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Search Results for " cem "

125

抑制剂 & 化合物

23

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T2331	Solithromycin 索利霉素,OP-1068,CEM-101	Antibacterial; Antibiotic	Microbiology/Virology
	Solithromycin (OP-1068) 是口服可生物利用的抗菌剂，抑制肺炎链球菌、葡萄球菌、金黄色葡萄球菌和流感嗜血杆菌的细胞活力、蛋白质合成和生长速率， IC50 值分别为 7.5 ng/mL、40 ng/mL 和 125 ng/mL。它可与核糖体的大 50S 亚基结合抑制蛋白质生物合成。
T39810	CEM114
	CEM114 is a potent chemical compound known as a chemical epigenetic modifier (CEM). It functions by employing CRISPR-Cas9 systems to harness endogenous chromatin machinery, thereby exerting its epigenetic modifying effects.
T9104	TJ191	Apoptosis	Apoptosis
	TJ191 是一种选择性抗癌试剂，靶向低 TβRIII 表达的恶性T 细胞白血病/淋巴瘤细胞，可研究癌症。
T20038	2-Fluoroadenine NSC-27364,NSC 27364,NSC27364,2-氟腺嘌呤	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	2-Fluoroadenine (NSC-27364) 对非增殖性和增殖性肿瘤细胞具有毒性。2-Fluoroadenine 可用于抗癌症的相关研究。
T6018	Zosuquidar trihydrochloride 唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride	P-gp	Membrane transporter/Ion channel; Neuroscience
	Zosuquidar trihydrochloride (LY-335979 trihydrochloride) 是一种P-糖蛋白抑制剂，Ki 值为 59 nM。
T0370	Pheniramine maleate Daneral,Inhiston,Trimetose,马来酸非尼拉敏	5-HT Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Pheniramine maleate (Trimetose) 是一种具有抗组胺和血管扩张特性的烷基胺衍生物，可与组胺 H1 受体结合，从而抑制磷脂酶 A2 和内皮源性松弛因子一氧化氮的产生。
T5858	Sertindole Lu 23-174,舍吲哚	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Sertindole (Lu 23-174) 是一种非典型抗精神病药，可与多巴胺 D2 受体和血清素受体亚型 5-HT1D、5-HT2A 和 5-HT2C 结合，Kd 值分别为 2.7、20、0.14 和 6 nM。
T9005	VPC-80051 racemate	Others	Others
	VPC-80051 是一种有效的 hnRNP A1 剪接活性抑制剂，靶向 hnRNP A1 RBD 并降低 22Rv1 CRPC 细胞系中的 AR-V7 信使水平。
T12400	Peliglitazar racemate (Rac)-Peliglitazar,(Rac)-BMS 426707-01,BMS 426707-01 racemate	PPAR	DNA Damage/DNA Repair; Metabolism
	Peliglitazar racemate(BMS 426707-01 racemate) 是 Peliglitazar 的外消旋体。Peliglitazar racemate 可作为潜在的抗糖尿病和抗肥胖剂。
T61477	dCeMM2	Molecular Glues	PROTAC
	dCeMM2 (Compound 2) 是一种胶降解剂。dCeMM2 促使 CDK12-cyclin K 与 CRL4B 连接酶复合物的相互作用，导致 cyclin K 的泛素化及降解。
T22988	MK-4827 Racemate Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide	PARP	Chromatin/Epigenetic; DNA Damage/DNA Repair
	MK-4827 Racemate (Niraparib Racemate) 是一种选择性 PARP1 和 PARP2 抑制剂，IC50 分别为 3.8 nM 和 2.1 nM，对 PARP3、V-PARP 和 Tank1 的选择性超过 330 倍。
T16731	Rentiapril racemate (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril	Angiotensin-converting Enzyme (ACE)	Metabolism
	Rentiapril racemate (SA-446 racemate) 是 Rentiapril 的外消旋体。Rentiapril racemate 具有抗炎活性，可用于研究青光眼。
T76750	Cemiplimab REGN-2810,SAR-439684	Others	Others
	Cemiplimab (Anti-Human PD-1) 是一种针对程序性细胞死亡受体 1 （PD-1）的人单克隆抗体，也是一种检查点抑制剂，可阻断 PD-1/PD-L1 介导的 T 细胞抑制，可用于转移性癌症和鳞状细胞皮肤癌研究。
T3562	Valrocemide TV1901,N-丙戊酰基甘氨酰胺,N-Valproylglycinamide,丙戊塞胺	Others	Others
	Valrocemide (TV1901) 是有前景的抗癫痫候选药物，具有广泛的抗惊厥特性。
T22253	AG-120 (racemic) 1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺	Dehydrogenase	Metabolism
	AG-120 (racemic) 是 AG-120 的外消旋混合物，是一种可口服的异柠檬酸脱氢酶 1 型 (IDH1) 抑制剂，具有潜在的抗肿瘤活性。
T11178L	ELN318463 racemate ELN318463 (racemate),ELN 318463 racemate	Gamma-secretase	Neuroscience; Proteases/Proteasome; Stem Cells
	ELN318463 racemate (ELN 318463 racemate) 是 ELN318463 的外消旋体，ELN318463 是一种淀粉样前体蛋白 (APP) 选择性 γ-分泌酶抑制剂。
T70407	cemadotin free base LU103793 free base	Microtubule Associated	Cytoskeletal Signaling
	Cemadotin free base(LU103793 free base) 是一种新型的抗限定性肽，是一种新型的抗有丝分裂肽，是Dolastatin 15的类似物。Dolastatin 15是一种天然存在的细胞毒肽，可阻断有丝分裂并抑制微管（管蛋白），Ki 为1μM。Cemadotin 用于研究抗癌。
T50055	Milacemide	MAO	Metabolism; Neuroscience
	Milacemide 是一种甘氨酸前药和 MAO-B 抑制剂。已经研究了米拉塞米对人类记忆的影响以及作为阿尔茨海默病症状的潜在治疗方法。
T3120	K858 (Racemic) K858 Racemic,K858	Apoptosis; Kinesin	Apoptosis; Cytoskeletal Signaling
	K858 Racemic (K858) 是一种选择性有丝分裂驱动蛋白 Eg5 抑制剂，以 ATP 非竞争性方式起作用，IC50值为 1.3 μM。
T20700	Racemetirosine	Others	Others
	Racemetirosine 是一种酪氨酸 3-单加氧酶抑制剂，因此会抑制儿茶酚胺的合成。
T6801	CeMMEC13	Carboxypeptidase; DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Proteases/Proteasome
	CeMMEC13 是一种异喹啉酮，可选择性抑制 TAF1 的第二个溴结构域，IC50为 2.1 μM。
T14864	Caracemide NSC-253272,卡醋胺	Others; DNA/RNA Synthesis; Antibacterial	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
	Caracemide (NSC-253272) 抑制大肠杆菌的核糖核苷酸还原酶。 Caracemide 可用于抗癌研究。
T6809	CPI-169 racemate CPI 169,CPI-169,CPI169	Epigenetic Reader Domain; Histone Methyltransferase	Chromatin/Epigenetic
	CPI-169 racemate (CPI 169) 是CPI-169的消旋体。CPI-169 是一种有效的选择性 EZH2 抑制剂，对 EZH2 WT、EZH2 Y641N 和 EZH1 的 IC50 分别为 0.24、0.51 和 6.1 nM。
T4345	CeMMEC1 CeMMEC1 HCl	Epigenetic Reader Domain; Carboxypeptidase; DNA/RNA Synthesis	Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
	CeMMEC1 是一种 BRD4 抑制剂，对 TAF1 有很好的亲和力，IC50为0.9 μM。
T6425	BTZ043 Racemate BTZ044,BTZ10526038,Benzothiazinone 10526038	Antibacterial; DprE1	Microbiology/Virology; Others
	BTZ043 Racemate (Benzothiazinone 10526038) 是一种癸二烯基磷酰-β-D-核糖 2'-差向异构酶(DprE1) 抑制剂，用作新的抗分枝杆菌剂。
T12215	Nexopamil racemate (Rac)-Nexopamil	Calcium Channel; 5-HT Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Nexopamil racemate（(Rac)-Nexopamil）是 Nexopamil 的外消旋体。Nexopamil racemate 具有潜在的抗哮喘和抗溃疡活性。
T67778	dCeMM1	Molecular Glues	PROTAC
	dCeMM1 是 RBM39 分子胶降解剂，可以降低 WT KBM7 细胞中 RBM39 水平的表达。dCeMM1 活性发挥通过重定向 CRL4DCAF15 连接酶进行。
T10464L	Atuveciclib Racemate BAY-1143572 Racemate,阿维西利	CDK	Cell Cycle/Checkpoint
	Atuveciclib Racemate (BAY-1143572 Racemate) 是 Atuveciclib 的外消旋混合物。 Atuveciclib 是口服有效的 P-TEFb/CDK9高选择性抑制剂，CDK9/CycT1的 IC50为13 nM。
T10591	BPO-27 racemate BPO-27 (racemate)	CFTR; Autophagy	Autophagy; Membrane transporter/Ion channel
	BPO-27 racemate (BPO-27(racemate)) 是一种CFTR 抑制剂，IC50为8 nM。
T2344L	LY 344864 racemate	5-HT Receptor	GPCR/G Protein; Neuroscience
	LY 344864 racemate 是一种 5-HT1F 受体激动剂。
T3534	Tetrabenazine Racemate Nitoman,丁苯那嗪外消旋体,丁苯那嗪,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE	Monoamine Transporter	Membrane transporter/Ion channel
	Tetrabenazine Racemate (Rubigen) 是一种选择性和可逆的囊泡单胺转运蛋白 2(VMAT-2) 抑制剂。它阻断神经递质吸收到肾上腺素能储存囊泡中，并已被用作囊泡运输系统的高亲和力标记。
T7359	CAY10471 Racemate TM30089 Racemate,3-[[(4-氟苯基)磺酰基]甲基氨基]-1,2,3,4-四氢-9H-咔唑-9-乙酸	GPR; Prostaglandin Receptor	Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
	CAY10471 Racemate (TM30089 Racemate) 是一种高选择性的 CRTH2/DP 2 受体拮抗剂，对 hCRTH2 的Ki 值为 0.6 nM，对其选择性远高于人血栓素 A2 受体 TP 或 PGD2 受体 DP。它对大小鼠的同源 CRTH2 也具有拮抗作用。
T3449	Bay 41-4109 racemate	HBV	Microbiology/Virology
	BAY 41-4109 racemate 是BAY 41-4109的消旋体。BAY 41-4109有效抑制人乙型肝炎病毒，IC50值为53 nM。
T7504	Necrostatin 2 racemate 5-[(7-氯-1H-吲哚-3-基)甲基]-3-甲基-2,4-咪唑烷二酮,Necrostatin-2 racemate	RIP kinase	Apoptosis; NF-κB
	Necrostatin 2 racemate (Necrostatin-2 racemate) 是一种特异性的RIPK1抑制剂，是一种稳定型 Nec-1。
T9758	dCeMM3 2-(1H-benzimidazol-2-ylsulfanyl)-N-(5-chloropyridin-2-yl)acetamide	Others	Others
	dCeMM3 (2-(1H-benzimidazol-2-ylsulfanyl)-N-(5-chloropyridin-2-yl)acetamide) 是一种胶降解剂，可以诱导 cyclin K 的泛素化和降解。机制是通过促进 CDK12-cyclin K 与 CRL4B 连接酶复合物的相互作用。
T27143	Delucemine Hydrochloride NPS 1506,Delucemine,Delucemine HCl,NPS1506,NPS-1506	NMDAR	Neuroscience
	Delucemine Hydrochloride (Delucemine) 是一种多胺NMDA受体拮抗剂，可用于研究抑郁症和阿尔茨海默症等神经系统疾病。
T1467	Acemetacin 阿西美辛,K-708,TVX 1322	COX	Immunology/Inflammation; Neuroscience
	Acemetacin (TVX 1322) 是一种非甾体抗炎类的化合物。
T60471	Lanicemine dihydrochloride
	Lanicemine (AZD6765) dihydrochloride 是NMDA 通道的低捕获拮抗剂，Ki 值为 0.56-2.1 μM，在CHO 和爪蟾卵母细胞的IC50分别为 4-7 μM 和 6.4 μM。Lanicemine (AZD6765) dihydrochloride 具有持续的抗抑郁功效。
T10481	BAY 73-6691 racemate	Others	Others
	BAY 73-6691 racemate is a phosphodiesterase 9 inhibitor.
T11859	Litronesib Racemate LY-2523355 Racemate,KF-89617 Racemate	Others	Others
	Litronesib is a selective, allosteric inhibitor of kinesin Eg5.Litronesib (Racemate) is the racemate of litronesib.
T13081	Taranabant racemate MK-0364 racemate	Cannabinoid Receptor	GPCR/G Protein
	Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
T16440	Ibrutinib Racemate PCI-32765 (Racemate)	Others	Others
	Ibrutinib is a selective, irreversible Btk inhibitor (IC50: 0.5 nM). Ibrutinib Racemate is the racemate of Ibrutinib.
T15829	L 888607 Racemate	Aurora Kinase	Cell Cycle/Checkpoint; Chromatin/Epigenetic
	L 888607 Racemate is a selective antagonist of prostaglandin D2 receptor subtype 1 (DP1) (Kis: 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively).
T13700	GDC-0927 Racemate SRN-927 Racemate	Others	Others
	GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.
T23949	Dacemazine hydrochloride Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001
	Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.
T72753	RSV604 racemate A-60444 racemate
	RSV604 (A-60444) racemate 是一种外消旋混合物，与 S-异构体相比，RSV604 racemate 对呼吸道合胞病毒(RSV)菌株的作用效果弱很多。
T13293	Veledimex racemate RG-115932 racemate,INXN-1001 racemate	Others	Others
	Veledimex racemate, the racemic form of veledimex, is an orally available, small-molecule ligand that activates the RheoSwitch Therapeutic System.
T13814	Pemafibrate (racemate) K13675 (racemate)	Others	Others
	Pemafibrate racemate is the racemate of pemafibrate
T62670	Cemdomespib
	Cemdomespib (KU-596) 是一种高效的二代 Hsp90 调节剂。Cemdomespib 能够诱导热休克反应，诱导 Hsp70 水平，具有神经保护作用。Cemdomespib 具有改善糖尿病周围神经病变模型感觉缺陷的疗效。
T12351	p53 and MDM2 proteins-interaction-inhibitor (racemic) p53-and-mdm2-proteins-interaction-inhibitor-racemic	Others	Others
	p53 and MDM2 proteins-interaction-inhibitor (racemic) is an inhibitor of the interaction between p53 and MDM2 proteins.

化合物

Cat.No: T2331

Synonym: 索利霉素,OP-1068,CEM-101

Target: Antibacterial, Antibiotic

Cat.No: T39810

Cat.No: T9104

Target: Apoptosis

2-Fluoroadenine

Cat.No: T20038

Synonym: NSC-27364,NSC 27364,NSC27364,2-氟腺嘌呤

Target: DNA/RNA Synthesis

Zosuquidar trihydrochloride

Cat.No: T6018

Synonym: 唑喹达三盐酸盐,Zosuquidar (LY335979) 3HCl,RS 33295-198 trihydrochloride,RS 33295-198 (D06387) 3HCl,Zosuquidar 3HCl,LY-335979 trihydrochloride

Target: P-gp

Pheniramine maleate

Cat.No: T0370

Synonym: Daneral,Inhiston,Trimetose,马来酸非尼拉敏

Target: 5-HT Receptor, Histamine Receptor

Cat.No: T5858

Synonym: Lu 23-174,舍吲哚

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Autophagy

VPC-80051 racemate

Cat.No: T9005

Target: Others

Peliglitazar racemate

Cat.No: T12400

Synonym: (Rac)-Peliglitazar,(Rac)-BMS 426707-01,BMS 426707-01 racemate

Target: PPAR

Cat.No: T61477

Target: Molecular Glues

MK-4827 Racemate

Cat.No: T22988

Synonym: Niraparib Racemate,2-(4-piperidin-3-ylphenyl)indazole-7-carboxamide

Target: PARP

Rentiapril racemate

Cat.No: T16731

Synonym: (Rac)-SA-446,SA-446 racemate,(Rac)-Rentiapril

Target: Angiotensin-converting Enzyme (ACE)

Cat.No: T76750

Synonym: REGN-2810,SAR-439684

Target: Others

Cat.No: T3562

Synonym: TV1901,N-丙戊酰基甘氨酰胺,N-Valproylglycinamide,丙戊塞胺

Target: Others

AG-120 (racemic)

Cat.No: T22253

Synonym: 1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺

Target: Dehydrogenase

ELN318463 racemate

Cat.No: T11178L

Synonym: ELN318463 (racemate),ELN 318463 racemate

Target: Gamma-secretase

cemadotin free base

Cat.No: T70407

Synonym: LU103793 free base

Target: Microtubule Associated

Cat.No: T50055

Target: MAO

Cat.No: T3120

Synonym: K858 Racemic,K858

Target: Apoptosis, Kinesin

Cat.No: T20700

Target: Others

Cat.No: T6801

Target: Carboxypeptidase, DNA/RNA Synthesis

Cat.No: T14864

Synonym: NSC-253272,卡醋胺

Target: Others, DNA/RNA Synthesis, Antibacterial

CPI-169 racemate

Cat.No: T6809

Synonym: CPI 169,CPI-169,CPI169

Target: Epigenetic Reader Domain, Histone Methyltransferase

Cat.No: T4345

Synonym: CeMMEC1 HCl

Target: Epigenetic Reader Domain, Carboxypeptidase, DNA/RNA Synthesis

BTZ043 Racemate

Cat.No: T6425

Synonym: BTZ044,BTZ10526038,Benzothiazinone 10526038

Target: Antibacterial, DprE1

Nexopamil racemate

Cat.No: T12215

Synonym: (Rac)-Nexopamil

Target: Calcium Channel, 5-HT Receptor

Cat.No: T67778

Target: Molecular Glues

Atuveciclib Racemate

Cat.No: T10464L

Synonym: BAY-1143572 Racemate,阿维西利

Target: CDK

BPO-27 racemate

Cat.No: T10591

Synonym: BPO-27 (racemate)

Target: CFTR, Autophagy

LY 344864 racemate

Cat.No: T2344L

Target: 5-HT Receptor

Tetrabenazine Racemate

Cat.No: T3534

Synonym: Nitoman,丁苯那嗪外消旋体,丁苯那嗪,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE

Target: Monoamine Transporter

CAY10471 Racemate

Cat.No: T7359

Synonym: TM30089 Racemate,3-[[(4-氟苯基)磺酰基]甲基氨基]-1,2,3,4-四氢-9H-咔唑-9-乙酸

Target: GPR, Prostaglandin Receptor

Bay 41-4109 racemate

Cat.No: T3449

Target: HBV

Necrostatin 2 racemate

Cat.No: T7504

Synonym: 5-[(7-氯-1H-吲哚-3-基)甲基]-3-甲基-2,4-咪唑烷二酮,Necrostatin-2 racemate

Target: RIP kinase

Cat.No: T9758

Synonym: 2-(1H-benzimidazol-2-ylsulfanyl)-N-(5-chloropyridin-2-yl)acetamide

Target: Others

Delucemine Hydrochloride

Cat.No: T27143

Synonym: NPS 1506,Delucemine,Delucemine HCl,NPS1506,NPS-1506

Target: NMDAR

Cat.No: T1467

Synonym: 阿西美辛,K-708,TVX 1322

Target: COX

Lanicemine dihydrochloride

Cat.No: T60471

BAY 73-6691 racemate

Cat.No: T10481

Target: Others

Litronesib Racemate

Cat.No: T11859

Synonym: LY-2523355 Racemate,KF-89617 Racemate

Target: Others

Taranabant racemate

Cat.No: T13081

Synonym: MK-0364 racemate

Target: Cannabinoid Receptor

Ibrutinib Racemate

Cat.No: T16440

Synonym: PCI-32765 (Racemate)

Target: Others

L 888607 Racemate

Cat.No: T15829

Target: Aurora Kinase

GDC-0927 Racemate

Cat.No: T13700

Synonym: SRN-927 Racemate

Target: Others

Dacemazine hydrochloride

Cat.No: T23949

Synonym: Ahistan HCl,Dacemazine HCl,Histantine HCl,UNII-DK78VKA001

RSV604 racemate

Cat.No: T72753

Synonym: A-60444 racemate

Veledimex racemate

Cat.No: T13293

Synonym: RG-115932 racemate,INXN-1001 racemate

Target: Others

Pemafibrate (racemate)

Cat.No: T13814

Synonym: K13675 (racemate)

Target: Others

Cat.No: T62670

p53 and MDM2 proteins-interaction-inhibitor (racemic)

Cat.No: T12351

Synonym: p53-and-mdm2-proteins-interaction-inhibitor-racemic

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T7220	Prohydrojasmon racemate Propyl dihydrojasmonate,茉莉酮,Prohydrojasmon	Others	Others
	Prohydrojasmon racemate (Propyl dihydrojasmonate) 是 Prohydrojasmon 的外消旋体。其中Prohydrojasmon 是合成的植物生长调节剂。
T2S1682	Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside	Amylase	Metabolism
	Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside 可抑制 α-淀粉酶活性，IC50值为0.03 umol/ml。
T2992	Pinocembrin 乔松素,5,7-Dihydroxyflavanone,Dihydrochrysin,Galangin flavanone,松属素	NF-κB; Reactive Oxygen Species; Antibacterial; Autophagy	Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
	Pinocembrin (5,7-Dihydroxyflavanone) 是从蜂胶中得到的黄酮类物质，是一种竞争性组氨酸脱羧酶抑制剂，也是抗过敏剂，具有抗氧化、抗菌、抗炎的作用。
TN2078	Pinocembrin chalcone 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone	Calcium Channel; Tyrosinase; Antibacterial; Antifection	Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome
	Pinocembrin chalcone 是一种具有抗诱变作用的酪氨酸酶抑制剂。 Pinocembrin 查尔酮可用于预防胃溃疡的研究。
T19720	Colcemid C 12669,C-12669,NSC-3096,Kolchicin,C12669,Demecolcine	Microtubule Associated	Cytoskeletal Signaling
	Colcemid (NSC-3096) 是一种微管聚合抑制剂，可诱导细胞凋亡，可用于肿瘤和胚胎克隆的研究。
T13514	5-MethoxyPinocembroside	Others	Others
	5-MethoxyPinocembroside 是一种黄酮类天然产物，存在于辣木 Moringa oleifera 的叶子中。
T5710	Pinocembrin-7-O-β-D-glucopyranoside Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷	Others	Others
	Pinocembrin-7-O-β-D-glucopyranoside (Pinocembrin 7-O-beta-D-glucoside) 是黄酮类化合物，能够提高脂质过氧化。
TN1499	Cimiracemoside C 千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Cimicifugoside M	AMPK	Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
	Cimiracemoside C (Cimicifugoside M) 是在升麻中发现的一种天然产物，可激活 AMPK 并具有抗糖尿病的潜在活性。
T5S1677	Cimiracemoside D	Others	Others
	Cimiracemoside D 是一种黑升麻植物提取的天然产物。
TN2077	(+/-)-Pinocembrin NSC 43318,(±)-5,7-Dihydroxyflavanone	GPR; Others	Endocrinology/Hormones; GPCR/G Protein; Others
	(+/-)-Pinocembrin (NSC-43318) 是一种来自腋松的天然产物，它是一种 GPR120 配体，能促进 HaCaT 细胞系的伤口愈合。
TN5509	(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside (2S)-Pinocembrin 7-O-[cinnamoyl(1→5)-β-D-apiosyl(1→2)]-β-D-glucoside
	(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5509，CAS号为 773899-29-9。
TN4792	Pinocembrin diacetate	Others	Others
	Pinocembrin diacetate 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4792，CAS号为 111441-88-4。
T72856	(+)-Cembrene A
	(+)-Cembrene A 是一种α-glucosidase 抑制剂，IC50为 30.31 μM。(+)-Cembrene A 对人正常肝细胞 (LO2) 无毒性。
TN4791	Pinocembrin 7-acetate	Others	Others
	Pinocembrin 7-acetate has antitumor activity.
T83379	2-Hydroxypinocembrin
	2-Hydroxypinocembrin 是一种具有 C-糖基转移酶活性的2-羟基黄烷酮类黄酮底物。
TN4423	Laxiracemosin H	Others	Others
	Laxiracemosin H is a natural product from Dysoxylum lenticellatum.
T72742	(-)-Pinocembrin (-)-乔松素
	(-)-Pinocembrin 对 H37Ra 结核分枝杆菌展示了抗菌活性，无论是休眠还是活跃期，其 IC50 值分别为1.11 mg/mL 和 1.21 mg/mL。作为一种抗增殖剂，(-)-Pinocembrin 对于 THP-1、A549、Panc-1、HeLa 和 MCF7 细胞系，IC50 值范围为 1.88 至 11.00 mg/mL。
T3815	Isoscopoletin 异莨菪亭,7-Methoxyesculetin,6-Hydroxy-7-methoxycoumarin	Others; HBV	Microbiology/Virology; Others
	Isoscopoletin (7-Methoxyesculetin) 是艾叶中的一种活性成分。它具有显著的细胞增殖抑制作用，对人类 CCRF-CEM 白血病细胞和耐药亚系 CEM/ADR5000 作用的 IC50值分别为 4.0 μM 和 1.6 μM。它具有抑制 HBV 复制的活性。
TN6512	Tectol	Transferase; Parasite	Metabolism; Microbiology/Virology
	Tectol 是从Lippia sidoides 中分离的，对人白血病细胞株 HL60 和 CEM 具有显著的抑制作用。它是法尼基转移酶抑制剂，在人和布氏锥虫的IC50分别为 2.09 和 1.73 μM。它具有抗疟原虫活性，是一种中等活性的生长抑制剂，IC50 为 3.44±0.20μM。
TN1674	Garcinone D 伽升沃 D	Reactive Oxygen Species; Nrf2; STAT	Immunology/Inflammation; JAK/STAT signaling; Metabolism; NF-κB; Stem Cells
	Garcinone D 是来自山竹的一种呫吨酮，可促进 C17.2 神经干细胞的增殖。它以浓度和时间依赖的方式增加磷酸化信号转导和转录激活因子 3 (p-STAT3)、Cyclin D1 和核因子红细胞 2 相关因子 (Nrf2)、以及血红素加氧酶-1 (HO-1) 的蛋白质水平。
TN4492	Mangostanol	AChR	Neuroscience
	Mangostanol is an acetylcholinesterase (AChE) selective inhibitor.Mangostanol has anti-cancer activity, it shows significant activities against the CEM-SS cell line, with IC50 values of 9.6 microg/ml.
TN3968	Epifriedelanol acetate	Others	Others
	Epifriedelanol exhibits antibacterial activities. It also can reduce cellular senescence in human primary cells and may be used to develop dietary supplements or cosmetics that modulate tissue aging or aging-associated diseases. Epifriedelanol and friedel
TN3438	Arborinine	HCV Protease; Antifection	Microbiology/Virology; Proteases/Proteasome
	Arborinine shows mild in vitro antibacterial activity, it possesses moderate levels of anti-hepatitis C virus(HCV) activities with the IC50 values being 6.4 ± 0.7 ug/ml. Arborinine shows antifeedant activity against Spodoptera frugiperda. Arborinin shows

天然产物

Prohydrojasmon racemate

Cat.No: T7220

Synonym: Propyl dihydrojasmonate,茉莉酮,Prohydrojasmon

Target: Others

Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside

Cat.No: T2S1682

Synonym: Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside

Target: Amylase

Cat.No: T2992

Synonym: 乔松素,5,7-Dihydroxyflavanone,Dihydrochrysin,Galangin flavanone,松属素

Target: NF-κB, Reactive Oxygen Species, Antibacterial, Autophagy

Pinocembrin chalcone

Cat.No: TN2078

Synonym: 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone

Target: Calcium Channel, Tyrosinase, Antibacterial, Antifection

Cat.No: T19720

Synonym: C 12669,C-12669,NSC-3096,Kolchicin,C12669,Demecolcine

Target: Microtubule Associated

5-MethoxyPinocembroside

Cat.No: T13514

Target: Others

Pinocembrin-7-O-β-D-glucopyranoside

Cat.No: T5710

Synonym: Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷

Target: Others

Cimiracemoside C

Cat.No: TN1499

Synonym: 千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Cimicifugoside M

Target: AMPK

Cimiracemoside D

Cat.No: T5S1677

Target: Others

(+/-)-Pinocembrin

Cat.No: TN2077

Synonym: NSC 43318,(±)-5,7-Dihydroxyflavanone

Target: GPR, Others

(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside

Cat.No: TN5509

Synonym: (2S)-Pinocembrin 7-O-[cinnamoyl(1→5)-β-D-apiosyl(1→2)]-β-D-glucoside

Pinocembrin diacetate

Cat.No: TN4792

Target: Others

(+)-Cembrene A

Cat.No: T72856

Pinocembrin 7-acetate

Cat.No: TN4791

Target: Others

2-Hydroxypinocembrin

Cat.No: T83379

Laxiracemosin H

Cat.No: TN4423

Target: Others

(-)-Pinocembrin

Cat.No: T72742

Synonym: (-)-乔松素

Cat.No: T3815

Synonym: 异莨菪亭,7-Methoxyesculetin,6-Hydroxy-7-methoxycoumarin

Target: Others, HBV

Cat.No: TN6512

Target: Transferase, Parasite

Cat.No: TN1674

Synonym: 伽升沃 D

Target: Reactive Oxygen Species, Nrf2, STAT

Cat.No: TN4492

Target: AChR

Epifriedelanol acetate

Cat.No: TN3968

Target: Others

Cat.No: TN3438

Target: HCV Protease, Antifection

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