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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T39986 LOX-IN-3 dihydrochloride

Lipoxygenase Metabolism
LOX-IN-3 dihydrochloride 是口服有效的赖氨酰氧化酶抑制剂,在纤维化,癌症和/或血管生成方面有研究价值。
T77528 5-LOX-IN-2

Apoptosis; Lipoxygenase Apoptosis; Metabolism
5-LOX-IN-2 是 一种 5-脂氧合酶抑制剂 (5-LOX )抑制剂,从体外实验测得的IC50 值为 0.33 μM。5-LOX-IN-2 以剂量依赖的方式抑制 5-LOX发挥作用。5-LOX-IN-2 可降低肾癌细胞的细胞活性并诱导凋亡 (apoptosis),可用于研究癌症。
T65427 5-LOX inhibitor

1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one

Lipoxygenase Metabolism
5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) 是伊曲康唑杂质之一,是一种选择性 LOX-5 抑制剂。
T77677 12R-LOX-IN-2

Lipoxygenase Metabolism
12R-LOX-IN-2 是一种 12R-脂氧合酶 (12R-LOX) 的抑制剂。12R-LOX-IN-2 抑制咪喹莫特 (IMQ) 诱导银屑病角质形成细胞过度增殖,并抑制细胞集落形成。12R-LOX-IN-2 还降低 IMQ 诱导细胞中 Ki67 的蛋白水平和 IL-17A 的 mRNA 表达。12R-LOX-IN-2 可用于牛皮癣和其他皮肤相关炎症性疾病的研究。
T38006 LOX-IN-3

LOX-IN-3, an orally active inhibitor of lysyl oxidase (LOX), holds potential application in the fields of fibrosis, cancer, and angiogenesis research[1].
T61211 5-LOX-IN-1

Lipoxygenase Metabolism
5-LOX-IN-1 是一种 5-Lipoxygenase(5-LOX)抑制剂(IC50: 2.3 μM)。5-LOX-IN-1 可用于研究癌症。
T36169 15-LOX-1 inhibitor 1

9c(i472) is an inhibitor of 15-lipoxygenase-1 (15-LO-1; IC50 = 0.19 μM).1 It decreases LPS- and IFN-γ-induced NF- B activity in RAW-Blue cells when used at concentrations of 0.2, 1, and 5 μM. 9c(i472) reduces LPS- and IFN-γ-induced increases in Nos2 expression and lipid peroxidation in RAW 264.7 cells when used at a concentration of 5 μM.
T83457 12R-LOX-IN-1

12R-LOX-IN-1(Compound 4a)是一种效能为IC50: 28.25 μM的12R-LOX抑制剂。该化合物能够有效抑制Imiquimod诱导的银屑病角质形成细胞的异常增殖和集落形成能力,同时减少活性氧、Ki67、IL-17A、TNF-α和IL-6的生成,适用于抗银屑病研究。
T8356 FPL 62064

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
FPL 62064 是 5-脂氧合酶和COX 双重抑制剂,具有抗炎活性,对 RBL-1 胞质 5-脂氧合酶和前列腺素合成酶 (环氧化酶) 的IC50值分别为 3.5 和 3.1 μM。
T78820 5-LOX-IN-5

Lipoxygenase Metabolism
5-LOX-IN-5(Compound 29)作为一种5-LOX抑制剂,拥有56 nM的半抑制浓度(IC50)。它主要被应用于神经退行性疾病的研究领域。
T79158 h15-LOX-2 inhibitor 1

Lipoxygenase Metabolism
h15-LOX-2 inhibitor 1(Comp 105)是一种针对人上皮细胞15-lipoxygenase-2 (h15-LOX-2)的抑制剂,表现出0.34 μM的IC50值。
T62350 XO/COX/LOX-IN-1

XO/COX/LOX-IN-1 是一种黄嘌呤氧化酶/环氧酶/脂氧合酶 XO/COX/LOX 的有效抑制剂。XO/COX/LOX-IN-1 能够用于研究炎症、癌症以及代谢性疾病。
T62998 COX-2/15-LOX-IN-1

COX-2/15-LOX-IN-1 (Compound 14) 是一种 COX-2 和 15-脂氧合酶 (15-LOX)抑制剂,可作用于 COX-1 (IC50: 10.65 μM)、COX-2 (IC50: 0.075 μM) 和 15-LOX (IC50: 2.98 μM)。COX-2-IN-25 具有抗炎作用。
T4347 ML355

Lipoxygenase Metabolism
ML355 是一种高选择性12-LOX 抑制剂,IC50=0.34 μM,对其他脂氧化酶和环氧化酶有很好的选择性,具有较好的药物动力学特征。
T79360 COX-2/15-LOX-IN-2

Lipoxygenase Metabolism
COX-2/15-LOX-IN-2 作为一种效能高的双重抑制剂,对COX-2和15-LOX的IC50值分别为0.065 μM和1.86 μM,显示出显著的抗氧化活性。
T61674 COX-2/5-LOX-IN-1

COX-2/5-LOX-IN-1 (compound 3a), a benzothiophen-2-yl pyrazole carboxylic acid derivative, is a potent and dual inhibitor of COX-2 / 5-LOX. It exhibits superior analgesic and anti-inflammatory properties compared to Celecoxib and Indomethacin. COX-2/5-LOX-IN-1 displays strong inhibitory activity against COX-1, COX-2, and 5-LOX, with IC50 values of 12.13 μM, 0.4 μM, and 4.96 μM, respectively [1].
T8950 CAY10698

Lipoxygenase Metabolism
CAY10698 是选择性的12-Lipoxygenase (12-LOX)抑制剂,IC50=5.1 μM。它对 5-LOX、15-LOX-1、15-LOX-2 和 COX-1/2 无活性。
T61352 COX-2/5-LOX-IN-3

COX-2/5-LOX-IN-3 (compound 5b) is a powerful and dual inhibitor of COX-2 and 5-LOX, with IC50 values of 45.73 μM, 5.45 μM, and 4.33 μM for COX-1, COX-2, and 5-LOX, respectively. This compound, COX-2/5-LOX-IN-3, shows promise for the investigation of inflammatory diseases [1].
T79362 COX-2/15-LOX-IN-4

Lipoxygenase Metabolism
COX-2/15-LOX-IN-4(compound 5i)是一种针对COX-2和15-LOX的双重抑制剂,其IC50值分别为0.075 μM和1.97 μM。该化合物能有效地阻止LPS诱发的细胞内促炎细胞因子(IL-6, ROS)的产生,表现出明确的抗炎活性。
T6243 U-73122

U73122

Phospholipase; Ferroptosis; Lipoxygenase Apoptosis; Metabolism
U-73122 (U73122) 是一种磷脂酶 C 和 5-脂氧合酶抑制剂,对磷脂酶 C 的 IC50值约为 1-2.1 µM。它是一种 PLC 抑制剂,可减少激动剂诱导的血小板和 PMN 中的 Ca2+ 增加。
T60630 COX/5-LOX-IN-1

COX/5-LOX-IN-1 (compound 6b) 是有效的COX/5-LOX 双重抑制剂,具有用于炎症性疾病研究的潜力。COX/5-LOX-IN-1 对于 COX-1、COX-2 和 5-LOX 酶的IC50值分别为 1.07、0.55 和 0.28 μM。
T61479 LOX-IN-3 dihydrochloride monohydrate

LOX-IN-3 dihydrochloride monohydrate (Compound 33) is a lysyl oxidase (LOX) inhibitor with oral activity. It is specifically designed for research purposes in the areas of fibrosis, cancer, and angiogenesis [1].
T9108 BI-0115

Lipoxygenase Metabolism
BI-0115 是LOX-1的选择性抑制剂,其IC50值为 5.4 µM,可以阻止细胞摄取氧化低密度脂蛋白。它通过形成同源二聚体配体结合域的二聚体来触发受体抑制。
T61910 COX-2/5-LOX-IN-2

COX-2/5-LOX-IN-2 是苯并噻吩-2-基吡唑羧酸衍生物。COX-2/5-LOX-IN-2 (5b) 对COX-2和5-LOX 均有抑制作用。COX-2/5-LOX-IN-2 抑制 COX-1、COX-2 和 5-LOX 的IC50s 分别为 5.40、0.01 和 1.78 μM。COX-2/5-LOX-IN-2 显示出超过塞来昔布和吲哚美辛的镇痛和抗炎活性。
T79361 COX-2/15-LOX-IN-3

Lipoxygenase Metabolism
COX-2/15-LOX-IN-3 (compound 5k) 为COX-2/15-LOX的一种双重抑制剂,具有分别为0.075 μM和1.97 μM的IC50值。该化合物能显著抑制LPS诱导的细胞产生促炎细胞因子(IL-6, ROS和NO),表明其具备显著的抗炎活性。
T16503 PF-4191834

PF-04191834

Lipoxygenase Metabolism
PF-4191834 是 5-Lipoxygenase (5-LOX) 的非铁螯合和非氧化还原抑制剂,IC50 为 229 nM。 PF-4191834 对 5-LOX 的特异性比 12-LOX 和 15-LOX 高约 300 倍,并且对环氧合酶没有活性。 PF-4191834 可用于炎症和疼痛的研究。
T6568 Licofelone

利克飞龙,ML-3000

Apoptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Licofelone (ML-3000) 是一种 COX/LOX 双重抑制剂,IC50分别为 0.21和0.18 μM,有潜力研究骨关节炎,具有抗炎和抗增殖作用。它可诱导细胞凋亡,减少促炎性白三烯和前列腺素的产生。
T21746 Terameprocol

tetramethyl Nordihydroguaiaretic Acid,EM-1421

HIV Protease Microbiology/Virology; Proteases/Proteasome
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。
T22398 Phenidone

菲尼酮,1-phenyl-3-pyrazolidinone

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenidone (1-phenyl-3-pyrazolidinone) 是可口服发环氧化酶和脂氧合酶双重抑制剂,可改善实验性自身免疫性脑脊髓炎大鼠的瘫痪,降低自发性高血压大鼠的血压,可用作照片显像剂。
T10098 PGS-IN-1

KME-4

Lipoxygenase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
PGS-IN-1 (KME-4)是一种前列腺素合成酶抑制剂,IC50=0.28 μM。它也可抑制5-脂肪氧合酶的活性,IC50=1.05 μM。
T7540 2,5-Di-tert-butylhydroquinone

BHQ,2,5-二特丁基对苯二酚

Calcium Channel; Lipoxygenase; COX Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
2,5-Di-tert-butylhydroquinone (BHQ) 是一种有效和选择性的内质网 Ca2+-ATPase 抑制剂,可调节5-LO 以及COX-2活性,IC50分别为 1.8 和 14.1 μM。
T21902 ML351

Lipoxygenase Metabolism
ML351 是一种高度特异的15-LOX-1抑制剂,其 IC50=200 nM。它对 T1D 非肥胖糖尿病小鼠模型的血糖异常和β细胞氧化应激有抑制作用。它对相关同工酶 (5-LOX、血小板 12-LOX、15-LOX-2、绵羊 COX-1 和人 COX-2) 表现出良好的选择性(>250倍)。
T8794 4-MMPB

15-Lipoxygenase Inhibitor 1

Apoptosis; Others; Lipoxygenase Apoptosis; Metabolism; Others
4-MMPB (15-Lipoxygenase Inhibitor 1) 是一种选择性15-脂氧合酶抑制剂,其 IC50值为 18 μM,具有前列腺癌的研究潜力。它对大豆 15-脂氧合酶和人 15-脂氧合酶-1 的 IC50 分别为 19.5 μM 和 19.1 μM。
T0477 Zileuton

Abbott 64077,齐留通,A 64077

Ferroptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Zileuton (A 64077) 是羟基脲的合成衍生物,是一种选择性的5-脂氧合酶抑制剂,具有平喘特性。
T6576 Malotilate

Malotilatum,NKK 105,马洛替酯,Kantec

Lipoxygenase Metabolism
Malotilate (Kantec) 是一种抗纤维化物质,是一种口服活性的促肝药,可选择性抑制5-lipoxygenase (5-LOX)(IC50=4.7 μM)。它通过降低肝脏乙醛水平并防止转铁蛋白保留在肝细胞中,从而预防了酒精-吡唑肝炎中肝细胞损伤的发展。
T5200 Indirubin-3'-monoxime

靛玉红-3' -单肟,Indirubin-3'-oxime

GSK-3; Lipoxygenase; CDK Cell Cycle/Checkpoint; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
Indirubin-3'-monoxime (Indirubin-3'-oxime) 是一种有效的 GSK3β 抑制剂,IC50值为 22 nM。它对 CDK5/p25、CDK1/cyclin B 和CDk2/cyclin E 也有作用,IC50值分别为 100、180 和 250 nM。
T7724 Tepoxalin

RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Tepoxalin (RWJ 20485) 是有效的5-脂氧合酶和环氧合酶抑制剂,表现出强大的抗炎活性和较小的胃肠道刺激性。
T6893 MK-886

MK886,L 663536

Apoptosis; Leukotriene Receptor; COX; PPAR; FLAP Apoptosis; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
MK-886 (L 663536)是一种细胞可渗透的,具有口服活性的 FLAP (IC50为 30 nM) 和白三烯生物合成 (完整白细胞和人全血中的IC50分别为 3 nM 和 1.1μM) 的抑制剂。它也是一种非竞争性PPARα拮抗剂,可以诱导细胞凋亡。
T27026 CJ-13,610

CJ 13610,CJ-13610

Lipoxygenase Metabolism
CJ-13,610 是一种具有口服活性的非氧化还原型 5-脂氧合酶 (5-LOX) 抑制剂。 CJ-13,610 抑制白三烯 B4 的生物合成并调节巨噬细胞中 IL-6 mRNA 的表达。
T67908 ThioLox

Lipoxygenase Metabolism
ThioLox 是一种竞争性 15-脂氧合酶-1 (15-LOX-1) 抑制剂(IC50值为12 μM)。ThioLox 显示抗炎和神经保护特性。具有抗炎和神经保护作用,对谷氨酸毒性有很强的保护作用。
T9319 Tosufloxacin

tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid

Others Others
Tosufloxacin (Ozex) 是一种喹诺酮类抗菌剂,是茶碱代谢的有效抑制剂。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T5323 Toloxatone

托洛沙酮,MD 69276

MAO; Monoamine Oxidase Metabolism; Neuroscience
Toloxatone (MD 69276) 是可逆的单胺氧化酶 A (MAOA) 抑制剂,是一种抗抑郁剂。
T3355 Naloxegol oxalate

NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate

P450 Metabolism
Naloxegol oxalate (NKTR-118) 是一种外周选择性 opioid 样物质拮抗剂,用于治疗 opioid 样物质引起的便秘。
T1001 Dicloxacillin Sodium hydrate

Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate

Antibacterial; Antibiotic Microbiology/Virology
Dicloxacillin Sodium hydrate 是一种青霉素类窄谱β内酰胺抗生素,可研究革兰氏阳性菌感染。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T15777 Loxoribine

RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾

Influenza Virus; TLR Immunology/Inflammation; Microbiology/Virology
Loxoribine (RWJ 21757) 是一种鸟苷类似物,是一种口服生物可利用的选择性 Toll 样受体 (TLR) 7 激动剂。 具有抗病毒和抗肿瘤活性。它是一种新型的强效免疫刺激剂,具有较广谱的免疫生物学活性。
T1466 Nadifloxacin

OPC7251,那氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Nadifloxacin (OPC7251) 是一种对粉刺有效的广谱氟喹诺酮类抗生素。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T1107 Sarafloxacin hydrochloride

Sarafloxacin HCl,盐酸沙拉沙星,A-56620 (hydrochloride),A-56620 HCl

Antibacterial; Antibiotic Microbiology/Virology
Sarafloxacin hydrochloride (A-56620 (hydrochloride)) 是一种抗菌化合物。

化合物

LOX-IN-3 dihydrochloride
Cat.No: T39986
Synonym:
Target: Lipoxygenase
5-LOX-IN-2
Cat.No: T77528
Synonym:
Target: Apoptosis, Lipoxygenase
5-LOX inhibitor
Cat.No: T65427
Synonym: 1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one
Target: Lipoxygenase
12R-LOX-IN-2
Cat.No: T77677
Synonym:
Target: Lipoxygenase
LOX-IN-3
Cat.No: T38006
Synonym:
Target:
5-LOX-IN-1
Cat.No: T61211
Synonym:
Target: Lipoxygenase
15-LOX-1 inhibitor 1
Cat.No: T36169
Synonym:
Target:
12R-LOX-IN-1
Cat.No: T83457
Synonym:
Target:
FPL 62064
Cat.No: T8356
Synonym:
Target: Lipoxygenase, COX
5-LOX-IN-5
Cat.No: T78820
Synonym:
Target: Lipoxygenase
h15-LOX-2 inhibitor 1
Cat.No: T79158
Synonym:
Target: Lipoxygenase
XO/COX/LOX-IN-1
Cat.No: T62350
Synonym:
Target:
COX-2/15-LOX-IN-1
Cat.No: T62998
Synonym:
Target:
ML355
Cat.No: T4347
Synonym:
Target: Lipoxygenase
COX-2/15-LOX-IN-2
Cat.No: T79360
Synonym:
Target: Lipoxygenase
COX-2/5-LOX-IN-1
Cat.No: T61674
Synonym:
Target:
CAY10698
Cat.No: T8950
Synonym:
Target: Lipoxygenase
COX-2/5-LOX-IN-3
Cat.No: T61352
Synonym:
Target:
COX-2/15-LOX-IN-4
Cat.No: T79362
Synonym:
Target: Lipoxygenase
U-73122
Cat.No: T6243
Synonym: U73122
Target: Phospholipase, Ferroptosis, Lipoxygenase
COX/5-LOX-IN-1
Cat.No: T60630
Synonym:
Target:
LOX-IN-3 dihydrochloride monohydrate
Cat.No: T61479
Synonym:
Target:
BI-0115
Cat.No: T9108
Synonym:
Target: Lipoxygenase
COX-2/5-LOX-IN-2
Cat.No: T61910
Synonym:
Target:
COX-2/15-LOX-IN-3
Cat.No: T79361
Synonym:
Target: Lipoxygenase
PF-4191834
Cat.No: T16503
Synonym: PF-04191834
Target: Lipoxygenase
Licofelone
Cat.No: T6568
Synonym: 利克飞龙,ML-3000
Target: Apoptosis, Lipoxygenase, COX
Terameprocol
Cat.No: T21746
Synonym: tetramethyl Nordihydroguaiaretic Acid,EM-1421
Target: HIV Protease
Phenidone
Cat.No: T22398
Synonym: 菲尼酮,1-phenyl-3-pyrazolidinone
Target: Lipoxygenase, COX
PGS-IN-1
Cat.No: T10098
Synonym: KME-4
Target: Lipoxygenase, Prostaglandin Receptor
2,5-Di-tert-butylhydroquinone
Cat.No: T7540
Synonym: BHQ,2,5-二特丁基对苯二酚
Target: Calcium Channel, Lipoxygenase, COX
ML351
Cat.No: T21902
Synonym:
Target: Lipoxygenase
4-MMPB
Cat.No: T8794
Synonym: 15-Lipoxygenase Inhibitor 1
Target: Apoptosis, Others, Lipoxygenase
Zileuton
Cat.No: T0477
Synonym: Abbott 64077,齐留通,A 64077
Target: Ferroptosis, Lipoxygenase, COX
Malotilate
Cat.No: T6576
Synonym: Malotilatum,NKK 105,马洛替酯,Kantec
Target: Lipoxygenase
Indirubin-3'-monoxime
Cat.No: T5200
Synonym: 靛玉红-3' -单肟,Indirubin-3'-oxime
Target: GSK-3, Lipoxygenase, CDK
Tepoxalin
Cat.No: T7724
Synonym: RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485
Target: Lipoxygenase, COX
MK-886
Cat.No: T6893
Synonym: MK886,L 663536
Target: Apoptosis, Leukotriene Receptor, COX, PPAR, FLAP
CJ-13,610
Cat.No: T27026
Synonym: CJ 13610,CJ-13610
Target: Lipoxygenase
ThioLox
Cat.No: T67908
Synonym:
Target: Lipoxygenase
Tosufloxacin
Cat.No: T9319
Synonym: tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid
Target: Others
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Toloxatone
Cat.No: T5323
Synonym: 托洛沙酮,MD 69276
Target: MAO, Monoamine Oxidase
Naloxegol oxalate
Cat.No: T3355
Synonym: NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate
Target: P450
Dicloxacillin Sodium hydrate
Cat.No: T1001
Synonym: Dicloxacillin sodium salt monohydrate,双氯西林钠,Dicloxacillin sodium monohydrate
Target: Antibacterial, Antibiotic
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Loxoribine
Cat.No: T15777
Synonym: RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾
Target: Influenza Virus, TLR
Nadifloxacin
Cat.No: T1466
Synonym: OPC7251,那氟沙星
Target: Antibacterial, Antibiotic
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Sarafloxacin hydrochloride
Cat.No: T1107
Synonym: Sarafloxacin HCl,盐酸沙拉沙星,A-56620 (hydrochloride),A-56620 HCl
Target: Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
T6S0413 Pectolinarigenin

柳穿鱼黄素,Pectolinaringenin

Others; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience; Others
Pectolinarigenin (Pectolinaringenin) 是 COX-2/5-LOX 的双重抑制剂,可抑制炎症病变中类花生酸的形成,具有抗炎活性。
T3399 Psoralidin

Others; Estrogen/progestogen Receptor; Reactive Oxygen Species; Lipoxygenase; Gamma-secretase; Akt; COX; Antibacterial Cytoskeletal Signaling; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。
T8260 4',5-Dihydroxyflavone

Lipoxygenase; Glucosidase Metabolism
4',5-Dihydroxyflavone 是大豆 LOX-1,Ki=102.6 μM。它也是一种酵母 α-葡萄糖苷酶抑制剂,IC50=66 μM。
TQ0180 Chebulagic acid

SARS-CoV; Influenza Virus; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Chebulagic acid 是从 Terminalia chebula Retz 中分离出来的一种 COX-LOX 双重抑制剂,有抗炎和抗感染作用。它抑制 SARS-CoV-2病毒的复制,EC50值为 9.76 μM。它还是 M2(S31N)抑制剂和抗流感病毒剂。
T8002 3-Hydroxycoumarin

Lipoxygenase Metabolism
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。
T2807 Caffeic Acid

Lipoxygenase; Endogenous Metabolite; TRP/TRPV Channel Membrane transporter/Ion channel; Metabolism
Caffeic acid 是5-脂氧合酶和 TRPV1离子通道的双重抑制剂。
TN5634 Aureusidin

Auresudidin,金鱼草素,Auresidin

Antioxidant; Reactive Oxygen Species; Lipoxygenase Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。
TN2330 Phenethyl ferulate

Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenethyl ferulate (Caffeic Acid 3-Methyl Phenethyl Ester) 对化学诱导的结肠癌具有化学预防特性,可增强偶氮甲烷诱导的结肠肿瘤的细胞凋亡。 它抑制环氧合酶(COX) 和 5-脂氧合酶 (5-LOX) ,IC50 值分别为 4.35 和 5.75 μM。
T5759 S-(+)-Marmesin

(+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
S-(+)-Marmesin (marmesin) 是一种从木橘成熟树皮中分离得到的香豆素,具有 COX-2/5-LOX 双重抑制活性。
T5714 5-O-Demethylnobiletin

5-DEMETHYLNOBILETIN,去甲基川陈皮素

Leukotriene Receptor; Lipoxygenase GPCR/G Protein; Metabolism
5-O-Demethylnobiletin (5-DEMETHYLNOBILETIN) 是从黄芪中分离出的多甲氧基黄酮,具有抗炎活性,可通过直接抑制 5-LOX 发挥作用,IC50为 0.1 μM。
T3S0153 Xanthatin

苍耳亭,叶黄制菌素

Apoptosis; VEGFR; Lipoxygenase; Wnt/beta-catenin; Antibacterial Angiogenesis; Apoptosis; Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Stem Cells; Tyrosine Kinase/Adaptors
Xanthatin 是一种从Xanthium strumarium 叶子中提取的天然产物,可诱导细胞凋亡。它抑制布鲁氏菌的IC50值为 2.63 μg/ mL,对寄生虫特异性锥虫硫磷还原酶具有不可逆的弱抑制作用。它通过抑制PGE2的合成和 5-脂氧合酶的活性而显示出抗炎活性。
TJS2190 Nordihydroguaiaretic acid

去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid

Antioxidant; Ferroptosis; Lipoxygenase; Autophagy Apoptosis; Autophagy; Metabolism; oxidation-reduction
Nordihydroguaiaretic acid (NDGA) 是从极叉开拉瑞阿提取出的一种天然产物,是脂氧合酶抑制剂,具有抗氧化和清除自由基的特性。
TN1097 β-Boswellic acid

Beta-boswellic acid,β-乳香酸

Lipoxygenase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
β-Boswellic acid (Beta-boswellic acid) 是从乳香的树胶脂中分离出来的一种天然产物。它是 5-脂氧合酶(5-LO) 产物形成的非还原型抑制剂,其直接与 5-LO 相互作用或阻断其易位。具有抗癌、抗肿瘤和抗高血脂活性。
TN1255 3-O-Acetyl-11-hydroxy-beta-boswellic acid

Lipoxygenase Metabolism
3-O-Acetyl-11-hydroxy-beta-boswellic acid 是 5-脂氧合酶抑制剂。
T3384 Wedelolactone

蟛蜞菊内酯,IKK Inhibitor II

Apoptosis; NF-κB; Lipoxygenase; Caspase Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物,通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录,具有抗癌,抗炎和抗氧化活性。
TN1182 11-​Keto-​beta-​boswellic acid

11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸

Leukotriene Receptor; NF-κB; Lipoxygenase GPCR/G Protein; Metabolism; NF-κB
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸,具有抗炎活性和剂量依赖性心脏保护作用,主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
T1276 Danofloxacin mesylate

甲磺酸达氟沙星,CP 76136-27

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。
T1121 Podofilox

鬼臼毒素,Podophyllotoxin,(+)-Shikonin

Microtubule Associated; Topoisomerase Cytoskeletal Signaling; DNA Damage/DNA Repair
Podofilox ((+)-Shikonin) 是从八角莲中分离的一种木脂素,是微管组装和 DNA 拓扑异构酶 II 抑制剂。它对皮肤和粘膜有很强的刺激性,具有角质溶解作用,可用于治疗疣和角化病,具有潜在的抗肿瘤特性。
TN1343 8-Geranyloxypsoralen

8-香叶草氧基补骨脂素

Anti-infection; P450; BACE Metabolism; Microbiology/Virology; Neuroscience
8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。
T4S1658 Benzoyloxypaeoniflorin

苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷

NF-κB; Tyrosinase NF-κB; Proteases/Proteasome
Benzoyloxypaeoniflorin (Benzoyloxypeoniflorin) 是一种酪氨酸酶抑制剂,分离于Paeonia suffruticosa 的根,对mushroom tyrosinase 的 IC50为 0.453 mM。它是一种NF-κB 抑制剂,它通过对血小板聚集和凝血的抑制作用,有助于改善血液循环。
T5744 7-Prenyloxycoumarin

7-(异戊烯基氧基)香豆素,Nsc267697,7-O-Prenylumbelliferone,7-异戊烯氧基香豆素

Antifungal Microbiology/Virology
7-Prenyloxycoumarin (Nsc267697) 是一种 Heracleum dissectum 的天然产物,对乳腺癌具有预防和治疗作用。
T1549 Raloxifene hydrochloride

LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl

Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
TN1025 3,29-O-Dibenzoyloxykarounidiol

Others Others
3,29-O-Dibenzoyloxykarounidiol 是一种苯甲酸三萜烯酯,从 Momordica grosvenori 果实中提取。它能够抑制肿瘤启动子 TPA 诱导的 EB 病毒早期抗原活化。
T8046 Tosufloxacin tosylate hydrate

Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) 是一个氟喹诺酮类抗菌剂。
T1306 Norfloxacin

氟哌酸,MK-0366,诺氟沙星

DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。
TN2627 14beta-Benzoyloxy-2-deacetylbaccatin VI

Others Others
14beta-Benzoyloxy-2-deacetylbaccatin VI是一种天然产物,属于红豆杉科红豆杉属,其产品编号为 TN2627,CAS号为 705973-69-9。14beta-Benzoyloxy-2-deacetylbaccatin VI可用作对照参考。
T83558 (3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone

(3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone(化合物3)是从丹参(Salvia miltiorrhiza)根提取的棕榈酸盐。该化合物展现出抗癌活性,对于不同的人类癌症细胞系具有显著的抑制效果,其DC50值分别为:HeLa细胞系25.5 μg/mL、HepG2细胞系37.5 μg/mL以及OVCAR-3细胞系30.2 μg/mL。
T83516 (Z)-2-Angeloyloxymethyl-2-butenoic

(Z)-2-Angeloyloxymethyl-2-butenoic acid 是 An anthriscus sylvestris Hoffm. 根部的一种天然产物。
T38658 3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione

3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione, also known as an anthraquinone, has been specifically extracted from Rubia cordifolia.
TN2938 3-Hydroxy-3-acetonyloxindole

Others Others
3-Hydroxy-3-acetonyloxindole是一种天然产物,属于萝藦科牛奶菜属,其产品编号为 TN2938,CAS号为 33417-17-3。3-Hydroxy-3-acetonyloxindole可用作对照参考。
TN5683 Ethyl 4-(rhamnosyloxy)benzylcarbamate

Ethyl 4-(rhamnosyloxy)benzylcarbamate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5683,CAS号为 208346-80-9。
TN5862 8-Hydroxy-9,10-diisobutyryloxythymol

8-Hydroxy-9,10-diisobutyryloxythymol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5862,CAS号为 22518-08-7。
TN3302 8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide

Others Others
8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3302,CAS号为 109770-86-7。
TN5613 3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid

ent-3β-Cinnamoyloxy-9α,17-dihydroxykaur-15-en-19-oic acid

3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5613,CAS号为 2186648-60-0。
TN3301 8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C

Others Others
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3301,CAS号为 93395-31-4。
TN3294 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate

NADPH-oxidase; P450; MAO Immunology/Inflammation; Metabolism; Neuroscience
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes.
T83233 8-Hydroxy-9-isobutyryloxy-10-(2-methylbutanoyl)thymol

8-Hydroxy9,10-diisobutyryloxy-thymol 是从Inula sericophylla中提取的有效萜类化合物。
T38657 2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester

2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester (compound 3) is a naturally occurring substance found in the dried roots of Rubia cordifolia.
TN5303 14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide

14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5303,CAS号为 1323952-04-0。
TN5555 7α-Galloyloxysweroside

7α-Galloyloxysweroside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5555,CAS号为 2222365-76-4。
TN6331 3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid

3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6331,CAS号为 1217268-13-7。
TN3810 Dehydroperilloxin

COX Immunology/Inflammation; Neuroscience
Dehydroperilloxin possesses inhibitory activity against cyclooxygenase-1, with the IC(50) value of 30.4 microM.
TN6207 7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin

7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6207,CAS号为 118584-19-3。
TN3295 8alpha-(2-Methylacryloyloxy)hirsutinolide

Others Others
8alpha-(2-Methylacryloyloxy)hirsutinolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3295,CAS号为 188293-70-1。
TMA2415 4-Prenyloxyresveratrol

4-异戊烯基氧基白藜芦醇,4'-Prenyloxyresveratrol

Others Others
4'-Prenyloxyresveratrol is a natural product from Morus wittiorum.
TN3299 8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide

Others Others
8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3299,CAS号为 142891-14-3。
T40636 8-(3-Ethoxy-2-hydroxy-3-methylbutyloxy)psoralen

8-(3-Ethoxy-2-hydroxy-3-methylbutyloxy)psoralen is a coumarin compound present in Heracleum pyrenaicum Lam.
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天然产物

Pectolinarigenin
Cat.No: T6S0413
Synonym: 柳穿鱼黄素,Pectolinaringenin
Target: Others, Lipoxygenase, COX
Psoralidin
Cat.No: T3399
Synonym:
Target: Others, Estrogen/progestogen Receptor, Reactive Oxygen Species, Lipoxygenase, Gamma-secretase, Akt, COX, Antibacterial
4',5-Dihydroxyflavone
Cat.No: T8260
Synonym:
Target: Lipoxygenase, Glucosidase
Chebulagic acid
Cat.No: TQ0180
Synonym:
Target: SARS-CoV, Influenza Virus, Lipoxygenase, COX
3-Hydroxycoumarin
Cat.No: T8002
Synonym:
Target: Lipoxygenase
Caffeic Acid
Cat.No: T2807
Synonym:
Target: Lipoxygenase, Endogenous Metabolite, TRP/TRPV Channel
Aureusidin
Cat.No: TN5634
Synonym: Auresudidin,金鱼草素,Auresidin
Target: Antioxidant, Reactive Oxygen Species, Lipoxygenase
Phenethyl ferulate
Cat.No: TN2330
Synonym: Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯
Target: Lipoxygenase, COX
S-(+)-Marmesin
Cat.No: T5759
Synonym: (+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin
Target: Lipoxygenase, COX
5-O-Demethylnobiletin
Cat.No: T5714
Synonym: 5-DEMETHYLNOBILETIN,去甲基川陈皮素
Target: Leukotriene Receptor, Lipoxygenase
Xanthatin
Cat.No: T3S0153
Synonym: 苍耳亭,叶黄制菌素
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
Nordihydroguaiaretic acid
Cat.No: TJS2190
Synonym: 去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid
Target: Antioxidant, Ferroptosis, Lipoxygenase, Autophagy
β-Boswellic acid
Cat.No: TN1097
Synonym: Beta-boswellic acid,β-乳香酸
Target: Lipoxygenase, DNA/RNA Synthesis
3-O-Acetyl-11-hydroxy-beta-boswellic acid
Cat.No: TN1255
Synonym:
Target: Lipoxygenase
Wedelolactone
Cat.No: T3384
Synonym: 蟛蜞菊内酯,IKK Inhibitor II
Target: Apoptosis, NF-κB, Lipoxygenase, Caspase
11-​Keto-​beta-​boswellic acid
Cat.No: TN1182
Synonym: 11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸
Target: Leukotriene Receptor, NF-κB, Lipoxygenase
Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Danofloxacin mesylate
Cat.No: T1276
Synonym: 甲磺酸达氟沙星,CP 76136-27
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Podofilox
Cat.No: T1121
Synonym: 鬼臼毒素,Podophyllotoxin,(+)-Shikonin
Target: Microtubule Associated, Topoisomerase
8-Geranyloxypsoralen
Cat.No: TN1343
Synonym: 8-香叶草氧基补骨脂素
Target: Anti-infection, P450, BACE
Benzoyloxypaeoniflorin
Cat.No: T4S1658
Synonym: 苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷
Target: NF-κB, Tyrosinase
7-Prenyloxycoumarin
Cat.No: T5744
Synonym: 7-(异戊烯基氧基)香豆素,Nsc267697,7-O-Prenylumbelliferone,7-异戊烯氧基香豆素
Target: Antifungal
Raloxifene hydrochloride
Cat.No: T1549
Synonym: LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
3,29-O-Dibenzoyloxykarounidiol
Cat.No: TN1025
Synonym:
Target: Others
Tosufloxacin tosylate hydrate
Cat.No: T8046
Synonym: Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate
Target: Others, Antibacterial, Antibiotic
Norfloxacin
Cat.No: T1306
Synonym: 氟哌酸,MK-0366,诺氟沙星
Target: DNA gyrase, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic
14beta-Benzoyloxy-2-deacetylbaccatin VI
Cat.No: TN2627
Synonym:
Target: Others
(3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone
Cat.No: T83558
Synonym:
Target:
(Z)-2-Angeloyloxymethyl-2-butenoic
Cat.No: T83516
Synonym:
Target:
3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione
Cat.No: T38658
Synonym:
Target:
3-Hydroxy-3-acetonyloxindole
Cat.No: TN2938
Synonym:
Target: Others
Ethyl 4-(rhamnosyloxy)benzylcarbamate
Cat.No: TN5683
Synonym:
Target:
8-Hydroxy-9,10-diisobutyryloxythymol
Cat.No: TN5862
Synonym:
Target:
8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide
Cat.No: TN3302
Synonym:
Target: Others
3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid
Cat.No: TN5613
Synonym: ent-3β-Cinnamoyloxy-9α,17-dihydroxykaur-15-en-19-oic acid
Target:
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C
Cat.No: TN3301
Synonym:
Target: Others
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
Cat.No: TN3294
Synonym:
Target: NADPH-oxidase, P450, MAO
8-Hydroxy-9-isobutyryloxy-10-(2-methylbutanoyl)thymol
Cat.No: T83233
Synonym:
Target:
2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester
Cat.No: T38657
Synonym:
Target:
14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide
Cat.No: TN5303
Synonym:
Target:
7α-Galloyloxysweroside
Cat.No: TN5555
Synonym:
Target:
3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid
Cat.No: TN6331
Synonym:
Target:
Dehydroperilloxin
Cat.No: TN3810
Synonym:
Target: COX
7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin
Cat.No: TN6207
Synonym:
Target:
8alpha-(2-Methylacryloyloxy)hirsutinolide
Cat.No: TN3295
Synonym:
Target: Others
4-Prenyloxyresveratrol
Cat.No: TMA2415
Synonym: 4-异戊烯基氧基白藜芦醇,4'-Prenyloxyresveratrol
Target: Others
8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide
Cat.No: TN3299
Synonym:
Target: Others
8-(3-Ethoxy-2-hydroxy-3-methylbutyloxy)psoralen
Cat.No: T40636
Synonym:
Target:
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