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Targets Recommended: HCV Protease SARS-CoV

56

抑制剂 & 化合物

49

天然产物

10

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T9331 Bemnifosbuvir hemisulfate

AT-527

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Bemnifosbuvir hemisulfate (AT-527) 是一种 HCV 病毒复制抑制剂。
T67812 Tenifatecan

SN2310

Tenifatecan (SN2310) 是一种高度亲脂性的7-乙基-10-羟基喜树碱(SN)制剂,具有潜在的抗肿瘤活性。
T1146 Nifedipine

BAY-a-1040,Procardia XL,Procardia,硝苯地平,Adalat

CaMK; Potassium Channel; Calcium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
Nifedipine (Procardia) 是一种二氢吡啶类钙通道阻滞剂,可抑制细胞外钙离子跨膜流入心肌和血管平滑肌细胞,导致主要冠状动脉和全身动脉扩张,降低心肌收缩力。它常用于心肌功能不全的相关研究。
T2514 Linifanib

利尼伐尼,ABT-869,RG3635,AL-39324

Apoptosis; c-Fms; VEGFR; FLT; CSF-1R; PDGFR; c-Kit; Autophagy Angiogenesis; Apoptosis; Autophagy; Tyrosine Kinase/Adaptors
Linifanib (AL-39324) 是一种高效口服的VEGFR 和PDGFR 家族多靶点抑制剂,具有显著的抗肿瘤活性。它对无关 RTKs、可溶性酪氨酸激酶或丝氨酸/苏氨酸激酶的活性要低得多。它是特异性 miR-10b 抑制剂,阻断miR-10b 的生物合成。
T2712 Nifekalant hydrochloride

Potassium Channel Membrane transporter/Ion channel
Nifekalant hydrochloride 是一种 IKr 钾通道阻滞剂,IC50为10 µM,属于 III 类抗心律不齐化合物,可用于快速室上性心律失常的研究。
T15271 Denifanstat

FASN-IN-2,TVB2640,TVB-2640

Fatty Acid Synthase Metabolism
Denifanstat (FASN-IN-2) 是一种口服具有活性的选择性 FASN 抑制剂,IC50=0.052 μM,EC50=0.072 μM。它有用于脂肪肝和癌症的研究潜力。
T8663 nifenalol.HCl

INPEA,1-(4-硝基苯基)-1-羟基-2-异丙基氨基乙烷盐酸盐

Adrenergic Receptor GPCR/G Protein; Neuroscience
Nifenalol.HCl(INPEA) 是β-肾上腺素能受体的拮抗剂。
T9341 Bemnifosbuvir

AT-511

Others; HCV Protease; SARS-CoV Microbiology/Virology; Others; Proteases/Proteasome
Bemnifosbuvir (AT-511) 是一种口服活性抑制剂,抑制 HCV 病毒复制,具有全基因型抗病毒活性。它有效抑制 SARS-CoV-2 (COVID-19)感染 (EC90=0.47 μM)。
T4503 Talniflumate

Somalgen,他尼氟酯

Chloride channel; COX; N-Acetylglucosaminyltransferase; Anion Exchanger Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Talniflumate (Somalgen) 是一种钙激活氯离子通道 (hCLCA1/mCLCA3) 阻滞剂,可减少动物模型和细胞培养中的粘蛋白合成和释放。它通过抑制环氧合酶,并抑制 Cl-/HCO3- 交换活性,具有抗炎作用。它还增加了远端肠梗阻综合征囊性纤维化小鼠模型的存活率。
T0693 Niflumic acid

氟尼酸,Nifluril,Forenol,Landruma

Others; Phospholipase; Chloride channel; COX; Monocarboxylate transporter; UGT Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Niflumic acid (Nifluril) 是钙离子激活的氯离子通道阻断剂,用于治疗类风湿性关节炎的镇痛剂和抗炎剂。
T5325 Nifurtimox

硝呋替莫,BAY-2502,BAY-A-2502

Dehydrogenase; Parasite Metabolism; Microbiology/Virology
Nifurtimox (BAY-A-2502) 是一种用于锥虫病的抗虫剂,可影响乳酸脱氢酶活性。它有潜力研究神经母细胞瘤细胞。
T19636 Morniflumate

马尼氟酯,Niflam,UP 164,UP-164,Morniflu,UP164

Others Others
Morniflumate (Niflam) 是一种非甾体抗炎药。它用于治疗炎症。
T0980 Nifenazone

尼芬那宗,Niapyrin,Nicodone,烟酰氨基比林,Nicazane

COX Immunology/Inflammation; Neuroscience
Nifenazone (Nicodone) 是吡唑类试剂,可用于研究各种风湿性疾病。
T77432 Anifrolumab

MDX-1333,MEDI-546

IFNAR Immunology/Inflammation
Anifrolumab(MEDI-546) 是一种有效的 I 型干扰素 (IFN) 受体拮抗剂,是一种靶向 IFN 的人源单克隆抗体。Anifrolumab 能抑制 I 型干扰素的活性,可用于预防和治疗系统性红斑狼疮 (SLE) 。
T36665 Dehydro Nifedipine

BAY-b 4759

Dehydro Nifedipine (BAY-b 4759) 是人血浆中硝苯地平的主要代谢物。Dehydro Nifedipine 抑制PC-12细胞葡萄糖摄取,IC50值为130 μM,硝苯地平是一种钙通道阻滞剂,用于治疗高血压和心绞痛。当硝苯地平被细胞色素P450 (CYP)异构体CYP3A4和CYP3A5代谢时形成脱氢硝苯地平。
T1563 Nifuroxazide

Diarlidan,硝呋齐特,Nifuroxazid,Dicoferin,硝呋酚酰肼

Antibacterial; Antibiotic; STAT JAK/STAT signaling; Microbiology/Virology; Stem Cells
Nifuroxazide (Diarlidan) 是STAT3抑制剂,具有抗转移和抗癌活性。
T7395 Lanifibranor

IVA337

PPAR DNA Damage/DNA Repair; Metabolism
Lanifibranor (IVA337) 是泛过氧化物酶体增殖物激活受体 (PPAR) 激动剂,对人类PPARα,PPARσ和PPARγ的EC50值分别为 1.5, 0.87 和 0.21 μM。
T6114 Nifursol

硝呋索尔,尼呋索尔

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Nifursol 是一种具有口服活性的兽用抗生素,用于预防组织口炎。它快速代谢形成代谢标记物 3,5-二硝基水杨酸环肼,并能持续很长时间。它可研究沙门氏菌感染的家禽、家禽和水生动物的大肠杆菌肠胃病。
T1526 Nifuratel

NF 113,SAP 113,硝呋太尔,Methylmercadone

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Nifuratel (SAP 113) 是广谱抗生素,有抗细菌、真菌和毛滴虫活性。
T7599 Sunifiram

桑尼菲拉姆,DM-235,桑尼非拉姆

iGluR Membrane transporter/Ion channel; Neuroscience
Sunifiram (DM-235) 是一种 ampakine 样促智剂。
T12223 Nifursemizone

NF161,5-Nitro-2-furancarbaldehyde 2-ethyl semicarbazone,硝呋米腙,Etafurazone

Antibiotic Microbiology/Virology
Nifursemizone (Etafurazone) 是抗原虫药。
T38192 Unifiram

Others Others
Unifiram 是一种认知增强剂。 Unifiram 诱导大鼠海马 CA1 区场兴奋性突触后电位 (fEPSP) 幅度的持久增加 (EC50= 27 nM) 并增加大鼠大脑皮层中乙酰胆碱 (ACh) 的释放。
T73198 Nifuroxime

Nifuroxime 是一种抗感染剂,可用于真菌感染相关的研究。
T73284 Vonifimod

Vonifimod 是一种免疫调节剂。
T26819 Binifibrate

WAC104,WAC 104,Antopal,WAC-104,Biniwas

Binifibrate is a hyperlipemiant drug used for the treatment of hyperlipidemia.
T125992 threo-Guaiacylglycerol β-dihydroconiferyl ether

threo-Guaiacylglycerol β-dihydroconiferyl ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125992。
T125621 erythro-Guaiacylglycerol β-coniferyl ether

erythro-Guaiacylglycerol β-coniferyl ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125621。
T35584 Hydroxydehydro Nifedipine Carboxylate

Hydroxydehydro nifedipine carboxylate is a metabolite of nifedipine .1 1.Roosemalen, M.C.M., Soons, P.A., Funaki, T., et al.High-performance liquid chromatographic determination of the polar metabolites of nifedipine in plasma, blood and urineJ. Chromatogr.565(1-2)516-522(1991)
TP2394 Nifalatide

Nifalatide is a analog of enkephalin.
T124473 threo-Guaiacylglycerol-beta-coniferyl aldehyde ether

threo-Guaiacylglycerol-beta-coniferyl aldehyde ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124473。
T68828 Chinifur

Chinifur is a selective inhibitor and subversive substrate" for Trypanosoma congolense trypanothione reductase"
T28610 Ronifibrate

Ronifibrate is a lipid modifying agent with antihyperlipidemic and antiarteriosclerotic activity.
T126480 (7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-xyloside

(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-xyloside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126480。
T22515 5'-Iodoresiniferatoxin

Others Others
TRPV1 (VR1) receptor antagonist
T74065 Nifurpirinol

Nifurpirinol (P-7138),一种硝基芳香型抗生素(antibiotic),作为细菌硝基还原酶(NTR)的底物。相较于甲硝唑,其作为一种prodrug,在表达硝基还原酶的转基因模型中引发细胞消融的效能更高。
T12222 Nifedipine-d6

硝苯地平 D6,Nifedipine D6,BAY-a-1040 D6

Others Others
Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.
T32766 Linifolin A

NSC 153859,NSC-153859,NSC153859,PF 57,PF-57

Linifolin A is a sesquiterpene lactone extracted from Helenium aromaticum.
T22527 6'-Iodoresiniferatoxin

Others Others
TRPV1 (VR1) vanilloid receptor partial agonist
T69021 Nifedipine HCl

Nifedipine HCl is a potent vasodilator agent with calcium antagonistic action. It is a useful anti-anginal agent that also lowers blood pressure.
T125568 Dihydroconiferin

Dihydroconiferin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125568,CAS号为 17609-06-2。
T33669 Nifurpipone

Rec-150122,Rec 150122,Rec150122

Nifurpipone is a biochemical existed in urine.
T33667 Nifrofam

Nifrofam is a fluorescent probe for imaging α4β2* nAChRs.
T71293 Nifuroxazide-d4

Nifuroxazide-d4 is intended for use as an internal standard for the quantification of nifuroxazide by GC- or LC-MS. Nifuroxazide is a nitrofuran antibiotic. It is active against strains of the enteropathogenic bacteria C. jejuni, Salmonella, Y. enterocolitica, Shigella, and E. coli. It inhibits quorum sensing and virulence factor production in P. aeruginosa. Nifuroxazide inhibits STAT3 activity in a reporter assay and decreases viability of U266 and INA-6 myeloma cells, which have constitutive S...
T124284 Erythro-Guaiacylglycerol-beta-coniferyl aldehyde ether

Erythro-Guaiacylglycerol-beta-coniferyl aldehyde ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124284。
T28171 Nifeviroc

TD-0232,TD 0232,尼非韦罗,TD0232

Nifeviroc, a CCR5 antagonist, is used potentially for treatment of inflammatory responses to HIV type-1 infection.
T11926 m-Nifedipine

Others Others
m-Nifedipine, an impurity of Nifedipine, serves as a potent calcium channel blocker and the preferred treatment option for cardiac insufficiencies.
T79836 Arbemnifosbuvir

SARS-CoV Microbiology/Virology
Arbemnifosbuvir 是用于干扰核病毒RdRp相关核苷酸基转移酶(NiRAN)非结构蛋白12(nsp12)的化合物,适用于SARS-CoVs感染的研究。
T126168 Pruniflorone R

Pruniflorone R 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126168。
T8663L Nifenalol

Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.
T25869 Nifurzide

Ricridene

Nifurzide is a nitrofuran derivative used as an intestinal antiinfectious agent. Low concentrations reduces growth rate while high concentrations completely inhibits growth.

化合物

Bemnifosbuvir hemisulfate
Cat.No: T9331
Synonym: AT-527
Target: HCV Protease, SARS-CoV
Tenifatecan
Cat.No: T67812
Synonym: SN2310
Target:
Nifedipine
Cat.No: T1146
Synonym: BAY-a-1040,Procardia XL,Procardia,硝苯地平,Adalat
Target: CaMK, Potassium Channel, Calcium Channel, Autophagy
Linifanib
Cat.No: T2514
Synonym: 利尼伐尼,ABT-869,RG3635,AL-39324
Target: Apoptosis, c-Fms, VEGFR, FLT, CSF-1R, PDGFR, c-Kit, Autophagy
Nifekalant hydrochloride
Cat.No: T2712
Synonym:
Target: Potassium Channel
Denifanstat
Cat.No: T15271
Synonym: FASN-IN-2,TVB2640,TVB-2640
Target: Fatty Acid Synthase
nifenalol.HCl
Cat.No: T8663
Synonym: INPEA,1-(4-硝基苯基)-1-羟基-2-异丙基氨基乙烷盐酸盐
Target: Adrenergic Receptor
Bemnifosbuvir
Cat.No: T9341
Synonym: AT-511
Target: Others, HCV Protease, SARS-CoV
Talniflumate
Cat.No: T4503
Synonym: Somalgen,他尼氟酯
Target: Chloride channel, COX, N-Acetylglucosaminyltransferase, Anion Exchanger
Niflumic acid
Cat.No: T0693
Synonym: 氟尼酸,Nifluril,Forenol,Landruma
Target: Others, Phospholipase, Chloride channel, COX, Monocarboxylate transporter, UGT
Nifurtimox
Cat.No: T5325
Synonym: 硝呋替莫,BAY-2502,BAY-A-2502
Target: Dehydrogenase, Parasite
Morniflumate
Cat.No: T19636
Synonym: 马尼氟酯,Niflam,UP 164,UP-164,Morniflu,UP164
Target: Others
Nifenazone
Cat.No: T0980
Synonym: 尼芬那宗,Niapyrin,Nicodone,烟酰氨基比林,Nicazane
Target: COX
Anifrolumab
Cat.No: T77432
Synonym: MDX-1333,MEDI-546
Target: IFNAR
Dehydro Nifedipine
Cat.No: T36665
Synonym: BAY-b 4759
Target:
Nifuroxazide
Cat.No: T1563
Synonym: Diarlidan,硝呋齐特,Nifuroxazid,Dicoferin,硝呋酚酰肼
Target: Antibacterial, Antibiotic, STAT
Lanifibranor
Cat.No: T7395
Synonym: IVA337
Target: PPAR
Nifursol
Cat.No: T6114
Synonym: 硝呋索尔,尼呋索尔
Target: Others, Antibacterial, Antibiotic
Nifuratel
Cat.No: T1526
Synonym: NF 113,SAP 113,硝呋太尔,Methylmercadone
Target: Antibacterial, Antibiotic, Parasite
Sunifiram
Cat.No: T7599
Synonym: 桑尼菲拉姆,DM-235,桑尼非拉姆
Target: iGluR
Nifursemizone
Cat.No: T12223
Synonym: NF161,5-Nitro-2-furancarbaldehyde 2-ethyl semicarbazone,硝呋米腙,Etafurazone
Target: Antibiotic
Unifiram
Cat.No: T38192
Synonym:
Target: Others
Nifuroxime
Cat.No: T73198
Synonym:
Target:
Vonifimod
Cat.No: T73284
Synonym:
Target:
Binifibrate
Cat.No: T26819
Synonym: WAC104,WAC 104,Antopal,WAC-104,Biniwas
Target:
threo-Guaiacylglycerol β-dihydroconiferyl ether
Cat.No: T125992
Synonym:
Target:
erythro-Guaiacylglycerol β-coniferyl ether
Cat.No: T125621
Synonym:
Target:
Hydroxydehydro Nifedipine Carboxylate
Cat.No: T35584
Synonym:
Target:
Nifalatide
Cat.No: TP2394
Synonym:
Target:
threo-Guaiacylglycerol-beta-coniferyl aldehyde ether
Cat.No: T124473
Synonym:
Target:
Chinifur
Cat.No: T68828
Synonym:
Target:
Ronifibrate
Cat.No: T28610
Synonym:
Target:
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-xyloside
Cat.No: T126480
Synonym:
Target:
5'-Iodoresiniferatoxin
Cat.No: T22515
Synonym:
Target: Others
Nifurpirinol
Cat.No: T74065
Synonym:
Target:
Nifedipine-d6
Cat.No: T12222
Synonym: 硝苯地平 D6,Nifedipine D6,BAY-a-1040 D6
Target: Others
Linifolin A
Cat.No: T32766
Synonym: NSC 153859,NSC-153859,NSC153859,PF 57,PF-57
Target:
6'-Iodoresiniferatoxin
Cat.No: T22527
Synonym:
Target: Others
Nifedipine HCl
Cat.No: T69021
Synonym:
Target:
Dihydroconiferin
Cat.No: T125568
Synonym:
Target:
Nifurpipone
Cat.No: T33669
Synonym: Rec-150122,Rec 150122,Rec150122
Target:
Nifrofam
Cat.No: T33667
Synonym:
Target:
Nifuroxazide-d4
Cat.No: T71293
Synonym:
Target:
Erythro-Guaiacylglycerol-beta-coniferyl aldehyde ether
Cat.No: T124284
Synonym:
Target:
Nifeviroc
Cat.No: T28171
Synonym: TD-0232,TD 0232,尼非韦罗,TD0232
Target:
m-Nifedipine
Cat.No: T11926
Synonym:
Target: Others
Arbemnifosbuvir
Cat.No: T79836
Synonym:
Target: SARS-CoV
Pruniflorone R
Cat.No: T126168
Synonym:
Target:
Nifenalol
Cat.No: T8663L
Synonym:
Target:
Nifurzide
Cat.No: T25869
Synonym: Ricridene
Target:
Cat. No. Product Name Target Signaling Pathways
T3S0012 coniferyl ferulate

P-gp; GST Membrane transporter/Ion channel; Neuroscience; oxidation-reduction
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。
T6S1652 Benzoylpaeoniflorin

COX Immunology/Inflammation; Neuroscience
Benzoylpaeoniflorin 是一种从白芍中提取的天然化合物,可以降低细胞凋亡,对冠心病具有潜在的研究价值。
T11218 ε-​Viniferin

epsilon-Viniferin,Epsilon-白藜芦醇脱氢二聚体

P450 Metabolism
ε-​Viniferin (epsilon-Viniferin) 提取自 Vitis vinifera,是 Resveratrol 的二聚体,能够抑制 CYP 家族,其 Ki=0.5~20 μM,具有抗氧化作用。
T2S1907 Coniferaldehyde

Ferulaldehyde,Ferulyl aldehyde,4-HYDROXY-3-METHOXYCINNAMALDEHYDE,松柏醛,Coniferyl aldehyde,松柏醛;4-羟基-3-甲氧基肉桂醛

Apoptosis; Antioxidant Apoptosis; oxidation-reduction
Coniferaldehyde (Ferulaldehyde) 是一种血红素加氧酶-1 的有效诱导剂,具有抗炎作用。在 RAW264.7 巨噬细胞中,它通过 PKCα/βII/Nrf-2/HO-1 依赖性途径来抑制 LPS 诱导的细胞凋亡。
TN3849 Dihydrodehydrodiconiferyl alcohol

TNF Apoptosis
Dihydrodehydrodiconiferyl alcohol 是 Liriodendron tulipifera 的甲醇提取物。
T4S1658 Benzoyloxypaeoniflorin

苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷

NF-κB; Tyrosinase NF-κB; Proteases/Proteasome
Benzoyloxypaeoniflorin (Benzoyloxypeoniflorin) 是一种酪氨酸酶抑制剂,分离于Paeonia suffruticosa 的根,对mushroom tyrosinase 的 IC50为 0.453 mM。它是一种NF-κB 抑制剂,它通过对血小板聚集和凝血的抑制作用,有助于改善血液循环。
T2230 Paeoniflorin

芍药苷,Peoniflorin

HSP; COX Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience
Paeoniflorin (Peoniflorin) 是从芍药根中提取的一种蒎烷单萜糖苷,具有抗癌作用、抗氧化应激、抗血小板聚集、血管扩张、降低血液粘度和抗炎活性等多种生物活性。它是一种热休克蛋白诱导剂,通过自噬途径保护 PC12 细胞免受 MPP+和酸性损伤。
TL0010 CONIFERYL ALCOHOL

松柏醇,Coniferol

Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology
Coniferyl alcohol (Coniferol) 是合成芪类和香豆素丁子香酚的中间体,有抗真菌功效。
TN1067 Galloylpaeoniflorin

6'-O-Galloyl paeoniflorin,没食子酰芍药苷

NF-κB; Androgen Receptor; ROS Endocrinology/Hormones; Immunology/Inflammation; NF-κB
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) 是 NF-κB 抑制剂,同时也是 DNA 裂解抑制剂。
TN3694 Coniferaldehyde

NOS; COX; Nrf2; PKC; Autophagy Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Neuroscience
Coniferaldehyde 能显着抑制酒球菌菌株的生长活力。 Coniferaldehyde 通过诱导血红素加氧酶 1 (HO-1) 发挥抗炎特性。
TN7097 Tetrahydrodehydrodiconiferyl alcohol

Others Others
Tetrahydrodehydrodiconiferyl alcohol 是一种天然产物。
T34295 Resiniferatoxin

RTX,[3H]resiniferatoxin,树脂毒素

IL Receptor Immunology/Inflammation
Resiniferatoxin ([3H]resiniferatoxin) 抑制 Th1 细胞因子的产生,有助于防御 T.spiralis 感染,并可用于免疫反应调节剂的研究。
TL0009 coniferin

Coniferoside,松柏苷,Abietin

Others; Antifungal Microbiology/Virology; Others
Coniferin (Abietin) 是一种松柏醇中的葡萄糖苷。它抑制真菌生长和黑化反应,具有 ATP 依赖性转运活性并具有抗氧化作用。
TN1174 Schinifoline

Apoptosis; cell cycle arrest Apoptosis; Cell Cycle/Checkpoint
Schinifoline 是从 Zanthoxylum schinifolium Sieb 中提取出来的一种喹啉酮衍生物,具有细胞毒性活性,可促进癌细胞放射敏感性,影响细胞循环周期和细胞凋亡。
T3773 Oxypaeoniflorin

氧化芍药苷,Oxypaeoniflora

Others Others
Oxypaeoniflorin (Oxypaeoniflora) 从 Paeoniae 中分离得到的单萜糖苷化合物,是一种抗氧化剂,是具有神经保护和抗炎作用。
TN1378 α-Viniferin

ALPHA-VINIFERIN,Alpha-葡萄素

P450; NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
α-Viniferin 也称为2-芳基苯并呋喃类黄酮,是前列腺素H2合成酶抑制剂。具有抗阿尔茨海默病、抗结核、抗肿瘤、抗炎、抗糖尿病等多种药理活性
TN1578 Dihydroconiferyl alcohol

Others Others
Dihydroconiferyl alcohol exhibits cytoprotective activity in cultured MCF-7 cells stressed by H2O2.
TN2844 (2R,3S)-Dihydrodehydroconiferyl alcohol

MAPK; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK
(2R,3S)-Dihydrodehydroconiferyl alcohol can induce neurite outgrowth and enhance NGF-induced neurite outgrowth from PC12 cells by amplifying up-stream steps such as MAPK and PKC.
TN2034 Paeoniflorigenone

Others; Caspase Apoptosis; Others; Proteases/Proteasome
Paeoniflorigenone is a depolarizing neuromuscular blocking agent, being similar to succinylcholine.
T82003 Juniferdin

Juniferdin是一种抑制Protein disulfide isomerase (PDI),IC50为3.5 μM,旨在阻断HIV传播的化合物。此外,Juniferdin展现出细胞毒性并能抑制血小板聚集。
TN3869 Dimeric coniferyl acetate

Others Others
Dimeric coniferyl acetate has anti-inflammary activity, it shows strong NO inhibition with IC50 values of 27.1 uM in lipopolysacchalide (LPS)-activated murine macrophage-like J774.1 cells. It exhibits significant inhibitory effects on the nitric oxide pro
TN3802 Dehydrodiconiferyl alcohol

Estrogen/progestogen Receptor Endocrinology/Hormones
Dehydrodiconiferyl alcohol (DHCA) 是一种从葫芦中分离出来的木脂素,通过作为雌激素受体激动剂抑制破骨细胞分化和卵巢切除术诱导的骨质流失。
T79976 Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside

HBV Microbiology/Virology
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside 作为一种抗HBV剂,在Hep G2.2.15细胞系上能够抑制HBsAg和HBeAg的分泌,其IC50值分别约为1.67 mM和>2.15 mM。
TN4004 Erythro-Guaiacylglycerol β-dihydroconiferyl ether

Erythro-Guaiacylglycerol β-dihydroconiferyl ether 是从加拿大枫糖浆中提取的,具有潜在的抗氧化活性,可用于研究营养保健品。
TN5406 threo-Guaiacylglycerol β-coniferyl ether

Threo-Guaiacylglycerol beta-coniferyl ether displays significant inhibitory effects on NO production.
T38524 Paeoniflorin sulfite

During the sulfur-fumigation process of Paeoniae Radix Alba, Paeoniflorin, which serves as a principal constituent, can be converted into Paeoniflorin sulfite.
T82594 Debenzoylpaeoniflorgenin

Debenzoylpaeoniflorgenin是从Paeonia lactiflora中分离得到的天然化合物,该植物是Guizhitang的一个组成成份。
TN2416 8-Debenzoylpaeoniflorin

Others Others
8-Debenzoylpaeoniflorin is a natural product from plants
T80776 Withasomniferolide A

Withasomniferolide A,属于睡茄内酯类化合物,通过对Withania somnifera根的GABAA受体阳性激活物进行甲醇提取分离得到。
T37962 Paeoniflorgenin

Paeoniflorgenin is a deglucosylated metabolite of Paeoniflorin[1]. [1]. Hsiu SL, et, al. A deglucosylated metabolite of paeoniflorin of the root of Paeonia lactiflora and its pharmacokinetics in rats. Planta Med. 2003 Dec; 69(12): 1113-8.
T79975 Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside

HBV Microbiology/Virology
Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside(化合物1)是一种具有抗HBV活性的木脂素类化合物。该化合物对HBV表面抗原(HBsAg)的IC50为0.58 mM,而对HBV e抗原(HBeAg)的IC50 > 2.4 mM。其可从八角茴香中提取分离。
TN5857 Debenzoylgalloylpaeoniflorin

Debenzoylgalloylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5857,CAS号为 262350-51-6。
TMA1203 Viniferol D

Others Others
Viniferol D is a natural product from Vitis vinifera.
TN5432 (7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucoside

(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5432,CAS号为 351346-10-6。
T40611 (E)-Dehydrodiconiferyl alcohol

(E)-Dehydrodiconiferyl alcohol is a potent dual inhibitor of hCA IX and hCA XII, effectively impeding the catalytic activity of both carbonic anhydrase isoforms. Additionally, (E)-Dehydrodiconiferyl alcohol exerts inhibitory effects on the nuclear translocation of NF-κB in the connective tissue of the healing area.
TN4687 O-Geranylconiferyl alcohol

Others Others
O-Geranylconiferyl alcohol是一种天然产物,属于芸香科花椒属,其产品编号为 TN4687,CAS号为 129350-09-0。O-Geranylconiferyl alcohol可用作对照参考。
T82431 Eupenifeldin

Eupenifeldin为五环双酚酮类化合物,源自Eupenicillium brefeldianum ATCC 74184培养物分离得到。该化合物对HCT-116细胞系展现细胞毒性,具有潜在的白血病研究价值。
TN6535 Somnifericin

Somnifericin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6535,CAS号为 173693-57-7。
T83310 4-O-Methyldebenzoylpaeoniflorin

4-O-Methyldebenzoylpaeoniflorin为自Paeonia albiflora提取的自然化合物。
TN4003 Erythro-Guaiacylglycerol beta-coniferyl ether

Glucosidase Metabolism
Erythro-Guaiacylglycerol beta-coniferyl ether 可以从绿豆的茎和叶中提取出来的化合物,对 α-糖苷酶有抑制作用,EC50 值为 18.71 μM。
TN5769 cis-ε-Viniferin

cis-ε-Viniferin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5769,CAS号为 62250-12-8。
T82028 Isomaltopaeoniflorin

Isomaltopaeoniflorin为舒郁中草药配方的代谢产物,该配方用以抑制抑郁症样疾病。
T40797 Essential oils, Melaleuca alternifolia

Melaleuca alternifolia essential oil, derived from the leaves of Melaleuca alternifolia, exhibits bactericidal and anti-inflammatory properties.
TN5416 threo-7-O-Methylguaiacylglycerol β-coniferyl ether

threo-7-O-Methylguaiacylglycerol β-coniferyl ether 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5416,CAS号为 150333-85-0。
T75557 Withasomniferolide B

Withasomniferolide B 是一种睡茄内酯。Withasomniferolide B 可以从 Withania somnifera 根部的 GABAA 受体阳性激活剂甲醇提取物中分离出来。
TN5855 2'-O-Benzoylpaeoniflorin

2'-O-Benzoylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5855,CAS号为 1456598-64-3。
T82555 Dihydrodehydrodiconiferyl alcohol 9-Oglucoside

Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucopyranoside (DHD) is an extractable compound from G. mangostana L.
TN1205 2,3-Didehydrosomnifericin

Others Others
2,3-Didehydrosomnifericin is a natural product
TL0011 Adonifoline

Others Others
Adonifoline is a hepatotoxic pyrrolizidine alkaloid.

天然产物

coniferyl ferulate
Cat.No: T3S0012
Synonym:
Target: P-gp, GST
Benzoylpaeoniflorin
Cat.No: T6S1652
Synonym:
Target: COX
ε-​Viniferin
Cat.No: T11218
Synonym: epsilon-Viniferin,Epsilon-白藜芦醇脱氢二聚体
Target: P450
Coniferaldehyde
Cat.No: T2S1907
Synonym: Ferulaldehyde,Ferulyl aldehyde,4-HYDROXY-3-METHOXYCINNAMALDEHYDE,松柏醛,Coniferyl aldehyde,松柏醛;4-羟基-3-甲氧基肉桂醛
Target: Apoptosis, Antioxidant
Dihydrodehydrodiconiferyl alcohol
Cat.No: TN3849
Synonym:
Target: TNF
Benzoyloxypaeoniflorin
Cat.No: T4S1658
Synonym: 苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷
Target: NF-κB, Tyrosinase
Paeoniflorin
Cat.No: T2230
Synonym: 芍药苷,Peoniflorin
Target: HSP, COX
CONIFERYL ALCOHOL
Cat.No: TL0010
Synonym: 松柏醇,Coniferol
Target: Endogenous Metabolite, Antifungal
Galloylpaeoniflorin
Cat.No: TN1067
Synonym: 6'-O-Galloyl paeoniflorin,没食子酰芍药苷
Target: NF-κB, Androgen Receptor, ROS
Coniferaldehyde
Cat.No: TN3694
Synonym:
Target: NOS, COX, Nrf2, PKC, Autophagy
Tetrahydrodehydrodiconiferyl alcohol
Cat.No: TN7097
Synonym:
Target: Others
Resiniferatoxin
Cat.No: T34295
Synonym: RTX,[3H]resiniferatoxin,树脂毒素
Target: IL Receptor
coniferin
Cat.No: TL0009
Synonym: Coniferoside,松柏苷,Abietin
Target: Others, Antifungal
Schinifoline
Cat.No: TN1174
Synonym:
Target: Apoptosis, cell cycle arrest
Oxypaeoniflorin
Cat.No: T3773
Synonym: 氧化芍药苷,Oxypaeoniflora
Target: Others
α-Viniferin
Cat.No: TN1378
Synonym: ALPHA-VINIFERIN,Alpha-葡萄素
Target: P450, NO Synthase, Prostaglandin Receptor
Dihydroconiferyl alcohol
Cat.No: TN1578
Synonym:
Target: Others
(2R,3S)-Dihydrodehydroconiferyl alcohol
Cat.No: TN2844
Synonym:
Target: MAPK, PKC
Paeoniflorigenone
Cat.No: TN2034
Synonym:
Target: Others, Caspase
Juniferdin
Cat.No: T82003
Synonym:
Target:
Dimeric coniferyl acetate
Cat.No: TN3869
Synonym:
Target: Others
Dehydrodiconiferyl alcohol
Cat.No: TN3802
Synonym:
Target: Estrogen/progestogen Receptor
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside
Cat.No: T79976
Synonym:
Target: HBV
Erythro-Guaiacylglycerol β-dihydroconiferyl ether
Cat.No: TN4004
Synonym:
Target:
threo-Guaiacylglycerol β-coniferyl ether
Cat.No: TN5406
Synonym:
Target:
Paeoniflorin sulfite
Cat.No: T38524
Synonym:
Target:
Debenzoylpaeoniflorgenin
Cat.No: T82594
Synonym:
Target:
8-Debenzoylpaeoniflorin
Cat.No: TN2416
Synonym:
Target: Others
Withasomniferolide A
Cat.No: T80776
Synonym:
Target:
Paeoniflorgenin
Cat.No: T37962
Synonym:
Target:
Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside
Cat.No: T79975
Synonym:
Target: HBV
Debenzoylgalloylpaeoniflorin
Cat.No: TN5857
Synonym:
Target:
Viniferol D
Cat.No: TMA1203
Synonym:
Target: Others
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucoside
Cat.No: TN5432
Synonym:
Target:
(E)-Dehydrodiconiferyl alcohol
Cat.No: T40611
Synonym:
Target:
O-Geranylconiferyl alcohol
Cat.No: TN4687
Synonym:
Target: Others
Eupenifeldin
Cat.No: T82431
Synonym:
Target:
Somnifericin
Cat.No: TN6535
Synonym:
Target:
4-O-Methyldebenzoylpaeoniflorin
Cat.No: T83310
Synonym:
Target:
Erythro-Guaiacylglycerol beta-coniferyl ether
Cat.No: TN4003
Synonym:
Target: Glucosidase
cis-ε-Viniferin
Cat.No: TN5769
Synonym:
Target:
Isomaltopaeoniflorin
Cat.No: T82028
Synonym:
Target:
Essential oils, Melaleuca alternifolia
Cat.No: T40797
Synonym:
Target:
threo-7-O-Methylguaiacylglycerol β-coniferyl ether
Cat.No: TN5416
Synonym:
Target:
Withasomniferolide B
Cat.No: T75557
Synonym:
Target:
2'-O-Benzoylpaeoniflorin
Cat.No: TN5855
Synonym:
Target:
Dihydrodehydrodiconiferyl alcohol 9-Oglucoside
Cat.No: T82555
Synonym:
Target:
2,3-Didehydrosomnifericin
Cat.No: TN1205
Synonym:
Target: Others
Adonifoline
Cat.No: TL0011
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-01357 S100A9 Protein, Human, Recombinant (His)

MRP14,P14,LIAG,CFAG,CGLB,CAGB,NIF,MIF,S100 calcium ...

Human Baculovirus Insect Cells
S100A9 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 14.6 kDa and the accession number is P06702.
TMPY-01356 S100A8 Protein, Human, Recombinant (His)

60B8AG,MRP-8,MA387,NIF,L1Ag,S100 calcium binding pr...

Human Baculovirus Insect Cells
S100A8 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 12.2 kDa and the accession number is P05109.
TMPY-01330 S100A9 Protein, Human, Recombinant

CAGB,MIF,60B8AG,S100 calcium binding protein A9,CGLB,L1AG,

Human E. coli
S100A9 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26 and 13 kDa and the accession number is P06702.
TMPH-03700 Hyaluronidase Protein, Vespa magnifica, Recombinant (His)

Vespa magnifica E. coli
Hydrolyzes high molecular weight hyaluronic acid to produce small oligosaccharides. Hyaluronidase Protein, Vespa magnifica, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is P86875.
TMPH-03704 Cytolysin Protein, Vibrio vulnificus, Recombinant (His & Myc)

Cytolysin,vvhA

Vibrio vulnificus E. coli
Bacterial hemolysins are exotoxins that attack blood cell membranes and cause cell rupture by mechanisms not clearly defined. Cytolysin Protein, Vibrio vulnificus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 55.8 kDa and the accession number is P19247.
TMPH-03407 NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc)

Rhizobium leguminosarum E. coli
The key enzymatic reactions in nitrogen fixation are catalyzed by the nitrogenase complex, which has 2 components: the iron protein and the molybdenum-iron protein. NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc) is expressed in E. coli expression system with N-10xHis-GST and C-Myc tag. The predicted molecular weight is 35.0 kDa and the accession number is P20623.
TMPH-00159 Subtilisin Carlsberg Protein, Bacillus licheniformis, Recombinant (His & SUMO)

Bacillus licheniformis E. coli
Subtilisin is an extracellular alkaline serine protease, it catalyzes the hydrolysis of proteins and peptide amides (Ref.4, PubMed:11109488). Shows high specificity for aromatic and hydrophobic amino acids in the P1 substrate position. May play an important role in the degradation of feather keratin. Subtilisin Carlsberg Protein, Bacillus licheniformis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO tag. The predicted molecular weight is 42.0 kDa and the ac...
TMPH-02460 nifH1 Protein, Methanobacterium ivanovii, Recombinant (His & Myc)

Methanobacterium ivanovii E. coli
The key enzymatic reactions in nitrogen fixation are catalyzed by the nitrogenase complex, which has 2 components: the iron protein and the molybdenum-iron protein. nifH1 Protein, Methanobacterium ivanovii, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.4 kDa and the accession number is P51602.
TMPH-03403 Renilla-type luciferase Protein, Renilla reniformis, Recombinant (His & Myc & SUMO)

Renilla reniformis E. coli
Renilla-type luciferase Protein, Renilla reniformis, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 56.0 kDa and the accession number is P27652.
TMPH-03705 NfuA Protein, Vibrio vulnificus, Recombinant

Vibrio vulnificus E. coli
Involved in iron-sulfur cluster biogenesis. Binds a 4Fe-4S cluster, can transfer this cluster to apoproteins, and thereby intervenes in the maturation of Fe/S proteins. Could also act as a scaffold/chaperone for damaged Fe/S proteins. NfuA Protein, Vibrio vulnificus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 21.0 kDa and the accession number is Q8DDU2.

重组蛋白

S100A9 Protein, Human, Recombinant (His)
Cat.No: TMPY-01357
Species: Human
Expression System: Baculovirus Insect Cells
S100A8 Protein, Human, Recombinant (His)
Cat.No: TMPY-01356
Species: Human
Expression System: Baculovirus Insect Cells
S100A9 Protein, Human, Recombinant
Cat.No: TMPY-01330
Species: Human
Expression System: E. coli
Hyaluronidase Protein, Vespa magnifica, Recombinant (His)
Cat.No: TMPH-03700
Species: Vespa magnifica
Expression System: E. coli
Cytolysin Protein, Vibrio vulnificus, Recombinant (His & Myc)
Cat.No: TMPH-03704
Species: Vibrio vulnificus
Expression System: E. coli
NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc)
Cat.No: TMPH-03407
Species: Rhizobium leguminosarum
Expression System: E. coli
Subtilisin Carlsberg Protein, Bacillus licheniformis, Recombinant (His & SUMO)
Cat.No: TMPH-00159
Species: Bacillus licheniformis
Expression System: E. coli
nifH1 Protein, Methanobacterium ivanovii, Recombinant (His & Myc)
Cat.No: TMPH-02460
Species: Methanobacterium ivanovii
Expression System: E. coli
Renilla-type luciferase Protein, Renilla reniformis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03403
Species: Renilla reniformis
Expression System: E. coli
NfuA Protein, Vibrio vulnificus, Recombinant
Cat.No: TMPH-03705
Species: Vibrio vulnificus
Expression System: E. coli
TargetMol Loading
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