56
49
10
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9331 |
Bemnifosbuvir hemisulfate
AT-527 |
HCV Protease; SARS-CoV | Microbiology/Virology; Proteases/Proteasome |
Bemnifosbuvir hemisulfate (AT-527) 是一种 HCV 病毒复制抑制剂。 | |||
T67812 |
Tenifatecan
SN2310 |
||
Tenifatecan (SN2310) 是一种高度亲脂性的7-乙基-10-羟基喜树碱(SN)制剂,具有潜在的抗肿瘤活性。 | |||
T1146 |
Nifedipine
BAY-a-1040,Procardia XL,Procardia,硝苯地平,Adalat |
CaMK; Potassium Channel; Calcium Channel; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Nifedipine (Procardia) 是一种二氢吡啶类钙通道阻滞剂,可抑制细胞外钙离子跨膜流入心肌和血管平滑肌细胞,导致主要冠状动脉和全身动脉扩张,降低心肌收缩力。它常用于心肌功能不全的相关研究。 | |||
T2514 |
Linifanib
利尼伐尼,ABT-869,RG3635,AL-39324 |
Apoptosis; c-Fms; VEGFR; FLT; CSF-1R; PDGFR; c-Kit; Autophagy | Angiogenesis; Apoptosis; Autophagy; Tyrosine Kinase/Adaptors |
Linifanib (AL-39324) 是一种高效口服的VEGFR 和PDGFR 家族多靶点抑制剂,具有显著的抗肿瘤活性。它对无关 RTKs、可溶性酪氨酸激酶或丝氨酸/苏氨酸激酶的活性要低得多。它是特异性 miR-10b 抑制剂,阻断miR-10b 的生物合成。 | |||
T2712 |
Nifekalant hydrochloride
|
Potassium Channel | Membrane transporter/Ion channel |
Nifekalant hydrochloride 是一种 IKr 钾通道阻滞剂,IC50为10 µM,属于 III 类抗心律不齐化合物,可用于快速室上性心律失常的研究。 | |||
T15271 |
Denifanstat
FASN-IN-2,TVB2640,TVB-2640 |
Fatty Acid Synthase | Metabolism |
Denifanstat (FASN-IN-2) 是一种口服具有活性的选择性 FASN 抑制剂,IC50=0.052 μM,EC50=0.072 μM。它有用于脂肪肝和癌症的研究潜力。 | |||
T8663 |
nifenalol.HCl
INPEA,1-(4-硝基苯基)-1-羟基-2-异丙基氨基乙烷盐酸盐 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Nifenalol.HCl(INPEA) 是β-肾上腺素能受体的拮抗剂。 | |||
T9341 |
Bemnifosbuvir
AT-511 |
Others; HCV Protease; SARS-CoV | Microbiology/Virology; Others; Proteases/Proteasome |
Bemnifosbuvir (AT-511) 是一种口服活性抑制剂,抑制 HCV 病毒复制,具有全基因型抗病毒活性。它有效抑制 SARS-CoV-2 (COVID-19)感染 (EC90=0.47 μM)。 | |||
T4503 |
Talniflumate
Somalgen,他尼氟酯 |
Chloride channel; COX; N-Acetylglucosaminyltransferase; Anion Exchanger | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Talniflumate (Somalgen) 是一种钙激活氯离子通道 (hCLCA1/mCLCA3) 阻滞剂,可减少动物模型和细胞培养中的粘蛋白合成和释放。它通过抑制环氧合酶,并抑制 Cl-/HCO3- 交换活性,具有抗炎作用。它还增加了远端肠梗阻综合征囊性纤维化小鼠模型的存活率。 | |||
T0693 |
Niflumic acid
氟尼酸,Nifluril,Forenol,Landruma |
Others; Phospholipase; Chloride channel; COX; Monocarboxylate transporter; UGT | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; Others |
Niflumic acid (Nifluril) 是钙离子激活的氯离子通道阻断剂,用于治疗类风湿性关节炎的镇痛剂和抗炎剂。 | |||
T5325 |
Nifurtimox
硝呋替莫,BAY-2502,BAY-A-2502 |
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
Nifurtimox (BAY-A-2502) 是一种用于锥虫病的抗虫剂,可影响乳酸脱氢酶活性。它有潜力研究神经母细胞瘤细胞。 | |||
T19636 |
Morniflumate
马尼氟酯,Niflam,UP 164,UP-164,Morniflu,UP164 |
Others | Others |
Morniflumate (Niflam) 是一种非甾体抗炎药。它用于治疗炎症。 | |||
T0980 |
Nifenazone
尼芬那宗,Niapyrin,Nicodone,烟酰氨基比林,Nicazane |
COX | Immunology/Inflammation; Neuroscience |
Nifenazone (Nicodone) 是吡唑类试剂,可用于研究各种风湿性疾病。 | |||
T77432 |
Anifrolumab
MDX-1333,MEDI-546 |
IFNAR | Immunology/Inflammation |
Anifrolumab(MEDI-546) 是一种有效的 I 型干扰素 (IFN) 受体拮抗剂,是一种靶向 IFN 的人源单克隆抗体。Anifrolumab 能抑制 I 型干扰素的活性,可用于预防和治疗系统性红斑狼疮 (SLE) 。 | |||
T36665 |
Dehydro Nifedipine
BAY-b 4759 |
||
Dehydro Nifedipine (BAY-b 4759) 是人血浆中硝苯地平的主要代谢物。Dehydro Nifedipine 抑制PC-12细胞葡萄糖摄取,IC50值为130 μM,硝苯地平是一种钙通道阻滞剂,用于治疗高血压和心绞痛。当硝苯地平被细胞色素P450 (CYP)异构体CYP3A4和CYP3A5代谢时形成脱氢硝苯地平。 | |||
T1563 |
Nifuroxazide
Diarlidan,硝呋齐特,Nifuroxazid,Dicoferin,硝呋酚酰肼 |
Antibacterial; Antibiotic; STAT | JAK/STAT signaling; Microbiology/Virology; Stem Cells |
Nifuroxazide (Diarlidan) 是STAT3抑制剂,具有抗转移和抗癌活性。 | |||
T7395 |
Lanifibranor
IVA337 |
PPAR | DNA Damage/DNA Repair; Metabolism |
Lanifibranor (IVA337) 是泛过氧化物酶体增殖物激活受体 (PPAR) 激动剂,对人类PPARα,PPARσ和PPARγ的EC50值分别为 1.5, 0.87 和 0.21 μM。 | |||
T6114 |
Nifursol
硝呋索尔,尼呋索尔 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Nifursol 是一种具有口服活性的兽用抗生素,用于预防组织口炎。它快速代谢形成代谢标记物 3,5-二硝基水杨酸环肼,并能持续很长时间。它可研究沙门氏菌感染的家禽、家禽和水生动物的大肠杆菌肠胃病。 | |||
T1526 |
Nifuratel
NF 113,SAP 113,硝呋太尔,Methylmercadone |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Nifuratel (SAP 113) 是广谱抗生素,有抗细菌、真菌和毛滴虫活性。 | |||
T7599 |
Sunifiram
桑尼菲拉姆,DM-235,桑尼非拉姆 |
iGluR | Membrane transporter/Ion channel; Neuroscience |
Sunifiram (DM-235) 是一种 ampakine 样促智剂。 | |||
T12223 |
Nifursemizone
NF161,5-Nitro-2-furancarbaldehyde 2-ethyl semicarbazone,硝呋米腙,Etafurazone |
Antibiotic | Microbiology/Virology |
Nifursemizone (Etafurazone) 是抗原虫药。 | |||
T38192 |
Unifiram
|
Others | Others |
Unifiram 是一种认知增强剂。 Unifiram 诱导大鼠海马 CA1 区场兴奋性突触后电位 (fEPSP) 幅度的持久增加 (EC50= 27 nM) 并增加大鼠大脑皮层中乙酰胆碱 (ACh) 的释放。 | |||
T73198 | Nifuroxime | ||
Nifuroxime 是一种抗感染剂,可用于真菌感染相关的研究。 | |||
T73284 |
Vonifimod
|
||
Vonifimod 是一种免疫调节剂。 | |||
T26819 |
Binifibrate
WAC104,WAC 104,Antopal,WAC-104,Biniwas |
||
Binifibrate is a hyperlipemiant drug used for the treatment of hyperlipidemia. | |||
T125992 |
threo-Guaiacylglycerol β-dihydroconiferyl ether
|
||
threo-Guaiacylglycerol β-dihydroconiferyl ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125992。 | |||
T125621 |
erythro-Guaiacylglycerol β-coniferyl ether
|
||
erythro-Guaiacylglycerol β-coniferyl ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125621。 | |||
T35584 |
Hydroxydehydro Nifedipine Carboxylate
|
||
Hydroxydehydro nifedipine carboxylate is a metabolite of nifedipine .1 1.Roosemalen, M.C.M., Soons, P.A., Funaki, T., et al.High-performance liquid chromatographic determination of the polar metabolites of nifedipine in plasma, blood and urineJ. Chromatogr.565(1-2)516-522(1991) | |||
TP2394 |
Nifalatide
|
||
Nifalatide is a analog of enkephalin. | |||
T124473 | threo-Guaiacylglycerol-beta-coniferyl aldehyde ether | ||
threo-Guaiacylglycerol-beta-coniferyl aldehyde ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124473。 | |||
T68828 |
Chinifur
|
||
Chinifur is a selective inhibitor and subversive substrate" for Trypanosoma congolense trypanothione reductase" | |||
T28610 |
Ronifibrate
|
||
Ronifibrate is a lipid modifying agent with antihyperlipidemic and antiarteriosclerotic activity. | |||
T126480 |
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-xyloside
|
||
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-xyloside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126480。 | |||
T22515 |
5'-Iodoresiniferatoxin
|
Others | Others |
TRPV1 (VR1) receptor antagonist | |||
T74065 |
Nifurpirinol
|
||
Nifurpirinol (P-7138),一种硝基芳香型抗生素(antibiotic),作为细菌硝基还原酶(NTR)的底物。相较于甲硝唑,其作为一种prodrug,在表达硝基还原酶的转基因模型中引发细胞消融的效能更高。 | |||
T12222 |
Nifedipine-d6
硝苯地平 D6,Nifedipine D6,BAY-a-1040 D6 |
Others | Others |
Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel. | |||
T32766 |
Linifolin A
NSC 153859,NSC-153859,NSC153859,PF 57,PF-57 |
||
Linifolin A is a sesquiterpene lactone extracted from Helenium aromaticum. | |||
T22527 | 6'-Iodoresiniferatoxin | Others | Others |
TRPV1 (VR1) vanilloid receptor partial agonist | |||
T69021 | Nifedipine HCl | ||
Nifedipine HCl is a potent vasodilator agent with calcium antagonistic action. It is a useful anti-anginal agent that also lowers blood pressure. | |||
T125568 |
Dihydroconiferin
|
||
Dihydroconiferin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125568,CAS号为 17609-06-2。 | |||
T33669 |
Nifurpipone
Rec-150122,Rec 150122,Rec150122 |
||
Nifurpipone is a biochemical existed in urine. | |||
T33667 |
Nifrofam
|
||
Nifrofam is a fluorescent probe for imaging α4β2* nAChRs. | |||
T71293 |
Nifuroxazide-d4
|
||
Nifuroxazide-d4 is intended for use as an internal standard for the quantification of nifuroxazide by GC- or LC-MS. Nifuroxazide is a nitrofuran antibiotic. It is active against strains of the enteropathogenic bacteria C. jejuni, Salmonella, Y. enterocolitica, Shigella, and E. coli. It inhibits quorum sensing and virulence factor production in P. aeruginosa. Nifuroxazide inhibits STAT3 activity in a reporter assay and decreases viability of U266 and INA-6 myeloma cells, which have constitutive S... | |||
T124284 | Erythro-Guaiacylglycerol-beta-coniferyl aldehyde ether | ||
Erythro-Guaiacylglycerol-beta-coniferyl aldehyde ether 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124284。 | |||
T28171 |
Nifeviroc
TD-0232,TD 0232,尼非韦罗,TD0232 |
||
Nifeviroc, a CCR5 antagonist, is used potentially for treatment of inflammatory responses to HIV type-1 infection. | |||
T11926 |
m-Nifedipine
|
Others | Others |
m-Nifedipine, an impurity of Nifedipine, serves as a potent calcium channel blocker and the preferred treatment option for cardiac insufficiencies. | |||
T79836 |
Arbemnifosbuvir
|
SARS-CoV | Microbiology/Virology |
Arbemnifosbuvir 是用于干扰核病毒RdRp相关核苷酸基转移酶(NiRAN)非结构蛋白12(nsp12)的化合物,适用于SARS-CoVs感染的研究。 | |||
T126168 |
Pruniflorone R
|
||
Pruniflorone R 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126168。 | |||
T8663L |
Nifenalol
|
||
Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina. | |||
T25869 |
Nifurzide
Ricridene |
||
Nifurzide is a nitrofuran derivative used as an intestinal antiinfectious agent. Low concentrations reduces growth rate while high concentrations completely inhibits growth. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3S0012 |
coniferyl ferulate
|
P-gp; GST | Membrane transporter/Ion channel; Neuroscience; oxidation-reduction |
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。 | |||
T6S1652 |
Benzoylpaeoniflorin
|
COX | Immunology/Inflammation; Neuroscience |
Benzoylpaeoniflorin 是一种从白芍中提取的天然化合物,可以降低细胞凋亡,对冠心病具有潜在的研究价值。 | |||
T11218 |
ε-Viniferin
epsilon-Viniferin,Epsilon-白藜芦醇脱氢二聚体 |
P450 | Metabolism |
ε-Viniferin (epsilon-Viniferin) 提取自 Vitis vinifera,是 Resveratrol 的二聚体,能够抑制 CYP 家族,其 Ki=0.5~20 μM,具有抗氧化作用。 | |||
T2S1907 |
Coniferaldehyde
Ferulaldehyde,Ferulyl aldehyde,4-HYDROXY-3-METHOXYCINNAMALDEHYDE,松柏醛,Coniferyl aldehyde,松柏醛;4-羟基-3-甲氧基肉桂醛 |
Apoptosis; Antioxidant | Apoptosis; oxidation-reduction |
Coniferaldehyde (Ferulaldehyde) 是一种血红素加氧酶-1 的有效诱导剂,具有抗炎作用。在 RAW264.7 巨噬细胞中,它通过 PKCα/βII/Nrf-2/HO-1 依赖性途径来抑制 LPS 诱导的细胞凋亡。 | |||
TN3849 |
Dihydrodehydrodiconiferyl alcohol
|
TNF | Apoptosis |
Dihydrodehydrodiconiferyl alcohol 是 Liriodendron tulipifera 的甲醇提取物。 | |||
T4S1658 |
Benzoyloxypaeoniflorin
苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷 |
NF-κB; Tyrosinase | NF-κB; Proteases/Proteasome |
Benzoyloxypaeoniflorin (Benzoyloxypeoniflorin) 是一种酪氨酸酶抑制剂,分离于Paeonia suffruticosa 的根,对mushroom tyrosinase 的 IC50为 0.453 mM。它是一种NF-κB 抑制剂,它通过对血小板聚集和凝血的抑制作用,有助于改善血液循环。 | |||
T2230 |
Paeoniflorin
芍药苷,Peoniflorin |
HSP; COX | Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience |
Paeoniflorin (Peoniflorin) 是从芍药根中提取的一种蒎烷单萜糖苷,具有抗癌作用、抗氧化应激、抗血小板聚集、血管扩张、降低血液粘度和抗炎活性等多种生物活性。它是一种热休克蛋白诱导剂,通过自噬途径保护 PC12 细胞免受 MPP+和酸性损伤。 | |||
TL0010 |
CONIFERYL ALCOHOL
松柏醇,Coniferol |
Endogenous Metabolite; Antifungal | Metabolism; Microbiology/Virology |
Coniferyl alcohol (Coniferol) 是合成芪类和香豆素丁子香酚的中间体,有抗真菌功效。 | |||
TN1067 |
Galloylpaeoniflorin
6'-O-Galloyl paeoniflorin,没食子酰芍药苷 |
NF-κB; Androgen Receptor; ROS | Endocrinology/Hormones; Immunology/Inflammation; NF-κB |
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) 是 NF-κB 抑制剂,同时也是 DNA 裂解抑制剂。 | |||
TN3694 |
Coniferaldehyde
|
NOS; COX; Nrf2; PKC; Autophagy | Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Neuroscience |
Coniferaldehyde 能显着抑制酒球菌菌株的生长活力。 Coniferaldehyde 通过诱导血红素加氧酶 1 (HO-1) 发挥抗炎特性。 | |||
TN7097 |
Tetrahydrodehydrodiconiferyl alcohol
|
Others | Others |
Tetrahydrodehydrodiconiferyl alcohol 是一种天然产物。 | |||
T34295 |
Resiniferatoxin
RTX,[3H]resiniferatoxin,树脂毒素 |
IL Receptor | Immunology/Inflammation |
Resiniferatoxin ([3H]resiniferatoxin) 抑制 Th1 细胞因子的产生,有助于防御 T.spiralis 感染,并可用于免疫反应调节剂的研究。 | |||
TL0009 |
coniferin
Coniferoside,松柏苷,Abietin |
Others; Antifungal | Microbiology/Virology; Others |
Coniferin (Abietin) 是一种松柏醇中的葡萄糖苷。它抑制真菌生长和黑化反应,具有 ATP 依赖性转运活性并具有抗氧化作用。 | |||
TN1174 |
Schinifoline
|
Apoptosis; cell cycle arrest | Apoptosis; Cell Cycle/Checkpoint |
Schinifoline 是从 Zanthoxylum schinifolium Sieb 中提取出来的一种喹啉酮衍生物,具有细胞毒性活性,可促进癌细胞放射敏感性,影响细胞循环周期和细胞凋亡。 | |||
T3773 |
Oxypaeoniflorin
氧化芍药苷,Oxypaeoniflora |
Others | Others |
Oxypaeoniflorin (Oxypaeoniflora) 从 Paeoniae 中分离得到的单萜糖苷化合物,是一种抗氧化剂,是具有神经保护和抗炎作用。 | |||
TN1378 |
α-Viniferin
ALPHA-VINIFERIN,Alpha-葡萄素 |
P450; NO Synthase; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Metabolism |
α-Viniferin 也称为2-芳基苯并呋喃类黄酮,是前列腺素H2合成酶抑制剂。具有抗阿尔茨海默病、抗结核、抗肿瘤、抗炎、抗糖尿病等多种药理活性 | |||
TN1578 |
Dihydroconiferyl alcohol
|
Others | Others |
Dihydroconiferyl alcohol exhibits cytoprotective activity in cultured MCF-7 cells stressed by H2O2. | |||
TN2844 |
(2R,3S)-Dihydrodehydroconiferyl alcohol
|
MAPK; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK |
(2R,3S)-Dihydrodehydroconiferyl alcohol can induce neurite outgrowth and enhance NGF-induced neurite outgrowth from PC12 cells by amplifying up-stream steps such as MAPK and PKC. | |||
TN2034 |
Paeoniflorigenone
|
Others; Caspase | Apoptosis; Others; Proteases/Proteasome |
Paeoniflorigenone is a depolarizing neuromuscular blocking agent, being similar to succinylcholine. | |||
T82003 |
Juniferdin
|
||
Juniferdin是一种抑制Protein disulfide isomerase (PDI),IC50为3.5 μM,旨在阻断HIV传播的化合物。此外,Juniferdin展现出细胞毒性并能抑制血小板聚集。 | |||
TN3869 |
Dimeric coniferyl acetate
|
Others | Others |
Dimeric coniferyl acetate has anti-inflammary activity, it shows strong NO inhibition with IC50 values of 27.1 uM in lipopolysacchalide (LPS)-activated murine macrophage-like J774.1 cells. It exhibits significant inhibitory effects on the nitric oxide pro | |||
TN3802 |
Dehydrodiconiferyl alcohol
|
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Dehydrodiconiferyl alcohol (DHCA) 是一种从葫芦中分离出来的木脂素,通过作为雌激素受体激动剂抑制破骨细胞分化和卵巢切除术诱导的骨质流失。 | |||
T79976 |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside
|
HBV | Microbiology/Virology |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside 作为一种抗HBV剂,在Hep G2.2.15细胞系上能够抑制HBsAg和HBeAg的分泌,其IC50值分别约为1.67 mM和>2.15 mM。 | |||
TN4004 |
Erythro-Guaiacylglycerol β-dihydroconiferyl ether
|
||
Erythro-Guaiacylglycerol β-dihydroconiferyl ether 是从加拿大枫糖浆中提取的,具有潜在的抗氧化活性,可用于研究营养保健品。 | |||
TN5406 |
threo-Guaiacylglycerol β-coniferyl ether
|
||
Threo-Guaiacylglycerol beta-coniferyl ether displays significant inhibitory effects on NO production. | |||
T38524 |
Paeoniflorin sulfite
|
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During the sulfur-fumigation process of Paeoniae Radix Alba, Paeoniflorin, which serves as a principal constituent, can be converted into Paeoniflorin sulfite. | |||
T82594 |
Debenzoylpaeoniflorgenin
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Debenzoylpaeoniflorgenin是从Paeonia lactiflora中分离得到的天然化合物,该植物是Guizhitang的一个组成成份。 | |||
TN2416 |
8-Debenzoylpaeoniflorin
|
Others | Others |
8-Debenzoylpaeoniflorin is a natural product from plants | |||
T80776 |
Withasomniferolide A
|
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Withasomniferolide A,属于睡茄内酯类化合物,通过对Withania somnifera根的GABAA受体阳性激活物进行甲醇提取分离得到。 | |||
T37962 |
Paeoniflorgenin
|
||
Paeoniflorgenin is a deglucosylated metabolite of Paeoniflorin[1]. [1]. Hsiu SL, et, al. A deglucosylated metabolite of paeoniflorin of the root of Paeonia lactiflora and its pharmacokinetics in rats. Planta Med. 2003 Dec; 69(12): 1113-8. | |||
T79975 |
Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside
|
HBV | Microbiology/Virology |
Dihydrodehydrodiconiferyl alcohol 9-O-α-L-rhamnopyranoside(化合物1)是一种具有抗HBV活性的木脂素类化合物。该化合物对HBV表面抗原(HBsAg)的IC50为0.58 mM,而对HBV e抗原(HBeAg)的IC50 > 2.4 mM。其可从八角茴香中提取分离。 | |||
TN5857 |
Debenzoylgalloylpaeoniflorin
|
||
Debenzoylgalloylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5857,CAS号为 262350-51-6。 | |||
TMA1203 |
Viniferol D
|
Others | Others |
Viniferol D is a natural product from Vitis vinifera. | |||
TN5432 |
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucoside
|
||
(7R,8R)-Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5432,CAS号为 351346-10-6。 | |||
T40611 |
(E)-Dehydrodiconiferyl alcohol
|
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(E)-Dehydrodiconiferyl alcohol is a potent dual inhibitor of hCA IX and hCA XII, effectively impeding the catalytic activity of both carbonic anhydrase isoforms. Additionally, (E)-Dehydrodiconiferyl alcohol exerts inhibitory effects on the nuclear translocation of NF-κB in the connective tissue of the healing area. | |||
TN4687 |
O-Geranylconiferyl alcohol
|
Others | Others |
O-Geranylconiferyl alcohol是一种天然产物,属于芸香科花椒属,其产品编号为 TN4687,CAS号为 129350-09-0。O-Geranylconiferyl alcohol可用作对照参考。 | |||
T82431 |
Eupenifeldin
|
||
Eupenifeldin为五环双酚酮类化合物,源自Eupenicillium brefeldianum ATCC 74184培养物分离得到。该化合物对HCT-116细胞系展现细胞毒性,具有潜在的白血病研究价值。 | |||
TN6535 |
Somnifericin
|
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Somnifericin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6535,CAS号为 173693-57-7。 | |||
T83310 |
4-O-Methyldebenzoylpaeoniflorin
|
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4-O-Methyldebenzoylpaeoniflorin为自Paeonia albiflora提取的自然化合物。 | |||
TN4003 |
Erythro-Guaiacylglycerol beta-coniferyl ether
|
Glucosidase | Metabolism |
Erythro-Guaiacylglycerol beta-coniferyl ether 可以从绿豆的茎和叶中提取出来的化合物,对 α-糖苷酶有抑制作用,EC50 值为 18.71 μM。 | |||
TN5769 |
cis-ε-Viniferin
|
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cis-ε-Viniferin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5769,CAS号为 62250-12-8。 | |||
T82028 |
Isomaltopaeoniflorin
|
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Isomaltopaeoniflorin为舒郁中草药配方的代谢产物,该配方用以抑制抑郁症样疾病。 | |||
T40797 | Essential oils, Melaleuca alternifolia | ||
Melaleuca alternifolia essential oil, derived from the leaves of Melaleuca alternifolia, exhibits bactericidal and anti-inflammatory properties. | |||
TN5416 | threo-7-O-Methylguaiacylglycerol β-coniferyl ether | ||
threo-7-O-Methylguaiacylglycerol β-coniferyl ether 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5416,CAS号为 150333-85-0。 | |||
T75557 | Withasomniferolide B | ||
Withasomniferolide B 是一种睡茄内酯。Withasomniferolide B 可以从 Withania somnifera 根部的 GABAA 受体阳性激活剂甲醇提取物中分离出来。 | |||
TN5855 |
2'-O-Benzoylpaeoniflorin
|
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2'-O-Benzoylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5855,CAS号为 1456598-64-3。 | |||
T82555 |
Dihydrodehydrodiconiferyl alcohol 9-Oglucoside
|
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Dihydrodehydrodiconiferyl alcohol 9-O-β-D-glucopyranoside (DHD) is an extractable compound from G. mangostana L. | |||
TN1205 |
2,3-Didehydrosomnifericin
|
Others | Others |
2,3-Didehydrosomnifericin is a natural product | |||
TL0011 |
Adonifoline
|
Others | Others |
Adonifoline is a hepatotoxic pyrrolizidine alkaloid. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01357 |
S100A9 Protein, Human, Recombinant (His)
MRP14,P14,LIAG,CFAG,CGLB,CAGB,NIF,MIF,S100 calcium ... |
Human | Baculovirus Insect Cells |
S100A9 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 14.6 kDa and the accession number is P06702. | |||
TMPY-01356 |
S100A8 Protein, Human, Recombinant (His)
60B8AG,MRP-8,MA387,NIF,L1Ag,S100 calcium binding pr... |
Human | Baculovirus Insect Cells |
S100A8 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 12.2 kDa and the accession number is P05109. | |||
TMPY-01330 |
S100A9 Protein, Human, Recombinant
CAGB,MIF,60B8AG,S100 calcium binding protein A9,CGLB,L1AG, |
Human | E. coli |
S100A9 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26 and 13 kDa and the accession number is P06702. | |||
TMPH-03700 |
Hyaluronidase Protein, Vespa magnifica, Recombinant (His)
|
Vespa magnifica | E. coli |
Hydrolyzes high molecular weight hyaluronic acid to produce small oligosaccharides. Hyaluronidase Protein, Vespa magnifica, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 45.1 kDa and the accession number is P86875. | |||
TMPH-03704 |
Cytolysin Protein, Vibrio vulnificus, Recombinant (His & Myc)
Cytolysin,vvhA |
Vibrio vulnificus | E. coli |
Bacterial hemolysins are exotoxins that attack blood cell membranes and cause cell rupture by mechanisms not clearly defined. Cytolysin Protein, Vibrio vulnificus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 55.8 kDa and the accession number is P19247. | |||
TMPH-03407 |
NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc)
|
Rhizobium leguminosarum | E. coli |
The key enzymatic reactions in nitrogen fixation are catalyzed by the nitrogenase complex, which has 2 components: the iron protein and the molybdenum-iron protein. NIFH Protein, Rhizobium leguminosarum, Recombinant (GST & His & Myc) is expressed in E. coli expression system with N-10xHis-GST and C-Myc tag. The predicted molecular weight is 35.0 kDa and the accession number is P20623. | |||
TMPH-00159 |
Subtilisin Carlsberg Protein, Bacillus licheniformis, Recombinant (His & SUMO)
|
Bacillus licheniformis | E. coli |
Subtilisin is an extracellular alkaline serine protease, it catalyzes the hydrolysis of proteins and peptide amides (Ref.4, PubMed:11109488). Shows high specificity for aromatic and hydrophobic amino acids in the P1 substrate position. May play an important role in the degradation of feather keratin. Subtilisin Carlsberg Protein, Bacillus licheniformis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO tag. The predicted molecular weight is 42.0 kDa and the ac... | |||
TMPH-02460 |
nifH1 Protein, Methanobacterium ivanovii, Recombinant (His & Myc)
|
Methanobacterium ivanovii | E. coli |
The key enzymatic reactions in nitrogen fixation are catalyzed by the nitrogenase complex, which has 2 components: the iron protein and the molybdenum-iron protein. nifH1 Protein, Methanobacterium ivanovii, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.4 kDa and the accession number is P51602. | |||
TMPH-03403 |
Renilla-type luciferase Protein, Renilla reniformis, Recombinant (His & Myc & SUMO)
|
Renilla reniformis | E. coli |
Renilla-type luciferase Protein, Renilla reniformis, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 56.0 kDa and the accession number is P27652. | |||
TMPH-03705 |
NfuA Protein, Vibrio vulnificus, Recombinant
|
Vibrio vulnificus | E. coli |
Involved in iron-sulfur cluster biogenesis. Binds a 4Fe-4S cluster, can transfer this cluster to apoproteins, and thereby intervenes in the maturation of Fe/S proteins. Could also act as a scaffold/chaperone for damaged Fe/S proteins. NfuA Protein, Vibrio vulnificus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 21.0 kDa and the accession number is Q8DDU2. |