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231

抑制剂 & 化合物

52

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1216 CaM kinase II inhibitor TFA salt

Autocamtide-2-related inhibitory peptide (TFA)

CaMK Neuroscience
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide(TFA)) 是一种高度特异性和有效的 CaMKII 抑制剂,IC50 为 40 nM。
T76690 Mavrilimumab

CAM 3001

Virus Protease; CSF-1R Microbiology/Virology; Tyrosine Kinase/Adaptors
Mavrilimumab (CAM 3001) 是一种单克隆抗体,具有抗病毒活性,对粒细胞-巨噬细胞集落刺激因子 (GM-CSF) 受体的 α 亚基有亲和力,并阻止 GM-CSF 下游细胞内信号传导。GM-CSF 可能与呼吸衰竭和死亡相关的过度活跃炎症反应有关,可用于研究类风湿性关节炎。
T41211 CAM 833

CAM 833 是一种有效的正位抑制剂,对 BRCA2 和 RAD51 之间相互作用具有抑制作用,对 ChimRAD51 蛋白的 Kd 为 366 nM。 CAM833 抑制 RAD51 的寡聚,促进 G2/M 阻滞细胞的凋亡 (apoptosis) 进程。
T70136 CAM 4750

CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist.
T70137 CAM 4515

CAM 4515 is a nonpeptide tachykinin NK1 receptor antagonist.
T70410 Cam 2445

Cam 2445 is a nonpeptide, alpha-methyltryptophan derivative; an NK1 neurokinin receptor antagonist that is a potentially useful treatment for arthritis, asthma, migraine, anxiety, psychosis, and emesis.
T28331 PD 136450

Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189

Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to elucidate the physiological role o
T70211 CAM741

CAM741 is a novel selective inhibitor of vascular cell adhesion molecule 1 (VCAM1) synthesis in endothelial cells, blocking the process of cotranslational translocation, which is dependent on the signal peptide of VCAM1.
T30442 Bialamicol Hydrochloride

Camoform hydrochloride,CAM 807,CAM-807,CI 301

Bialomicol Hydrochloride is a bio-active chemical.
T41184 Clocinnamox mesylate

C-CAM,NIH 10443

Clocinnamox mesylate is a systemically active, irreversibleμ-opioid receptor antagonist (apparent Kivalues are 0.7, 1.9 and 5.7 nM for mouseμ,δandκreceptors respectively).
T69909 CAM4066

CAM4066 is a novel potent and selective CK2alpha inhibitor.
T16366 NVR 3-778

HBV Microbiology/Virology
NVR 3-778 是一种 SBA 类的口服有效HBV CAM 衣壳组装调制剂,具有抗 HBV 活性。
T69908 Pidnarulex HCl

Pidnarulex HCl is the salt form of CX-5461, a first-in-class non-genotoxic small molecule targeted inhibitor of RNA polymerase I (Pol I) that activates the p53 pathway without causing DNA damage. CX-5461 selectively inhibits rRNA synthesis by Pol I in the nucleolus, but does not inhibit mRNA synthesis by RNA Polymerase II (Pol II) and does not inhibit DNA replication or protein synthesis. Inhibition of Pol I results in nucleolar stress and release of ribosomal proteins (RP) from the nucleolus. T...
T70210 FT-1101 free base

FT-1101 is an orally bioavailable, potent and selective BET inhibitor. FT-1101 binds to the acetylated lysine recognition motifs in the bromodomain sites of BET proteins, thereby preventing the interaction between the BET proteins and acetylated histones. This disrupts chromatin remodeling and gene expression. Prevention of the expression of certain growth-promoting genes may lead to the inhibition of tumor cell growth. BET proteins, comprised of BRD2, BRD3, BRD4 and BRDT, are transcriptional r...
T23525 W-9 hydrochloride

N-(6-aminohexyl)-5-chloronaphthalene-2-sulfonamide hydrochloride

CaMK Neuroscience
W-9 hydrochloride 是一种钙调蛋白拮抗剂。
T70135 Nepaprazole sodium dihydrate

Nepaprazole sodium dihydrate is a proton pump inhibitor potentially for treatment of gastric ulcers.
T70409 6alpha-Fluorotestosterone

6alpha-Fluorotestosterone is a synthetic nonaromatizable androgen analog of testosterone. It binds to and activates specific nuclear receptors inhibits and is equipotent to testosterone.
T63717 CAM833

CAM833 是有效的抑制 BRCA2 和 RAD51 之间相互作用的正位抑制剂,也能够抑制 RAD51 的寡聚,能够作用于 ChimRAD51 蛋白 (Kd: 366 nM)。
T20792 W-7 hydrochloride

N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W 7 HCl,W7 HCl,W-7 HCl

CaMK; Apoptosis; Myosin; PDE Apoptosis; Cytoskeletal Signaling; Metabolism; Neuroscience
W-7 hydrochloride (W-7 HCl) 是一种选择性的钙调蛋白拮抗剂。它抑制Ca2+-钙调蛋白依赖性磷酸二酯酶和肌球蛋白轻链激酶,IC50值分别为 28 μM 和 51 μM。它可诱导细胞凋亡,具有抗癌活性。
TP1921L1 Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)

CaMK; Autophagy Autophagy; Neuroscience
Autocamtide-2-related inhibitory peptide, myristoylated acetate 是CaM 激酶II 抑制剂;是 Autocamtide-2相关抑制肽的增强细胞渗透性衍生物。
T1586 Tenoxicam

Ro-12-0068,替诺昔康,Tenoxicamum,Mobiflex,Tilcotil

COX Immunology/Inflammation; Neuroscience
Tenoxicam (Tilcotil) 是一种抗炎化合物,具有退热止痛作用。
T35033L (S)-Vamicamide

(S)-Vamicamide (Iso-132373-81-0)

AChE Neuroscience
(S)-Vamicamide 是一种新型抗抗胆碱能化合物。Vamicamide 在 32 mg/kg 或更高 (p.o.) 时增加小鼠的自发运动活动,并在 100 mg/kg 时抑制小鼠强直性惊厥。
TP2310 Autocamtide-2-related inhibitory peptide

CaMK; Autophagy Autophagy; Neuroscience
Autocamtide-2-related inhibitory peptide 是一种高度特异性和有效的 CaMKII 抑制剂,IC50 为 40 nM。
TP2057L Camstatin acetate

NO Synthase Immunology/Inflammation
Camstatin acetate 结合钙调蛋白并抑制神经元一氧化氮合酶。它是 PEP-19 的单一钙调蛋白结合 IQ 基序的具有功能活性的 25 个残基片段。
T9048 Ecamsule

Others Others
Ecamsule 是一种亚苄基樟脑衍生物,其中许多以其出色的光稳定性而闻名。 可添加到防晒霜中以过滤掉 UVA 射线。
T11237 Camizestrant

Estrogen receptor antagonist 2

Estrogen Receptor/ERR Endocrinology/Hormones
Camizestrant (Estrogen receptor antagonist 2) 是一种雌激素受体拮抗剂,可用于 ER+ HER2 晚期乳腺癌的研究[1]。
T35033 Vamicamide

FK 176,FK-176,FK176

AChE Neuroscience
Vamicamide (FK 176)是一种新型抗胆碱能化合物。Vamicamide 在 32 mg/kg (p.o.)或更高时增加小鼠的自发运动活动,并在 100 mg/kg 时抑制小鼠强直性惊厥。
T15050 Danicamtiv

MYK-491,SAR 440181

Myosin Cytoskeletal Signaling
Danicamtiv (MYK-491) 是一种正性肌力药物,也是一种心肌肌球蛋白的选择性变构激活剂,可增加心脏收缩功能并保持机械效率。
T0818 Decamethonium bromide

十烃溴铵,Decacuran,溴化十烃季胺,Syncurine

AChR; AChE Neuroscience
Decamethonium bromide (Syncurine) 是神经肌肉阻滞剂和烟碱型 AChR 部分激动剂。
T18990 Fluorescamine

荧光胺,Ro 20-7234

Others Others
Fluorescamine (Ro 20-7234) 是一种螺环化合物,其本身无荧光性质,但与初级胺反应后可形成荧光,因此可用于胺和肽的检测。
T2159 CaMKP Inhibitor

CaMK Neuroscience
CaMKP Inhibitor 可以抑制 CaMKP。
T67795 Camonagrel

Camonagrel 是一种化合物,对Prostaglandin E2具有抑制作用。
T9258 Aficamten

Others Others
Aficamten 是一种可研究肥厚型心肌病的新型心肌肌球蛋白抑制剂,IC50为 1.4 μM。
T16807 Rucaparib monocamsylate

瑞卡帕布樟脑磺酸盐,Rucaparib Camsylate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Rucaparib monocamsylate (Rucaparib Camsylate) 是一种口服有效的 PARP 蛋白抑制剂,对 PARP-1 的Ki 为 1.4 nM。它是六磷酸己糖脱氢酶 (H6PD) 抑制剂,有用于去势抵抗性前列腺癌 (CRPC) 的研究潜力。
T4111 Blarcamesine hydrochloride

Anavex 2-73,AVex-73 hydrochloride,AE-37 hydrochloride

Sigma receptor GPCR/G Protein
Blarcamesine hydrochloride (AVex-73 hydrochloride) 是一个sigma-1受体激动剂,IC50值为 860 nM。
T38845 Dodecamethylpentasiloxane

Parasite Microbiology/Virology
Dodecamethylpentasiloxane 可用作臭虫杀虫剂。 Dodecamethylpentasiloxane 是硅氧烷的一种成分,可用作硅油。
T20713 Flonicamid

UNII-9500W2Z53J,N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide

Others Others
Flonicamid (N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide) 是一种吡啶甲酰胺杀虫剂,在食用日本萝卜叶的过程中抑制蚜虫(M.persicae)的唾液分泌和汁液摄入。它对棉蚜、红蚜、巴迪蚜、禾谷蚜和大鼠产生毒性。
T2391 Camostat mesylate

FOY-S980,甲磺酸卡莫司他,FOY305,Camostat mesilate

Serine/threonin kinase; SARS-CoV; Sodium Channel Cell Cycle/Checkpoint; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Camostat mesylate (FOY-S980) 是口服活性合成的丝氨酸蛋白酶抑制剂,用于慢性胰腺炎。它是TMPRSS2的抑制剂,对SARS-CoV-2具有抗病毒活性。它抑制前列腺素、胰蛋白酶和苦参多糖的活性。
T62083 Camonsertib

ATR inhibitor 4,RP-3500

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Camonsertib (RP-3500) 是一种选择性的、口服具有活力的 ATR 激酶抑制剂 (ATRi),在生化试验中的 IC50: 1.00 nM,表现出有效的抗肿瘤作用。RP-3500 对 ATR 的选择性是 mTOR 的 30 倍 (IC50: 120 nM),是 ATM、DNA-PK 和 PI3Kα 激酶的 2,000 倍以上。
T13147 ICAM-1-IN-1

Integrin Cytoskeletal Signaling
ICAM-1-IN-1 是选择性的 ICAM-1和 E-selectin 抑制剂,IC50值分别为5和7 nM。
T7465 4-Methylbenzylidene camphor

Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC

AChE Neuroscience
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。
T37535 Camrelizumab

SHR-1210

Camrelizumab (SHR-1210) 是一种具有高亲和力且针对 PD-1的人源 IgG4-κ单克隆抗体。Camrelizumab 与 PD-1 的结合亲和力高达 3 nM,对 PD-1/PD-L1具有抑制作用, IC50 为 0.70 nM。Camrelizumab 具有抗肿瘤活性和耐受性,可用于研究包括 NSC-LC、ESCC、霍奇金淋巴瘤和晚期 HCC 等的癌症。
TP1217L Autocamtide 2 TFA(129198-88-5 free base)

CaMK Neuroscience
Autocamtide 2 TFA(129198-88-5 free base) 是钙/钙调蛋白依赖性蛋白激酶 II (CaMKII) 的高选择性肽底物。 Autocamtide 2 TFA 可用于 CaMKII 活性测定。
T2006 Omecamtiv mecarbil

CK-1827452

ATPase; Myosin Cytoskeletal Signaling; Membrane transporter/Ion channel
Omecamtiv mecarbil (CK-1827452) 是一种心脏特异性的肌球蛋白激活剂,用于研究心脏相关疾病。
T20856 Dicamba

Dianat,麦草畏,Mediben,Banlen,Banvel

Others Others
Dicamba (Banvel) 是一种氯化有机除草剂。 Dicamba 可用于防治阔叶杂草。
T1673 Acamprosate calcium

calcium acetylhomotaurinate,N-Acetylhomotaurine Calcium,Alcomed,阿坎酸钙,Sobriol,Campral EC,Calcium N-acetylhomotaurinate

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Acamprosate calcium (Campral EC) 是 GABA 受体激动剂和谷氨酸能系统调节剂,用于治疗酒精依赖。
T11508L Camicinal hydrochloride

GSK962040 hydrochloride

Others; Motilin Receptor GPCR/G Protein; Others
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。
T27209 Droxicam

Droxicamum,屈昔康

Others Others
Droxicam (Droxicamum) 是一种非甾体抗炎化合物,可用于缓解肌肉骨骼疾病的炎症和疼痛的研究。
T7780 Blarcamesine

AE-37,AVex-73

AChR Neuroscience
Blarcamesine (AVex-73) 是一种毒蕈碱 M1 激动剂,具有抗惊厥、抗失忆、神经保护和抗抑郁的特性,可能用于治疗阿尔茨海默病。
T73718 N-methyl-N-dithiocarboxyglucamine sodium

N-methyl-N-dithiocarboxyglucamine (MDCG) sodium 在小鼠模型中动员并促进金属硫蛋白结合109Cd的排泄,显著降低肝脏和肾脏中的镉含量。肝脏和肾脏为镉诱导毒性影响的主要易感器官。

化合物

CaM kinase II inhibitor TFA salt
Cat.No: TP1216
Synonym: Autocamtide-2-related inhibitory peptide (TFA)
Target: CaMK
Mavrilimumab
Cat.No: T76690
Synonym: CAM 3001
Target: Virus Protease, CSF-1R
CAM 833
Cat.No: T41211
Synonym:
Target:
CAM 4750
Cat.No: T70136
Synonym:
Target:
CAM 4515
Cat.No: T70137
Synonym:
Target:
Cam 2445
Cat.No: T70410
Synonym:
Target:
PD 136450
Cat.No: T28331
Synonym: Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
Target:
CAM741
Cat.No: T70211
Synonym:
Target:
Bialamicol Hydrochloride
Cat.No: T30442
Synonym: Camoform hydrochloride,CAM 807,CAM-807,CI 301
Target:
Clocinnamox mesylate
Cat.No: T41184
Synonym: C-CAM,NIH 10443
Target:
CAM4066
Cat.No: T69909
Synonym:
Target:
NVR 3-778
Cat.No: T16366
Synonym:
Target: HBV
Pidnarulex HCl
Cat.No: T69908
Synonym:
Target:
FT-1101 free base
Cat.No: T70210
Synonym:
Target:
W-9 hydrochloride
Cat.No: T23525
Synonym: N-(6-aminohexyl)-5-chloronaphthalene-2-sulfonamide hydrochloride
Target: CaMK
Nepaprazole sodium dihydrate
Cat.No: T70135
Synonym:
Target:
6alpha-Fluorotestosterone
Cat.No: T70409
Synonym:
Target:
CAM833
Cat.No: T63717
Synonym:
Target:
W-7 hydrochloride
Cat.No: T20792
Synonym: N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W 7 HCl,W7 HCl,W-7 HCl
Target: CaMK, Apoptosis, Myosin, PDE
Autocamtide-2-related inhibitory peptide, myristoylated acetate(201422-04-0 free base)
Cat.No: TP1921L1
Synonym:
Target: CaMK, Autophagy
Tenoxicam
Cat.No: T1586
Synonym: Ro-12-0068,替诺昔康,Tenoxicamum,Mobiflex,Tilcotil
Target: COX
(S)-Vamicamide
Cat.No: T35033L
Synonym: (S)-Vamicamide (Iso-132373-81-0)
Target: AChE
Autocamtide-2-related inhibitory peptide
Cat.No: TP2310
Synonym:
Target: CaMK, Autophagy
Camstatin acetate
Cat.No: TP2057L
Synonym:
Target: NO Synthase
Ecamsule
Cat.No: T9048
Synonym:
Target: Others
Camizestrant
Cat.No: T11237
Synonym: Estrogen receptor antagonist 2
Target: Estrogen Receptor/ERR
Vamicamide
Cat.No: T35033
Synonym: FK 176,FK-176,FK176
Target: AChE
Danicamtiv
Cat.No: T15050
Synonym: MYK-491,SAR 440181
Target: Myosin
Decamethonium bromide
Cat.No: T0818
Synonym: 十烃溴铵,Decacuran,溴化十烃季胺,Syncurine
Target: AChR, AChE
Fluorescamine
Cat.No: T18990
Synonym: 荧光胺,Ro 20-7234
Target: Others
CaMKP Inhibitor
Cat.No: T2159
Synonym:
Target: CaMK
Camonagrel
Cat.No: T67795
Synonym:
Target:
Aficamten
Cat.No: T9258
Synonym:
Target: Others
Rucaparib monocamsylate
Cat.No: T16807
Synonym: 瑞卡帕布樟脑磺酸盐,Rucaparib Camsylate
Target: PARP
Blarcamesine hydrochloride
Cat.No: T4111
Synonym: Anavex 2-73,AVex-73 hydrochloride,AE-37 hydrochloride
Target: Sigma receptor
Dodecamethylpentasiloxane
Cat.No: T38845
Synonym:
Target: Parasite
Flonicamid
Cat.No: T20713
Synonym: UNII-9500W2Z53J,N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide
Target: Others
Camostat mesylate
Cat.No: T2391
Synonym: FOY-S980,甲磺酸卡莫司他,FOY305,Camostat mesilate
Target: Serine/threonin kinase, SARS-CoV, Sodium Channel
Camonsertib
Cat.No: T62083
Synonym: ATR inhibitor 4,RP-3500
Target: ATM/ATR
ICAM-1-IN-1
Cat.No: T13147
Synonym:
Target: Integrin
4-Methylbenzylidene camphor
Cat.No: T7465
Synonym: Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC
Target: AChE
Camrelizumab
Cat.No: T37535
Synonym: SHR-1210
Target:
Autocamtide 2 TFA(129198-88-5 free base)
Cat.No: TP1217L
Synonym:
Target: CaMK
Omecamtiv mecarbil
Cat.No: T2006
Synonym: CK-1827452
Target: ATPase, Myosin
Dicamba
Cat.No: T20856
Synonym: Dianat,麦草畏,Mediben,Banlen,Banvel
Target: Others
Acamprosate calcium
Cat.No: T1673
Synonym: calcium acetylhomotaurinate,N-Acetylhomotaurine Calcium,Alcomed,阿坎酸钙,Sobriol,Campral EC,Calcium N-acetylhomotaurinate
Target: GABA Receptor
Camicinal hydrochloride
Cat.No: T11508L
Synonym: GSK962040 hydrochloride
Target: Others, Motilin Receptor
Droxicam
Cat.No: T27209
Synonym: Droxicamum,屈昔康
Target: Others
Blarcamesine
Cat.No: T7780
Synonym: AE-37,AVex-73
Target: AChR
N-methyl-N-dithiocarboxyglucamine sodium
Cat.No: T73718
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1008 Psoralenoside

CaMK; Calcium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T8846 beta-Escin

B-escin,AESCINE,beta-七叶素

Immunology/Inflammation related Immunology/Inflammation
beta-Escin 是七叶树种子的主要活性成分。它可抑制碱性成纤维细胞生长因子所诱导的增殖、迁移、管形成以及体内 CAM 血管生成。它具有研究抗血管生成作用的分子机制的潜力。
TMS2262 (-)-CAMPHOR

L-Camphor,左旋樟脑

Others Others
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。
T5S1952 9-Methoxycamptothecin

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
9-Methoxycamptothecin 是从臭味假柴龙树中分离得到的一种天然产物,通过抑制拓扑异构酶起到抗肿瘤作用,具有强效的诱导 G2/M 期细胞和癌细胞凋亡的作用。
T2764 (S)-10-Hydroxycamptothecin

10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。
T4S2157 Campesterol

菜油甾醇,(24R)-5-Ergosten-3β-ol

Endogenous Metabolite Metabolism
Campesterol ((24R)-5-Ergosten-3β-ol) 是一种植物甾醇,具有降胆固醇和抗癌的活性。
T1123 Camptothecin

NSC-100880,Campathecin,喜树碱,(S)-(+)-Camptothecin,CPT

Apoptosis; Influenza Virus; Topoisomerase; Antibiotic; Antifungal Apoptosis; DNA Damage/DNA Repair; Microbiology/Virology
Camptothecin (CPT) 属于生物碱类天然产物,是一种 DNA 拓扑异构酶 I (Topo I) 的抑制剂 (IC50=679 nM),具有特异性。Camptothecin 具有抗肿瘤活性,可以诱导细胞凋亡。
T5037 Midecamycin

Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A

Antibacterial; Antibiotic Microbiology/Virology
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。
T3S1955 7-Ethylcamptothecin

Others Others
7-Ethylcamptothecin 是一种喜树碱类似物。其中喜树碱是一种细胞毒性生物碱,从喜树中分离出得到,对 L1210 白血病和 Walker 256 癌肉瘤模型具有很强的抗肿瘤活性。
T4S1951 10-Methoxycamptothecin

Others Others
10-Methoxycamptothecin 是分离自喜树的喜树碱衍生物,具有高抗癌特性。通过对 2774 细胞系的抗肿瘤活性测定,发现它比 10-羟基喜树碱的细胞毒性更高。
T17143 Toyocamycin

丰加霉素,Vengicide

Apoptosis; Others; IRE1; Antibiotic; Antifungal Apoptosis; Cell Cycle/Checkpoint; Microbiology/Virology; Others
Toyocamycin (Vengicide) 是放线菌类产生的腺苷类似物,为 X 盒结合蛋白 1 (XBP1) 抑制剂,抑制 IRE1α 诱导的 ATP 依赖性 XBP1 mRNA 的断裂,IC50值为 80 nM。它还诱导凋亡。
T14329 Ascamycin

Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。
T3853 Camelliaside B

山茶苷 B,山茶甙B

Others Others
Camelliaside B 是一种类黄酮,来自于油茶种子残渣的甲醇提取物。
T1468 Lornoxicam

Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康

COX; Endogenous Metabolite Immunology/Inflammation; Metabolism; Neuroscience
Lornoxicam (Chlortenoxicam) 是一种新型非甾体抗炎药,是高活性 COX-1 和 COX-2 抑制剂,IC50 分别为 5 和 8 nM。
T20191 (-)-Camphoric acid

(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

GluR Neuroscience
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。
T67867 Mycaminosyltylonolide

Antibacterial Microbiology/Virology
Mycaminosyltylonolide 是一种大环内酯类抗生素,它是 tyololide 在位置5上具有β - d -mycaminosyl 残基。Mycaminosyltylonolide 是一种有效的抗生素,具有抗菌活性和抑制荧光素酶的合成。
T7959 (+)-ISOPINOCAMPHEOL

Others Others
(+)-ISOPINOCAMPHEOL 是一种天然产物。
T10668 Camalexin

Reactive Oxygen Species; ROS; Antibacterial; Antifungal Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Camalexin 是从Camelina sativa 和Arabidopsis 中分离出来的一种植物抗毒素,可诱导活性氧的产生,具有抗菌、抗真菌、抗增殖和抗癌活性。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T40179 Sodium Camptothecin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Sodium Camptothecin 是一种植物生物碱,具有抗肿瘤活性。它是可逆 RNA 合成抑制剂,可以抑制腺病毒的复制。它能抑制 DNA 合成,并引起细胞内预形成的病毒 DNA 断裂。
T0882 (+)-Camphor

D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor

Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。
T3854 Camelliaside A

山茶苷 A,山茶甙A

Others Others
Camelliaside A 是一种的类黄酮化合物,来源于油茶种子残渣的甲醇提取物中。
T2952 Camphor

樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa

Influenza Virus; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。
T2S0271 Voacamine

老刺木胺,Voacanginine

Cannabinoid Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Voacamine (Voacanginine) 是非洲马铃果中的一种吲哚生物碱,可抑制多药耐药肿瘤细胞中的 P-糖蛋白作用,具有强效的大麻素 CB1受体拮抗活性。
T1286 Vincamine

Angiopac,Oxybral,Devincan,Novicet,Equipur,长春胺,Perval

GPR; Others Endocrinology/Hormones; GPCR/G Protein; Others
Vincamine (Perval) 是从长春花中提取的单萜类吲哚生物碱,可作为外周血管扩张剂,对脑微血管循环有选择性的血管调节作用。它可改善体内葡萄糖稳态,对 2 型糖尿病具有研究潜力。它是GPR40激动剂,通过改善 β 细胞功能障碍和促进葡萄糖刺激型胰岛素分泌发挥 β 细胞保护作用。
T82786 Campneoside II

Campneoside II, 分离自毛泡桐,展现出显著的抗补体活性。
TN4025 Eucamalduside A

Others Others
Eucamalduside A is a natural product from Eucalyptus camaldulensis var. obtusa.
T4952 9-Hydroxycamptothecin

9-HCPT,9-羟基喜树碱,10-Hydroxycampothecin

Topoisomerase DNA Damage/DNA Repair
9-Hydroxycampothecin 是具有抗癌活性的喜树碱衍生物。
T82002 Juniper camphor

Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。
TN3573 Camaric acid

Antifection Microbiology/Virology
Camaric acid shows antibacterial activity against Staphylococcus aureus and methicillin resistant S. aureus with IC50 values 8.74 and 8.09 uM, respectively, it also shows moderate antileishmanial activity and highly potent antitrypanosomal activity. Camar
T1521 (±)-10-Hydroxycamptothecin

Hydroxy Camptothecine,10-羟基喜树碱,10-Hydroxycamptothecin

Topoisomerase DNA Damage/DNA Repair
(±)-10-Hydroxycamptothecin (Hydroxy Camptothecine) 是一种从喜树茎木中分离出来的生物碱,抑制拓扑异构酶 I 活性,具有广谱抗肿瘤活性。
TN2620 14,15-Didehydrovincamenine

Others Others
14,15-Didehydrovincamenine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2620,CAS号为 112219-48-4。
T21098 Decamethylcyclopentasiloxane

Dekamethylcyklopentasiloxan,Cyclopentasiloxane, decamethyl-

Decamethylcyclopentasiloxane is a cyclic methylsiloxane with volatile properties.
TN5954 Camaldulenic acid

Camaldulenic acid是一种天然产物,属于唇形科鼠尾草属,其产品编号为 TN5954,CAS号为 71850-15-2。Camaldulenic acid可用作对照参考。
TN5830 Campsiketalin

Rengyoxide dimethyl ketal

Campsiketalin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5830,CAS号为 93675-96-8。
TN4471 Lysicamine

IL Receptor; Antifection Immunology/Inflammation; Microbiology/Virology
Lysicamine shows significant antioxidant capacity in the ORAC(FL) assay and it is active against S. epidermidis and C. dubliniensis, with MIC values in the range 12.5-100 microg mL(-1). Lysicamine has antimicrobial and anti-inflammation activity, the mini
T21047 Apovincamine

cis-Apovincamine

Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity.
TN1464 Camellianin A

RAAS Endocrinology/Hormones
Camellianin A has anticancer activity, it can inhibit the proliferation of the human hepatocellular liver carcinoma Hep G2 and human breast adenocarcinoma MCF-7 cell lines in a dose-dependent manner and induce the significant increase of the G0/G1 cell po
TN1176 10-Nitro-camptothecin

9-硝基喜树碱

Others Others
10-Nitro-camptothecin is a natural product
T38481 Camellianin B

Camellianin B, a flavonoid compound and metabolite of Camellianin A, exhibits antioxidant properties and acts as an angiotensin converting enzyme (ACE) inhibitor.
TN2681 Elasticamide

2-(2'-Hydroxytetracosanoylamino)-octadecane-1,3,4-triol

Others Others
(2S,3S,4R,2'R)-2-(2'-hydroxytetracosanoylamino)octadecane-1,3,4-triol shows selectively inhibitory activity against phospholipase A 2 (PLA 2) secreted from Crotalus adamenteus venom at concentration of 100 ug/mL.
TN4667 Norcamphor

Others Others
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。
T16726 Rebeccamycin

Topoisomerase DNA Damage/DNA Repair
Rebeccamycin is an antitumor antibiotic+ inhibits DNA topoisomerase I. Rebeccamycin appears to exert its primary antineoplastic effect by poisoning topoisomerase I. It also has a negligible effect on protein kinase C and topoisomerase II.
T31651 Epicoccamide

Epicoccamide is a marine fungal metabolite originally isolated from E. purpurascens.
TN2642 16,17-Dihydroapovincamine

Others Others
16,17-Dihydroapovincamine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2642,CAS号为 57130-30-0。
TN4026 Eucamalol

Others Others
Eucamolol exhibits significant repellent activity against Aedes albopictus, and inhibits its feeding as well as DEET, is effective repellent (75%) up to 3 h after exposure to mosquito.
T83520 (S)-Campesterol

5-Ergosten-3β-ol

(S)-Campesterol (5-Ergosten-3β-ol),一种植物甾醇,存在于多种食物和植物源中,对人体健康具有潜在益处。
TN2460 12-Ethyl-9-hydroxycamptothecin

7-乙基-10-羟基喜树碱,7-Ethyl-10-Hydroxy-Camptothecin

Others Others
12-Ethyl-9-hydroxycamptothecin 是一种 Camptothecin 的衍生物。其中Camptothecin (CPT) 是一种生物碱,也是 DNA 拓扑异构酶I 抑制剂(IC50:679 nM)。
T38299 Tunicamycin V

Tunicamycin 15:1 is a mixture of tunicamycin structural isomers that contains a 15-carbon N-acyl chain with variable branching patterns.References Tunicamycin 15:1 is a mixture of tunicamycin structural isomers that contains a 15-carbon N-acyl chain with variable branching patterns. References
T74198 Beauverolide Ja

Beauverolide Ja 是一种环四缩酚肽,是一种有效的钙调蛋白 (CaM) 抑制剂,对 Ca2+-CaM 的Kd 为 0.078 μM,Ki 为 0.39 μM。Beauverolide Ja 是Isaria fumosorosea 的次级代谢产物。
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天然产物

Psoralenoside
Cat.No: TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
beta-Escin
Cat.No: T8846
Synonym: B-escin,AESCINE,beta-七叶素
Target: Immunology/Inflammation related
(-)-CAMPHOR
Cat.No: TMS2262
Synonym: L-Camphor,左旋樟脑
Target: Others
9-Methoxycamptothecin
Cat.No: T5S1952
Synonym:
Target: Apoptosis, Topoisomerase
(S)-10-Hydroxycamptothecin
Cat.No: T2764
Synonym: 10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT
Target: Apoptosis, Topoisomerase
Campesterol
Cat.No: T4S2157
Synonym: 菜油甾醇,(24R)-5-Ergosten-3β-ol
Target: Endogenous Metabolite
Camptothecin
Cat.No: T1123
Synonym: NSC-100880,Campathecin,喜树碱,(S)-(+)-Camptothecin,CPT
Target: Apoptosis, Influenza Virus, Topoisomerase, Antibiotic, Antifungal
Midecamycin
Cat.No: T5037
Synonym: Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A
Target: Antibacterial, Antibiotic
7-Ethylcamptothecin
Cat.No: T3S1955
Synonym:
Target: Others
10-Methoxycamptothecin
Cat.No: T4S1951
Synonym:
Target: Others
Toyocamycin
Cat.No: T17143
Synonym: 丰加霉素,Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
Ascamycin
Cat.No: T14329
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Antibacterial, Antibiotic
Camelliaside B
Cat.No: T3853
Synonym: 山茶苷 B,山茶甙B
Target: Others
Lornoxicam
Cat.No: T1468
Synonym: Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康
Target: COX, Endogenous Metabolite
(-)-Camphoric acid
Cat.No: T20191
Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-
Target: GluR
Mycaminosyltylonolide
Cat.No: T67867
Synonym:
Target: Antibacterial
(+)-ISOPINOCAMPHEOL
Cat.No: T7959
Synonym:
Target: Others
Camalexin
Cat.No: T10668
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antifungal
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Sodium Camptothecin
Cat.No: T40179
Synonym:
Target: DNA/RNA Synthesis
(+)-Camphor
Cat.No: T0882
Synonym: D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor
Target: Antibacterial, TRP/TRPV Channel
Camelliaside A
Cat.No: T3854
Synonym: 山茶苷 A,山茶甙A
Target: Others
Camphor
Cat.No: T2952
Synonym: 樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa
Target: Influenza Virus, TRP/TRPV Channel
Voacamine
Cat.No: T2S0271
Synonym: 老刺木胺,Voacanginine
Target: Cannabinoid Receptor, P-gp
Vincamine
Cat.No: T1286
Synonym: Angiopac,Oxybral,Devincan,Novicet,Equipur,长春胺,Perval
Target: GPR, Others
Campneoside II
Cat.No: T82786
Synonym:
Target:
Eucamalduside A
Cat.No: TN4025
Synonym:
Target: Others
9-Hydroxycamptothecin
Cat.No: T4952
Synonym: 9-HCPT,9-羟基喜树碱,10-Hydroxycampothecin
Target: Topoisomerase
Juniper camphor
Cat.No: T82002
Synonym:
Target:
Camaric acid
Cat.No: TN3573
Synonym:
Target: Antifection
(±)-10-Hydroxycamptothecin
Cat.No: T1521
Synonym: Hydroxy Camptothecine,10-羟基喜树碱,10-Hydroxycamptothecin
Target: Topoisomerase
14,15-Didehydrovincamenine
Cat.No: TN2620
Synonym:
Target: Others
Decamethylcyclopentasiloxane
Cat.No: T21098
Synonym: Dekamethylcyklopentasiloxan,Cyclopentasiloxane, decamethyl-
Target:
Camaldulenic acid
Cat.No: TN5954
Synonym:
Target:
Campsiketalin
Cat.No: TN5830
Synonym: Rengyoxide dimethyl ketal
Target:
Lysicamine
Cat.No: TN4471
Synonym:
Target: IL Receptor, Antifection
Apovincamine
Cat.No: T21047
Synonym: cis-Apovincamine
Target:
Camellianin A
Cat.No: TN1464
Synonym:
Target: RAAS
10-Nitro-camptothecin
Cat.No: TN1176
Synonym: 9-硝基喜树碱
Target: Others
Camellianin B
Cat.No: T38481
Synonym:
Target:
Elasticamide
Cat.No: TN2681
Synonym: 2-(2'-Hydroxytetracosanoylamino)-octadecane-1,3,4-triol
Target: Others
Norcamphor
Cat.No: TN4667
Synonym:
Target: Others
Rebeccamycin
Cat.No: T16726
Synonym:
Target: Topoisomerase
Epicoccamide
Cat.No: T31651
Synonym:
Target:
16,17-Dihydroapovincamine
Cat.No: TN2642
Synonym:
Target: Others
Eucamalol
Cat.No: TN4026
Synonym:
Target: Others
(S)-Campesterol
Cat.No: T83520
Synonym: 5-Ergosten-3β-ol
Target:
12-Ethyl-9-hydroxycamptothecin
Cat.No: TN2460
Synonym: 7-乙基-10-羟基喜树碱,7-Ethyl-10-Hydroxy-Camptothecin
Target: Others
Tunicamycin V
Cat.No: T38299
Synonym:
Target:
Beauverolide Ja
Cat.No: T74198
Synonym:
Target:
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