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84

抑制剂 & 化合物

30

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T1909	L-701324 7-氯-4-羟基-3-(3-苯氧基)苯基-2(1H)-喹啉,L701324	NMDAR; iGluR	Membrane transporter/Ion channel; Neuroscience
	L-701324 是一种 NMDA 受体，对甘氨酸位点具有高亲和力和选择性，用作口服活性和长效抗惊厥药。
T3268	Mildronate Kvaterin,米屈肼,Meldonium,Quaterin	Hydroxylase	Metabolism
	Mildronate (Meldonium) 是心血管保护药，能够竞争性的抑制 BBOX1和 OCTN2。作用于人重组 BBOX 的(IC50:34-62 μM)、人 OCTN2 (EC50:21 μM)。它 n 能够诱导长链脂肪酸代谢从线粒体向过氧化物酶体的重定向。
T15733	Lemildipine NB-818,NPK-1886	Others	Others
	Lemildipine is a new blocker of dihydropyridine calcium entry.
T0227	Bromisoval 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral	Others	Others
	Bromisoval (Isobromyl) 具有抗炎活性。
T19841	Tribenoside Glyvenol,Glyvenal,Ba 2140,BG-356,Glivenol,三苄糖苷,TBGF	Others	Others
	Tribenoside (BG-356) 是血管保护剂，能够温和的镇痛、抗炎及伤口愈合，可用研究痔疮。
T1884	CX516 Ampakine CX516,BDP 12,Ampalex,安帕来斯	GluR; iGluR	Membrane transporter/Ion channel; Neuroscience
	CX516 (Ampalex) 是AMPA 受体正向调节剂，可用于研究阿尔茨海默病，精神分裂等。
T7114	GALANTHAMINONE (-)-Narwedine,氢溴酸加兰他敏,Narwedin	AChE	Neuroscience
	Galanthaminone ((-)-Narwedine) 是一种竞争性的、可逆的胆碱酯酶抑制剂，可作用于多种记忆障碍疾病的研究。
T77054	Lecanemab BAN-2401	Beta Amyloid	Neuroscience
	Lecanemab (BAN-2401) 是一种靶向可溶性聚集性 β 淀粉样蛋白（Abeta）的 IgG1 单克隆抗体，对寡聚体、原纤维和不溶性原纤维具有活性，可用于研究阿尔茨海默病（AD）引起的轻度认知障碍和轻度 AD 痴呆。
T0669	Chloramine-T Chloralone,氯胺 T,Chlorasan,Chlorozone	Others; Antibacterial	Microbiology/Virology; Others
	Chloramine-T (Chloralone) 是一种 N-氯化和 N-去质子化磺胺，用作杀生物剂和温和消毒剂。
T2222	Carbinoxamine Maleate Salt Lergefin,马来酸罗托沙敏,CarbinoxaMine Maleate	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Carbinoxamine Maleate Salt (Lergefin) 是一种乙醇胺类 H1 抗组胺药，具有温和的抗毒蕈碱和镇静作用。
T24451	Mepyramine NSC-13136,NSC13136,NSC 13136
	Mepyramine is a histamine H1 antagonist. It has mild hypnotic properties and some local anesthetic action and is used for allergies both parenterally and locally.
T68036	Carprazidil	Others	Others
	Carprazidil 是一种强效的血管扩张剂，可用于治疗严重高血压和轻度心力衰竭。
T13689	Ethylene dimethanesulfonate	Apoptosis	Apoptosis
	Ethylene dimethanesulfonate 是温和的烷基化乙二醇非挥发性甲烷磺酸二酯，对 LC 具有选择性的促凋亡作用。
T26526	Abt-288 ABT 288,ABT288	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	ABT-288 是一种具有选择性和高效性的 H3 拮抗剂，可用于治疗轻度至中度阿尔茨海默氏痴呆。
T5500	DORA-22	OX Receptor	GPCR/G Protein; Neuroscience
	DORA-22 是一种双食欲素受体拮抗剂，可改善轻度压力引起的失眠，对记忆的影响很小。
T0240	Trimetozine Sedoxazine,Trioxazin,三甲氧啉	Others	Others
	Trimetozine (Sedoxazine) 是一种镇静剂，自 1959 年以来一直在欧洲上市。它具有温和的镇静作用，已用于治疗焦虑症。
T14377	AZD5423	Glucocorticoid Receptor	Endocrinology/Hormones
	AZD5423 是可吸入的非甾体糖皮质激素受体选择性调节剂，能够有效降改善轻度过敏性哮喘患者的过敏原诱导反应。
T7887	8-Hydroxyquinoline hemisulfate 8-羟基喹啉硫酸盐,Oxyquinoline sulfate	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	8-Hydroxyquinoline hemisulfate (Oxyquinoline sulfate) 是一种单质子双齿螯合剂，具有温和的抑菌、驱虫和杀螨作用。
T33711L	Nolomirole HCl CHF 1035 HCl,CHF 1035,CHF1035,CHF1035 HCl,CHF-1035 HCl,CHF-1035,Nolomirole Hydrochloride	Dopamine Receptor; Norepinephrine	GPCR/G Protein; Neuroscience
	Nolomirole HCl（CHF 1035）是一种具有口服活性的新型选择性多巴胺激动剂，对去甲肾上腺素的释放有抑制作用，可用于研究轻度慢性心力衰竭。
T31482	Diloxanide Diloxanid,RD 3803,RD3803,RD-3803,Diloxanida,二氯尼特	Parasite	Microbiology/Virology
	Diloxanide (RD3803) 是一种抗原虫制剂，可研究组织学内阿米巴原虫或者其他原虫感染引起的无症状肠道阿米巴病。它是一种活性的鲁米那抗阿米巴试剂，是由其前药二氯尼特糠酸酯在胃肠道中水解得来的。
T7041	Donepezil E2020,Donepezilo,Aricept,多奈哌齐	AChE	Neuroscience
	Donepezil (Aricept) 是一种AChE 抑制剂，对牛 AChE 和人 AChE 的IC50分别为 8.12 nM 和 11.6 nM。
T2507	Azeliragon TTP488,阿齐瑞格	Beta Amyloid; advanced glycation end products	Neuroscience; Others
	Azeliragon (TTP488) 是一种生物可利用的、可穿过血脑屏障 (BBB)的晚期糖基化终产物 (RAGE) 受体抑制剂，可缓解轻度阿尔茨海默病 (AD) 的发展。
T21434	Sulfacetamide NSC 63871,磺胺醋酰,NSC-63871,Sebizon,Region,NSC63871,Sulphacetamide,Acetosulfamine	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Sulfacetamide (NSC-63871) 是一种抗生素，通过限制细菌生存所需的叶酸的存在来治疗睑缘炎或结膜炎，有潜力用于眼部感染的研究。
T20982	Sodium 3-nitrobenzenesulfonate	Others	Others
	Sodium 3-nitrobenzenesulfonate 是一种温和的氧化剂。 Sodium 3-nitrobenzenesulfonate 在轧染印花或蒸汽印花时可以保护色光，并抵消还原物质的作用。
T4615	Balsalazide sodium hydrate 巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium	STAT; Interleukin	Immunology/Inflammation; JAK/STAT signaling; Stem Cells
	Balsalazide sodium hydrate (Balsalazide disodium) 可通过调节IL-6/STAT3通路起抑癌作用，可用于治疗炎症性肠病。
T67886	Girard's Reagent T Trimethylacetohydrazideammonium Chloride	Others	Others
	Girard's Reagent T (Trimethylacetohydrazideammonium Chloride) 是生化试剂。Girard's Reagent T 在温和的酸性或碱性条件下，与含有α-二羰基官能团的醛类和酮类反应，生成强吸收紫外线的加成化合物
TP2500	Cholecystokinin (26-33) free acid CCK (26-33) free acid	cholecystokinin	GPCR/G Protein
	Cholecystokinin (26-33) free acid 是胆囊收缩素 (CCK) 的一部分，是脊椎动物中枢神经系统中存在的 CCKB 型受体的高选择性配体，可诱导大鼠轻度味觉厌恶条件反射。
T1232	Mepyramine maleate 马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Mepyramine maleate (Pyrilamine maleate) 是一种组胺 H1 拮抗剂，对 H1、H2 和 H3 受体的 Kd 值分别为 0.8、5200 和大于 3000 nM，对 H1 受体的 pKd 值为 9.4。它是感冒药的常见成分，具有温和的催眠特性和局部麻醉作用，可用于胃肠外和局部过敏。
T33589	Nanterinone UK-61260,UK61260,UK 61260	PDE	Metabolism
	Nanterinone (UK 61260) 是一种口服的部分磷酸二酯酶抑制剂，是一种新型的正性肌力和平衡血管扩张化合物。Nanterinone 口服后，可使急性血流动力学得到明显改善，这可能取决于先前存在的左心室充盈压。
T0331	Moxifloxacin hydrochloride 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl	Topoisomerase; Antibacterial; Antibiotic	DNA Damage/DNA Repair; Microbiology/Virology
	Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物，可研究感染性肺炎，急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
T1951	Asenapine Maleate Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐	5-HT Receptor	GPCR/G Protein; Neuroscience
	Asenapine Maleate (Org 5222 maleate) 是5-HT 和D2的拮抗剂，Ki 值分别为 0.03-4.0 nM, 1.3 nM。它也是抗精神病药物，用于治疗与双相 1 型障碍相关的精神分裂症和躁狂或混合发作。
T34081	Piromelatine NEU-P-11,NEU-P 11,NEU-P11	P2X Receptor; 5-HT Receptor; MT Receptor; Sodium Channel; TRP/TRPV Channel	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Piromelatine 是褪黑激素 MT1/MT2 受体、5-HT1A 和 5-HT1D 的激动剂，也是 5-HT2B 的拮抗剂。Piromelatine 具有抗痛觉活性，对 P2X3、TRPV1 和 Nav1.7 通道有抑制作用，可用于促进睡眠、缓解疼痛、抗神经退行性疾病和抗抑郁疾病的研究。
T0976	Propoxur 残杀威,Aprocarb,Propoxure,Baygon	AChR; Antifungal	Microbiology/Virology; Neuroscience
	Propoxur (Propoxure) 是一种氨基甲酸酯类杀虫剂，用于控制蟑螂、苍蝇、蚊子以及草坪和草坪昆虫。
T11043	Dihydroergocristine mesylate 甲磺酸双氢麦角汀,DHEC (mesylate)	Beta Amyloid	Neuroscience
	Dihydroergocristine mesylate (DHEC (mesylate)) 是一种 γ-secretase (GSI) 的抑制剂，能够阿尔茨海默氏病淀粉样蛋白 β 肽 (amyloid-β) 的产生，与 γ-secretase 和 Nicastrin 结合的平衡解离常数 (Kd) 值分别为 25.7 nM 和 9.8 μM。
T22232	Alfuzosin
	Alfuzosin 是选择性和竞争性的α1肾上腺素受体拮抗剂，可用于良性前列腺增生（BPH）的研究。
T13152	Thymol iodide	Others	Others
	Thymol iodide is a compound of Iodide and Thymol. It is mostly used as mild antiseptic and fungicide.
T24899	Trimosulfa Trimethoprim-sulfamethoxazole,Sulfamethoxazole-trimethoprim,TMP-SMX,Trimforte,Trimethoprimsulfa
	Trimosulfa is a fixed antibiotic combination that widely used for mild-to-moderate bacterial infections and as prophylaxis against opportunistic infections.
T21247	Carbinoxamine Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine
	Carbinoxamine, an anticholinergic and antihistamine agent, is used for hay fever, angioedema, vasomotor rhinitis, mild urticaria, dermatographism and allergic conjunctivitis. It is a histamine antagonist, specifically an H1-antagonist.
T37622	F13714 fumarate F13714 fumarate
	F13714 fumarate, a selective biased agonist of the 5-HT1A receptor, exhibits antidepressant-like effects upon single administration in the mouse model of chronic mild stress[1].
T33424	MK-0952 MK 0952
	MK-0952 is a selective PDE4 inhibitor used to treat long-term memory loss and mild cognitive impairment. It is an intrinsically potent inhibitor and has shown limited whole blood activity.
T24450	Mephenoxalone Lenetran Lenetran,TAB Lenetranat
	Mephenoxalone is a muscle relaxant and mild anxiolytic. It inhibits neuron transmission and relaxing skeletal muscles by inhibiting the reflex arc.
T22268	Benzyldimethylstearylammonium chloride Benzyldimethylstearylammonium Chloride Hydrate,十八烷基二甲基苄基氯化铵	Others	Others
	Benzyl dimethyl stearyl ammonium chloride hydrate is a kind of mild smell chemical
T24787	SGE-201
	SGE-201 is an allosteric modulator of N-methyl-D-aspartate receptors. SGE-201 also unmasked differences among the blockers in neuronal networks - measured either by suppression of activity in multi-electrode arrays or by neuroprotection against a mild exc
T20167	Cilazapril Ro-34-2848,Ro 34-2848,Cilazapril (anhydrous),Ro34-2848,西拉普利
	Cilazapril is an angiotensin-converting enzyme inhibitor. It has been researched for mild to moderate essential hypertension.
T68707	DJ 7141
	DJ 7141 is a unique alpha-2 agonist which shows high affinity to peripheral alpha-2 adrenoceptors but only a mild hypotensive activity.
T15131	Diloxanide furoate	Others	Others
	Diloxanide furoate is a luminal amebicide used in the treatment of Amebiasis. Amebiasis is considered the luminal agent of choice for mild intestinal amebiasis or asymptomatic cyst carriers.
T20427	Dichloramine-T NSC 1130,NSC1130,NSC-1130
	Tosylchloramide sodium salt is a N-chlorinated and N-deprotonated sulfonamide used as a biocide and a mild disinfectant.
T79855	Nevadistinel NYX-458,NYX-3054	iGluR	Membrane transporter/Ion channel; Neuroscience
	Nevadistinel (NYX-458; NYX-3054) 是一种NMDA受体的正变构调节剂，主要应用于抑制与神经退行性疾病相关的认知障碍，疾病包括轻度认知障碍、轻度阿尔茨海默病、帕金森病和路易体病。
T39575	Janelia Fluor® 669, SE JF669, SE,JF669,NHS,Janelia Fluor? 669, SE
	Janelia Fluor 669, SE (JF669, SE), a red fluorescent dye, can be directly reacted with the available thiol-containing HaloTag ligand under mild conditions (DIEA, DMF) to afford a JF669 HaloTag ligand in a single step (Ex = 669 nm; Em = 682 nm).
T32154	Indapamide hemihydrate Tenaxil,Indapamide hydrate,D06401,UNII-W0LY35K007
	Indapamide semi-hydrate (Sandoz) is a drug that contains the active ingredient of indapamide. It can be used alone or in combination with other drugs to treat mild to moderate hypertension. The effect of this drug is to deprive the body of excess water an

化合物

Cat.No: T1909

Synonym: 7-氯-4-羟基-3-(3-苯氧基)苯基-2(1H)-喹啉,L701324

Target: NMDAR, iGluR

Cat.No: T3268

Synonym: Kvaterin,米屈肼,Meldonium,Quaterin

Target: Hydroxylase

Cat.No: T15733

Synonym: NB-818,NPK-1886

Target: Others

Cat.No: T0227

Synonym: 2-Bromo-N-carbamoyl-3-methylbutanamide,Isobromyl,溴米那,BRN 1773255,Bromovalerylurea,溴米索伐,Bromaral

Target: Others

Cat.No: T19841

Synonym: Glyvenol,Glyvenal,Ba 2140,BG-356,Glivenol,三苄糖苷,TBGF

Target: Others

Cat.No: T1884

Synonym: Ampakine CX516,BDP 12,Ampalex,安帕来斯

Target: GluR, iGluR

Cat.No: T7114

Synonym: (-)-Narwedine,氢溴酸加兰他敏,Narwedin

Target: AChE

Cat.No: T77054

Synonym: BAN-2401

Target: Beta Amyloid

Cat.No: T0669

Synonym: Chloralone,氯胺 T,Chlorasan,Chlorozone

Target: Others, Antibacterial

Carbinoxamine Maleate Salt

Cat.No: T2222

Synonym: Lergefin,马来酸罗托沙敏,CarbinoxaMine Maleate

Target: Histamine Receptor

Cat.No: T24451

Synonym: NSC-13136,NSC13136,NSC 13136

Cat.No: T68036

Target: Others

Ethylene dimethanesulfonate

Cat.No: T13689

Target: Apoptosis

Cat.No: T26526

Synonym: ABT 288,ABT288

Target: Histamine Receptor

Cat.No: T5500

Target: OX Receptor

Cat.No: T0240

Synonym: Sedoxazine,Trioxazin,三甲氧啉

Target: Others

Cat.No: T14377

Target: Glucocorticoid Receptor

8-Hydroxyquinoline hemisulfate

Cat.No: T7887

Synonym: 8-羟基喹啉硫酸盐,Oxyquinoline sulfate

Target: Others, Antibacterial, Antibiotic

Cat.No: T33711L

Synonym: CHF 1035 HCl,CHF 1035,CHF1035,CHF1035 HCl,CHF-1035 HCl,CHF-1035,Nolomirole Hydrochloride

Target: Dopamine Receptor, Norepinephrine

Cat.No: T31482

Synonym: Diloxanid,RD 3803,RD3803,RD-3803,Diloxanida,二氯尼特

Target: Parasite

Cat.No: T7041

Synonym: E2020,Donepezilo,Aricept,多奈哌齐

Target: AChE

Cat.No: T2507

Synonym: TTP488,阿齐瑞格

Target: Beta Amyloid, advanced glycation end products

Cat.No: T21434

Synonym: NSC 63871,磺胺醋酰,NSC-63871,Sebizon,Region,NSC63871,Sulphacetamide,Acetosulfamine

Target: Others, Antibacterial, Antibiotic

Sodium 3-nitrobenzenesulfonate

Cat.No: T20982

Target: Others

Balsalazide sodium hydrate

Cat.No: T4615

Synonym: 巴柳氮钠水合物,Balsalazide disodium dihydrate,巴柳氮钠,Balsalazide disodium salt dihydrate,Balsalazide disodium

Target: STAT, Interleukin

Girard's Reagent T

Cat.No: T67886

Synonym: Trimethylacetohydrazideammonium Chloride

Target: Others

Cholecystokinin (26-33) free acid

Cat.No: TP2500

Synonym: CCK (26-33) free acid

Target: cholecystokinin

Mepyramine maleate

Cat.No: T1232

Synonym: 马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐

Target: Histamine Receptor

Cat.No: T33589

Synonym: UK-61260,UK61260,UK 61260

Target: PDE

Moxifloxacin hydrochloride

Cat.No: T0331

Synonym: 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Target: Topoisomerase, Antibacterial, Antibiotic

Asenapine Maleate

Cat.No: T1951

Synonym: Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐

Target: 5-HT Receptor

Cat.No: T34081

Synonym: NEU-P-11,NEU-P 11,NEU-P11

Target: P2X Receptor, 5-HT Receptor, MT Receptor, Sodium Channel, TRP/TRPV Channel

Cat.No: T0976

Synonym: 残杀威,Aprocarb,Propoxure,Baygon

Target: AChR, Antifungal

Dihydroergocristine mesylate

Cat.No: T11043

Synonym: 甲磺酸双氢麦角汀,DHEC (mesylate)

Target: Beta Amyloid

Cat.No: T22232

Cat.No: T13152

Target: Others

Cat.No: T24899

Synonym: Trimethoprim-sulfamethoxazole,Sulfamethoxazole-trimethoprim,TMP-SMX,Trimforte,Trimethoprimsulfa

Cat.No: T21247

Synonym: Allergefon,(+-)-Carbinoxamine,Paracarbinoxamine

F13714 fumarate

Cat.No: T37622

Synonym: F13714 fumarate

Cat.No: T33424

Synonym: MK 0952

Cat.No: T24450

Synonym: Lenetran Lenetran,TAB Lenetranat

Benzyldimethylstearylammonium chloride

Cat.No: T22268

Synonym: Benzyldimethylstearylammonium Chloride Hydrate,十八烷基二甲基苄基氯化铵

Target: Others

Cat.No: T24787

Cat.No: T20167

Synonym: Ro-34-2848,Ro 34-2848,Cilazapril (anhydrous),Ro34-2848,西拉普利

Cat.No: T68707

Diloxanide furoate

Cat.No: T15131

Target: Others

Cat.No: T20427

Synonym: NSC 1130,NSC1130,NSC-1130

Cat.No: T79855

Synonym: NYX-458,NYX-3054

Target: iGluR

Janelia Fluor® 669, SE

Cat.No: T39575

Synonym: JF669, SE,JF669,NHS,Janelia Fluor? 669, SE

Indapamide hemihydrate

Cat.No: T32154

Synonym: Tenaxil,Indapamide hydrate,D06401,UNII-W0LY35K007

Cat. No.	Product Name	Target	Signaling Pathways
T2721	Digitonin	Others	Others
	Digitonin 属于糖苷类天然产物，是一种去垢剂。Digitonin 具有抗肿瘤活性，可以与胆固醇分子结合从而增加细胞膜的通透性，对多种细胞的细胞膜具有裂解活性。
T75489	Mildiomycin
	Mildiomycin是一种针对大麦白粉病具有活性的链轮丝菌抗生素。该化合物能够抑制部分分枝杆菌和红桃菌的生长，然而，对大部分真菌和细菌则显示出无效性。
T8026	(-)-Limonene l-Limonene,(S)-(−)-Limonene,(-)-柠檬烯	Endogenous Metabolite	Metabolism
	(S)-(-)-Limonene (l-Limonene) 是一种存在多种松针油和松节油中的单萜烯，能轻微的引起支气管收缩。
T0732	Benzyl alcohol Benzoyl alcohol,苯甲醇,Benzenemethanol,Phenylcarbinol,Phenylmethanol	Dehydrogenase	Metabolism
	Benzyl alcohol (Benzenemethanol) 是一种无色液体，是一种芳香醇，带有温和的芳香气味。
TQ0298	Fagomine D-Fagomine	ROS; glycosidase	Immunology/Inflammation; Metabolism
	Fagomine (D-Fagomine) 是一种温和的糖苷酶 (glycosidase) 抑制剂，是1-脱氧野尻霉素（DNJ）的类似物，具有降血糖活性，Fagomine 降低了细胞内活性氧（ROS）的产生和丙二醛（MDA）水平。
T2S0491	Isoeugenol acetate 乙酸异丁香酚酯,Isoeugenyl acetate,Acetisoeugenol,Acetylisoeugenol,乙酸异丁香酚酯，乙酰基异丁香酚;2-甲氧基-4-丙烯基苯基乙酸酯	AChE; Antifungal	Microbiology/Virology; Neuroscience
	Isoeugenol acetate (Acetylisoeugenol) 是肉豆蔻，丁香和肉桂的精油成分，对某些代谢酶如乙酰胆碱酯酶，能够抑制α-糖苷酶和 α-淀粉酶。它用于医疗和化妆品工业，具有抗氧化，抗癌，抗菌和抗炎作用。
T5266	Tricaprilin Glycerol Tri-n-octanoate,三辛酸甘油酯,trioctanoin,tricaprylic glyceride,Glyceryl trioctanoate	Others; Endogenous Metabolite	Metabolism; Others
	Tricaprilin (Glycerol Tri-n-octanoate) 能够用于研究轻度到中度阿尔茨海默病患者，具有抗惊厥和植物代谢产物的活性。
T1126	Penicillin V Potassium 青霉素V钾,Penicillin V potassium salt,Phenoxymethylpenicillin potassium salt	Antibacterial; Antibiotic	Microbiology/Virology
	Penicillin V Potassium (Phenoxymethylpenicillin potassium salt) 是一种有口服活性的抗生素。它可抑制链球菌，艰难梭菌和金黄色葡萄球菌的生长，可研究中耳炎，鼻窦炎，咽炎和扁桃体炎。
TN1727	Helichrysetin 4,2',4'-三羟基-6'-甲氧基查耳酮,蜡菊亭	Apoptosis; HIV Protease	Apoptosis; Microbiology/Virology; Proteases/Proteasome
	Helichrysetin 是从豆蔻果实中分离出的一种天然产物，是一种 DNA 结合抑制剂，可抑制原位导管癌DCIS 的形成。它抑制细胞生长，可诱导 A549 细胞凋亡。
T3S0381	Chrysophanol 8-O-glucoside	Serine Protease	Proteases/Proteasome
	Chrysophanol 8-O-glucoside 来自Rumex acetosa 根部，具有中等的弹性蛋白酶抑制特性。它具有温和的细胞毒性和抗糖尿病特性，能够在胰岛素刺激的葡萄糖转运途径中发挥代谢作用。
T0690	Quinine 奎宁树	Potassium Channel; Platelet aggregation; Parasite	Membrane transporter/Ion channel; Microbiology/Virology; Others
	Quinine 是一种从金鸡纳树皮中提取的生物碱，用于预防和治疗疟疾。它也用于特发性肌肉痉挛，可抑制电压脉冲引起的 MT mSlo3 (KCa5.1) 通道 +100 mV 电流, 其IC50值为 169 μM，是一种钾离子通道抑制剂。
T5558	Chelidonic acid Jervaic acid,Jerva acid,白屈菜酸,γ-Pyrone-2,6-dicarboxylic acid	NF-κB; Caspase	Apoptosis; NF-κB; Proteases/Proteasome
	Chelidonic acid (Jervaic acid) 是从白屈菜中分到的酸类物质，用作温和的镇痛剂、抗菌剂和中枢神经系统镇静剂。它是谷氨酸脱羧酶抑制剂，Ki 值为 1.2 μM。它可能通过抑制 NF-κB 和caspase-1来降低 IL-6 的产生抗炎作用。
T2O2777	L-Threonine 苏氨酸,threonine,L-苏氨酸	Others; Endogenous Metabolite	Metabolism; Others
	L-Threonine (threonine) 是人体必需氨基酸，是神经系统的重要氨基酸。L-Threonine 在卟啉和脂肪代谢中也起着重要作用，防止肝脏脂肪堆积。L-Threonine 可用于治疗肠道疾病和消化不良，也可用于缓解焦虑和轻度抑郁。
T2175	Apigenin C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400	P450; Autophagy	Autophagy; Metabolism
	Apigenin (NSC 83244) 是从韩信草中提取的一种天然产物，是一种竞争性CYP2C9抑制剂，Ki 为 2 μM。它被用作镇静剂、温和的镇痛剂和安眠药。
T0224	Meropenem 美罗培南,SM 7338	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Meropenem (SM 7338) 是一种具有广谱抗菌活性的碳青霉烯抗生素，对敏感和耐药的淋病奈瑟氏球菌，流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL，0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T4716	Pyrrole-2-carboxylic acid 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline	Endogenous Metabolite	Metabolism
	Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类，从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。
T4947	3-Hydroxybutyric acid Butanoic acid,3-羟基丁酸	Endogenous Metabolite	Metabolism
	3-Hydroxybutyric acid (Butanoic acid) 是一种人内源性代谢物，在 I 型糖尿病中升高。它能够调节膜脂的性质。
TN5117	Taxiphyllin	Tyrosinase; Antifection	Microbiology/Virology; Proteases/Proteasome
	Taxiphyllin can inhibit tyrosinase activity in vitro significantly and is a potent tyrosinase inhibitor. Taxiphyllin displays mild antibacterial activity against Staphylococcus aureus.
T20854	Isethionic acid Hydroxyethylsulfonic acid,Ethanolsulfonic acid
	Isethionic acid, a major metabolite in F. cylindrus, is an organosulfur compound containing a short-chain alkane sulfonate linked to a hydroxyl group. It is a water-soluble liquid for the manufacture of mild, biodegradable, and high-foaming anionic surfac
TN4438	Ligucyperonol	Others	Others
	Ligucyperonol exhibits significant activities on protecting muscle cells from mild to moderate oxidative stress.
TN3742	Cycloeucalenol	Others	Others
	Cycloeucalenol produces mild cardiotonic effects. Cycloeucalenol and its regio-isomer were present in a ratio of 1.04:1, a dose-dependent decrease in cell viability was observed.
T83257	7(8)-Dehydroschisandrol A
	7(8)-Dehydroschisandrol A (Compound 4a)为从Schizandra chinensis Baill分离的木脂素，对激性胃溃疡表现出较弱抑制效果。
TN4570	Minumicrolin	Others	Others
	Minumicrolin is a plant growth inhibitor against the 2nd leaf sheath elongation of rice seedlings. Murrangatin exhibits cytotoxicity against cholangiocarcinoma cell line, KKU-100, it might be valuable anti-tumor-promoting agents. Minumicrolin shows mild butyrylcholinesterase inhibition activity.
TN3721	Cryptofolione	Antifection	Microbiology/Virology
	Z-Cryptofolione and Cryptomoscatone D2 as highly efficacious inhibitors of the G(2) checkpoint, G(2) checkpoint inhibitors can force cells arrested in G(2) phase by DNA damage to enter mitosis. Cryptofolione shows moderate cytotoxicity in both macrophages and T. cruzi amastigotes, it also displays a mild inhibitory effect on the promastigote form of Leishmania spp.
TN6028	Gardneramine
	Gardneramine has a mild central depressive effect. Gardneramine and hirsutine show a local anesthetic action, they also can inhibit the ganglionic transmission of the dog urinary bladder and that the blockade of the nicotinic receptor plays a main role.
TN3438	Arborinine	HCV Protease; Antifection	Microbiology/Virology; Proteases/Proteasome
	Arborinine shows mild in vitro antibacterial activity, it possesses moderate levels of anti-hepatitis C virus(HCV) activities with the IC50 values being 6.4 ± 0.7 ug/ml. Arborinine shows antifeedant activity against Spodoptera frugiperda. Arborinin shows
T82445	Erinacine P
	Erinacine P（化合物1）为担子菌猴头菇YB4-6237菌丝体分离得到的木犀草素亲代代谢产物。其在温和条件下可化学转化为猴头素B，继而可转化为猴头素A。
T82219	Heilaohuguosu F
	Heilaohuguosu F (compound 6)为一类四氢呋喃木脂素，表现出轻度肝脏保护效果。该化合物对于APAP诱导的HepG2细胞所呈现的肝毒性具有微弱的防护作用。
TN1834	Kobusin 去甲槟郎碱,自旋七叶素	Others; NOS; NF-κB	Immunology/Inflammation; NF-κB; Others
	Kobusin, a Calmodulin inhibitor, shows mild antiplasmodial,anti-inflammatory, and cytotoxic activities; it may be beneficial for the treatment of neuro-inflammatory diseases through the inhibition of iNOS expression and peroxynitrite scavenging potential. Kobusin can mildly reduce gastrointestinal motility in mice, it activates CFTR and CaCCgie chloride channel activities in mouse colonic epithelia and shows inhibitory effects toward ANO1/CaCC-mediated short-circuit currents in ANO1/CaCC-express...
T83117	Angeloylbinankadsurin A
	Angeloylbinankadsurin A（化合物7）是一种从黑虎胡的EtOAc和CH2Cl2提取物中分离出的抗RA试剂，它在RA-FLS细胞上显示出显著的抑制活性（IC50=11.70 μM），同时对人类癌细胞系（Hela和BGC-823）表现出较低的毒性（IC50分别为19.9 μM和21.93 μM）。

天然产物

Cat.No: T2721

Target: Others

Cat.No: T75489

Cat.No: T8026

Synonym: l-Limonene,(S)-(−)-Limonene,(-)-柠檬烯

Target: Endogenous Metabolite

Cat.No: T0732

Synonym: Benzoyl alcohol,苯甲醇,Benzenemethanol,Phenylcarbinol,Phenylmethanol

Target: Dehydrogenase

Cat.No: TQ0298

Synonym: D-Fagomine

Target: ROS, glycosidase

Isoeugenol acetate

Cat.No: T2S0491

Synonym: 乙酸异丁香酚酯,Isoeugenyl acetate,Acetisoeugenol,Acetylisoeugenol,乙酸异丁香酚酯，乙酰基异丁香酚;2-甲氧基-4-丙烯基苯基乙酸酯

Target: AChE, Antifungal

Cat.No: T5266

Synonym: Glycerol Tri-n-octanoate,三辛酸甘油酯,trioctanoin,tricaprylic glyceride,Glyceryl trioctanoate

Target: Others, Endogenous Metabolite

Penicillin V Potassium

Cat.No: T1126

Synonym: 青霉素V钾,Penicillin V potassium salt,Phenoxymethylpenicillin potassium salt

Target: Antibacterial, Antibiotic

Cat.No: TN1727

Synonym: 4,2',4'-三羟基-6'-甲氧基查耳酮,蜡菊亭

Target: Apoptosis, HIV Protease

Chrysophanol 8-O-glucoside

Cat.No: T3S0381

Target: Serine Protease

Cat.No: T0690

Synonym: 奎宁树

Target: Potassium Channel, Platelet aggregation, Parasite

Chelidonic acid

Cat.No: T5558

Synonym: Jervaic acid,Jerva acid,白屈菜酸,γ-Pyrone-2,6-dicarboxylic acid

Target: NF-κB, Caspase

Cat.No: T2O2777

Synonym: 苏氨酸,threonine,L-苏氨酸

Target: Others, Endogenous Metabolite

Cat.No: T2175

Synonym: C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400

Target: P450, Autophagy

Cat.No: T0224

Synonym: 美罗培南,SM 7338

Target: Others, Antibacterial, Antibiotic

Pyrrole-2-carboxylic acid

Cat.No: T4716

Synonym: 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline

Target: Endogenous Metabolite

3-Hydroxybutyric acid

Cat.No: T4947

Synonym: Butanoic acid,3-羟基丁酸

Target: Endogenous Metabolite

Cat.No: TN5117

Target: Tyrosinase, Antifection

Isethionic acid

Cat.No: T20854

Synonym: Hydroxyethylsulfonic acid,Ethanolsulfonic acid

Cat.No: TN4438

Target: Others

Cat.No: TN3742

Target: Others

7(8)-Dehydroschisandrol A

Cat.No: T83257

Cat.No: TN4570

Target: Others

Cat.No: TN3721

Target: Antifection

Cat.No: TN6028

Cat.No: TN3438

Target: HCV Protease, Antifection

Cat.No: T82445

Heilaohuguosu F

Cat.No: T82219

Cat.No: TN1834

Synonym: 去甲槟郎碱,自旋七叶素

Target: Others, NOS, NF-κB

Angeloylbinankadsurin A

Cat.No: T83117

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