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92

抑制剂 & 化合物

21

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T38117	WSP-5 Washington State Probe-5,WSP-5
	Hydrogen sulfide (H2S) is an important gaseous mediator, like nitric oxide, that has significant effects on the immunological, neurological, cardiovascular and pulmonary systems of mammals. WSP-5 is a reactive disulfide-containing, fluorescent probe designed for fast detection of H2S in biological samples and cells. Through a reaction-based fluorescent turn-on strategy, WSP-5 selectively and rapidly reacts with H2S, generating a fluorophore with excitation and emission maxima of 502 and 525 nm, ...
T7414	ARS-853	Apoptosis; Raf; Ras	Apoptosis; GPCR/G Protein; MAPK
	ARS-853 是一种选择性共价KRAS G12C 抑制剂，IC50为 2.5 μM。它通过与 GDP 结合的癌蛋白结合并阻止激活来抑制突变 KRAS 驱动的信号传导。
T22675	Co 102862 V 102862	Others; Sodium Channel	Membrane transporter/Ion channel; Others
	Co 102862 是一种电压门控钠通道阻滞剂。 Co 102862 可用于抗惊厥的研究。
T10826	CK-666	HIV Protease; Microtubule Associated	Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
	CK-666 是一种肌动蛋白相关蛋白 Arp2/3 复合物的细胞渗透性抑制剂。它与 Arp2/3 复合物结合，稳定复合物的非活性状态，阻止 Arp2 和 Arp3 亚基进入活化的丝状短节距构象。
T8369	Adagrasib MRTX849	Ras	GPCR/G Protein; MAPK
	Adagrasib (MRTX849) 是一种 KRAS G12C 共价抑制剂，具有口服活性和选择性。Adagrasib 与 KRAS G12C 非活性构象的 GDP 状态结合，抑制 KRAS 及其下游信号的传导。Adagrasib 对 KRAS G12C 突变肿瘤具有抑制活性。
T12519	Sodium metatungstate POM-1,聚钨酸钠,Sodium polyoxotungstate	Phosphatase	Metabolism
	Sodium metatungstate (Sodium polyoxotungstate) 是一种外核苷三磷酸二磷酸水解酶抑制剂，能够抑制 ATP 的分解，并阻断中枢突触传递，这是独立于抑制 NTPDase 而发挥作用的。
T64830	Tetrapotassium decatungstate
	Tetrapotassium decatungstate 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T64830。
T64838	Tetrabutylphonium decatungstate
	Tetrabutylphonium decatungstate 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T64838。
T30154	Ascorbyl myristate Ascorbyl monomyristate,6-tetradecanoate,L-Ascorbic acid
	Ascorbyl myristate is a bioactive chemical.
T33791	Oleyl myristate
	Oleyl myristate is a bioactive chemical.
T64775	Sodium tungstate(VI)
	Sodium tungstate(VI) 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T64775。
T23189	prostate apoptosis response protein PAR-4 (2-7) [Homo sapiens]	Others	Others
	Prostate apoptosis response protein PAR-4 (2-7) [Homo sapiens] is a peptide with the sequence H2N-Ala-Thr-Gly-Gly-Tyr-Arg-OH, MW= 623.66.
T64579	Tetrabutylammonium decatungstate
	Tetrabutylammonium decatungstate 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T64579。
T80552	Prostate Specific Antigen Substrate
	Prostate Specific Antigen Substrate为前列腺特异性抗原（PSA）的荧光底物，专用于检测PSA的酶活性。
T21339	Peramivir RWJ 270201,BCX1812,BCX 1812,帕拉米韦,RWJ270201
	Peramivir, a neuraminidase inhibitor, acts as a transition-state analogue inhibitor of influenza neuraminidase and thereby preventing new viruses from emerging from infected cells. It is used as an antiviral drug for the treatment of influenza.
T5370	DTT 二硫苏糖醇,DL-Dithiothreitol	Others	Others
	DTT (DL-Dithiothreitol) 是一种强还原剂。它被氧化后，会形成带有内部二硫键的稳定六元环。
T13925	THS-044 N-[2-Nitro-4-(Trifluoromethyl)phenyl]morpholin-4-Amine,N-Morpholino-2-nitro-4-(trifluoromethyl)aniline	HIF	Angiogenesis; Chromatin/Epigenetic
	THS-044 (N-[2-Nitro-4-(Trifluoromethyl)phenyl]morpholin-4-Amine) 的结合可稳定 HIF2α PAS-B 折叠状态，kd 为 2 μM，并在内源性和临床环境中调节 HIF2 活性。
T8700	TKIM	Potassium Channel	Membrane transporter/Ion channel
	TKIM 是一种 TWIK 相关的钾通道 1 (TREK-1) 抑制剂，与 TREK-1 的中间 (IM) 状态的口袋结合。
T21769L	β-Pompilidotoxin Acetate β-Pompilidotoxin Acetate(216064-36-7 Free base)	Sodium Channel	Membrane transporter/Ion channel
	β-Pompilidotoxin Acetate 是一种黄蜂毒肽。它可以减缓钠通道的失活并增加细胞中的稳态钠电流。
T15711	Larazotide acetate	Gap Junction Protein	Cytoskeletal Signaling
	Larazotide acetate 是合成肽，它起到紧密连接调节器的作用，并将泄漏连接反转到它们的常闭状态。
T19352	HBC620	Others	Others
	HBC620 在 Pepper 结合状态下显示出明亮的荧光，可以可视化活细胞中的 RNA 动力学。 HBC620 是一种类似 HBC 的荧光团。
T26287	Transcainide R54718,R 54718,R-54718	Sodium Channel	Membrane transporter/Ion channel
	Transcainide(R 54718) 是一种新的利多卡因类似物，是具有口服活性的抗心律失常剂。Transcainide 可阻断牛心脏和大鼠骨骼肌中 BTX 激活的钠通道的开放状态。
T2635	Org 27569	Cannabinoid Receptor	GPCR/G Protein
	Org 27569 是一种 CB1 receptor 别构调节剂，可以增加激动剂与 CB1 结合，能够抑制激动剂诱导的 CB1 信号通路。
T2169	Zebularine NSC309132,4-Deoxyuridine	DNA Methyltransferase; Autophagy	Autophagy; Chromatin/Epigenetic
	Zebularine (4-Deoxyuridine) 是一种 DNA 甲基化抑制剂，还抑制胞苷脱氨酶。它通过以共价水合物的形式与活性大小结合，充当胞苷脱氨酶的过渡态类似物抑制剂。
T29037	UC-781 NSC 675186,UC781,UC 781	Antiviral; HIV Protease	Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
	UC-781 (NSC-675186) 是一种高效且具有选择性的人类免疫缺陷病毒 HIV-1 非核苷类逆转录酶(NNRTI)I抑制剂，C50 值为 5 nM。UC-781 具有抗病毒活性和耐药性。UC-781状态稳定，较低的 PH 或不同温度对其影响较小。
T8711	PF-05186462 PF-05150122	Sodium Channel	Membrane transporter/Ion channel
	PF-05186462 (PF-05150122)是选择性的人Nav1.7电压依赖性钠通道抑制剂，IC50为 21 nM，与其他钠通道 (Nav 1.1、1.2、1.3、1.4、1.5、1.6 和 1.8) 相比，它对 Nav1.7显示出显著的选择性。PF-05186462在急性或慢性疼痛中具有研究价值。
T33816	Ordopidine ACR-325,ACR 325,ACR325	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Ordopidine (ACR325) 是一种多巴胺能稳定剂，可抑制精神刺激剂引起的多动症，并在不活动时刺激行为。Ordopidine 在体外作为多巴胺 D2 受体拮抗剂起作用，尽管亲和力低，但其依赖于特定状态的行为效应特征是 D2 受体拮抗剂所不具备的。
T8684	Sotorasib AMG-510	Ras	GPCR/G Protein; MAPK
	Sotorasib (AMG-510) 是一种 KRAS G12C 共价抑制剂，具有口服活性和选择性。Sotorasib 与 KRAS G12C 非活性构象的 GDP 状态结合，抑制 KRAS 及其下游信号的传导。Sotorasib 对 KRAS G12C 突变肿瘤具有抑制活性。
T24754	Hh-Ag1.5 SAG-1.5,SAG1.5,SAG 1.5	Hedgehog/Smoothened	GPCR/G Protein; Stem Cells
	Hh-Ag1.5 (SAG-1.5) 是一种高效的 Hedgehog (Hh) 激动剂(EC50： 1 nM)和Smoothened (Smo)受体激动剂，对Smo的 EC50 为 1 nM、 Ki值在 0.5 和 2.3 nM 之间。Hh-Ag1.5 介导的重编程打破了非损伤肝脏干细胞的静止状态，从而挽救了肝衰竭。Hh-Ag1.5 诱导 hiPSCs 分化为皮肤前体细胞、脊髓运动神经元和脊髓感觉神经元。
T13983	0990CL	cAMP; Others	GPCR/G Protein; Others
	0990CL 是一种有效的异三聚体Gαi subunit 特异性抑制剂，可与纯化的Go±在gdp 结合状态下相互作用，能够阻断α2AR 介导的cAMP 调控。在细胞模型中低浓度0990CL 能够部分恢复cAMP 水平，高浓度的0990CL (10 μM)下，开始对细胞活力产生负面影响。
T9972	Divarasib GDC-6036	Ras	GPCR/G Protein; MAPK
	Divarasib (GDC-6036) (GDC-6036)是一种正在研究的、口服的、高效力和选择性的 KRAS G12C 抑制剂，IC50 为 <0.01 μM。Divarasib 不可逆地将 KRAS G12C 癌蛋白锁定在非活性状态，抑制肿瘤细胞生长。它正在被研究用于实体肿瘤，包括非小细胞肺癌和结肠直肠癌及其他类型的癌症。
T2408	Ostarine MK-2866,GTX-024,Enobosarm	Androgen Receptor	Endocrinology/Hormones
	Ostarine (MK-2866) 是一种具有合成代谢活性的非甾体药物。选择性雄激素受体调节剂 (SARM) GTx-024 旨在像睾酮一样发挥作用，从而促进和/或维持性欲、生育能力、前列腺生长以及肌肉生长和力量。模仿睾酮的作用，这种药物可以增加瘦体重，从而改善癌症恶病质高代谢状态下的肌肉萎缩。
T14884	CBR-5884	Others; Dehydrogenase	Metabolism; Others
	CBR-5884 是一种磷酸甘油酸脱氢酶抑制剂，IC50为 33 μM。它抑制癌细胞中的丝氨酸合成，选择性地抑制黑素瘤和乳腺癌细胞系的增殖，对具有高丝氨酸生物合成活性的癌细胞系有选择性毒性。
T37807	JTV 519 fumarate
	Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo. Hunt et al (2007) K201 (JTV519) suppresses spontaneous Ca2+ release and [3H]ryanodine binding to RyR2 irrespective of FKBP12.6 association. Biochem.J. 404 431 PMID:17313373 \|Chen et al (2008) Effect of K201, a novel antiarrhythmic drug on calcium handling and arrhythmogenic activity of pulmonary vein cardiomyocytes. Br.J.Pharmacol. 153 915 PMID:17994112 \|...
T24902	TROX-1 TROX1,TROX 1
	TROX-1 is the activation state-dependent Cav2 channel antagonist.
T14992	Raxatrigine hydrochloride GSK-1014802 hydrochloride,CNV1014802 (hydrochloride)	Others	Others
	Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.
T30827	Cgp 33304 Cgp-33304,Cgp33304
	CGP 33304 is a dual leukotriene receptor antagonist and phospholipase A2 inhibitor. It prevents hypoxia secondary to bronchial constriction induced by leukotriene in a shocking state.
T25896	Octicidine ASOHO
	Octicidine is derived from phaseolotoxin by the removal of C-terminal dipeptide. It is a transition state analog that irreversibly suppresses ornithine carbamoyltransferase.
T25184	Butalamine Butalamina
	Butalamine is a vasodilator (peripheral) with local anesthetic effects. It suppresses state 3 respiration and decreases ADP/O in the rat liver.
T34665	SN-1 SN1
	SN-1 is a zinc chelator which increases steady-state expression level of A3G in the presence of Vif.
T81459	Pinacyanol iodide
	Pinacyanol iodide，一种具有超快激发态异构化特性的荧光花青染料。
T25184L	Butalamine HCl LA 1221,Hemotrope,Butalamine hydrochloride,Adrevil
	Butalamine HCl is a vasodilator (peripheral) with local anesthetic effects. It suppresses state 3 respiration and decreases ADP/O in the rat liver.
T36587	8-Aminopyrene-1,3,6-trisulfonic Acid sodium salt	Others	Others
	8-Aminopyrene-1,3,6-trisulfonic Acid sodium salt 是一种阴离子荧光染料，用作葡萄糖传感和检测其他糖类的报告分子。激发/发射光谱为 425/503 nm。它可以在溶液中使用，也可以通过还原胺化连接醛官能化单体来固定，而不会显著改变荧光强度。
T71239	CNV-2197944
	CNV-2197944 is a novel, small molecule, state-dependent calcium channel blocker, designed to selectively inhibit highly active Cav2.2 channels.
T70543	U 92163
	U 92163 is synthetic peptidic transition state analog inhibitor that was used to determine the crystallographic structure of the protease from human immunodeficiency virus type 2.
T7352L	Pridopidine hydrochloride ASP2314 HCl,Pridopidine HCl,FR310826,ASP-2314 hydrochloride
	Pridopidine Hydrochloride is a dopaminergic stabilizer that has been shown to improve a variety of neurological and psychiatric disorders, including Huntington's disease. Pridopidine Hydrochloride stabilizes psychomotor activity in a state-dependent way t
T23506	Viomycin	Others	Others
	Viomycin is a member of the tuberactinomycin family of antibiotics. Viomycin also inhibits group I intron splicing and prokaryotic protein synthesis. Freezes bacterial ribosomes in either the pre- or post-translational state. Facilitates trans-cleavage of
T19351	HBC599	Others	Others
	HBC599 is an HBC-like fluorophore. HBC599 shows brightly fluoresced in the Pepper bound state and can be visualized RNA dynamics in live cells.
T10374	ARS-1323-alkyne	Ras	GPCR/G Protein; MAPK
	ARS-1323-alkyne 是switch-II pocket (S-IIP)抑制剂，能够特异性报告活体细胞中 KRASG12C 核苷酸的状态。
TP1977	187-1, N-WASP inhibitor
	Inhibits neural Wiskott-Aldrich syndrome protein (N-WASP) by stabilizing the autoinhibited state of the protein. Blocks phosphatidylinositol 4,5-bisphosphate (PIP2)-stimulated actin assembly (IC50 ~ 2 μM) but does not directly inhibit actin polymerization

化合物

Cat.No: T38117

Synonym: Washington State Probe-5,WSP-5

Cat.No: T7414

Target: Apoptosis, Raf, Ras

Cat.No: T22675

Synonym: V 102862

Target: Others, Sodium Channel

Cat.No: T10826

Target: HIV Protease, Microtubule Associated

Cat.No: T8369

Synonym: MRTX849

Target: Ras

Sodium metatungstate

Cat.No: T12519

Synonym: POM-1,聚钨酸钠,Sodium polyoxotungstate

Target: Phosphatase

Tetrapotassium decatungstate

Cat.No: T64830

Tetrabutylphonium decatungstate

Cat.No: T64838

Ascorbyl myristate

Cat.No: T30154

Synonym: Ascorbyl monomyristate,6-tetradecanoate,L-Ascorbic acid

Oleyl myristate

Cat.No: T33791

Sodium tungstate(VI)

Cat.No: T64775

prostate apoptosis response protein PAR-4 (2-7) [Homo sapiens]

Cat.No: T23189

Target: Others

Tetrabutylammonium decatungstate

Cat.No: T64579

Prostate Specific Antigen Substrate

Cat.No: T80552

Cat.No: T21339

Synonym: RWJ 270201,BCX1812,BCX 1812,帕拉米韦,RWJ270201

Cat.No: T5370

Synonym: 二硫苏糖醇,DL-Dithiothreitol

Target: Others

Cat.No: T13925

Synonym: N-[2-Nitro-4-(Trifluoromethyl)phenyl]morpholin-4-Amine,N-Morpholino-2-nitro-4-(trifluoromethyl)aniline

Target: HIF

Cat.No: T8700

Target: Potassium Channel

β-Pompilidotoxin Acetate

Cat.No: T21769L

Synonym: β-Pompilidotoxin Acetate(216064-36-7 Free base)

Target: Sodium Channel

Larazotide acetate

Cat.No: T15711

Target: Gap Junction Protein

Cat.No: T19352

Target: Others

Cat.No: T26287

Synonym: R54718,R 54718,R-54718

Target: Sodium Channel

Cat.No: T2635

Target: Cannabinoid Receptor

Cat.No: T2169

Synonym: NSC309132,4-Deoxyuridine

Target: DNA Methyltransferase, Autophagy

Cat.No: T29037

Synonym: NSC 675186,UC781,UC 781

Target: Antiviral, HIV Protease

Cat.No: T8711

Synonym: PF-05150122

Target: Sodium Channel

Cat.No: T33816

Synonym: ACR-325,ACR 325,ACR325

Target: Dopamine Receptor

Cat.No: T8684

Synonym: AMG-510

Target: Ras

Cat.No: T24754

Synonym: SAG-1.5,SAG1.5,SAG 1.5

Target: Hedgehog/Smoothened

Cat.No: T13983

Target: cAMP, Others

Cat.No: T9972

Synonym: GDC-6036

Target: Ras

Cat.No: T2408

Synonym: MK-2866,GTX-024,Enobosarm

Target: Androgen Receptor

Cat.No: T14884

Target: Others, Dehydrogenase

JTV 519 fumarate

Cat.No: T37807

Cat.No: T24902

Synonym: TROX1,TROX 1

Raxatrigine hydrochloride

Cat.No: T14992

Synonym: GSK-1014802 hydrochloride,CNV1014802 (hydrochloride)

Target: Others

Cat.No: T30827

Synonym: Cgp-33304,Cgp33304

Cat.No: T25896

Synonym: ASOHO

Cat.No: T25184

Synonym: Butalamina

Cat.No: T34665

Synonym: SN1

Pinacyanol iodide

Cat.No: T81459

Cat.No: T25184L

Synonym: LA 1221,Hemotrope,Butalamine hydrochloride,Adrevil

8-Aminopyrene-1,3,6-trisulfonic Acid sodium salt

Cat.No: T36587

Target: Others

Cat.No: T71239

Cat.No: T70543

Pridopidine hydrochloride

Cat.No: T7352L

Synonym: ASP2314 HCl,Pridopidine HCl,FR310826,ASP-2314 hydrochloride

Cat.No: T23506

Target: Others

Cat.No: T19351

Target: Others

ARS-1323-alkyne

Cat.No: T10374

Target: Ras

187-1, N-WASP inhibitor

Cat.No: TP1977

Cat. No.	Product Name	Target	Signaling Pathways
TQ0198	Phorbol 12-myristate 13-acetate 佛波醇12-十四酸酯13-乙酸酯,PMA	NF-κB; S1P Receptor; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; NF-κB
	Phorbol 12-myristate 13-acetate (PMA) 属于佛波酯类天然产物，是一种 PKC、SphK、NF-κB 的激活剂。Phorbol 12-myristate 13-acetate 可诱导 THP1 细胞分化。
T20005	Isopropyl myristate IPM,Isomyst,HSDB 626,肉豆蔻酸异丙酯,FEMA No. 3556,十四酸异丙酯,NSC 406280,Stepan D-50	Others	Others
	Isopropyl myristate (IPM) 是异丙醇和肉豆蔻酸的酯。它是一种可用于化妆品和外用药物制剂中的极性润肤剂。
TN6901	Methyl myristate 肉豆蔻酸甲酯,methyl tetradecanoate	Others	Others
	Methyl myristate (methyl tetradecanoate) 是一种肉豆蔻酸经酯化反应得到的饱和脂肪酸甲酯。对 B16F10 黑色素瘤具有显著的诱导作用。
T8040	Cholesterol myristate 胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate	Others; Potassium Channel; GABA Receptor; Endogenous Metabolite; AChR	Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
	Cholesterol myristate (Cholesteryl myristate) 是粗吻海龙中的一种类固醇，可与多种离子通道结合，例如nAChR、GABAA 受体和内向整流钾离子通道。
TN6994	Ethyl Myristate
	Ethyl Myristate is a natural product.
TN4546	Methyl isocostate	Others	Others
	Methyl isocostate 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4546，CAS号为 132342-55-3。
T10023	1-Naphthol NSC 9586,Nako TRB,1-萘酚,Furro ER	Endogenous Metabolite	Metabolism
	1-Naphthol (Furro ER) 是激发态质子转移荧光分子探针。
T4884	alpha-D-glucose α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose	Others; Endogenous Metabolite	Metabolism; Others
	alpha-D-glucose (α-Dextrose) 是内源性代谢产物的一种。
T0887	D-Glucose Dextrose,D-无水葡萄糖,Glucopyranose,Grape sugar,葡萄糖,D(+)-Glucose	Endogenous Metabolite	Metabolism
	D-Glucose (Glucopyranose) 是一种单糖。D-Glucose 是甜味剂，是一般代谢的关键组成部分，并作为与细胞代谢状态以及生物和非生物应激反应有关的关键信号分子。
T8733	Antrodin A (2-氯苯基)二苯基甲醇,camphorataanhydride A	Others	Others
	Antrodin A (camphorataanhydride A) 是固体发酵樟脑菌菌丝体的一种主要活性成分。它能够增强肝脏的抗炎及抗氧化能力，维持肠道菌群的稳定，避免酒精对肝脏的损伤。
T67685	4-Methylumbelliferyl-β-D-xylopyranoside 4-Methylumbelliferyl-β-D-xyloside
	4-Methylumbelliferyl-β-D-xylopyranoside (4-Methylumbelliferyl-β-D-xyloside)在生物实验中展现出爆裂的稳态动力学，这支持底物4-Methylumbelliferyl-β-D-xylopyranoside 糖苷键快速水解的结论。4-Methylumbelliferyl-β-D-xylopyranoside 可用于 β- 木糖苷酶活性研究。
T2910	Flavonol 3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone	Others; Endogenous Metabolite	Metabolism; Others
	Flavonol (3-Hydroxyflavone) 是内源性代谢产物的一种。
TN1163	2'-Hydroxychalcone	Others	Others
	2'-Hydroxychalcone 是一种药物合成中间体，可用于合成黄酮类化合物。负载在纳米乳液中的2'-Hydroxychalcone 在Danio rerio 模型对副球孢子菌显示出杀真菌活性。2'-Hydroxychalcone 通过负载脂质的Hepg2细胞中的氧化应激诱导细胞毒性。2'-Hydroxychalcone 抑制通过逆转录聚合酶链反应确定的肿瘤坏死因子-α诱导ICAM-1，VCAM-1和E-选择素的稳态转录水平，因此可能会干扰其基因的转录。
T38108	Fulvic Acid	Antioxidant; PDE	Metabolism; oxidation-reduction
	Fulvic Acid 是一种来自土壤、沉积物或水生环境中微生物产生的腐殖质的天然产物，是一种首次青霉菌中分离出的酚酸和真菌代谢产物。Fulvic Acid 抑制淀粉样蛋白b (17-42) (AB17-42)二聚化，破坏预先形成的AB17-42三聚体，并结合到磷酸二酯酶5A (PDE5A)的催化位点，可以调节机体免疫系统，影响细胞的氧化状态，改善胃肠功能。Fulvic Acid 可作为氧化剂或还原剂，具有研究糖尿病等慢性炎症性疾病的潜力。
T38395	Pyrrole-2-carboxaldehyde
	Pyrrole-2-carboxaldehyde exhibits distinctive vibrational and electronic properties which serve to validate its dimeric state in the solid phase and monomeric state in the solution phase.
T19565	Streptolysin O	Others	Others
	Streptolysin O causes both lysis of cells and cardiotoxicity. Streptolysin O is widely used for the controlled permeabilization of cell membranes. Streptolysin O exists in two forms, a reduced active state and an oxidized reversibly inactive state .
TN2830	26-Nor-8-oxo-alpha-onocerin	Others	Others
	26-Nor-8-oxo-alpha-onocerin can promote the osteoblast proliferation rate, the effect is time-dependent,concentration-dependent and differentiation state-dependent.
TN3844	Didrovaltrate	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Didrovaltrate shows cytotoxic against human cancer cell lines. Didrovaltrate blocks I(Ca-L) in a concentration-dependent manner and probably inhibits I(Ca-L) in its inactive state, which may contribute to its cardiovascular effect.
TN1912	Marinobufogenin 南美蟾毒精,Marinobufagenin	ATPase; EGFR	Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
	Marinobufagenin, a cardiotonic steroid, its increased concentrations are important in the cardiac disease and oxidant stress state seen with renal failure.
T71750	Quinolactacin A1
	Quinolactacin A1 是一种有效的乙酰胆碱酯酶 (AChE) 抑制剂，可从Penicillium citrinum 中得到。Quinolactacin A1 可用于阿尔茨海默病的研究。
TN3541	Broussonin E	ERK; p38 MAPK; TNF; JAK; STAT	Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; MAPK; Stem Cells
	Broussonin E could suppress inflammation by modulating macrophages activation state via inhibiting the ERK and p38 MAPK and enhancing JAK2-STAT3 signaling pathway, and can be further developed as a promising drug for the treatment of inflammation-related

天然产物

Phorbol 12-myristate 13-acetate

Cat.No: TQ0198

Synonym: 佛波醇12-十四酸酯13-乙酸酯,PMA

Target: NF-κB, S1P Receptor, PKC

Isopropyl myristate

Cat.No: T20005

Synonym: IPM,Isomyst,HSDB 626,肉豆蔻酸异丙酯,FEMA No. 3556,十四酸异丙酯,NSC 406280,Stepan D-50

Target: Others

Methyl myristate

Cat.No: TN6901

Synonym: 肉豆蔻酸甲酯,methyl tetradecanoate

Target: Others

Cholesterol myristate

Cat.No: T8040

Synonym: 胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate

Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR

Ethyl Myristate

Cat.No: TN6994

Methyl isocostate

Cat.No: TN4546

Target: Others

Cat.No: T10023

Synonym: NSC 9586,Nako TRB,1-萘酚,Furro ER

Target: Endogenous Metabolite

alpha-D-glucose

Cat.No: T4884

Synonym: α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose

Target: Others, Endogenous Metabolite

Cat.No: T0887

Synonym: Dextrose,D-无水葡萄糖,Glucopyranose,Grape sugar,葡萄糖,D(+)-Glucose

Target: Endogenous Metabolite

Cat.No: T8733

Synonym: (2-氯苯基)二苯基甲醇,camphorataanhydride A

Target: Others

4-Methylumbelliferyl-β-D-xylopyranoside

Cat.No: T67685

Synonym: 4-Methylumbelliferyl-β-D-xyloside

Cat.No: T2910

Synonym: 3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone

Target: Others, Endogenous Metabolite

2'-Hydroxychalcone

Cat.No: TN1163

Target: Others

Cat.No: T38108

Target: Antioxidant, PDE

Pyrrole-2-carboxaldehyde

Cat.No: T38395

Cat.No: T19565

Target: Others

26-Nor-8-oxo-alpha-onocerin

Cat.No: TN2830

Target: Others

Cat.No: TN3844

Target: Calcium Channel

Marinobufogenin

Cat.No: TN1912

Synonym: 南美蟾毒精,Marinobufagenin

Target: ATPase, EGFR

Quinolactacin A1

Cat.No: T71750

Cat.No: TN3541

Target: ERK, p38 MAPK, TNF, JAK, STAT

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