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43

抑制剂 & 化合物

11

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Cat. No. Product Name Target Signaling Pathways
T8423 ML417

Dopamine Receptor; Arrestin GPCR/G Protein; Neuroscience
ML417 是选择性的,可透过血脑屏障的 D3 多巴胺受体激动剂,EC50=38 nM。它能够促进 D3R 介导的 β-arrestin 易位、G 蛋白介导的信号传导和 pERK 磷酸化,对其他 GPCR 介导的信号传导影响小。它对毒素诱导的多巴胺能神经元变性具有神经保护活性。
T8887 2'MeO6MF

GABA Receptor Membrane transporter/Ion channel; Neuroscience
2'MeO6MF 是可透过血脑屏障的α2β1γ2L 和所有含α1的GABAA 受体的正变构调节剂。它也可以直接激活α2β2/3和α2β2/3γ2L GABAA 受体。它具有抗焦虑和促进安定作用。它可提供神经保护作用并改善功能恢复,还可抑制中风诱发的炎症反应。
T21551 2-hexyl-4-Pentynoic Acid

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
2-Hexyl-4-pentynoic acid 是一种丙戊酸 (VPA) 衍生物,可以抑制HDAC(IC50=13 µM) 和诱导HSP70。它可引起培养神经元的组蛋白高度乙酰化,防止谷氨酸诱导的兴奋性毒性,具有强大的神经保护作用。
T1476 Pramipexole

SND 919,普拉克索

Dopamine Receptor GPCR/G Protein; Neuroscience
Pramipexole (SND 919) 是能够透过血脑屏障的 D2 型多巴胺受体的选择性激动剂,对 D2 型受体、D2、D3、D4亚型受体的Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM。它可用于研究帕金森综合症和腿多动综合征。
T7644 DPN

Diarylpropionitrile,2,3-双(4-羟苯基)丙腈

Apoptosis; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones
DPN (Diarylpropionitrile) 是一种非甾体雌激素受体 ERβ选择性配体,其 EC50值为 0.85 nM。DPN 在许多神经系统疾病具有神经保护作用。
T1057 Azilsartan

TAK-536,阿齐沙坦

RAAS Endocrinology/Hormones
Azilsartan (TAK-536) 是一种高活性的血管紧张素Ⅱ1型受体特异性拮抗剂(IC50:2.6 nM)。
T6540 Ibuprofen Lysine

布洛芬赖氨酸盐,Neoprofen

COX Immunology/Inflammation; Neuroscience
Ibuprofen Lysine (Neoprofen) 是一种非甾体抗炎药。
T3198L PRE-084 hydrochloride

Sigma receptor GPCR/G Protein
PRE-084 hydrochloride 是 σ1 的选择性激动剂在sigma 受体检测中,IC50值为44 nM。
T1394 Ibuprofen

Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil

COX Immunology/Inflammation; Neuroscience
Ibuprofen (Advil) 是一种丙酸衍生物和非甾体抗炎药 (NSAID),具有抗炎、镇痛和解热作用。它是COX-1和COX-2的抑制剂,IC50值分别为 13 和 370 μM,导致前列腺素和血栓素前体的形成减少。
T8505 SC-236

4-(5-(4-氯苯基)-3-(三氟甲基)-1H-,Sc 236

Apoptosis; COX; PPAR Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience
SC-236 (Sc 236) 是一种具有口服活性的COX-2特异性抑制剂和PPARγ激动剂。它可通过 c-Jun 氨基端抑制激活蛋白-1活性,在小鼠模型中通过抑制 ERK 的磷酸化发挥抗炎作用。
T0334 Rosiglitazone

BRL49653,罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone (BRL49653) 是一种 PPARγ 激动剂、TRPC5 激活剂和 TRPM3 抑制剂,具有口服活性。Rosiglitazone 也是一种降糖剂,是噻唑烷二酮类胰岛素增敏剂。
T2226 Pergolide mesylate

甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。
T6951 Pramipexole dihydrochloride hydrate

Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索

Dopamine Receptor GPCR/G Protein; Neuroscience
Pramipexole dihydrochloride hydrate (Mirapex) 是选择性的,具有血脑屏障 (BBB) 渗透性的 D2 型多巴胺受体激动剂,对 D2 型受体、D2、D3、D4亚型受体的 Ki 分别为 2.2 nM、3.9 nM、0.5 nM、1.3 nM,可用于研究帕金森综合症和腿多动综合征。
T6646 Rosiglitazone hydrochloride

盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone hydrochloride (BRL-49653 HCl) 是一种降血糖药物,通过与脂肪细胞中的 PPAR 受体结合来刺激胰岛素分泌。它对 PPARγ1、PPARγ2 和 PPARγ 的EC50值分别为 30 nM、100 nM 和 60 nM。它也是TRPC5的激活剂和TRPM3的抑制剂。
T9956 VK-28

Mitochondrial Metabolism; Lipid Metabolism
VK-28 是一种具有神经保护作用的脑渗透性铁螯合剂。 VK-28 抑制基础以及铁诱导的线粒体脂质过氧化。
T22900 L-701252

L-701,252

NMDAR Neuroscience
L-701252 是一种有效的甘氨酸位点 NMDA 受体拮抗剂,IC50 值为 420 nM。L-701252 对全脑缺血提供小范围的神经保护。
T10212 A2AR-agonist-1

N-(2-(1H-Indol-3-yl)ethyl)adenosine

Others; Adenosine Receptor GPCR/G Protein; Neuroscience; Others
A2AR-agonist-1 (N-(2-(1H-Indol-3-yl)ethyl)adenosine)是一种有效的 A2AR 和 ENT1激动剂, Ki 值 分别为 4.39 μM 和 3.47 μM。
T27748L KRP-199 sodium

KRP-199 sodium(221164-28-9 Free base)

GluR Neuroscience
KRP-199 sodium 在体外对AMPA-R具有很高的效力和选择性,在体内表现出良好的神经保护作用。
T21757 BRL 52537 hydrochloride

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
BRL 52537 hydrochloride 是一种选择性和特异性 KOR 激动剂,与缺血性神经元损伤的神经保护有关。它用于研究中风和心脏病发作的潜在治疗方法以及更一般的大脑研究。
T76863 Elezanumab

AE12-1Y-QL,ABT-555

TGF-beta/Smad Stem Cells
Elezanumab(ABT-555) 是一种有效的人抗 RGMa 单克隆抗体。Elezanumab 通过 SMAD1/5/8 通路发挥对 RGMa 介导的 BMP 信号传导的抑制作用,IC50 约为 97 pM。在神经元损伤和脱髓鞘模型中,Elezanumab 促进神经再生、神经保护和神经恢复。Elezanumab 促进皮质脊髓轴突生长为脊髓灰质,并增强腹角的血清素能神经支配,形成颈部病变尾部的突触连接。
T1993 J-147

J147

Epigenetic Reader Domain; Dopamine Receptor; Monoamine Oxidase Chromatin/Epigenetic; GPCR/G Protein; Neuroscience
J-147 是一种高效的、具有口服活性的、可透过血脑屏障神经保护剂,可增强认知能力。它抑制单胺氧化酶 B 和多巴胺转运体,EC50分别为 1.88 μM 和 0.649 μM。它有研究阿尔茨海默氏症的潜力。
TP1079 (Arg)9 TFA (143413-47-2 free base)

Nona-L-arginine (TFA),(Arg)9 TFA,Peptide R9 (TFA)

Others Others
(Arg)9 TFA (Peptide R9 TFA) 是一种可渗透细胞的多肽,在谷氨酸模型实验模型中保护神经(IC50:0.78 μM)。
T23736 AND-302

AND 302

AND-302 is a potent agent of anticonvulsant. It also has in vitro neuroprotection.
T28117 MSN-50

MSN50,MSN 50

MSN-50, an inhibitor of Bax and Bak oligomerization, inhibits liposome permeabilization, prevents genotoxic cell death and promotes neuroprotection.
T24529 Neuroprotectant-7

Neuroprotectant7

Neuroprotectant-7 is a neuroprotectant for Alzheimer's disease. It displays significant neuroprotection and antioxidative properties. It also can cross the blood-brain barrier.
T16292 NFPS

Thrombin Proteases/Proteasome
NFPS exerts neuroprotection via glyR alpha1 subunit in the rat model of transient focal cerebral ischaemia and reperfusion. NFPS is a selective and non-competitive glycine transporter-1 (GlyT1) inhibitor (IC50s: 2.8 nM and 9.8 nM for hGlyT1 and rGlyT1, respectively).
T24787 SGE-201

SGE-201 is an allosteric modulator of N-methyl-D-aspartate receptors. SGE-201 also unmasked differences among the blockers in neuronal networks - measured either by suppression of activity in multi-electrode arrays or by neuroprotection against a mild exc
T78681 ITH12711

Phosphatase Metabolism
ITH12711为PP2A配体,具有穿透血脑屏障(BBB)的能力,其神经保护机制是通过恢复PP2A磷酸酶活性来实现。
T28894 SZV558

SZV 558,SZV-558

SZV558 is a potent inhibitor of both human and rodent MAO-B. SZV558 is safe in high doses with no hERG and mutagenic activities and demonstrated neuroprotection in an in vivo chronic model of PD.
T21470 Davunetide

AL-208,AL 208,AL 108,AL-108

Davunetide is an eight amino acid peptide (NAPVSIPQ) with potent neuroprotection in vitro and in vivo. Davunetide has been shown to enhance functional daily behaviors in schizophrenia patients and to increase memory scores in patients suffering from amnes
T35889 PB2

PB2, a tris(2-carboxyethyl)phosphine (TCEP) analogue, enhances the survival of retinal ganglion cells (RGCs) following axotomy in vitro. Even at nanomolar and picomolar concentrations, PB2 demonstrates pronounced efficacy in promoting RGC survival. Notably, PB2 exhibits superior permeability compared to TCEP. Serving as a potent reducing agent, PB2 provides robust neuroprotection for RGCs[1].
T41058 Nelonemdaz potassium

Neu2000potassium,Salfaprodil

Nelonemdaz potassium (also known as Salfaprodil) is a potent NR2B-selective and uncompetitive antagonist of N-methyl-D-aspartate (NMDA). This compound exhibits remarkable neuroprotection against cell death induced by both NMDA and free radicals, in addition to its role as a free radical scavenger.
T75408 Batroxobin

Batroxobin (DF-521),一种从Bothrops atrox moojeni获得的蛇毒,能促进血栓溶解,防止血栓复发并具有神经保护作用,显示出在脑静脉血栓性疾病研究中的潜力。
T78094 Eglumegad hydrochloride

LY354740 hydrochloride,Eglumetad hydrochloride

Eglumegad (LY354740) hydrochloride是一种高效且选择性的group II (mGlu2/3) receptor激动剂,其对人mGlu2和mGlu3受体的IC50值分别是5和24 nM。该化合物能够保护神经元不受NMDA毒性影响,并表现出抗焦虑及抗精神病样作用。
T60695 DPQ

DPQ 是PARP-1的有效抑制剂,可用于研究神经保护。DPQ 可降低 N-甲基-D-天冬氨酸(NMDA) 诱导的 PARP 激活,将 ATP 恢复至接近正常水平,并且显著减轻 NMDA 暴露模型中的神经元损伤。
T62743 AChE-IN-10

AChE-IN-10 (Compound 24r) 是一种 AChE 的有效抑制剂,其 IC50 值为 2.4 nM。AChE-IN-10 在 AChE 存在下能够降低淀粉样蛋白的聚集。AChE-IN-10 对 AChE 表现出有效抑制作用,可以降低 S396 残基的 tau 磷酸化,挽救神经元形态和增加细胞活力,进而提供神经保护作用。
T80210 TAT-GluN2BCTM

DAPK Apoptosis
TAT-GluN2BCTM 是一种靶向DAPK1的膜透性肽,能够促使活性DAPK1定向降解于溶酶体。该化合物通过降低DAPK1的表达,有助于防护神经元免遭氧化应激和NMDAR-介导的兴奋毒性。TAT-GluN2BCTM常用于神经保护性研究领域。
T83963 Z-DEVD-FMK Caspase-3 Inhibitor

Z-DEVD-FMK Caspase-3 Inhibitor 是一种可渗透细胞膜的、不可逆的 caspase-3/CPP32 抑制剂,能够抑制肿瘤细胞的凋亡。在动物体内,它在大鼠发作后的海马区具有神经保护作用,且显著减少创伤后的细胞凋亡,并在诱发的大鼠创伤性脑损伤之前和之后改善神经学恢复情况。
T79569 AChE/Aβ-IN-1

AChE/Aβ-IN-1(compound 32)是一种双功能化合物,既表现出高效的AChE抑制活性,IC50值为86 nM,又能作为NMDA受体(GluN1-1b/GluN2B亚基组合)的拮抗剂,其IC50为3.876 μM。此外,它能够抑制Aβ聚集,且表现出优秀的血脑屏障穿透能力和神经保护效果,能在大鼠模型中显著改善认知和空间记忆障碍。
T73989 Tirilazad

Tirilazad是一种21-氨基类固醇非糖皮质激素,具有抑制脂质过氧化的能力。它对于脑或脊髓中因创伤、中风、缺血再灌注损伤所致的损害有减轻作用。此外,Tirilazad还展现出针对新型肺炎病毒的抗病毒活性,并在缺血性中风中提供神经保护,适用于蛛网膜下腔出血研究场景。
T16797 RPR104632

NMDAR Neuroscience
RPR104632 是一种新型有效的位于 NMDA 甘氨酸位点的拮抗剂,具有神经保护活性。
T13976 (Arg)9

Peptide R9,Nona-L-arginine

Others Others
(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).
T64672 Colivelin TFA

Colivelin (sequence SALLRSIPAPAGASRLLLLTGEIDLP) is composed of activity-dependent neurotrophic factor (ADNF) C-terminally fused to AGA-(C8R)HNG17, a potent HN derivative. It works as a neuroprotective peptide and activator of STAT3. Colivelin-induced neuroprotection has been confirmed to occur via two neuroprotective pathways: one mediated by Ca2+/calmodulin-dependent protein kinase IV, triggered by ADNF, and one mediated by signal transducer and activator of transcription 3, triggered by HN. Co...

化合物

ML417
Cat.No: T8423
Synonym:
Target: Dopamine Receptor, Arrestin
2'MeO6MF
Cat.No: T8887
Synonym:
Target: GABA Receptor
2-hexyl-4-Pentynoic Acid
Cat.No: T21551
Synonym:
Target: HDAC
Pramipexole
Cat.No: T1476
Synonym: SND 919,普拉克索
Target: Dopamine Receptor
DPN
Cat.No: T7644
Synonym: Diarylpropionitrile,2,3-双(4-羟苯基)丙腈
Target: Apoptosis, Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Autophagy
Azilsartan
Cat.No: T1057
Synonym: TAK-536,阿齐沙坦
Target: RAAS
Ibuprofen Lysine
Cat.No: T6540
Synonym: 布洛芬赖氨酸盐,Neoprofen
Target: COX
PRE-084 hydrochloride
Cat.No: T3198L
Synonym:
Target: Sigma receptor
Ibuprofen
Cat.No: T1394
Synonym: Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil
Target: COX
SC-236
Cat.No: T8505
Synonym: 4-(5-(4-氯苯基)-3-(三氟甲基)-1H-,Sc 236
Target: Apoptosis, COX, PPAR
Rosiglitazone
Cat.No: T0334
Synonym: BRL49653,罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Pergolide mesylate
Cat.No: T2226
Synonym: 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Pramipexole dihydrochloride hydrate
Cat.No: T6951
Synonym: Pramipexole 2HCl Monohydrate,普拉克索盐酸盐水合物,Mirapex,普拉克索
Target: Dopamine Receptor
Rosiglitazone hydrochloride
Cat.No: T6646
Synonym: 盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
VK-28
Cat.No: T9956
Synonym:
Target: Mitochondrial Metabolism, Lipid
L-701252
Cat.No: T22900
Synonym: L-701,252
Target: NMDAR
A2AR-agonist-1
Cat.No: T10212
Synonym: N-(2-(1H-Indol-3-yl)ethyl)adenosine
Target: Others, Adenosine Receptor
KRP-199 sodium
Cat.No: T27748L
Synonym: KRP-199 sodium(221164-28-9 Free base)
Target: GluR
BRL 52537 hydrochloride
Cat.No: T21757
Synonym:
Target: Opioid Receptor
Elezanumab
Cat.No: T76863
Synonym: AE12-1Y-QL,ABT-555
Target: TGF-beta/Smad
J-147
Cat.No: T1993
Synonym: J147
Target: Epigenetic Reader Domain, Dopamine Receptor, Monoamine Oxidase
(Arg)9 TFA (143413-47-2 free base)
Cat.No: TP1079
Synonym: Nona-L-arginine (TFA),(Arg)9 TFA,Peptide R9 (TFA)
Target: Others
AND-302
Cat.No: T23736
Synonym: AND 302
Target:
MSN-50
Cat.No: T28117
Synonym: MSN50,MSN 50
Target:
Neuroprotectant-7
Cat.No: T24529
Synonym: Neuroprotectant7
Target:
NFPS
Cat.No: T16292
Synonym:
Target: Thrombin
SGE-201
Cat.No: T24787
Synonym:
Target:
ITH12711
Cat.No: T78681
Synonym:
Target: Phosphatase
SZV558
Cat.No: T28894
Synonym: SZV 558,SZV-558
Target:
Davunetide
Cat.No: T21470
Synonym: AL-208,AL 208,AL 108,AL-108
Target:
PB2
Cat.No: T35889
Synonym:
Target:
Nelonemdaz potassium
Cat.No: T41058
Synonym: Neu2000potassium,Salfaprodil
Target:
Batroxobin
Cat.No: T75408
Synonym:
Target:
Eglumegad hydrochloride
Cat.No: T78094
Synonym: LY354740 hydrochloride,Eglumetad hydrochloride
Target:
DPQ
Cat.No: T60695
Synonym:
Target:
AChE-IN-10
Cat.No: T62743
Synonym:
Target:
TAT-GluN2BCTM
Cat.No: T80210
Synonym:
Target: DAPK
Z-DEVD-FMK Caspase-3 Inhibitor
Cat.No: T83963
Synonym:
Target:
AChE/Aβ-IN-1
Cat.No: T79569
Synonym:
Target:
Tirilazad
Cat.No: T73989
Synonym:
Target:
RPR104632
Cat.No: T16797
Synonym:
Target: NMDAR
(Arg)9
Cat.No: T13976
Synonym: Peptide R9,Nona-L-arginine
Target: Others
Colivelin TFA
Cat.No: T64672
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2919 Sesamin

Fagarol,Fsesamin,芝麻素

Others Others
Sesamin (Fsesamin) 是多不饱和脂肪酸生物合成中的选择性delta 5 去饱和酶抑制剂,是在芝麻油中存在丰富的木脂素。它对脑缺血具有有效的神经保护作用。
T0683 Mevastatin

Compactin,ML236B,美伐他汀

Apoptosis; Antibacterial; Antibiotic; HMG-CoA Reductase; Autophagy; Lipid Apoptosis; Autophagy; Metabolism; Microbiology/Virology
Mevastatin (ML236B) 是他汀类 HMG-CoA 还原酶抑制剂。它是一种降脂药,可诱导细胞凋亡,将癌细胞阻滞在 G0/G1期。它还可增加内皮型一氧化氮合酶的 mRNA 和蛋白质水平。它有抗肿瘤活性,用于心血管疾病的研究。
T0883 Tramiprosate

Homotaurine,3-Amino-1-propanesulfonic acid,Alzhemed,高牛黄酸

Beta Amyloid; GABA Receptor Membrane transporter/Ion channel; Neuroscience
Tramiprosate (Alzhemed) 是一种具有口服活性的、可透过血脑屏障的天然氨基酸,存在于各种红色海藻中,能够可溶性 Aβ 结合并以非原纤维形式维持 Aβ。它是一种 GABA 类似物,具有神经保护,抗惊厥和抗高血压的活性。
T4024 Norharmane

2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满

DNA; Endogenous Metabolite; Monoamine Oxidase DNA Damage/DNA Repair; Metabolism; Neuroscience
Norharmane (β-Carboline) 是一种有效的选择性单胺氧化酶 A (MAO-A) 抑制剂,Ki=3.34 μM。
T2961 Notoginsenoside R1

Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1

Apoptosis; ERK; Beta Amyloid Apoptosis; MAPK; Neuroscience
Notoginsenoside R1 (Sanchinoside R1) 是一种从三七中分离出来的皂苷,具有抗氧化、抗炎、抗血管生成和抗凋亡的活性。它有神经保护和抗缺血/再灌注损伤的心脏保护作用。
T2163 Dihydrocapsaicin

CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide

Others; TRP/TRPV Channel Membrane transporter/Ion channel; Others
Dihydrocapsaicin (CCRIS1589) 是一种天然来源的辣椒素,是TRPV1的选择性激动剂,同时可以增加 p-Akt 水平。它可以增强低温诱导的神经保护。
T6S1587 Notoginsenoside R2

三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2

Others; Nrf2 Immunology/Inflammation; Others
Notoginsenoside R2 (20(S)-Notoginsenoside R2) 是一种新分离三七皂苷,表现出对6-OHDA 诱导的氧化应激及细胞凋亡的保护作用。
T2879 Fisetin

漆黄素,非瑟酮

TNF; Sirtuin; PPAR Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Fisetin 是在许多水果和蔬菜中发现的一种天然黄酮醇,有抗氧化、抗癌和神经保护作用。
T6S0721 Orientin

荭草苷,Lutexin,Luteolin-8-glucoside

Others Others
Orientin (Luteolin-8-glucoside) 是天然存在的生物活性类黄酮,是一种有前景的神经保护剂,具有多种生物特性,如抗炎、抗肿瘤、抗氧化、保护心脏等。它有用于神经性疼痛研究潜力。
T2808 Bilobalide

白果内酯,银杏内酯,(-)-Bilobalide

Apoptosis; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism
Bilobalide ((-)-Bilobalide) 是银杏叶中的的一种倍半萜三内酯成分,抑制 NMDA 诱导的胆碱流出,IC50值为 2.3 µM。它通过激活 SH-SY5Y 细胞中的 PI3K/Akt 通路来防止细胞凋亡。对神经元发挥保护和营养作用。
TN5639 Rocaglaol

Ferrugin,Aglaiastatin A

Rocaglaol is a potent anticancer drug that induces apoptosis of LNCaP cells through the mitochondrial pathway and its G2/M-phase cell cycle arrest is associated with the down-regulation of Cdc25C and the dephosphorylation of Cdc2. Rocaglaol can reduce tis

天然产物

Sesamin
Cat.No: T2919
Synonym: Fagarol,Fsesamin,芝麻素
Target: Others
Mevastatin
Cat.No: T0683
Synonym: Compactin,ML236B,美伐他汀
Target: Apoptosis, Antibacterial, Antibiotic, HMG-CoA Reductase, Autophagy, Lipid
Tramiprosate
Cat.No: T0883
Synonym: Homotaurine,3-Amino-1-propanesulfonic acid,Alzhemed,高牛黄酸
Target: Beta Amyloid, GABA Receptor
Norharmane
Cat.No: T4024
Synonym: 2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满
Target: DNA, Endogenous Metabolite, Monoamine Oxidase
Notoginsenoside R1
Cat.No: T2961
Synonym: Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1
Target: Apoptosis, ERK, Beta Amyloid
Dihydrocapsaicin
Cat.No: T2163
Synonym: CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide
Target: Others, TRP/TRPV Channel
Notoginsenoside R2
Cat.No: T6S1587
Synonym: 三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2
Target: Others, Nrf2
Fisetin
Cat.No: T2879
Synonym: 漆黄素,非瑟酮
Target: TNF, Sirtuin, PPAR
Orientin
Cat.No: T6S0721
Synonym: 荭草苷,Lutexin,Luteolin-8-glucoside
Target: Others
Bilobalide
Cat.No: T2808
Synonym: 白果内酯,银杏内酯,(-)-Bilobalide
Target: Apoptosis, Endogenous Metabolite, Autophagy
Rocaglaol
Cat.No: TN5639
Synonym: Ferrugin,Aglaiastatin A
Target:
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