具有潜在的拮抗活性。与 PGF2α 相比,它与绵羊黄体细胞上的 FP 受体结合的相对效力为 756%。
T6228 Irinotecan

CPT-11,Topotecin,伊立替康,(+)-Irinotecan

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan (CPT-11) 是喜树碱的衍生物,是一种 DNA 拓扑异构酶 I (Topo I) 的抑制剂。Irinotecan 通过与 Topo I 复合物结合来阻止 DNA 链的重新连接,并导致双链 DNA 断裂和细胞死亡,具有抗肿瘤活性。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T5530 Mithramycin A

Plicamycin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Mithramycin A (Plicamycin) 是一种dna 结合的抗肿瘤抗生素,选择性特异性蛋白1 (Sp1)抑制剂,通过降低Sp1蛋白抑制多种肿瘤的生长。特异性蛋白1 (Sp1)是一种锌指转录因子,调节多种细胞功能,促进肿瘤进展。
T4893 Spermidine

N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane

Endogenous Metabolite Metabolism
Spermidine (N-(3-Aminopropyl)-1,4-diaminobutane) 能够维持细胞膜稳定性,提高抗氧化酶活性,改善光系统 II 以及相关基因表达。它结合并激活 NMDA,并已显示以浓度依赖性方式增强 NMDA 诱导的电流。
T3862 Irigenin

NF-κB; Integrin Cytoskeletal Signaling; NF-κB
Irigenin 可通过特异性和选择性地阻断 Extra Domain A 域的 C-C 环上α9β1和α4β1整合素结合位点,介导其抗转移作用。可通过增强胃癌细胞中促凋亡分子的表达来敏化 TRAIL 诱导的凋亡,具有抗癌作用。
T0912 Tetracycline hydrochloride

NCI-c55561,盐酸四环素,Tetracycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。
T5244 Aminomalonic acid

2-Aminopropanedioic Acid,氨基丙二酸,Aminomalonate

Others; Endogenous Metabolite Metabolism; Others
Aminomalonic acid (Aminomalonate) 是氨基内源性代谢产物,在体外能作为来源 Leukemia 5178Y/AR 和小鼠胰腺的 L- 天冬酰胺合成酶的高效抑制剂 (Leukemia 5178Y/AR:Ki= 0.0023 M,小鼠胰腺:Ki= 0.0015 M)。它有潜力用作区分黑素瘤转移的不同阶段生物标志物。
T5S0994 N-Methylcytisine

N-甲基野靛碱,Caulophylline

Others; AChR Neuroscience; Others
N-Methylcytisine (Caulophylline) 是苦参中的一种三环喹啉类生物碱,具有降血糖、缓解疼痛和抗炎活性。它是中枢神经系统中乙酰胆碱烟碱受体的选择性配体,对鱿鱼视神经节中的烟碱乙酰胆碱受体具有很高的亲和力,Kd 为 50 nM。
T2220 2-Methoxyestradiol

2-甲氧雌二醇,二甲氧基雌二醇,NSC-659853,2-MeOE2,2-ME2

Apoptosis; Reactive Oxygen Species; Microtubule Associated; Endogenous Metabolite; HIF; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB
2-Methoxyestradiol (2-ME2) 是一种口服生物可利用的雌二醇代谢物,具有抗肿瘤活性。它通过减少内皮细胞增殖和诱导内皮细胞凋亡来抑制血管生成,也可破坏微管的稳定。它可诱导半胱天冬酶活化,导致细胞周期停滞在 G2 期、DNA 断裂和细胞凋亡。
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天然产物

Kamebakaurin
Cat.No: TWS1977
Synonym: 尾叶香茶菜丙素,Kamebakaurine
Target: NF-κB
Ochromycinone
Cat.No: T6995
Synonym: STA 21,STA21,STA-21
Target: Antibacterial, STAT
Tacrolimus
Cat.No: T2144
Synonym: 他克莫司,Fujimycin,FK506,FR900506
Target: Phosphatase, Others, Antibacterial, Antibiotic, mTOR, Autophagy
Mimosine
Cat.No: T6569
Synonym: Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine
Target: Others
Ascomycin
Cat.No: T2481
Synonym: FK520,Immunomycin,子囊霉素,FR-900520
Target: Phosphatase, Others, Antibiotic, Parasite, Antifungal
Rapamycin
Cat.No: T1537
Synonym: Sirolimus,AY 22989,雷帕霉素,NSC-2260804
Target: Others, Endogenous Metabolite, Antibiotic, mTOR, Autophagy, Antifungal
Tacrolimus monohydrate
Cat.No: T20879
Synonym: FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506
Target: Phosphatase, Others, Antibacterial, Antibiotic, Autophagy
Fustin
Cat.No: TN1653
Synonym:
Target: ERK, Beta Amyloid, AChR
Hypaphorine
Cat.No: T5S0273
Synonym: Lenticin,Glyyunnanenine,Tryptophan Betaine,刺桐碱
Target: Others
Maytansine
Cat.No: T21351
Synonym: NSC-153858,NSC153858,Maitansina,NSC 153858,Maitansine,美坦新
Target: Microtubule Associated, Antibiotic
Terminolic acid
Cat.No: TN6722
Synonym: 2α,6β,23-trihydroxyl oleanolic acid
Target: Antibacterial
Cytochalasin B
Cat.No: T7097
Synonym: Phomin,细胞松弛素 B,细胞松弛素B
Target: Arp2/3 Complex
Ac-Ala-OH
Cat.No: T4839
Synonym: N-Acetylalanine,N-Acetyl-L-alanine,N-乙酰-L-丙氨酸
Target: Others, Endogenous Metabolite
Calf thymus DNA
Cat.No: T13592
Synonym: DNA from calf thymus, Thymonucleic acid
Target: DNA/RNA Synthesis
(-)-α-Pinene
Cat.No: TN1202
Synonym: 左旋-α-蒎烯,左旋-alpha-蒎烯,(1S)-(-)-Alpha-Pinene
Target: Virus Protease, GABA Receptor, Endogenous Metabolite, Antibacterial
Tetracycline
Cat.No: T0912L
Synonym: Deschlorobiomycin,Tetracyclinum,Tetracyclin,四环素
Target: Others, ribosome, Antibacterial, Antibiotic
Anthragallol
Cat.No: T30086
Synonym: Anthragallic acid,1,2,3-Trihydroxyanthraquinone
Target: Others
Pleuromutilin
Cat.No: T16552
Synonym: Mutilin 14-glycolate,Drosophilin B,截短侧耳素
Target: Antibacterial, Antibiotic
Liothyronine
Cat.No: T1653
Synonym: Tresitope,O-(4-Hydroxy-3-iodophenyl)-3,5-diiodo-L-tyrosine,碘噻罗宁,Triiodothyronine,三碘甲状腺原氨酸,L-3,3',5-Triiodothyronine,3,3',5-Triiodo-L-thyronine,Lyothyronine
Target: Thyroid hormone receptor(THR), Endogenous Metabolite
Edrophonium chloride
Cat.No: T5855
Synonym:
Target: AChE
kaempferide
Cat.No: T3806
Synonym: Kaempferol 4'-O-methyl ether,山奈素,Kaempferol 4'-methyl ether,4'-Methylkaempferol,4'-O-Methylkaempferol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Influenza Virus, Antibacterial, Autophagy
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
Adenine monohydrochloride hemihydrate
Cat.No: T5081
Synonym: 腺嘌呤盐酸盐,Adenine hydrochloride hydrate,6-Aminopurine hydrochloride hydrate
Target: Endogenous Metabolite, Adenosine Receptor
Cyclen
Cat.No: TJS1183
Synonym: 轮环藤宁,1,4,7,10-tetraazacyclododecane
Target: Others
Clausine E
Cat.No: TN6779
Synonym:
Target: Others
Puromycin dihydrochloride
Cat.No: T2219
Synonym: CL13900 dihydrochloride,Puromycin 2HCl,嘌呤霉素二盐酸盐水合物,嘌呤霉素二盐酸盐
Target: ribosome, DNA/RNA Synthesis, Antibacterial, Antibiotic
3-Oxo-5β-cholanoic acid
Cat.No: T13502
Synonym: 3-氧代-5β-胆烷酸,Dehydrolithocholic acid
Target: ROR
Rubrofusarin gentiobioside
Cat.No: TN2165
Synonym: Rubrofusarin-6-O-beta-D-gentiobioside,红链霉素-龙胆二糖苷,芸苔红素龙胆苷
Target: ERK, NF-κB, TGF-beta/Smad
Saikosaponin B2
Cat.No: T3810
Synonym: 柴胡皂苷 B2,柴胡皂甙 B2
Target: Others, HCV Protease
P-Hydroxyphenethyl trans-ferulate
Cat.No: TN2030
Synonym: 反式-阿魏酸对羟基苯乙酯
Target: 5-HT Receptor
Ginsenoside F3
Cat.No: T3829
Synonym: 人参皂苷F3
Target: Others, IFNAR, Interleukin
Tetramethylcurcumin
Cat.No: TN2269
Synonym:
Target: Apoptosis, STAT
Oxytetracycline Hydrochloride
Cat.No: T21430
Synonym: Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin
Target: Antiviral, Endogenous Metabolite, Antibacterial, HSV
Tartaric acid disodium dihydrate
Cat.No: T65128
Synonym: Disodium L-(+)-Tartrate Dihydrate
Target: Phosphatase, Endogenous Metabolite
N-Benzoyl-(2R,3S)-3-phenylisoserine
Cat.No: T7054
Synonym: N-苯甲酰基-(2R,3S)-3-苯基异丝氨酸,taxol side chain
Target: Antiviral
(2S)-6-Prenylnaringenin
Cat.No: TN1325
Synonym: (2S)-6-异戊烯基柚皮素,6-异戊二烯基柚皮素,6-Prenylnaringenin,6-PN
Target: GABA Receptor
Anacardic Acid
Cat.No: T6389
Synonym: 漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid
Target: Others, Epigenetic Reader Domain, Histone Acetyltransferase, Antibacterial
25-Hydroxycholesterol
Cat.No: T4717
Synonym: 25-羟基胆固醇,25-羟基胆甾醇
Target: Others, Endogenous Metabolite, HMG-CoA Reductase
Raspberry ketone
Cat.No: T2S0633
Synonym: Oxyphenalon,Rasketone,Aloenin,4-(4-Hydroxyphenyl)-2-butanone,p-Hydroxybenzyl acetone,Frambinone,覆盆子酮
Target: PPAR
4-methoxylonchocarpin
Cat.No: TN7235
Synonym:
Target: TNF, NF-κB
Bimatoprost acid
Cat.No: T20939
Synonym: 17-phenyl trinor PGF2α,17-phenyl trinor Prostaglandin F2α
Target: GPR
Irinotecan
Cat.No: T6228
Synonym: CPT-11,Topotecin,伊立替康,(+)-Irinotecan
Target: Topoisomerase, Autophagy
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Mithramycin A
Cat.No: T5530
Synonym: Plicamycin
Target: DNA/RNA Synthesis
Spermidine
Cat.No: T4893
Synonym: N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane
Target: Endogenous Metabolite
Irigenin
Cat.No: T3862
Synonym:
Target: NF-κB, Integrin
Tetracycline hydrochloride
Cat.No: T0912
Synonym: NCI-c55561,盐酸四环素,Tetracycline HCl
Target: ribosome, Antibacterial, Antibiotic
Aminomalonic acid
Cat.No: T5244
Synonym: 2-Aminopropanedioic Acid,氨基丙二酸,Aminomalonate
Target: Others, Endogenous Metabolite
N-Methylcytisine
Cat.No: T5S0994
Synonym: N-甲基野靛碱,Caulophylline
Target: Others, AChR
2-Methoxyestradiol
Cat.No: T2220
Synonym: 2-甲氧雌二醇,二甲氧基雌二醇,NSC-659853,2-MeOE2,2-ME2
Target: Apoptosis, Reactive Oxygen Species, Microtubule Associated, Endogenous Metabolite, HIF, Autophagy
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