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125

抑制剂 & 化合物

6

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T12064	Niraparib (R-enantiomer) MK 4827 (R-enantiomer),Niraparib R-enantiomer	PARP	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Niraparib R-enantiomer (MK 4827 R-enantiomer) 是一种 PARP1抑制剂，IC50为 2.4 nM。
T12831	SAR405 R enantiomer	Others	Others
	SAR405 R enantiomer 是一种 PIK3C3/Vps34 抑制剂，也是活性低于 SAR405 的对映体。
T15263	Selisistat R-enantiomer EX-527 (R-enantiomer)	Sirtuin	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Selisistat R-enantiomer (EX-527 (R-enantiomer)) 是 Selisistat R 型对映体。Selisistat 是SIRT1的选择性抑制剂，IC50为98 nM。
T12697	Refametinib R enantiomer RDEA119 R enantiomer,Refametinib R enantiomer,BAY 869766 R enantiomer	MEK	MAPK
	Refametinib R enantiomer (RDEA119 R enantiomer) 是一种 MEK 抑制剂，EC50为 2.0-15 nM。Refametinib R enantiomer 具有抗癌活性，可用于研究癌症。
T13140	Umbralisib R-enantiomer TGR-1202 R-enantiomer,RP5264 R-enantiomer	PI3K	PI3K/Akt/mTOR signaling
	Umbralisib R-enantiomer (RP5264 R-enantiomer) 是 PI3K 的δ型抑制剂，是 TGR-1202 活性较低的对映体。Umbralisib R-enantiomer 对δ型 pi3激酶的 IC50，至少比抑制剂对其他 PI3K 亚型(A， β和γ)的 IC50低20倍。
T19618	(R)-(-)-JQ1 Enantiomer (R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯	Epigenetic Reader Domain	Chromatin/Epigenetic
	(R)-(-)-JQ1 Enantiomer 是 (+)-JQ1 的立体异构体。 (+)-JQ1 是一种 BET 溴结构域抑制剂，对BRD4(1/2)的IC50 为 77 和 33 nM。
T11129L	Duvelisib (R enantiomer) hydrochloride IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl	PI3K	PI3K/Akt/mTOR signaling
	Duvelisib (R enantiomer) hydrochloride (INK1197 R enantiomer HCl) 是 PI3K 抑制剂。Duvelisib (R enantiomer) hydrochloride 是 Duvelisib 的活性较低的对映体。
T39541	THK5351 (R enantiomer)
	THK5351 R enantiomer is an R enantiomer of THK5351.
T17102	Tipifarnib (S enantiomer) Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer	Transferase	Metabolism
	Tipifarnib S enantiomer ((S)-(-)-R-115777) 是Tipifarnib 的 S 型对映体，它比 Tipifarnib 特性低。其中 Tipifarnib 是farnesyltransferase 高效特异性抑制剂，IC50=0.6 nM。
T12274	Siremadlin (R Enantiomer) Siremadlin R Enantiomer,HDM201 R Enantiomer,NVP-HDM201 R Enantiomer	Others	Others
	Siremadlin R Enantiomer is the R enantiomer of Siremadlin. Siremadlin is a potent and highly specific inhibitor of MDM-2/p53.
T11334	Fulvestrant (R enantiomer) ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer	Others	Others
	Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T13120	Tenalisib R Enantiomer RP6530 R Enantiomer	Others	Others
	Tenalisib R Enantiomer is an R enantiomer of Tenalisib .
T11129	Duvelisib (R enantiomer) Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer	PI3K	PI3K/Akt/mTOR signaling
	Duvelisib R enantiomer (IPI-145 R enantiomer) 是一种 Duvelisib 的对映异构体，活性较低。它是一种 PI3K 抑制剂。
T13422L	Talarozole (R enantiomer) (R)-Talarozole,Talarozole R enantiomer	Others	Others
	Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.
T10552	Bitopertin (R enantiomer) RO4917838 (R enantiomer),RG1678 (R enantiomer),Bitopertin R enantiomer	GlyT	Neuroscience
	Bitopertin R enantiomer (RG1678 R enantiomer) is the R-enantiomer of Bitopertin. Bitopertin is a noncompetitive glycine reuptake inhibitor and inhibits glycine uptake at human GlyT1 (IC50: 25 nM).
T11410	GLPG0492 (R enantiomer) GLPG0492 R enantiomer	Others	Others
	GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.
T12775	RSV604 (R enantiomer) RSV604 R enantiomer	Others	Others
	RSV604 R enantiomer is the R-enantiomer of RSV604. RSV604 is a respiratory syncytial virus (RSV) replication inhibitor.
T67881	Acalabrutinib enantiomer R-Acalabrutinib	BTK	Angiogenesis; Tyrosine Kinase/Adaptors
	Acalabrutinib enantiomer (R-Acalabrutinib) 是一类属于布鲁顿酪氨酸激酶(BTK)抑制剂的化合物。Acalabrutinib enantiomer 可用于癌症、自身免疫性疾病和慢性炎症等领域的研究。
T10856	Cobimetinib (R-enantiomer) 考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer	Others	Others
	Cobimetinib R-enantiomer is the less active R-enantiomer of Cobimetinib which is a selective MEK inhibitor.
T13312	Seviteronel R enantiomer VT-464 (R enantiomer)	Others	Others
	Seviteronel R enantiomer is the R enantiomer of Seviteronel and is a potent inhibitor of CYP17 lyase (IC50: 69 nM for h-Lyase).
T12723	Ribocil-C R enantiomer	Others	Others
	Ribocil-C R enantiomer is the R enantiomer of Ribocil-C. Ribocil-C is a highly selective bacterial riboflavin riboswitches inhibitor.
T11841	Leu-AMS R enantiomer	Others	Others
	Leu-AMS R enantiomer 是 Leu-AMS 的 R 对映体。 Leu-AMS 是一种有效的亮氨酰-tRNA 合成酶 (LRS) 抑制剂，可抑制细菌的生长。
T11662	INT-777 R-enantiomer S-EMCA R enantiomer	Others	Others
	INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5.
T11627	IACS-8968 R-enantiomer IDO/TDO Inhibitor (R-enantiomer)	IDO	Metabolism
	IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T12096	Morinidazole (R enantiomer) R-Morinidazole,R-吗啉硝唑	Others	Others
	Morinidazole (R enantiomer) is the R-enantiomer of Morinidazole.
T12612	(R)-Apremilast R-阿普斯特,(R)-CC-10004	Others	Others
	(R)-Apremilast ((R)-CC-10004) 是一种 Apremilast 的异构体。
T20898	(R)-Propranolol hydrochloride Dexpropranolol hydrochloride,(R)-(+)-Propranolol,盐酸普奈洛尔	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) 是一种抗肾上腺素受体拮抗剂，是一种普萘洛尔的活性较低的对映体。Dexpropranolol 是一种非选择性的β-adrenergic receptor 拮抗剂，对 β1AR 和 β2AR 具有高亲和力。
T10608	BRD5648 (R)-BRD0705	GSK-3	PI3K/Akt/mTOR signaling; Stem Cells
	BRD5648 ((R)-BRD0705) 是 BRD0705 的阴性对照，BRD0705 是旁系选择性和口服有效的 GSK3α 抑制剂，Kd 为 4.8 μM，IC50为 66 nM。与 GSK3β (IC50为 515 nM) 相比，BRD0705 对 GSK3α 的选择性更高 (8 倍)。BRD0705 可用于急性髓细胞性白血病。
T27210	DRX-065 DRX 065,DRX065,deuterated R-enantiomer of pioglitazone
	DRX-065 is a stabilized and deuterated R-enantiomer of pioglitazone. DRX-065 has pharmacological properties desirable for the treatment of NASH (mitochondrial function modulation, non-steroidal anti-inflammatory effects, and glucose lowering effects) with
T13448	(R)-(-)-Rolipram (R)-Rolipram,(-)-Rolipram	DNA-PK; Others	DNA Damage/DNA Repair; Others; PI3K/Akt/mTOR signaling
	(R)-(-)-Rolipram ((-)-Rolipram) 是一种 PDE4 抑制剂 Rolipram 的 R-对映异构体。
T12624	(R)-Ketorolac (+)-Ketorolac,(1R)-5-苯基-2,3-二氢-1H-吡啶-1-羧酸	Others	Others
	(R)-Ketorolac ((+)-Ketorolac) 是一种 Ketorolac 的 R 型对应体，对 COX 无作用，具有镇痛作用，并可以减少溃疡的发生。
T36839	(R)-Mephenytoin R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin	Others	Others
	(R)-Mephenytoin ((–)-Mephenytoin) 是 Mephenytoin 的 R-对映体，Mephenytoin 是一种抗惊厥药。
T70388L	(R)-Enitociclib	CDK	Cell Cycle/Checkpoint
	(R)-Enitociclib 是 BAY-1251152的一个对映体，是 CDK9 抑制剂，具有抗癌活性。
T17309	(R)-(-)-Ibuprofen levibuprofen,(R)-Ibuprofen	NF-κB	NF-κB
	(R)-(-)-Ibuprofen ((R)-Ibuprofen) 是 Ibuprofen 的 R 型异构体，对 COX 无作用，可以抑制 NF-κB 的活化；(R)-(-)-Ibuprofen 具有抗炎作用，可用于缓解疼痛的研究。
T5843	Tarenflurbil MPC7869,(R)-Flurbiprofen,R-flurbiprofen,氟比洛芬,R-氟比洛芬	Retinoid Receptor; Autophagy	Autophagy; Metabolism
	Tarenflurbil ((R)-Flurbiprofen) 是 Flurbiprofen 的 R 型对映体，可抑制 [3H]9-cis-RA 结合到 RXRαLBD，IC50为 75 μM。它可研究阿尔兹海默症。
T10012	P7C3-OMe	Others	Others
	P7C3-OMe 是促神经原性化合物，其 R-对映体活性远高于 S-对映体。可以用于研究神经精神疾病和神经退行性疾病。
T12632L	(S)-Mirtazapine (S)-6-Azamianserin,(S)-Org3770	5-HT Receptor	GPCR/G Protein; Neuroscience
	(S)-Mirtazapine ((S)-Org3770) 是 Mirtazapine 的 S(+)-对映体。(S)-Mirtazapine 是一种选择性 5-HT2 受体拮抗剂,具有促痛觉作用,常与Mirtazapine 的 R(-)-对映体混合使用来研究抑郁症。
T10003	α1 adrenoceptor-MO-1	Others	Others
	α1 adrenoceptor-MO-1（S 对映体）对α1肾上腺素受体具有亲和力，具有抗α-肾上腺素能和镇痛作用。α1 adrenoceptor-MO-1比R 对映体更具活性。
T12632	(R)-Mirtazapine (R)-Org3770,(R)-6-Azamianserin	5-HT Receptor	GPCR/G Protein; Neuroscience
	(R)-Mirtazapine ((R)-Org3770) 是 Mirtazapine 的 R(-)-对映体，在急性热痛觉动物模型中具有抗伤害感受的特性。(R)-Mirtazapine 是 5-HT3 受体的拮抗剂，是一种潜在的镇痛剂。
T22148	(S)-Lisofylline	Others	Others
	(S)-Lisofylline 是抗炎剂 (R)-lisofylline 的非活性光学对映异构体。 (S)-Lisofylline 在人肝微粒体中专门转化为己酮可可碱。
T10174	5-R-Rivaroxaban	Factor Xa	Metabolism
	5-R-Rivaroxaban 是一种 Rivaroxaban 的 R 型对映体。其中 Rivaroxaban 是选择性的Factor Xa(FXa) 抑制剂。
T12628	(R)-MG-132 (S,R,S)-(-)-MG-132,N-[(苯基甲氧基)羰基]-L-亮氨酰-N-[(1S)-1-甲酰基-3-甲基丁基]-D-亮氨酰胺,Z-Leu-D-leu-leu-al	Proteasome	Proteases/Proteasome; Ubiquitination
	(R)-MG-132 (Z-Leu-D-leu-leu-al) 是一种 MG-132 的对映异构体，是一种蛋白酶体 (proteasome) 抑制剂，细胞毒性比 MG-132 弱，是一种比 MG-132 更有效的proteasome 抑制剂。
T4295	(R)-GNE-140 GNE-140	Dehydrogenase	Metabolism
	(R)-GNE-140 (GNE-140) 是 LDHA 抑制剂，能够作用于 LDHA (IC50:3 nM) 和 LDHB (IC50:3 nM)。它的活性是 S 型异构体的 18 倍。
T12643	(R)-Terazosin (R)-特拉唑嗪,盐酸特拉唑嗪	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	(R)-Terazosin 是一种 Terazosin 的活性 R 型对映体, 是 α1-肾上腺素受体拮抗剂，对 α1a，α1b 和α1d-肾上腺素受体的Ki 分别为 6.51 nM，1.01 nM 和 1.97 nM。
T13428	(5R)-BW-4030W92	Sodium Channel	Membrane transporter/Ion channel
	(5R)-BW-4030W92是 R 型的 BW-4030W92 ，是具有活性的对映体。(5R)-BW-4030W92 是一种可口服的非选择性、电压依赖性和使用依赖性的钠离子通道 (sodium channel) 拮抗剂，可用于研究神经系统疾病。
T22354	Levocetirizine Dihydrochloride Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydrochloride is the R-enantiomer of Cetirizine, which gives it a higher affinity for the H1-receptor than the S-enantiomer. Due to this enhanced affinity, Levocetirizine Dihydrochloride is effective in treating allergic rhinitis and chronic idiopathic urticaria.
T6396	(R)-(-)-Gossypol acetic acid (-)-Gossypol acetic acid,AT-101 (acetic acid),(R)-Gossypol acetic acid,AT101醋酸,AT101,AT101 acetate	BCL; Autophagy	Apoptosis; Autophagy
	(R)-(-)-Gossypol acetic acid (AT101 acetate) 是天然产物 Gossypol 的左旋异构体，与 Bcl-2、Bcl-xL 和 Mcl-1 结合，Ki 为 0.32 μM、0.48 μM 和 0.18 μM。
T10776	CFTR corrector 4	CFTR	Membrane transporter/Ion channel
	CFTR corrector 4是一种高效且可口服的囊性纤维化跨膜电导调节剂 (CFTR)，是一种有效的 (R，R) 型活性对映体。CFTR corrector 4 可以增加细胞表面的 CFTR 水平，是用来研究囊性纤维化的潜在化合物。
T6649	(S)-(+)-Rolipram (S)-Rolipram,(+)-Rolipram,盐酸环胞苷,S- (+)-Rolipram	Apoptosis; PDE	Apoptosis; Metabolism
	(S)-(+)-Rolipram ((+)-Rolipram) 是一种 cAMP 依赖性磷酸二酯酶 4 (PDE4) 抑制剂，IC50=1100 nM。它能够抑制人单核细胞产生的肿瘤坏死因子 α (TNFα)。
T20828	Citalopram Cipram,Lu 10-171,Lu-10-171 Lu10-171	5-HT Receptor	GPCR/G Protein; Neuroscience
	Citalopram (Lu 10-171) 是一种具有口服活性的、选择性的血清素再摄取抑制剂 (SSRI)，是一种选择性5-羟色胺再摄取抑制剂，是一种 S(+)-对映体 (Escitalopram) 和 R(-)-对映体的外消旋混合物。Citalopram 具有抗抑郁活性，可增强血清素能神经传递，可用于研究老年痴呆。

化合物

Niraparib (R-enantiomer)

Cat.No: T12064

Synonym: MK 4827 (R-enantiomer),Niraparib R-enantiomer

Target: PARP

SAR405 R enantiomer

Cat.No: T12831

Target: Others

Selisistat R-enantiomer

Cat.No: T15263

Synonym: EX-527 (R-enantiomer)

Target: Sirtuin

Refametinib R enantiomer

Cat.No: T12697

Synonym: RDEA119 R enantiomer,Refametinib R enantiomer,BAY 869766 R enantiomer

Target: MEK

Umbralisib R-enantiomer

Cat.No: T13140

Synonym: TGR-1202 R-enantiomer,RP5264 R-enantiomer

Target: PI3K

(R)-(-)-JQ1 Enantiomer

Cat.No: T19618

Synonym: (R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯

Target: Epigenetic Reader Domain

Duvelisib (R enantiomer) hydrochloride

Cat.No: T11129L

Synonym: IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl

Target: PI3K

THK5351 (R enantiomer)

Cat.No: T39541

Tipifarnib (S enantiomer)

Cat.No: T17102

Synonym: Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer

Target: Transferase

Siremadlin (R Enantiomer)

Cat.No: T12274

Synonym: Siremadlin R Enantiomer,HDM201 R Enantiomer,NVP-HDM201 R Enantiomer

Target: Others

Fulvestrant (R enantiomer)

Cat.No: T11334

Synonym: ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer

Target: Others

Tenalisib R Enantiomer

Cat.No: T13120

Synonym: RP6530 R Enantiomer

Target: Others

Duvelisib (R enantiomer)

Cat.No: T11129

Synonym: Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer

Target: PI3K

Talarozole (R enantiomer)

Cat.No: T13422L

Synonym: (R)-Talarozole,Talarozole R enantiomer

Target: Others

Bitopertin (R enantiomer)

Cat.No: T10552

Synonym: RO4917838 (R enantiomer),RG1678 (R enantiomer),Bitopertin R enantiomer

Target: GlyT

GLPG0492 (R enantiomer)

Cat.No: T11410

Synonym: GLPG0492 R enantiomer

Target: Others

RSV604 (R enantiomer)

Cat.No: T12775

Synonym: RSV604 R enantiomer

Target: Others

Acalabrutinib enantiomer

Cat.No: T67881

Synonym: R-Acalabrutinib

Target: BTK

Cobimetinib (R-enantiomer)

Cat.No: T10856

Synonym: 考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer

Target: Others

Seviteronel R enantiomer

Cat.No: T13312

Synonym: VT-464 (R enantiomer)

Target: Others

Ribocil-C R enantiomer

Cat.No: T12723

Target: Others

Leu-AMS R enantiomer

Cat.No: T11841

Target: Others

INT-777 R-enantiomer

Cat.No: T11662

Synonym: S-EMCA R enantiomer

Target: Others

IACS-8968 R-enantiomer

Cat.No: T11627

Synonym: IDO/TDO Inhibitor (R-enantiomer)

Target: IDO

Morinidazole (R enantiomer)

Cat.No: T12096

Synonym: R-Morinidazole,R-吗啉硝唑

Target: Others

Cat.No: T12612

Synonym: R-阿普斯特,(R)-CC-10004

Target: Others

(R)-Propranolol hydrochloride

Cat.No: T20898

Synonym: Dexpropranolol hydrochloride,(R)-(+)-Propranolol,盐酸普奈洛尔

Target: Adrenergic Receptor

Cat.No: T10608

Synonym: (R)-BRD0705

Target: GSK-3

Cat.No: T27210

Synonym: DRX 065,DRX065,deuterated R-enantiomer of pioglitazone

(R)-(-)-Rolipram

Cat.No: T13448

Synonym: (R)-Rolipram,(-)-Rolipram

Target: DNA-PK, Others

Cat.No: T12624

Synonym: (+)-Ketorolac,(1R)-5-苯基-2,3-二氢-1H-吡啶-1-羧酸

Target: Others

(R)-Mephenytoin

Cat.No: T36839

Synonym: R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin

Target: Others

(R)-Enitociclib

Cat.No: T70388L

Target: CDK

(R)-(-)-Ibuprofen

Cat.No: T17309

Synonym: levibuprofen,(R)-Ibuprofen

Target: NF-κB

Cat.No: T5843

Synonym: MPC7869,(R)-Flurbiprofen,R-flurbiprofen,氟比洛芬,R-氟比洛芬

Target: Retinoid Receptor, Autophagy

Cat.No: T10012

Target: Others

(S)-Mirtazapine

Cat.No: T12632L

Synonym: (S)-6-Azamianserin,(S)-Org3770

Target: 5-HT Receptor

α1 adrenoceptor-MO-1

Cat.No: T10003

Target: Others

(R)-Mirtazapine

Cat.No: T12632

Synonym: (R)-Org3770,(R)-6-Azamianserin

Target: 5-HT Receptor

(S)-Lisofylline

Cat.No: T22148

Target: Others

5-R-Rivaroxaban

Cat.No: T10174

Target: Factor Xa

Cat.No: T12628

Synonym: (S,R,S)-(-)-MG-132,N-[(苯基甲氧基)羰基]-L-亮氨酰-N-[(1S)-1-甲酰基-3-甲基丁基]-D-亮氨酰胺,Z-Leu-D-leu-leu-al

Target: Proteasome

Cat.No: T4295

Synonym: GNE-140

Target: Dehydrogenase

Cat.No: T12643

Synonym: (R)-特拉唑嗪,盐酸特拉唑嗪

Target: Adrenergic Receptor

(5R)-BW-4030W92

Cat.No: T13428

Target: Sodium Channel

Levocetirizine Dihydrochloride

Cat.No: T22354

Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride

Target: Histamine Receptor

(R)-(-)-Gossypol acetic acid

Cat.No: T6396

Synonym: (-)-Gossypol acetic acid,AT-101 (acetic acid),(R)-Gossypol acetic acid,AT101醋酸,AT101,AT101 acetate

Target: BCL, Autophagy

CFTR corrector 4

Cat.No: T10776

Target: CFTR

(S)-(+)-Rolipram

Cat.No: T6649

Synonym: (S)-Rolipram,(+)-Rolipram,盐酸环胞苷,S- (+)-Rolipram

Target: Apoptosis, PDE

Cat.No: T20828

Synonym: Cipram,Lu 10-171,Lu-10-171 Lu10-171

Target: 5-HT Receptor

Cat. No.	Product Name	Target	Signaling Pathways
T10935	D-Glutamic acid (R)-Glutamic acid,D-谷氨酸	Endogenous Metabolite	Metabolism
	D-Glutamic acid ((R)-Glutamic acid) 是一种广泛用于药物和食品中的L-glutamic acid 对映异构体。
T4000	(±)-Equol Equol,(±)-雌马酚,(R,S)-Equol	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Drug Metabolite	Endocrinology/Hormones; Metabolism
	(±)-Equol ((R,S)-Equol) 是 equol 的外消旋体。它对 ERα 和 ERβ 的 EC50s of 分别为 200 和 74 nM。Equol 是大豆异黄酮黄豆苷和大豆黄素的代谢产物。
T6491	(-)-(S)-Equol (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) 是雌激素受体β的高亲和力配体。
T0185	Escitalopram Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体，是一种选择性 5-羟色胺再摄取抑制剂，Ki=0.89 nM，比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性，是一种研究抑郁症的抗抑郁药。
T40529	(R)-(-)-1,2-Propanediol
	(R)-(-)-1,2-Propanediol is the (R)-enantiomer of 1,2-Propanediol, which is derived from glucose through the expression of NADH-linked glycerol dehydrogenase genes in Escherichia coli.
T40576	(S)-Salsolidine
	(S)-Salsolidine, a chemical compound, functions as a weak inhibitor of monoamine oxidase (MAO), exhibiting an inhibition constant (K i ) of 63 μM. R enantiomer demonstrating a greater efficacy than (S)-Salsolidine, boasting a K i value of 26 μM compared to the S form.

天然产物

D-Glutamic acid

Cat.No: T10935

Synonym: (R)-Glutamic acid,D-谷氨酸

Target: Endogenous Metabolite

Cat.No: T4000

Synonym: Equol,(±)-雌马酚,(R,S)-Equol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite

Cat.No: T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Cat.No: T0185

Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor

(R)-(-)-1,2-Propanediol

Cat.No: T40529

(S)-Salsolidine

Cat.No: T40576

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