9
365
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1380 |
Alodan
Cyclodan,Nodon,冰片丹,Chlorbicyclen |
Others | Others |
Alodan (Nodon) 是一种有机氯化物杀虫剂。 | |||
T72024 |
ZIM
|
||
ZIM,一种从4-Aminoantipyrine衍生的降冰片烯,有效诱导DNA损伤,造成基因组及染色体损害,进而引发细胞死亡和激活吞噬。其化疗潜力适用于癌症研究。 | |||
T36898 |
Sandacanol
Sandranol,2-Ethyl-4-(2,2,3-trimethylcyclopent-3-en-yl)-but-2-en-1-ol |
Apoptosis | Apoptosis |
Sandacanol(Sandranol) 是一种选择性嗅觉受体(OR10H1)激动剂。Sandacanol可诱导膀胱癌细胞的细胞周期停止和部分凋亡,可降低细胞迁移率和增殖率。 | |||
T27563 |
Hydroxypropyl-beta-cyclodextrin
HP-beta-CyD,VTS-270,HP-beta-CD,Hydroxypropyl-beta-cyclodextri,THPB,HPbCD |
||
Hydroxypropyl-beta-cyclodextrin, also known as Hydroxypropyl-beta-cyclodextrin; THPB; HP-beta-CD; HPbCD; HP-beta-CyD; VTS-270; HPbetaCD; HPbetaCyD, is a drug candidate potentially for the treatment of Niemann-Pick type C diseases. In April 2009, hydroxypr | |||
T37680 |
3-hydroxy Palmitic Acid methyl ester
|
||
3-hydroxy Palmitic acid methyl ester (3-hydroxy PAME) is an esterized long-chain fatty acid involved in quorum sensing in R. solanacearum, a bacteria that causes lethal wilting in plants. 3-hydroxy-PAME (175 nM) increases levels of PhcA-regulated virulence factors, greater than 20-, 30-, and 25-fold for EPS I, EGL, and PME, respectively, in the AW1-83 strain of R. solanacearum. | |||
T37555 |
Cardanol triene
|
||
Cardanol triene is a phenol found in cashew nut shell liquid that reversibly inhibits tyrosinase with an IC50 value of 40.5 μM in vitro. A mixture of cardanol mono-, di-, and triene is used to synthesize cardanol-metal complexes that inhibit uropathogenic E. coli biofilm formation. | |||
T24776 |
Secologanate
Secologanic Acid |
||
Secologanate is an inhibitor of plant growth. | |||
T21096 |
Decamethylene glycol
alpha,omega-Decanediol,Decamethylenediol,1,10-Dihydroxydecane,Decane-1,10-diol |
||
Decamethylene glycol is a substance used as a reagent in the biological study of modified oligonucleotide with in vivo antitumoral activity. Also used in the pharmaceutical study on the composition of essential oils obtained from myrrh and frankincense an | |||
T32269 |
Jasmone, (E)-
EINECS 228-410-7 |
||
Jasmone, (E)- is a type of perfuming agent. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3741 |
(-)-borneol
L-Borneol,冰片 |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
(-)-borneol (L-Borneol) 对 GABA 受体具有高效的正向调节作用,EC50 为 237 μM。 | |||
T5734 |
(+)-BORNEOL
d-Borneol,(+)-冰片 |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
(+)-BORNEOL (d-Borneol) 是一种天然的双环单萜,在中药中用于镇痛和麻醉;增强 GABA 受体活性,EC50 为 248 μM。 | |||
T8283 |
(+)-Bornyl Acetate
Bornyl acetate,1-乙酸冰片酯,(+)-乙酸龙脑酯 |
Others | Others |
(+)-Bornyl Acetate 存在于 Pichtae 精油 (西伯利亚冷杉针油) 中。它能够显著抑制拟南芥幼苗根系生长。 | |||
T7983 |
Isoborneol
DL-Isoborneol,异冰片,异龙脑 |
HSV | Microbiology/Virology |
Isoborneol (DL-Isoborneol) 是存在于许多药用植物精油中的一种单萜醇,具有抗氧化和抗病毒特性,是 1 型单纯疱疹病毒(HSV-1)的有效抑制剂。 | |||
TN1448 |
(-)-Bornyl acetate
L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯 |
p38 MAPK; NF-κB; JNK; Antifungal | MAPK; Microbiology/Virology; NF-κB |
(-)-Bornyl acetate (L-(-)-Bornyl acetate) 是存在于牛膝草油中的一种具有抗真菌活性的 (+)-Bornyl acetate 低活性异构体。 | |||
T1246 |
Bornyl acetate
乙酸冰片酯,Bornyl acetic ether,2-Camphanol acetate,乙酸龙脑酯,Isobornyl acetate |
Apoptosis; IL Receptor | Apoptosis; Immunology/Inflammation |
Bornyl acetate (Isobornyl acetate) 是一种强效的芳香剂,是功效最强大的风味稀释因子之一,具有抗肿瘤活性。 | |||
TN2364 |
Sudan IV
苏丹红Ⅳ,Solvent Red 24,C.I. 26105 |
Others | Others |
Sudan IV (Solvent Red 24) 是脂溶性重氮染料,可用于冰冻或石蜡切片上,能够将脂类、甘油三酯和脂蛋白染色。 | |||
T2981 |
Xanthoxylin
Brevifolin,Xanthoxyline,花椒素,2'-Hydroxy-4',6'-dimethoxyacetophenone |
Others; Antifungal | Microbiology/Virology; Others |
Xanthoxylin (Brevifolin)e 是从Zanthoxylum simulans 中分离出来的是一种冰片和樟脑味化合物,有抗真菌和抗癫痫作用。 | |||
TN2058 |
Persicogenin
|
Anti-infection | Microbiology/Virology |
Persicogenin 是分离自 Rhus retinorrhoea 中,具有抗癌作用。 | |||
T4S1114 |
Dryocrassin ABBA
东北贯众素,Dryocrassin |
Influenza Virus; Antibacterial | Microbiology/Virology |
Dryocrassin ABBA (Dryocrassin) 是一种从苦参中提取的黄酮类天然产物,具有抗病毒和抗菌活性。它抑制树突状细胞的免疫刺激功能,延长同种异体皮肤移植成活率。 | |||
T2900 |
Paeonol
丹皮酚,Peonol |
MAO; Autophagy; Monoamine Oxidase | Autophagy; Metabolism; Neuroscience |
Paeonol (Peonol) 是一种从牡丹中提取的活性物质,可抑制 MAO-A 和 MAO-B,IC50 分别为 54.6 μM 和 42.5 μM。 | |||
TN6945 |
Lactic acid
2-hydroxypropanoic acid |
Others | Others |
Lactic acid (2-hydroxypropanoic acid) 是糖酵解的产物,广泛存在与自然界中。Lactate acid 在体内收缩骨骼肌缺氧时会产生,可在完全有氧条件下被去除。Lactic acid 可作为危重病人的血流动力学指标。Lactic acid 具有抗肿瘤活性。 | |||
T5687 |
WITHAFERIN A
醉茄素 A,醉茄素A |
Ferroptosis; NF-κB | Apoptosis; NF-κB |
Withaferin A 是从南非醉茄中分离到的一种甾体内酯,是内皮蛋白 C 受体脱落抑制剂,可以抑制NF-kB 的活性,具有抗炎,抗肿瘤等作用。它是一种新型 NFkappaB 抑制剂,有望成为治疗各种炎症性疾病和癌症的新型抗炎药。 | |||
T4S0998 |
Trifolirhizin
红车轴草根甙/三叶豆紫檀苷,三叶豆紫檀苷 |
TNF; Tyrosinase | Apoptosis; Proteases/Proteasome |
Trifolirhizin 是一种从苦参根中分离出的 pterocarpan 黄酮类化合物。它具有酪氨酸酶高抑制活性,IC50=506 μM。它具有抗炎和抗癌的潜能。 | |||
T1664 |
Meglutol
Dicrotalic acid,3-Hydroxy-3-methylglutaric acid,美格鲁托 |
Endogenous Metabolite; HMG-CoA Reductase; Autophagy | Autophagy; Metabolism |
Meglutol (3-Hydroxy-3-methylglutaric acid) 是一种抗血脂剂,可降低胆固醇、甘油三酯、血清 β-脂蛋白和磷脂。它抑制胆固醇生物合成中的限速酶羟甲基戊二酰辅酶 A 还原酶的活性。 | |||
T3233 |
Sophoricoside
Genistein sophoricoside,槐苷 |
Others | Others |
Sophoricoside (Genistein sophoricoside) 是一种异黄酮糖苷,从槐花中分离得到,具有抗炎,抗癌和免疫抑制作活性。 | |||
T2P2923 |
Stearic acid
硬脂酸,Isostearic acid,Octadecanoic acid,Cetylacetic acid |
Phosphatase; Endogenous Metabolite | Metabolism |
Stearic acid (Cetylacetic acid) 是长链饱和脂肪酸,存在于许多动植物油脂中。 | |||
T3738 |
3-(4-Hydroxyphenyl)-1-propanol
|
LTR | Immunology/Inflammation |
3-(4-Hydroxyphenyl)-1-propanol 能够用于合成 (-)-centrolobine。 | |||
T2786 |
Oxysophocarpine
氧化槐树碱,氧卡地平 |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Oxysophocarpine 是提取自海藻的生物碱。它抑制口腔鳞状细胞癌的生长和转移。它对中枢神经系统和周围神经系统具有神经保护作用和抗伤害感受作用。 | |||
T3321 |
Oleanonic acid
3-Oxooleanolic acid,3-Oxoolean-12-en-28-oic Acid,Oleanonic Acid,齐墩果酮酸,3-Ketooleanolic Acid |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Oleanonic acid (3-Ketooleanolic Acid) 是一种三萜,可以抑制 HIV-1 对细胞的感染。它具有保肝作用,并具有抗肿瘤和抗病毒特性。 | |||
TN6709 |
6,7-DIMETHOXY-3,4-DIHYDRO-2H-ISOQUINOLIN
|
Others | Others |
6,7-DIMETHOXY-3,4-DIHYDRO-2H-ISOQUINOLIN 是一种从毛豆中分离出来的天然产物。 | |||
T8165 |
Erythrodiol
|
Endogenous Metabolite; ABC | Membrane transporter/Ion channel; Metabolism |
Erythrodiol 是一种橄榄油的成分,能够选择性抑制ABCA1蛋白的降解来促进胆固醇外流,有用于动脉粥样硬化的研究潜力。 | |||
TN3522 |
Blumeatin B
|
Xanthine Oxidase | Metabolism |
Blumeatin shows XO inhibitory activity. | |||
TN5944 |
Hedragonic acid
24-Nor-3-oxoolean-12-en-28-oic acid |
||
Hedragonic acid is a natural product from Dryobalanops aromatica. | |||
TN3867 |
Dihydrotamarixetin
|
Others | Others |
Dihydrotamarixetin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3867,CAS号为 70411-27-7。 | |||
T6S1768 |
Narcissin
水仙苷,Isorhamnetin 3-Rutinoside,Narcissoside |
Antioxidant | oxidation-reduction |
Narcissin (Isorhamnetin 3-Rutinoside) 是一种黄连糖苷,能够清除 ONOO-(IC50:3.5 μM)和 SIN-1 衍生的 ONOO-(IC50:9.6 μM),具有抗氧化作用。 | |||
T5716 |
4'-Methoxyresveratrol
白藜芦醇-4'-甲醚,4'-O-Methylresveratrol |
advanced glycation end products | Others |
4'-Methoxyresveratrol (4'-O-Methylresveratrol) 是一种多酚类化合物,来源于双翅目植物中,具有抗雄激素、抗真菌和抗炎症作用。它能抑制 RAGE- 介导的 MAPK/NF-κB 信号通路,并激活 NLRP3 炎性体,从而缓解 AGE- 诱导的炎症。 | |||
T0966 |
Sennoside A
番泻苷A,NSC 112929,番泻苷 A |
MAO; HIV Protease | Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Sennoside A (NSC-112929) 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷,抑制 HIV-1 复制。 | |||
T2734 |
Sennoside B
番泻苷 B,番泻苷B |
PDGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
Sennoside B 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷。它可通过与 PDGF-BB 及其受体结合并下调 PDGFR-β 信号传导途径来抑制 PDGF 刺激的细胞增殖。 | |||
TN1722 |
Hamamelitannin
|
Antifection | Microbiology/Virology |
Hamamelitannin 是分离自 Hamamelis virginiana 树皮的一种多酚,是群体感应抑制剂。它通过影响肽聚糖生物合成和 eDNA 释放增加金黄色葡萄球菌生物膜的抗生素敏感性。 | |||
T3776 |
Rhapontigenin
丹叶大黄素,Protigenin |
P450; Antibacterial; Antifungal | Metabolism; Microbiology/Virology |
Rhapontigenin (Protigenin) 是一种基于机制的选择性细胞色素 P450 1A1 (IC50: 400 nM) 灭活剂。它是一种芳烃羟化酶,可激活作为致癌物质的多环芳烃。它是白藜芦醇的天然类似物,具有抗癌,抗氧化剂,抗真菌和抗菌活性。 | |||
T1558 |
Resveratrol
白藜芦醇,trans-Resveratrol,SRT 501 |
Apoptosis; Mitophagy; IκB/IKK; Lipoxygenase; Sirtuin; COX; NADPH; DNA/RNA Synthesis; Nrf2; Antibacterial; Antibiotic; Autophagy; Antifungal | Apoptosis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB |
Resveratrol (SRT 501) 属于多酚类天然产物,是一种植物抗毒素,具有抗氧化和化学预防活性。Resveratrol 的靶点广泛,包括 COX、SIRT、LOC 等。Resveratrol 可以诱导细胞自噬和凋亡。 | |||
TN2437 |
Serotonin
5-羟基色胺,5-hydroxytryptamine,血清素,五羟色胺,5-HT |
Others; 5-HT Receptor; Endogenous Metabolite; Transferase | GPCR/G Protein; Metabolism; Neuroscience; Others |
Serotonin (5-hydroxytryptamine) 是 CNS 中的单胺神经递质和内源性5-HT 受体激动剂。它也是儿茶酚 O-甲基转移酶(COMT) 的抑制剂,Ki 值为 44 μM。 | |||
TN2277 |
Torachrysone-8-O-b-D-glucoside
芦荟大黄素 8-葡萄糖甙,Torachrysone 8-O-glucoside |
Antifection | Microbiology/Virology |
Torachrysone-8-O-b-D-glucoside 可从 Polygonum multiflorum 分离得到。它对 DPCs(真皮乳头细胞)的增殖具有促进作用。 | |||
T1273 |
Diacerein
双醋瑞因,Diacerhein,Fisiodar,Diacetylrhein |
IL Receptor; Interleukin | Immunology/Inflammation |
Diacerein (Fisiodar) 是一种慢效具有白介素-1β 抑制效果的蒽醌类化合物。 | |||
TN3875 |
Dipterocarpol
|
P450; AChR | Metabolism; Neuroscience |
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng. Dipterocarpol A shows moderate acetylcholinesterase inhibitory activity with the IC50 value of 8.28 uM. | |||
T2S0967 |
Sennoside C
|
Others | Others |
Sennoside C 是从番泻叶和豆荚中提取的蒽醌甙,对小鼠的通便作用有辅助作用。 | |||
T0877 |
Gallic acid
3,4,5-Trihydroxybenzoic acid,Gallate,没食子酸,Benzoic acid |
Apoptosis; Ferroptosis; Reactive Oxygen Species; ROS; COX; Endogenous Metabolite | Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
Gallic acid (Benzoic acid) 是一种天然多羟基酚类化合物,具有抑制环氧合酶-2 的自由基清除作用,还具有抗菌、抗氧化、抗菌、抗炎和抗肿瘤活性。 | |||
T2S0968 |
Sennoside D
|
Others | Others |
Sennoside D 是一种从番泻 Cassia angustifolia 的叶子和豆荚中提取的蒽醌苷。 | |||
TN1052 |
Lindleyin
|
Estrogen Receptor/ERR; Estrogen/progestogen Receptor | Endocrinology/Hormones |
Lindleyin 是从 Rhei rhizoma 中分离得到,通过雌激素受体介导激素作用。它能够与 ERα结合,有类似雌激素的作用。 | |||
T0610 |
Piceatannol
白皮杉醇,trans-Piceatannol,Astringenin |
Apoptosis; Serine/threonin kinase; PKA; Syk; PKC; Autophagy | Angiogenesis; Apoptosis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Tyrosine Kinase/Adaptors |
Piceatannol (Astringenin) 是一种Syk 抑制剂,可降低由 TNF 诱导的 iNOS 表达,可研究急性肺损伤。它是存在于各种水果和蔬菜中天然存在的多酚二苯乙烯,可诱导细胞自噬和凋亡,具有抗癌和抗炎特性。 | |||
T2177 |
Kaempferol
Kempferol,山柰酚,山奈酚,Robigenin |
Apoptosis; Estrogen Receptor/ERR; Mitophagy; Estrogen/progestogen Receptor; HIV Protease; Endogenous Metabolite; Parasite; Autophagy | Apoptosis; Autophagy; Endocrinology/Hormones; Metabolism; Microbiology/Virology; Proteases/Proteasome |
Kaempferol (Robigenin) 属于天然类黄酮,是一种 ERRα 和 ERRγ 的反向激动剂。Kaempferol 具有抗肿瘤、抗炎、抗氧化、抗菌和抗病毒等多种活性。 | |||
TN6774 |
Emodin 6-O-β-D-glucoside
大黄素-6-O-β-D-葡萄糖苷,Glucoemodin |
Others | Others |
Emodin 6-O-β-D-glucoside (Glucoemodin) 是一种从 Reynoutria japonica 中提取的活性化合物。它具有显著的抗炎和屏障保护活性,可用于研究动脉粥样硬化及糖尿病并发症。 | |||
TQ0205 |
Procyanidin B1
原花青素B1,原花青素 B1 |
TLR | Immunology/Inflammation |
Procyanidin B1 是水果中常见的多酚类黄酮,能够与TLR4/MD-2复合体结合,具有抗炎活性。 | |||
TMA1403 |
Cyclo(Ile-Ala)
|
Others | Others |
Cyclo(Ile-Ala) 是存在于海洋放线菌11014 I.中的天然产物。 | |||
T6S1587 |
Notoginsenoside R2
三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2 |
Others; Nrf2 | Immunology/Inflammation; Others |
Notoginsenoside R2 (20(S)-Notoginsenoside R2) 是一种新分离三七皂苷,表现出对6-OHDA 诱导的氧化应激及细胞凋亡的保护作用。 | |||
T6S1367 |
Procyanidin B2
原花青素 B2,Proanthocyanidin B2 |
Reactive Oxygen Species; NOD | Immunology/Inflammation; Metabolism; NF-κB |
Procyanidin B2 (Proanthocyanidin B2) 是天然黄酮类物质,具有抗肿瘤,抗氧化等活性。 | |||
TN1017 |
Physion 8-O-β-D-glucoside
大黄素甲醚-8-o-β-D-葡萄糖苷,Physcion 1-O-beta-D-glucoside |
Others | Others |
Physion 8-O-β-D-glucoside 是一种 Fallopia multiflora 的活性成分,可用于头晕的研究。 | |||
T3S0381 |
Chrysophanol 8-O-glucoside
|
Serine Protease | Proteases/Proteasome |
Chrysophanol 8-O-glucoside 来自Rumex acetosa 根部,具有中等的弹性蛋白酶抑制特性。它具有温和的细胞毒性和抗糖尿病特性,能够在胰岛素刺激的葡萄糖转运途径中发挥代谢作用。 | |||
T4S0795 |
Berberrubine chloride
9-Berberoline Chloride,Beroline,Beroline Chloride,小檗红碱,Berberrubine,9-Berberoline |
IL Receptor | Immunology/Inflammation |
Berberrubine chloride (9-Berberoline Chloride) 是一种黄连素的有效代谢物,能够改善动物模型中溃疡性结肠炎的症状。 | |||
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