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13

抑制剂 & 化合物

273

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0058 2-Ethoxybenzamide

Ethenzamide,Anovigam,止痛灵,2-乙氧基苯甲酰胺

COX Immunology/Inflammation; Neuroscience
2-Ethoxybenzamide (Anovigam) 常作为解热镇痛药。
T40564 Neoabietic acid

Neoabietic acid is an abietic-type acid isolated from the oleoresin and rosin of Pinus palustris . Neoabietic acid is highly susceptible to mineral acid. Neoabietic acid has antibacterial activity in vitro.
T21125 Decane, 1-iodo-

1-Iododecane

Decane, 1-iodo- is used as an intermediate in organic synthesis. Through palladium-catalyzed carbonylative cross-coupling reaction with 9-octyl-9-borabicyclo[3.3.l]nonane, it is also used as a precursor to prepare 9-nonadecanone.
T19557 Sanshool

Others Others
Sanshool is a natural product isolated from Zanthoxylum bungeanum. Sanshool improves UVB-induced skin photodamage by targeting JAK2/STAT3-dependent autophagy.
T31323 Decane, 2,4-dimethyl-

2,4-dimethyl-decane

Decane, 2,4-dimethyl- is a biochemical.
T31846 Foresticine

Longtouconitine B

Foresticine is an alkaloid.
T31529 d-Isothujone

d-Isothujone is a biochemical.
T22913 L-CCG-lll

Others Others
inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate.
T36412 Multiflorenol

Multiflorenol is a triterpene that has been found in T. kirilowii seeds.1 It inhibits in vitro activation of Epstein-Barr virus early antigen (EBV-EA) induced by the tumor promoter phorbol 12-myristate 13-acetate in a concentration-dependent manner. |1. Akihisa, T., Tokuda, H., Ichiishi, E., et al. Anti-tumor promoting effects of multiflorane-type triterpenoids and cytotoxic activity of karounidiol against human cancer cell lines. Cancer Lett. 173(1), 9-14 (2001).
T35285 Yuccagenone

Yuccagenone is a biochemical.
T38189 2-hydroxy Lignoceric Acid

2-hydroxy Lignoceric acid is an α-hydroxy very long chain fatty acid that is normally present in the mammalian nervous system. In the brain, 2-hydroxy lignoceric acid is derived from lignoceric acid and further converted to ceramides and cerebrosides during the process of nerve sheath myelination. 2-hydroxy Lignoceric acid is produced by the α-oxidation of lignoceric acid in the peroxisome and defects in this pathway are associated with disorders such as Zellweger syndrome.
T10163 4'-Methylchrysoeriol

Others Others
4'-Methylchrysoeriol is a potent inhibitor of cytochrome P450 enzymes (IC50: 19 nM for human P450 1B1-dependent EROD).
T35646 4-oxo-2-Nonenal

4-oxo-2-Nonenal,4-ONE

4-hydroxy Nonenal is a lipid peroxidation product derived from oxidized ω-6 polyunsaturated fatty acids such as arachidonic acid and linoleic acid. [1] [2] It exhibits various biological activities such as cytotoxicity, growth inhibiting activity, genotoxicity, and chemotactic activity and has been widely used as a marker of lipid peroxidation.[1][2][3] 4-oxo-2-Nonenal is a more recently identified product of lipid peroxidation.[4][5][6] It actively modifies histidine and lysine residues on prot...

化合物

2-Ethoxybenzamide
Cat.No: T0058
Synonym: Ethenzamide,Anovigam,止痛灵,2-乙氧基苯甲酰胺
Target: COX
Neoabietic acid
Cat.No: T40564
Synonym:
Target:
Decane, 1-iodo-
Cat.No: T21125
Synonym: 1-Iododecane
Target:
Sanshool
Cat.No: T19557
Synonym:
Target: Others
Decane, 2,4-dimethyl-
Cat.No: T31323
Synonym: 2,4-dimethyl-decane
Target:
Foresticine
Cat.No: T31846
Synonym: Longtouconitine B
Target:
d-Isothujone
Cat.No: T31529
Synonym:
Target:
L-CCG-lll
Cat.No: T22913
Synonym:
Target: Others
Multiflorenol
Cat.No: T36412
Synonym:
Target:
Yuccagenone
Cat.No: T35285
Synonym:
Target:
2-hydroxy Lignoceric Acid
Cat.No: T38189
Synonym:
Target:
4'-Methylchrysoeriol
Cat.No: T10163
Synonym:
Target: Others
4-oxo-2-Nonenal
Cat.No: T35646
Synonym: 4-oxo-2-Nonenal,4-ONE
Target:
Cat. No. Product Name Target Signaling Pathways
TN1768 Iriflophenone

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Iriflophenone 是从 Aquilaria sinensis 中分离得到,能诱导 MCF-7 和 T-47D 人乳腺癌细胞增殖。
TN1621 Eriodictyol-7-O-glucoside

Nrf2 Immunology/Inflammation
Eriodictyol-7-O-glucoside 是一种 Nrf2 激活剂,可防止顺铂诱导的毒性。 Eriodictyol-7-O-glucoside 是一种类黄酮和自由基清除剂,在开心果皮中具有抗氧化活性。
T3379 Decanoic Acid

Decoic acid,CAPRIC ACID,Caprynic acid,癸酸

GluR; iGluR Membrane transporter/Ion channel; Neuroscience
Decanoic Acid (Caprynic acid) 是中链甘油三酯中的成分,是非竞争性和可透过血脑屏障的 AMPA 受体抑制剂,具有抗癫痫作用。
T1738 Taxifolin

(+)-Taxifolin,紫杉叶素,Dihydroquercetin,二氢槲皮素,(+)-Dihydroquercetin

VEGFR; TNF; Tyrosinase; Adrenergic Receptor; Autophagy Angiogenesis; Apoptosis; Autophagy; GPCR/G Protein; Neuroscience; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Taxifolin (Dihydroquercetin) 是一种天然类黄酮,具有抗纤维化作用。它是一种自由基清除剂,具有抗氧化能力。它有效抑制胶原酶,IC50为 193.3 μM,具有重要的抗酪氨酸酶活性。
T6S0232 Eriodictyol

圣草酚,Huazhongilexone

Influenza Virus; DNA/RNA Synthesis; Nrf2; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology
Eriodictyol (Huazhongilexone) 是从中草药中得到的一种黄酮类天然产物,具有抗氧化、抗炎和抗糖尿病作用。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 18 nM。它可诱导Nrf2信号通路。
T2755 Rhoifolin

野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside

Others; p38 MAPK; NF-κB; transporter; IGF-1R; Autophagy Autophagy; MAPK; Metabolism; NF-κB; Others; Tyrosine Kinase/Adaptors
Rhoifolin (Apigenin 7-O-neohesperidoside) 是从琯溪蜜柚叶子分离的一种黄酮糖苷。它通过 RANKL 诱导的NF-κB 和MAPK 途径改善钛颗粒刺激的骨溶解并减少破骨细胞生成。它通过增强脂联素分泌,胰岛素受体-β的酪氨酸磷酸化和GLUT4易位有助于治疗糖尿病并发症。
TN1877 Lonicerin

忍冬苦苷,金银花

Apoptosis; Antibacterial Apoptosis; Microbiology/Virology
Lonicerin 是一种抗藻酸盐分泌蛋白的黄酮类化合物,对铜绿假单胞菌有抑制作用。它可预防脂多糖诱导的急性肺损伤的炎症和细胞凋亡。
T2838 Naringenin

柚皮素,Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875

P450; Influenza Virus; Reactive Oxygen Species; Endogenous Metabolite; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Naringenin (NSC-11855) 是葡萄柚中主要的黄烷酮,可作为抗氧化剂、自由基清除剂、抗炎剂、碳水化合物代谢促进剂、免疫系统调节剂。
T6S1885 Benzoylmesaconine

Mesaconine 14-benzoate,苯甲酰新乌头原碱

Others Others
Benzoylmesaconine (Mesaconine 14-benzoate) 是乌头汤最丰富的组分。其中乌头汤可用于研究类风湿性关节炎。
T5710 Pinocembrin-7-O-β-D-glucopyranoside

Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷

Others Others
Pinocembrin-7-O-β-D-glucopyranoside (Pinocembrin 7-O-beta-D-glucoside) 是黄酮类化合物,能够提高脂质过氧化。
TN4675 Nortrachelogenin

(-)-Wikstromol,(-)-Nortrachelogenin

Apoptosis; Antifungal Apoptosis; Microbiology/Virology
Nortrachelogenin ((-)-Wikstromol) 可从 Partrinia scabiosaefolia 提取得到,具有抗真菌活性,可诱导膜破坏和半胱天冬酶依赖性细胞凋亡.
T0970 Racanisodamine

山莨菪碱,Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine,消旋山莨菪碱

Adrenergic Receptor; AChR GPCR/G Protein; Neuroscience
Racanisodamine (7β-Hydroxyhyoscyamine) 是 anisodamine 的消旋体,是非选择性的毒蕈碱拮抗剂,是近视控制滴眼液的有效成分。
T4S0295 Apigenin 7-glucoside

波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Apigenin 7-glucoside (Cosmosiin) 是一种 ROS 清除剂,具有抗增殖、抗氧化作用。
TQ0089 Juglanin

Apoptosis; JNK; Autophagy Apoptosis; Autophagy; MAPK
Juglanin 是来自金鸡脚的一种黄酮类天然产物,是一种 JNK 的激活剂,能诱导人乳腺癌细胞的凋亡和自噬,具有炎症和抗肿瘤活性。
TN3340 Acetylatractylodinol

Tractylodinol acetate,乙酰基仓术呋喃烃醇

Others Others
Acetylatractylodinol (Tractylodinol acetate) 是分离自Atractylodes lancea 中,具有抗氧化作用。
T0473 Arbutin

Uva,p-Arbutin,p-Arbutin,熊果苷,β-Arbutin

Tyrosinase Proteases/Proteasome
Arbutin (p-Arbutin) 是一种从熊果植物 Arctostaphylos uvaursi 中分离出的天然多酚,具有抗氧化,抗炎和抗肿瘤特性。它是一种脱色剂,也是一种黑色素细胞中酪氨酸酶的竞争性抑制剂,对单酚酶的 Kiapp 值为 1.42 mM;对二酚酶Kiapp 的值为 0.9 mM。
T3888 Scopolin

Murrayin,东莨菪甙,Scopoloside,东莨菪苷

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Scopolin (Scopoloside) 是从拟南芥根中分离出来的香豆素,可通过激活SIRT1介导的信号级联反应减轻了肝脂肪变性。
T2848 Osthole

Osthol,NSC 31868,蛇床子素,Ostol

Apoptosis; HBV; Parasite; Histamine Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Osthole (Osthol) 是一种天然抗组胺药替代试剂,可刺激成骨细胞增殖和分化。它可抑制组胺 H1受体活性,还可抑制细胞培养物中 HBV 的分泌。
T2S0765 Epibetulinic acid

NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Epibetulinic acid 对细菌内毒素刺激的小鼠巨噬细胞 (RAW 264.7) 中 NO 和前列腺素 E(2) 的产生具有有效的抑制作用,IC50分别为 0.7 和 0.6 μM,具有抗炎活性。
TN6797 Isoneochamaejasmin A

Others Others
Isoneochamaejasmin A 是一种双黄酮类化合物,是一种广泛使用的中药 stellera chamaejasme L. 干燥根中的主要活性成分之一。
TN1482 Chamaechromone

P450; HBV Metabolism; Microbiology/Virology
Chamaechromone 是从 Stellera chamaejasme L. 的根中分离出来的天然产物。 Chamaechromone 具有抗 HBV 和杀虫活性。
TN6743 ETHYL OCTANOATE

辛酸乙酯,CAPRYLIC ACID ETHYL ESTER

Others Others
ETHYL OCTANOATE (CAPRYLIC ACID ETHYL ESTER) 是一种天然产物。
TN1819 Kaempferol 3-neohesperidoside

Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷

GSK-3; MEK; PI3K MAPK; PI3K/Akt/mTOR signaling; Stem Cells
Kaempferol 3-neohesperidoside (Kaempferol 3-O-neohesperidoside) 是一种类黄酮,对大鼠比目鱼肌具有拟胰岛素作用。
T5S0168 Atractylenolide II

2-Atractylenolide,Asterolide,苍术内酯II

Apoptosis; ERK; p38 MAPK; Akt; STAT Apoptosis; Cytoskeletal Signaling; JAK/STAT signaling; MAPK; PI3K/Akt/mTOR signaling; Stem Cells
Atractylenolide II (2-Atractylenolide) 是一种从白术干燥根茎分离的倍半萜类天然产物,具有抗增殖活性。
T0878 Diosmin

Venosmine,Diosmil,Barosmin,地奥司明,地奥司明(7-芸香糖甙)

Aryl Hydrocarbon Receptor; Norepinephrine Immunology/Inflammation; Neuroscience
Diosmin (Venosmine) 是在各种柑橘类水果中发现的类黄酮,也是芳烃受体激动剂,有增强血管壁的作用。
TN1142 8-Oxocoptisine

8-Oxycoptisine,8-氧黄连碱

Others Others
8-Oxocoptisine (8-Oxycoptisine) 是天然原小檗碱生物碱,具有抗癌作用。
T5S0055 Chelidonine

Helidonine,Khelidonin,白屈菜碱,Stylophorin

Apoptosis; Others; Influenza Virus Apoptosis; Microbiology/Virology; Others
Chelidonine (Stylophorin) 是白屈菜中的一种异喹啉生物碱,有抗肿瘤和抗病毒作用。它可导致细胞周期 G2/M 停滞,诱导 caspase 依赖和非依赖性的细胞凋亡。
T6S1879 Indaconitine

Others Others
Indaconitine 可分离自乌头植物根茎。
T2883 Syringic acid

3,5-dimethyl ether Gallic Acid,SYRA,3,5-dimethoxy-4-hydroxy Benzoic Acid,丁香酸,NSC 2129

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
Syringic acid (3,5-dimethoxy-4-hydroxy Benzoic Acid) 能抑制低密度脂蛋白的氧化。
TN1772 Isoastilbin

Anti-infection; Tyrosinase; Antibacterial Microbiology/Virology; Proteases/Proteasome
Isoastilbin 是Rhizoma Smilacis glabrae 和Astragalus membranaceus 中的二氢黄酮醇糖苷。它抑制酪氨酸酶活性,还抑制葡萄糖基转移酶,IC50值为 54.3 μg/mL。它具有神经保护、抗氧化、抗微生物和抗凋亡活性,可研究阿尔茨海默氏病。
T4S1881 Aconine

乌头原碱,Jesaconine

Others; NF-κB NF-κB; Others
Aconine (Jesaconine) 是一种退热药,有胃麻醉作用,能够抑制核因子 κB 受体活化剂配体诱导的 NF-κB 激活。
T3001 Honokiol

和厚朴酚,NSC 293100

ERK; HCV Protease; MEK; Akt; Autophagy Autophagy; Cytoskeletal Signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Honokiol (NSC-293100) 是厚朴提取物的活性成分,靶向多种信号分子,具有抗氧化,抗炎,抗血管生成和抗癌活性。它可抑制 Akt 的激活并增强 ERK1/ERK2 的磷酸化。
TJS2216 Aurantiamide acetate

金色酰胺醇酯,Asperglaucide

Cysteine Protease Proteases/Proteasome
Aurantiamide acetate (Asperglaucide) 是抑制口服有活性的 cathepsin 选择性抑制剂,分离自 Portulaca oleracea L。它具有抗炎作用,可用于研究炎性相关疾病。
T3S0717 Thymol

2-isopropyl-5-methylphenol,Pseudoaspidin,Thymic Acid,Thyme Camphor,百里酚

Antibacterial Microbiology/Virology
Thymol (Pseudoaspidin) 是从唇形科植物以及如马鞭草科、玄参科、毛茛科等其他植物中分离出来的精油中的主要单萜酚。它具有抗炎、抗菌、抗氧化和抗真菌作用。
T5S1959 (-)-Asarinin

Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin

Antibacterial Microbiology/Virology
(-)-Asarinin (Eleutheroside B4) 是一种主要从 Zanthoxylum armatum 根部提取到的木脂素。
TQ0160 Hydrastine

北美黄连碱,(-)-β-Hydrastine,(1R,9S)-β-Hydrastine

Others Others
Hydrastine ((-)-β-Hydrastine) 是一种天然生物碱,存在于Hydrastis canadensis 和Ranunculaceae 家族其他植物。
T2972 Rutaecarpine

Rutacarpine,吴茱萸次碱,Rhetine,Rutecarpine

COX Immunology/Inflammation; Neuroscience
Rutaecarpine (Rhetine) 是从槐木中提取的一种生物碱,是 COX-2的抑制剂,IC50值为0.28 μM。
T8859 NITIDINE

Others Others
NITIDINE 是一种从花椒根中分离出来的具有生物活性的植物苯并菲啶生物碱。它具有抗癌、神经保护、抗疟疾、抗 HIV、镇痛、抗炎和抗真菌活性。
T0965 Histamine

Ergamine,组胺

5-HT Receptor; Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine (Ergamine) 是通过组胺的酶促脱羧衍生的胺。它是一种强大的胃分泌兴奋剂、支气管平滑肌的收缩剂、血管扩张剂以及中枢作用的神经递质。
T3095 Tyramine

4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine

MAO; Endogenous Metabolite Metabolism; Neuroscience
Tyramine (Uteramine) 是天然存在于体内或某些食物中的氨基酸。Tyramine 有助于调节血压。
T0847 Chenodeoxycholic acid

CDCA,鹅去氧胆酸,Chenodiol

Potassium Channel; FXR; Endogenous Metabolite; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Chenodeoxycholic acid (CDCA) 是一种胆汁酸,通常与甘氨酸或牛磺酸结合。它作为清洁剂溶解脂肪以供肠道吸收,并被小肠重新吸收。它被用作利胆剂、利胆泻药,以及预防或溶解胆结石。
TN1905 Magnolioside

七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷

Antifection Microbiology/Virology
Magnolioside 是分离自Angelica gigas Nakai(Umbelliferae) 中,对谷氨酸诱导的毒性有显著的神经保护作用。 它显示出对金黄色葡萄球菌 CIP 53.154 的中等抗菌活性。它具有抗疟原虫活性,对氯喹敏感的恶性疟原虫菌株具有强烈的生长抑制作用。
T3000 Magnolol

NSC 293099,厚朴酚,5,5'-Diallyl-2,2'-biphenyldiol

NF-κB; Retinoid Receptor; Antibacterial; PPAR; p53; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB
Magnolol (5,5'-Diallyl-2,2'-biphenyldiol) 是RXRα和PPARγ的激动剂,EC50值分别为 10.4 µM 和 17.7 µM。他是从厚朴的树皮中分离得到的一种木脂素。
TN4943 Sanguisorbigenin

地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid

Antibacterial Microbiology/Virology
Sanguisorbigenin (Tomentosolic acid) 抑制耐甲氧西林金黄色葡萄球菌,是一种天然抗菌剂。
TN2719 2',4'-Dihydroxy-6'-methoxyacetophenone

Antibacterial Microbiology/Virology
2',4'-Dihydroxy-6'-methoxyacetophenone 是从豆科植物和菊科植物中提取的酚类苯乙酮,具有抗菌活性,可用于合成吡喃镰酮。
T3798 Ziyuglycoside I

Gouguside 7,Ziyu-glycoside I,3-O-alpha-L-Arabinopyranosylpomolic acid beta-D-glucopyranosyl ester,地榆皂苷 I,苦丁冬青甙 H,Zigu-glucoside I,Kudinoside H

Apoptosis; Others Apoptosis; Others
Ziyuglycoside I (Gouguside 7) 是从地榆根中分离的一种天然产物。它可用作化妆品的有效成分,具有抗皱活性,并增加 I 型胶原蛋白的表达。它引发p53介导的细胞周期阻滞和凋亡,可用于三阴乳腺癌的相关研究。
T3828 (-)-Gallocatechin

(2S,3R)-gallocatechin,(−)-GC,(-)-棓儿茶酸;没食子儿茶素,没食子儿茶素

Others Others
(-)-Gallocatechin ((−)-GC) 是一种 (-)-Epigallocatechin (EGC) 的差向异构体,常存在于各种茶产品中,具有抗氧化特性。
T0439 L-Tryptophan

(S)-Tryptophan,Tryptophan,L-Tryptophane,Tryptophane,L-色氨酸

Amino Acids and Derivatives; Endogenous Metabolite Metabolism
L-Tryptophan (Tryptophane) 是一种必需氨基酸,是褪黑素、血清素和维生素B3的前体。
T3S1892 Crassicauline A

粗茎乌头碱甲,Crassicauline I

Others Others
Crassicauline A (Crassicauline I) 是一种乌头根中具有生物活性的生物碱。它对赤拟谷盗成虫具有拒食剂作用,其 EC50=1134.5 ppm。
T4S1876 3-Deoxyaconitine

Sodium Channel Membrane transporter/Ion channel
3-Deoxyaconitine 是一种二萜类生物碱,对钠离子通道有激活作用。
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天然产物

Iriflophenone
Cat.No: TN1768
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Eriodictyol-7-O-glucoside
Cat.No: TN1621
Synonym:
Target: Nrf2
Decanoic Acid
Cat.No: T3379
Synonym: Decoic acid,CAPRIC ACID,Caprynic acid,癸酸
Target: GluR, iGluR
Taxifolin
Cat.No: T1738
Synonym: (+)-Taxifolin,紫杉叶素,Dihydroquercetin,二氢槲皮素,(+)-Dihydroquercetin
Target: VEGFR, TNF, Tyrosinase, Adrenergic Receptor, Autophagy
Eriodictyol
Cat.No: T6S0232
Synonym: 圣草酚,Huazhongilexone
Target: Influenza Virus, DNA/RNA Synthesis, Nrf2, Endogenous Metabolite
Rhoifolin
Cat.No: T2755
Synonym: 野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside
Target: Others, p38 MAPK, NF-κB, transporter, IGF-1R, Autophagy
Lonicerin
Cat.No: TN1877
Synonym: 忍冬苦苷,金银花
Target: Apoptosis, Antibacterial
Naringenin
Cat.No: T2838
Synonym: 柚皮素,Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875
Target: P450, Influenza Virus, Reactive Oxygen Species, Endogenous Metabolite, PPAR
Benzoylmesaconine
Cat.No: T6S1885
Synonym: Mesaconine 14-benzoate,苯甲酰新乌头原碱
Target: Others
Pinocembrin-7-O-β-D-glucopyranoside
Cat.No: T5710
Synonym: Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷
Target: Others
Nortrachelogenin
Cat.No: TN4675
Synonym: (-)-Wikstromol,(-)-Nortrachelogenin
Target: Apoptosis, Antifungal
Racanisodamine
Cat.No: T0970
Synonym: 山莨菪碱,Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine,消旋山莨菪碱
Target: Adrenergic Receptor, AChR
Apigenin 7-glucoside
Cat.No: T4S0295
Synonym: 波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin
Target: Reactive Oxygen Species, HIV Protease
Juglanin
Cat.No: TQ0089
Synonym:
Target: Apoptosis, JNK, Autophagy
Acetylatractylodinol
Cat.No: TN3340
Synonym: Tractylodinol acetate,乙酰基仓术呋喃烃醇
Target: Others
Arbutin
Cat.No: T0473
Synonym: Uva,p-Arbutin,p-Arbutin,熊果苷,β-Arbutin
Target: Tyrosinase
Scopolin
Cat.No: T3888
Synonym: Murrayin,东莨菪甙,Scopoloside,东莨菪苷
Target: Sirtuin
Osthole
Cat.No: T2848
Synonym: Osthol,NSC 31868,蛇床子素,Ostol
Target: Apoptosis, HBV, Parasite, Histamine Receptor
Epibetulinic acid
Cat.No: T2S0765
Synonym:
Target: NO Synthase, Prostaglandin Receptor
Isoneochamaejasmin A
Cat.No: TN6797
Synonym:
Target: Others
Chamaechromone
Cat.No: TN1482
Synonym:
Target: P450, HBV
ETHYL OCTANOATE
Cat.No: TN6743
Synonym: 辛酸乙酯,CAPRYLIC ACID ETHYL ESTER
Target: Others
Kaempferol 3-neohesperidoside
Cat.No: TN1819
Synonym: Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷
Target: GSK-3, MEK, PI3K
Atractylenolide II
Cat.No: T5S0168
Synonym: 2-Atractylenolide,Asterolide,苍术内酯II
Target: Apoptosis, ERK, p38 MAPK, Akt, STAT
Diosmin
Cat.No: T0878
Synonym: Venosmine,Diosmil,Barosmin,地奥司明,地奥司明(7-芸香糖甙)
Target: Aryl Hydrocarbon Receptor, Norepinephrine
8-Oxocoptisine
Cat.No: TN1142
Synonym: 8-Oxycoptisine,8-氧黄连碱
Target: Others
Chelidonine
Cat.No: T5S0055
Synonym: Helidonine,Khelidonin,白屈菜碱,Stylophorin
Target: Apoptosis, Others, Influenza Virus
Indaconitine
Cat.No: T6S1879
Synonym:
Target: Others
Syringic acid
Cat.No: T2883
Synonym: 3,5-dimethyl ether Gallic Acid,SYRA,3,5-dimethoxy-4-hydroxy Benzoic Acid,丁香酸,NSC 2129
Target: Others, Endogenous Metabolite, Antibacterial
Isoastilbin
Cat.No: TN1772
Synonym:
Target: Anti-infection, Tyrosinase, Antibacterial
Aconine
Cat.No: T4S1881
Synonym: 乌头原碱,Jesaconine
Target: Others, NF-κB
Honokiol
Cat.No: T3001
Synonym: 和厚朴酚,NSC 293100
Target: ERK, HCV Protease, MEK, Akt, Autophagy
Aurantiamide acetate
Cat.No: TJS2216
Synonym: 金色酰胺醇酯,Asperglaucide
Target: Cysteine Protease
Thymol
Cat.No: T3S0717
Synonym: 2-isopropyl-5-methylphenol,Pseudoaspidin,Thymic Acid,Thyme Camphor,百里酚
Target: Antibacterial
(-)-Asarinin
Cat.No: T5S1959
Synonym: Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin
Target: Antibacterial
Hydrastine
Cat.No: TQ0160
Synonym: 北美黄连碱,(-)-β-Hydrastine,(1R,9S)-β-Hydrastine
Target: Others
Rutaecarpine
Cat.No: T2972
Synonym: Rutacarpine,吴茱萸次碱,Rhetine,Rutecarpine
Target: COX
NITIDINE
Cat.No: T8859
Synonym:
Target: Others
Histamine
Cat.No: T0965
Synonym: Ergamine,组胺
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Tyramine
Cat.No: T3095
Synonym: 4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine
Target: MAO, Endogenous Metabolite
Chenodeoxycholic acid
Cat.No: T0847
Synonym: CDCA,鹅去氧胆酸,Chenodiol
Target: Potassium Channel, FXR, Endogenous Metabolite, Autophagy
Magnolioside
Cat.No: TN1905
Synonym: 七叶苷甲基醚,6-甲氧基香豆素-7-0-BETA-D-吡喃葡萄糖苷
Target: Antifection
Magnolol
Cat.No: T3000
Synonym: NSC 293099,厚朴酚,5,5'-Diallyl-2,2'-biphenyldiol
Target: NF-κB, Retinoid Receptor, Antibacterial, PPAR, p53, Autophagy
Sanguisorbigenin
Cat.No: TN4943
Synonym: 地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid
Target: Antibacterial
2',4'-Dihydroxy-6'-methoxyacetophenone
Cat.No: TN2719
Synonym:
Target: Antibacterial
Ziyuglycoside I
Cat.No: T3798
Synonym: Gouguside 7,Ziyu-glycoside I,3-O-alpha-L-Arabinopyranosylpomolic acid beta-D-glucopyranosyl ester,地榆皂苷 I,苦丁冬青甙 H,Zigu-glucoside I,Kudinoside H
Target: Apoptosis, Others
(-)-Gallocatechin
Cat.No: T3828
Synonym: (2S,3R)-gallocatechin,(−)-GC,(-)-棓儿茶酸;没食子儿茶素,没食子儿茶素
Target: Others
L-Tryptophan
Cat.No: T0439
Synonym: (S)-Tryptophan,Tryptophan,L-Tryptophane,Tryptophane,L-色氨酸
Target: Amino Acids and Derivatives, Endogenous Metabolite
Crassicauline A
Cat.No: T3S1892
Synonym: 粗茎乌头碱甲,Crassicauline I
Target: Others
3-Deoxyaconitine
Cat.No: T4S1876
Synonym:
Target: Sodium Channel
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