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Cat. No. | Product Name | ||
---|---|---|---|
L9300 | 大环化合物库 | 210 compounds | |
210 种活性已知的大环化合物,用于高通量、高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T33816 |
Ordopidine
ACR-325,ACR 325,ACR325 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Ordopidine (ACR325) 是一种多巴胺能稳定剂,可抑制精神刺激剂引起的多动症,并在不活动时刺激行为。Ordopidine 在体外作为多巴胺 D2 受体拮抗剂起作用,尽管亲和力低,但其依赖于特定状态的行为效应特征是 D2 受体拮抗剂所不具备的。 | |||
T34616 |
Seridopidine
ACR-343,ACR 343,ACR343 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Seridopidine (ACR343) 是一种多巴胺能活性调节剂,可作为精神分裂症、帕金森病和抽动秽语综合征的口服疗法。 | |||
T34210 |
Pyrophosphoric acid, chloromethyl trimethyl ester
ACR-58-26,ACR58-26,ACR 58-26 |
||
Pyrophosphoric acid, chloromethyl trimethyl ester is an agricultural and biochemical product. | |||
T7352 |
Pridopidine
ACR16,ASP2314,FR310826,4-[3-(甲磺酰基)苯基]-1-丙基哌啶 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Pridopidine (FR310826) 是多巴胺稳定剂,是一种低亲和力的多巴胺 D2 受体拮抗剂。它高亲和力作用于 sigma 1受体,Ki=70-80 nM,比其对 D2R 的亲和力高约 100 倍。 | |||
T65288 |
Methacrylic anhydride
|
Others | Others |
Methacrylic anhydride 是一种可聚合 1,6- 二烯烃的化合物,可以通过自由基引发形成可溶的环己烷聚合物。Methacrylic anhydride 可以通过乙烯基自发聚合, 2-6- 二叔丁基 4- 甲基苯酚对此有抑制作用。Methacrylic anhydride 可用于研究新型水凝胶。 | |||
T5373 |
Acrizanib
LHA510 |
VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
Acrizanib (LHA510) 是一种 VEGFR-2 的抑制剂,其对 BaF3-VEGFR-2 的 IC50 值为 17.4 nM。 | |||
T14118 |
Acridine Orange hydrochloride
吖啶橙,3,6-双(二甲基氨基)吖啶 |
Others | Others |
Acridine Orange hydrochloride 是可透过细胞的荧光染料。 它与核酸结合,导致光谱发射发生改变。它被用作超活体染色剂和荧光细胞化学。 它可能导致微生物发生突变。 | |||
T77682 |
(E)-3-(Naphth-1-yl)acrylic acid
3-(1-Naphthyl)acrylic acid |
Others | Others |
(E)-3-(Naphth-1-yl)acrylic acid (3-(1-Naphthyl)acrylic acid) 是一种生化试剂,可用于合成多种化合物,参与机体的很多反应。 | |||
T21439 |
Tacrine
他克林,CS 12602,Tacrinum,Tetrahydroaminocrine |
AChR | Neuroscience |
Tacrine (CS 12602) 一种间接胆碱能激动剂和中枢作用的抗胆碱酯酶。它被批准用于治疗阿尔茨海默病。 | |||
T24214 |
Phenamacril
JS39919,苯那普利,JS399 19 |
Myosin; Antifungal | Cytoskeletal Signaling; Microbiology/Virology |
Phenamacril (JS39919) 是一种氰基丙烯酸酯类杀菌剂,对镰刀菌,特别是禾谷镰刀菌有很强的抑制作用。它是一种特异性镰刀菌肌球蛋白 I 抑制剂。 | |||
T12137 |
N-(2-Hydroxypropyl)methacrylamide
|
Parasite | Microbiology/Virology |
N-(2-Hydroxypropyl)methacrylamide 用于合成共聚物,用于靶向递送内脏利什曼病中的抗寄生虫剂。 | |||
T2191 |
Tacrine hydrochloride (hydrate)
Tacrine,他克林盐酸盐水合物,Tacrine hydrochloride hydrate,Tetrahydroaminacrine,Tetrahydroaminoacridine |
AChR; AChE | Neuroscience |
Tacrine hydrochloride hydrate (Tetrahydroaminacrine) 是一种乙酰胆碱酯酶 (AChE) 和丁酰胆碱酯酶 (BChE) 的抑制剂,它们的IC50值分别为 31 nM 和 25.6 nM。 | |||
T5820 |
Amsacrine hydrochloride
acridinyl anisidide hydrochloride,盐酸胺苯吖啶,m-AMSA hydrochloride |
Topoisomerase; Autophagy | Autophagy; DNA Damage/DNA Repair |
Amsacrine hydrochloride (acridinyl anisidide hydrochloride) 是一种拓扑异构酶 II 抑制剂,用于治疗急性髓细胞性白血病。 | |||
T19832 |
Acriflavine Hydrochloride
盐酸吖啶黄,Acriflavine HCl |
HIF | Angiogenesis; Chromatin/Epigenetic |
Acriflavine Hydrochloride (Acriflavine HCl) 是一种 HIF-1α 抑制剂。它通过靶向 HIF-1α 介导的途径并在体外和体内降低 PGK1、VEGF 和 HIF-1α 的水平发挥作用。 | |||
T24449 |
Mepacrine
Haffkinine,Erion |
Others | Others |
Mepacrine (Erion) 是一种吖啶衍生物,以前广泛用作抗疟药。它在细胞生物学实验中用作磷脂酶A2的抑制剂。 | |||
T1206 |
Amsacrine
AMSA,m-AMSA,安吖啶,CI-880,acridinyl anisidide |
Potassium Channel; Topoisomerase; Autophagy | Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel |
Amsacrine (AMSA) 是一种抗肿瘤剂,可以嵌入到肿瘤细胞的 DNA 中。它还表达拓扑异构酶抑制剂活性,特异性抑制拓扑异构酶 II。 | |||
T9322 |
N-Phenylacrylamide
|
Others | Others |
N-Phenylacrylamide 通过荧光转酰胺法抑制人重组 TGM2。 | |||
T8321 |
10-methyl-9-(phenoxycarbonyl) Acridinium
|
Others | Others |
10-methyl-9-(phenoxycarbonyl) Acridinium 是一种吖啶鎓酯,在碱性条件下与过氧化氢、过硫酸盐和其他氧化剂氧化后会产生荧光 10-methyl-9-acridone。 | |||
T2657 |
Elacridar
GW0918,依克立达,GW120918,GF120918,GG918 |
BCRP; P-gp | Membrane transporter/Ion channel; Neuroscience |
Elacridar (GG918) 是一种有效的 P-糖蛋白和BCRP 的抑制剂。 | |||
T6020 |
Pacritinib
SB1518 |
FLT; Tyrosine Kinases; JAK | Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors |
Pacritinib (SB1518) 是一种野生型 JAK2和 JAK2V617F 突变型抑制剂,IC50分别为 23 和 19 nM。它也抑制 FLT3及其突变型 FLT3D835Y,IC50分别为 22 和 6 nM。 | |||
T4557 |
Amylmetacresol
戊甲酚,5-Methyl-2-Pentylphenol |
Others; HIV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
Amylmetacresol (5-Methyl-2-Pentylphenol) 是一种有潜力研究咽喉痛相关疾病的抗病毒化合物。 | |||
T21556 |
Hydroxytacrine maleate
Velnacrine maleate,HP 029 maleate |
AChE | Neuroscience |
Hydroxytacrine maleate (Velnacrine maleate) 是一种胆碱酯酶(cholinesterase) 抑制剂,可增强啮齿动物的记忆力,可用于研究阿尔茨海默型老年性痴呆(SDAT)。 | |||
T0289 |
9-Aminoacridine
Aminacrine,9-氨基吖啶 |
Others; HIV Protease; Antibacterial | Microbiology/Virology; Others; Proteases/Proteasome |
9-Aminoacridine 是一种具有龋齿传播特性的抗菌剂,可用作局部消毒剂。它也是一种高度荧光染料,实验用作一种诱变剂,是细胞内 pH 的指示剂。 | |||
T9307 |
(E)-3-(3,4-dichlorophenyl)-N-(2-(4-(methylsulfonyl)piperazin-1-yl)-2-oxoethyl)acrylamide
|
Others | Others |
SR18662 又名 SR18662 ,是一种KLF5 抑制剂, 基于ML264结构的优化而得。它在体内外抑制结直肠癌的生长。 | |||
T18882 |
2-Aminoacridone
|
Others | Others |
2-Aminoacridone 是一种荧光团 (λexc= 428nm, λem= 525nm),普遍用于标记不饱和二糖。 | |||
T4564 |
Ethacrynic acid
Edecrin,利尿酸,Etacrynic Acid,Hydromedin |
Others; Calcium Channel; NF-κB; GST | Membrane transporter/Ion channel; Metabolism; NF-κB; Others; oxidation-reduction |
Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂,也是NF-κB 信号传导途径的有效抑制剂,并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道,从而导致气道平滑肌细胞松弛。它是利尿剂,具有抗炎特性,可减轻类维生素 A 诱导的小鼠耳部水肿。 | |||
T8636 |
Ibrutinib deacryloylpiperidine
IBT4A,5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine,伊布替尼中间体N-2 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Ibrutinib deacryloylpiperidine (IBT4A) 是 Ibrutinib 的杂质之一。它是一种不可逆的、选择性的 Btk 抑制剂 (IC50:0.5 nM)。 | |||
T5446 |
CIBACRON BLUE 3G-A
|
Others | Others |
Cibacron Blue 3G-A 是蒽醌染料,能够抑制 R46β-lactamase(Ki:1.2 uM)。 | |||
T28226 |
Octahydroaminoacridine succinate
|
Others | Others |
Octahydroaminoacridine succinate 是一种乙酰胆碱酯酶抑制剂,可用于治疗阿尔茨海默病。 | |||
T28475 |
Pyrazoloacridine
PD-115934,NSC 366140,NSC-366140,PD 115,934,PD 115934 |
Apoptosis; Topoisomerase | Apoptosis; DNA Damage/DNA Repair |
Pyrazoloacridine (PD 115934) 是一种核酸结合剂,在 K562 细胞中抑制 topo I 和 II 的活性,IC50 为 1.25 μM。 Pyrazoloacridine 具有抗癌活性。 | |||
T0942 |
Quinacrine dihydrochloride
疟疾平,Mepacrine dihydrochloride,阿的平,SN-390,Quinacrine 2HCl |
Apoptosis; Mitophagy; DNA; Phospholipase; Parasite; Autophagy; Histamine Receptor | Apoptosis; Autophagy; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience |
Quinacrine dihydrochloride (Mepacrine dihydrochloride) 是一种具有口服活性的抗疟剂,抑制 NF-κB 并激活 p53 信号转导,诱导肿瘤细胞发生凋亡,具有抗肿瘤和抗寄生虫活性。 | |||
T7891 |
Ipidacrine
伊匹达克林,NIK‐247 |
Others | Others |
Ipidacrine (NIK‐247) 是一种具有益智作用的化合物,也是一种胆碱酯酶抑制剂,具有药物活性,可用于阿尔茨海默病的治疗。 | |||
T77704 |
N-Isopropylacrylamide
|
Others | Others |
N-Isopropylacrylamide 具有热响应效应,被生物医学领域广泛应用。 | |||
T1440 |
Ethacridine lactate monohydrate
乳酸依沙吖啶一水物,利凡诺 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ethacridine lactate monohydrate 是一种聚 (ADP-核糖) 糖基水解酶 (PARG) 抑制剂,有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。它也是抗菌剂和流产剂。 | |||
T18911 |
Acriflavine
Acriflavinium chloride 3,6-Acridinediamine mix |
SARS-CoV; Antibacterial | Microbiology/Virology |
Acriflavine (Acriflavinium chloride 3,6-Acridinediamine mix) 是木瓜蛋白酶样蛋白酶(PL(pro))抑制剂,是一种用于标记高分子量 RNA 的荧光染料,具有抗菌抗癌活性,抑制 SARS-CoV-2 和其他 β 冠状病毒,可用于研究白血病。 | |||
T4551 |
Acrivastine
Acrivastin,阿伐斯汀,BW825C,Semprex |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Acrivastine (Acrivastin) 是一种短效组胺 1 受体拮抗剂,可用于研究过敏性鼻炎。 | |||
T5967 |
Ethacridine lactate
乳酸依沙吖啶,Acrinol,6,9-DIAMINO-2-ETHOXYACRIDINE LACTATE |
Others; Antibacterial | Microbiology/Virology; Others |
Ethacridine lactate (Acrinol) 是一种聚 (ADP-核糖) 糖水解酶 (PARG) 抑制剂,也是一种抗菌剂和流产剂。它有抗金黄色葡萄球菌和其他革兰氏阳性球菌的活性。 | |||
T67772 |
Phos-tag Acrylamide AAL-107
|
||
Phos-tag Acrylamide AAL-107 是一种丙烯酰胺悬垂物,可用作可视化磷酸化蛋白质的工具。 | |||
T64829 | N-(5-((4-(1-Methyl-1H-indol-3-yl)pyridin-2-yl)amino)-2-(2-methylpyrrolidin-1-yl)phenyl)acrylamide | ||
N-(5-((4-(1-Methyl-1H-indol-3-yl)pyridin-2-yl)amino)-2-(2-methylpyrrolidin-1-yl)phenyl)acrylamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64829。 | |||
T66278 | Methyl 3-(4-(bromomethyl)phenyl)acrylate | ||
Methyl 3-(4-(bromomethyl)phenyl)acrylate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66278,CAS号为 946-99-6。 | |||
T64918 | Ethylene diacrylate | ||
Ethylene diacrylate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64918。 | |||
T125276 | Acronyculatin Q | ||
Acronyculatin Q 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125276。 | |||
T29622 |
Acridine, 2,6-diamino- (8CI)
Acramine Red,Diflavine |
||
Acridine, 2,6-diamino- (8CI) is a biochemical. | |||
T29625 |
Acridine-9-carboxamide, 1,2,3,4-tetrahydro-N,N-diethyl-
O=C(C1=C(CCCC2)C2=NC3=CC=CC=C31)N(CC)CC |
||
Acridine-9-carboxamide, 1,2,3,5-tetrahydro-N,N-diethyl- is a biochemcial. | |||
T65342 | N,N′-Methylenebisacrylamide | ||
N,N′-Methylenebisacrylamide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65342。 | |||
T26555 |
Acreozast
TYB 2285,TYB-2285,TYB2285 |
||
Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis. | |||
T14117 |
Acridine Orange 10-Nonyl Bromide
Nonylacridine orange,10-壬基溴代吖啶橙 |
Others | Others |
Acridine Orange 10-Nonyl Bromide is a cardiolipin fluorescent probe (λex: 489 nm, λem: 525 nm). | |||
T37031 |
Quinacrine mustard hydrochloride
Quinacrine mustard HCl |
Autophagy | Autophagy |
Quinacrine mustard hydrochloride 是一种荧光染料,也 是一种多环芳香剂,可作为诱变剂诱导细菌的突变体。Quinacrine mustard hydrochloride 能选择性地与腺嘌呤-胸腺嘧啶(AT)碱基对结合,而不 是与鸟嘌呤-胞嘧啶(GC)碱基对结合,诱导细胞周期停滞在 G2/M 期。Quinacrine mustard (hydrochloride) 已被用于标记移相染色体,以通过自动放射摄影技术进行核型分析。 | |||
T40978 |
Acrylodan
|
||
Acrylodan, when subjected to thiol reactions, exhibits sensitivity to the dipolarity and dynamics of its surrounding binding pocket, specifically those surrounding Cys 34. | |||
T29619 |
Acridine Yellow
Acridine Yellow Base |
||
Acridine yellow, also known as acridine yellow G, acridine yellow H107, basic yellow K, and 3,6-diamino-2,7-dimethylacridine, is a yellow dye with strong bluish-green fluorescence. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2266 |
SantacruzaMate A
CAY-10683 |
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
SantacruzaMate A (CAY-10683) 是一种高效选择性的HDAC2抑制剂,IC50为 119 pM。 | |||
T4S1990 |
Carvacrol
香荆芥酚,Karvakrol,O-Thymol,cymophenol,香芹酚 |
Apoptosis; Others; Gamma-secretase; Endogenous Metabolite; Antifungal | Apoptosis; Metabolism; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Stem Cells |
Carvacrol (O-Thymol) 是唇形科植物中的一种单萜酚类天然产物,具有镇痛、抗焦虑、抗抑郁、抗氧化、抗炎和抗癌作用。 | |||
T2144 |
Tacrolimus
他克莫司,Fujimycin,FK506,FR900506 |
Phosphatase; Others; Antibacterial; Antibiotic; mTOR; Autophagy | Autophagy; Metabolism; Microbiology/Virology; Others; PI3K/Akt/mTOR signaling |
Tacrolimus (Fujimycin) 可与 FKBP12 结合形成高亲和力复合物 (Ki: 0.2 nM),抑制钙/钙调蛋白依赖性蛋白磷酸酶的活性。 | |||
T3S2325 |
Ardisiacrispin A
百两金素,Saxifragifolin B,LTS-4,Deglucocyclamin |
HSV | Microbiology/Virology |
Ardisiacrispin A (Deglucocyclamin) 是一种常见的三萜皂苷,来自于紫金牛属物种。 它与来自紫金牛属的 A. crenata 中的一些三萜皂苷具有相似的生物学特性,如对肿瘤细胞具有细胞毒活性、免疫调节和抗病毒活性。 | |||
TN6780 |
Carvacrol methyl ether
Methyl carvacrol,Methyl carvacryl ether |
Antibacterial | Microbiology/Virology |
Carvacrol methyl ether 来源于植物挥发油,具有抗菌活性。 | |||
T3858 |
macranthoidin A
灰毡毛忍冬皂苷甲,金银花 |
Others | Others |
Macranthoidin A 是一种具有口服活性的、提取于金银花中的皂苷。它对四氯化碳,对乙酰氨基酚和镉所致的肝损伤具有保护作用,对耳巴豆油的溶胀具有明显的抑制作用。 | |||
T41095 |
(E)-3-(4-Methoxyphenyl)acrylic acid
(E)-3-(4-甲氧基苯基)丙烯酸 |
Glucosidase | Metabolism |
(E)-3-(4-Methoxyphenyl)acrylic acid 是从 Etlingera pavieana (Pierre ex Gagnep.) R. M. Sm. 的根茎中分离出来的一种小分子化合物。它是一种新型 α-葡萄糖苷酶抑制剂。(E)-3-(4-甲氧基苯基)丙烯酸具有保肝活性、抗失水活性、增强认知效果,并可用于降低血压血糖。 | |||
T67710 |
3-Indoleacrylic acid
|
Endogenous Metabolite | Metabolism |
3-Indoleacrylic acid 是由链球菌属产生的色氨酸的代谢产物。3-Indoleacrylic acid 对肠上皮屏障功能有有益作用,并减轻免疫细胞的炎症反应。 | |||
TN1159 |
(1(10)E,2R*,4R*)-2-Methoxy-8,12-epoxygermacra-1(10),7,11-trien-6-one
[(1(10)E,2R,4R)]-2-Methoxy-8,12-epoxygemacra-1(10),7,11-trien-6-one |
Others | Others |
(1(10)E,2R*,4R*)-2-Methoxy-8,12-epoxygermacra-1(10),7,11-trien-6-one ([(1(10)E,2R,4R)]-2-Methoxy-8,12-epoxygemacra-1(10),7,11-trien-6-one) 是一种来自姜黄的倍半萜。 | |||
T5703 |
β,β-Dimethylacrylalkannin
|
Others | Others |
β,β-Dimethylacrylalkannin 是一种萘醌类化合物,分离自紫草属植物中,可以提高皮肤细胞中胶原蛋白和内披蛋白的含量。 | |||
T19412 |
Macrozamin
甲基氧化偶氮甲醇樱草糖苷,大泽明素 |
Others | Others |
Macrozamin 是苏铁的一种主要成分,表现出致癌,致畸,诱变和神经毒性作用。 | |||
T5787 |
Macranthoside B
金银花,灰毡毛忍冬次皂苷乙 |
Antibacterial | Microbiology/Virology |
Macranthoside B 是一种从金银花中分离出来的天然产物,具有抗菌活性。 | |||
T5262 |
trans-3-Indoleacrylic acid
(E)-3-吲哚丙烯酸,反式-3-吲哚丙烯酸,trans-IAA |
Others; Endogenous Metabolite | Metabolism; Others |
trans-3-Indoleacrylic acid (trans-IAA) 是内源性代谢产物的一种。 | |||
T2945 |
Germacrone
|
P450; Antiviral; Influenza Virus | Immunology/Inflammation; Metabolism; Microbiology/Virology |
Germacrone 提取自姜黄,具有抗炎、抗雄激素和抗病毒活性。 它还通过促进细胞凋亡来抑制胶质瘤细胞的增殖。 | |||
T3S2344 |
β,β-Dimethylacrylshikonin
β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin |
ERK; HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; MAPK; Metabolism |
β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) 是一种萘醌衍生物,从 Arnebia nobilis 中提取得到。它利用 PI3K 通路诱导 eNOS、VEGF 和 HIF-1α 的表达,促进血管生成,具有抗肿瘤活性。 | |||
T3367 |
Macranthoidin B
灰毡毛忍冬皂苷乙,金银花,Macranthoiside I |
Others | Others |
Macranthoidin B (Macranthoiside I) 是一种活性天然皂苷。 | |||
T20879 |
Tacrolimus monohydrate
FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506 |
Phosphatase; Others; Antibacterial; Antibiotic; Autophagy | Autophagy; Metabolism; Microbiology/Virology; Others |
Tacrolimus monohydrate (LCP-Tacro) 是大环内酯类化合物,它与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶,从而抑制 T 淋巴细胞信号转导和 IL-2 转录。具有强免疫抑制特性。 | |||
TN7113 |
Methacrylamide
|
Others | Others |
Methacrylamide 是一种具有染色性的天然产物。 | |||
TN1831 |
Macranthoside A
Kalopanaxsaponin H |
Antioxidant | oxidation-reduction |
Macranthoside A (Kalopanaxsaponin H) 是一种从地黄中提取的三萜糖苷,属于环烯醚萜类化合。Macranthoside A 具有抗炎、抗氧化、抗菌和神经保护活性,抑制促炎细胞因子的产生和抑制炎症信号通路的激活,有助于中和有害的自由基,保护细胞免受氧化损伤,可以促进神经元的存活和生长,并防止氧化应激或神经毒性化合物引起的神经元细胞死亡,具有治疗神经退行性疾病、心血管疾病和肝损伤的潜力。 | |||
TN4478 | Macrocarpal H | Antifection | Microbiology/Virology |
Macrocarpal H has anti-glucosyltransferase, and anti-bacterial activities. | |||
TN4474 |
Macrocarpal B
|
c-Met/HGFR | Tyrosine Kinase/Adaptors |
The intestinal absorption of M-A, Macrocarpal B, and Cy-C was passive diffusion as the dominating process and Cy-C was partly ATP-dependent. | |||
TN6402 |
Methyl 3-methoxyacrylate
|
||
Methyl 3-methoxyacrylate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6402,CAS号为 34846-90-7。 | |||
TN4556 |
Methyl trans-3-(3,4,5-trimethoxyphenyl)acrylate
|
Others | Others |
Methyl trans-3-(3,4,5-trimethoxyphenyl)acrylate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4556,CAS号为 20329-96-8。 | |||
T8253 |
Carvacryl acetate
|
Others | Others |
Carvacryl acetate 是抗炎和抗氧化剂。 | |||
TN3294 |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
|
NADPH-oxidase; P450; MAO | Immunology/Inflammation; Metabolism; Neuroscience |
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. | |||
TN2997 |
4(15),5,10(14)-Germacratrien-1-ol
|
Others | Others |
4(15),5,10(14)-Germacratrien-1-ol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2997,CAS号为 81968-62-9。 | |||
T81887 |
Macrostemonoside I
|
||
Macrostemonoside I,一种从Allium macrostemon分离得到的呋甾烷醇皂苷。 | |||
TN4928 |
Rutacridone
|
P450 | Metabolism |
Rutacridone has mutagenicity. | |||
TN6917 |
Macrostemonoside J
|
||
Macrostemonoside J is a natural product. | |||
TN6492 | (1E)-3-methoxy-8,12-epoxygermacra-1,7,10,11-tetraen-6-one | ||
(1E)-3-methoxy-8,12-epoxygermacra-1,7,10,11-tetraen-6-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6492,CAS号为 1393342-06-7。 | |||
TN2538 | 1-Hydroxy-N-methylacridone | Others | Others |
1-Hydroxy-N-methylacridone is a natural product from Ruta chalepensis. | |||
TN2520 | 1,7-Dihydroxyacridone | Others | Others |
1,7-Dihydroxyacridone is a natural product from Boenninghausenia albiflora. | |||
TN6066 | 1-Hydroxyacridone | ||
1-Hydroxyacridone has potential antiviral activity. | |||
TN3293 | 8alpha-(2-Methylacryloyloxy)-1-O-methylhirsutinolide 13-O-acetate | Others | Others |
8alpha-(2-Methylacryloyloxy)-1-O-methylhirsutinolide 13-O-acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3293,CAS号为 883872-71-7。 | |||
TN4476 |
Macrocarpal D
|
Antifection | Microbiology/Virology |
Macrocarpal D is a HIV-RTase inhibitor. It has antibacterial activity. | |||
T83551 |
(9S)-Macrocidin B
|
||
(9S)-Macrocidin B 的除草活性不如macrocidin A。 | |||
TN4480 |
Macrocarpal J
|
Antifection | Microbiology/Virology |
Macrocarpal J has anti-bacterial activity, it also has anti-glucosyltransferase activity. | |||
T72731 |
Acremoxanthone C
|
||
Acremoxantone C 是一种有效的钙调素(CaM)抑制剂,存在于 Purpureocillium lilacinum 中。Acremoxantone C 与人钙调素 (hCaM) 生物传感器 hCaM M124C mBBr 结合,Kd 为 18.25 nM。 | |||
TN6021 |
Daphmacropodine
|
||
Daphmacropodine是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN6021,CAS号为 39729-21-0。Daphmacropodine可用作对照参考。 | |||
TN4866 | Pyracrenic acid | Others | Others |
Pyracrenic acid is a potent elastase inhibitor with an IC50 value of 1.5 mg/mL. Pyracrenic acid shows DPPH radical scavenging activity. It also shows significant cytotoxic activities against human cancer cells COLO 205 and AGS. | |||
TN4481 |
Macrocarpal K
|
Others | Others |
Macrocarpal K 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4481,CAS号为 218290-59-6。 | |||
TN3295 |
8alpha-(2-Methylacryloyloxy)hirsutinolide
|
Others | Others |
8alpha-(2-Methylacryloyloxy)hirsutinolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3295,CAS号为 188293-70-1。 | |||
T21032 |
Germacrene D
1(10),4(14),5-Germacratriene |
||
Germacrene D, a natural essential oil, has antioxidant activity and cytotoxicity on tumor cells. | |||
TN4479 |
Macrocarpal I
|
Antifection | Microbiology/Virology |
Macrocarpal I has anti-glucosyltransferase, and anti-bacterial activities. | |||
T72902 |
Acremonidin A
|
||
Acremonidin A 是一种有效的钙调素(CaM)抑制剂,存在于Purpureocillium lilacinum 中。Acremonidin A 与人钙调素 (hCaM) 生物传感器 hCaM M124C mBBr 结合,Kd 为 19.40 nM。 | |||
T37552 |
(+)-Macrosphelide A
|
||
(+)-Macrosphelide A is a fungal metabolite originally isolated from Microsphaeropsis. It inhibits adhesion of HL-60 human leukemia cells to human umbilical vein endothelial cells (HUVECs) in a concentration-dependent manner. It also inhibits the growth of SKOV3 ovarian cancer cells in a concentration-dependent manner. (+)-Macrosphelide A inhibits the growth of Gram-positive bacteria, including B. subtilis, M. luteus, B. thuringiensis, and S. aureus (MICs = 143, 143, 57, and 57 μg/ml, respectivel... | |||
TN1397 |
Ardisiacrispin B
|
Others | Others |
Ardisiacrispin B displays cytotoxic effects in multi-factorial drug resistant cancer cells via ferroptotic and apoptotic cell death. | |||
TN5345 |
8α-Methacryloyloxybalchanin
|
||
8α-Methacryloyloxybalchanin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5345,CAS号为 104021-39-8。 | |||
TN3299 |
8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide
|
Others | Others |
8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3299,CAS号为 142891-14-3。 | |||
TN4130 | Germacrone 4,5-epoxide | gp120/CD4; IL Receptor; P450 | Immunology/Inflammation; Metabolism |
(4S,5S)-(+)-Germacrone-4,5-epoxide inhibits certain subtypes of cytochrome P450 (CYP). | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02990 |
Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (His)
14 kDa antigen,Acr,16 kDa antigen,HSP 16.3 |
Mycobacterium bovis | Baculovirus Insect Cells |
Acts as a chaperone. Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (His) is expressed in Baculovirus insect cells with C-9xHis tag. The predicted molecular weight is 18.1 kDa and the accession number is P0A5B8. | |||
TMPH-02991 |
Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (E. coli, His)
14 kDa antigen,Acr,16 kDa antigen,HSP 16.3 |
Mycobacterium bovis | E. coli |
Acts as a chaperone. Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 20.1 kDa and the accession number is P0A5B8. | |||
TMPY-02208 |
Peroxiredoxin 5 Protein, Human, Recombinant (His)
B166,HEL-S-55,prx-V,ACR1,PMP20,AOEB166,SBBI10,PRXV,... |
Human | E. coli |
Peroxiredoxin 5 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 18.5 kDa and the accession number is P30044-2. | |||
TMPY-01813 |
ACRV1 Protein, Human, Recombinant (His)
SP-10,SPACA2,D11S4365,acrosomal vesicle protein 1 |
Human | HEK293 Cells |
Acrosomal protein SP-1, also known as Acrosomal vesicle protein 1 and ACRV1, is a testis-specific, differentiation antigen, that arises within the acrosomal vesicle during spermatogenesis, and is associated with the acrosomal membranes and matrix of mature sperm. Regulation of cell type-specific gene transcription is central to cellular differentiation and development. During spermatogenesis, a number of testis-specific genes are expressed in a precise spatiotemporal order. The longest tr... | |||
TMPH-01279 |
CRACR2B Protein, Human, Recombinant (His)
CRACR2B,EFCAB4A,EF-hand calcium-binding domain-cont... |
Human | E. coli |
Plays a role in store-operated Ca(2+) entry (SOCE). | |||
TMPH-02147 |
TACR1 Protein, Human, Recombinant (GST)
|
Human | E. coli |
This is a receptor for the tachykinin neuropeptide substance P. It is probably associated with G proteins that activate a phosphatidylinositol-calcium second messenger system. The rank order of affinity of this receptor to tachykinins is: substance P > substance K > neuromedin-K. TACR1 Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 30.1 kDa and the accession number is P25103. | |||
TMPH-02455 |
Acrosin Protein, Meleagris gallopavo, Recombinant (His & Myc)
EC:3.4.21.10,Proacrosin,Proacro1 |
Meleagris gallopavo | E. coli |
Serine protease of trypsin-like cleavage specificity. Synthesized in a zymogen form, proacrosin and stored in the acrosome. Acrosin Protein, Meleagris gallopavo, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 43.1 kDa and the accession number is Q2UVH8. | |||
TMPH-00908 |
MACROD1 Protein, Human, Recombinant (His & Myc)
|
Human | Baculovirus Insect Cells |
MACROD1 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus. | |||
TMPH-00907 |
MACROD1 Protein, Human, Recombinant (His)
|
Human | E. coli |
MACROD1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 41.5 kDa and the accession number is Q9BQ69. | |||
TMPY-05059 |
LACRT Protein, Human, Recombinant (His)
lacritin |
Human | HEK293 Cells |
LACRT Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13.7 kDa and the accession number is Q9GZZ8. | |||
TMPY-02063 |
Alpha-2-macroglobulin Protein, Human, Recombinant (His)
α-2-macroglobulin,FWP007,CPAMD5,A2MD,S863-7,alpha-2... |
Human | Baculovirus Insect Cells |
alpha-2-macroglobulin, also known as α2-macroglobulin (α2M and A2M), is an abundant protein of the plasma of vertebrates and members of several invertebrate phyla and functions as a broad-spectrum protease-binding protein. alpha-2-macroglobulin is produced by the liver, and is a major component of the alpha-2 band in protein electrophoresis. alpha-2-macroglobulin is a large plasma glycoprotein that has long been known as an irreversible inhibitor of a variety of proteinases. More recently, it ha... |