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Targets Recommended: GABA Receptor

218

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6355 (R)-baclofen

STX209,Arbaclofen,(R)-巴氯芬

GABA Receptor Membrane transporter/Ion channel; Neuroscience
(R)-baclofen (STX209) 是一种选择性GABAB 受体激动剂。
T5843L (S)-Flurbiprofen

esflurbiprofen,(S)-氟比洛芬

COX; PGE Synthase Immunology/Inflammation; Neuroscience
Esflurbiprofen 是 Flurbiprofen 的活性对映体,是 COX-1 和 COX-2 的抑制剂,对 COX-1和 COX-2的 IC50分别为0.48 和 0.47 μM。
T11071 Dofequidar fumarate

MS-209

P-gp Membrane transporter/Ion channel; Neuroscience
Dofequidar fumarate (MS-209) 是口服活性的喹啉化合物,通过抑制 ABCB1/P-gp 和 ABCC1/MDR 相关蛋白 1 来克服 MDR。
T25956 Piketoprofen

Calmatel

Others Others
Piketoprofen (Calmatel) 是一种局部非甾体抗炎药。
T4384 Halofenozide

Others Others
Halofenozide 是一种新的昆虫生长调节剂 (IGR),具有苯甲酰肼结构,也是一种蜕皮激素 (ecdysteroid) 激动剂。可模拟天然昆虫蜕皮激素 20-羟基蜕皮激素的作用,
T16022 Arhalofenate

JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102

PPAR DNA Damage/DNA Repair; Metabolism
Arhalofenate (JNJ 39659100) 是一种选择性的(PPAR)-γ部分激动剂,用于研究 2 型糖尿病。
T4466 Pitofenone hydrochloride

Baralgin Ketone Hydrochloride,Pitophenone hydrochloride,吡托非农盐酸盐

AChE Neuroscience
Pitofenone hydrochloride (Pitophenone hydrochloride) 是一种能够抑制乙酰胆碱酯酶活性的解痉化合物,对于来自牛红细胞和电鳗的乙酰胆碱酯酶的Ki 分别为 36 和 45 μM。
T0839 Ketoprofen

酮基布洛芬,RP-19583,酮洛芬

Apoptosis; COX; MRP Apoptosis; Immunology/Inflammation; Neuroscience
Ketoprofen (RP-19583) 是一种非甾体抗炎剂,能够有效地抑制COX 的活性,在人血单核细胞中,对 COX-1 和 COX-2 的IC50值分别为 2 nM 和 26 nM。
T4440 Saclofen

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Saclofen 是竞争性GABAB 受体拮抗剂(IC50:7.8 μM)。它可研究 GABAB 受体调节大脑中缓慢抑制性突触后电位的功能。
T0291 Flurbiprofen

氟比洛芬,dl-Flurbiprofen

Apoptosis; COX; MRP Apoptosis; Immunology/Inflammation; Neuroscience
Flurbiprofen (dl-Flurbiprofen) 是一种高效的,具有口服活性的非甾体抗炎化合物,有退热止痛活性, 常用于炎症性疾病的研究。它是一种非选择性的环氧合酶抑制剂,可研究结肠癌。
T6476 Dofetilide

UK 68789,UK-68798,Tikosyn,多非利特

Potassium Channel Membrane transporter/Ion channel
Dofetilide (UK 68789) 是一种具有口服活性、有效的且特异性的IKr 阻滞剂,作为 III 类抗心律失常药物。Dofetilide 可用于心血管疾病研究。
T6470 Diclofenac Potassium

双氯芬酸钾,CGP-45840B,Cataflam,Voltfast

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Diclofenac Potassium (CGP-45840B) 是一种非甾体抗炎药,用于减轻炎症并在某些情况下作为镇痛剂减轻疼痛。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的IC50值分别为 5.1 μM 和0.84 μM。
T5030 Zofenopril calcium

SQ26991,佐芬普利钙,Zofenopril (calcium)

RAAS; Reactive Oxygen Species Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
Zofenopril calcium (SQ26991) 是一种抗氧化剂和血管紧张素转化酶 (ACE) 抑制剂。
T4994 Tocofersolan

Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯

Others Others
Tocofersolan (TPGS) 是合成的 α-生育酚的聚乙二醇衍生物。
T36683 Vedaprofen

Quadrisol,PM 150,维达洛芬,CERM 10202

COX; Antibacterial; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Vedaprofen (PM 150) 抑制 COX-1 并通过抗炎活性减少前列腺素 H2 的合成。 Vedaprofen 是一种大肠杆菌滑动钳抑制剂,IC50 为 222 μM,Ki 为 131 μM。
T0321 Indoprofen

吲哚洛芬,(±)-Indoprofe,茚酮苯丙酸

COX Immunology/Inflammation; Neuroscience
Indoprofen ((±)-Indoprofe) 是非甾体类抗炎药, 可用于研究脊髓性肌萎缩。
T0184 Fenoprofen calcium dihydrate

COX Immunology/Inflammation; Neuroscience
Fenoprofen calcium dihydrate 是一种丙酸衍生物,用作非甾体抗炎剂。
T50053 Lofemizole

P450 Metabolism
Lofemizole 是 CYP1A2 的拮抗剂。
T1065 Baclofen

巴氯芬,Lioresal

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Baclofen (Lioresal) 是 γ-氨基丁酸 (GABA) 的亲脂性衍生物,是可口服的选择性代谢型 GABA-B 受体激动剂,具有高血脑屏障渗透率,用于治疗因脊髓损伤和多发性硬化引起的痉挛。
T6540 Ibuprofen Lysine

布洛芬赖氨酸盐,Neoprofen

COX Immunology/Inflammation; Neuroscience
Ibuprofen Lysine (Neoprofen) 是一种非甾体抗炎药。
T12987 Spirodiclofen

BAJ-2740,螺螨酯

Parasite Microbiology/Virology
Spirodiclofen (BAJ-2740) 是选择性非系统性的杀螨剂,来自新的化学类特酮酸衍生物, 与目前市面上的杀螨剂无交叉耐药, 具有额外的杀虫性能。
T8364 Mebrofenin

N-(3-溴-2,4,6-三甲基苯基甲酰甲基)乙酰乙酸,SQ 26962

Others Others
Mebrofenin (SQ 26962) 是一种亚氨基二乙酸 (IDA) ,可用作 Tc-99m 的放射性标记试剂盒。其中Tc-99m Mebrofenin 是一种诊断剂,用于肝胆显像,也是评价肝功能的首选放射性药物。
T6568 Licofelone

利克飞龙,ML-3000

Apoptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Licofelone (ML-3000) 是一种 COX/LOX 双重抑制剂,IC50分别为 0.21和0.18 μM,有潜力研究骨关节炎,具有抗炎和抗增殖作用。它可诱导细胞凋亡,减少促炎性白三烯和前列腺素的产生。
T0643 Diclofenac Amide

Others Others
Diclofenac Amide 用作Diclofenac 的中间体。
T15300 Fluorofenidone

AKF-PD

Others Others
Fluorofenidone (AKF-PD) 是 AMR69 的类似物,抗纤维化活性与 AMR69相同,但 Fluorofenidone 的毒性更低,半衰期长。它部分通过 PI3K/Akt 信号通路抑制 NADPH 氧化酶和细胞外基质 (ECM) 的沉积,能够减少肾间质纤维化的发生。
T37482 Diclofenac methyl ester

Others Others
Diclofenac methyl ester 是双氯芬酸(diclofenac)的疏水性前药形式,它是一种非甾体抗炎药 (NSAID)。它比双氯芬酸更易溶于肉豆蔻酸异丙酯,但毒性更高。
T16329 Nitroflurbiprofen

NO-flurbiprofen,Nitroxybutyl flurbiprofen,硝基氟比洛芬,HCT 1206

COX Immunology/Inflammation; Neuroscience
Nitroflurbiprofen (Nitroxybutyl flurbiprofen) 是一种释放 NO 的环氧合酶抑制剂,可调节门脉高压性肝硬化大鼠肝内血管张力的增加。
T1185 Rofecoxib

MK 966,罗非昔布,罗非考昔,MK-0966

COX Immunology/Inflammation; Neuroscience
Rofecoxib (MK 966) 是可口服的 COX-2特异性抑制剂,具有抗炎、解热和镇痛特性以及潜在的抗肿瘤特性。在人骨肉瘤细胞和中国仓鼠卵巢细胞中,对人 COX-2 的 IC50值分别为 26 和 18 nM。
T5460 Mofezolac

莫苯唑酸,莫非佐酸

COX Immunology/Inflammation; Neuroscience
Mofezolac 是一种非甾体类抗炎药,可缓解疼痛并具有抗炎活性,抑制 COX-1和COX-2的IC50为 1.44 和 447 nM。
T2553 Etofenamate

COX Immunology/Inflammation; Neuroscience
Etofenamate 是非甾体类抗炎小分子,也是非选择性的 COX 抑制剂,具有抗风湿和解热抗炎作用,可用于缓解疼痛、关节炎等炎症相关疾病的研究。
T0463 Loxoprofen

Loxoprofene,洛索洛芬,Loxoprofeno,Koloxo

COX Immunology/Inflammation; Neuroscience
Loxoprofen (Koloxo) 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX 抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
T0159 Pranoprofen

普拉洛芬,Pyranoprofen

Apoptosis; COX; PGE Synthase; Prostaglandin Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pranoprofen (Pyranoprofen) 可抑制COX1/2酶,阻断花生四烯酸转化为二十烷醇,减少前列腺素的合成。它是一种用于眼科的非甾体抗炎试剂。
T0196 Diclofenac

双氯芬酸,奥尔芬,Diclofenacum,Voltaren

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac (Diclofenacum) 是一种具有抗炎活性的非甾体苯乙酸衍生物,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T6687 Suprofen

Maldocil,Suprol,TN-762,舒洛芬,Profenal

COX; PGE Synthase Immunology/Inflammation; Neuroscience
Suprofen (Suprol) 是一种非甾体抗炎化合物,对前列腺素合成具有抑制作用。
T7363 Ibuprofen Piconol

U75630,匹美诺芬,布洛芬吡啶甲醇

Others Others
Ibuprofen Piconol (U75630) 是非甾体抗炎药物,局部使用可缓解原发性热灼伤和晒伤。
T6497 Fenoprofen Calcium

Others; COX Immunology/Inflammation; Neuroscience; Others
Fenoprofen Calcium 是一种非甾体类抗炎药,可治疗关节炎。
T34268 Raxofelast

IRFI016,IRFI-016,IRFI 016

Raxofelast (IRFI-016) 具有治疗糖尿病并发症和动脉粥样硬化的潜力
T27572 Ibuprofen diethylaminoethyl ester

Brufen diethylaminoethyl ester,BF-DEAE,BF DEAE

Others Others
Ibuprofen diethylaminoethyl ester (BF DEAE) 具有抗炎活性,可作为局部麻醉剂,可用于研究麻风性神经炎等神经系统疾病。
T3496 Buprofezin

噻嗪酮,NNI 750,Applaud,Buprofezine

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Buprofezin (Applaud) 是一种杀虫剂,通过抑制几丁质合成起作用,在体外还可以剂量依赖性地增加活性氧的产生。
T19679 Benoxaprofen

氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459

COX Immunology/Inflammation; Neuroscience
Benoxaprofen (NSC-299582) 是长效的、强效的抗炎和解热化合物,在体外具有较弱的对环氧合酶的抑制作用,也可以抑制脂氧合酶,在一些炎症动物模型中抑制单核细胞迁移。
T39280 Nitrofen

Others Others
Nitrofen 是选择性接触除草剂,也是视原卟啉原氧化酶和网膜脱氢酶抑制剂。
T9472 Rebamipide mofetil

COX Immunology/Inflammation; Neuroscience
Rebamipide mofetil 是 Rebamipide 的口服活性前药,是一种粘膜保护剂。
T1555 Diclofenac sodium

GP 45840,双氯芬酸钠

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac sodium (GP 45840) 是一种非选择性抗炎剂,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T6053 Turofexorate Isopropyl

XL335,FXR-450,WAY-362450,妥芬异丙酯

FXR; Autophagy Autophagy; Metabolism
Turofexorate Isopropyl (XL335) 是一种口服有效的,选择性 FXR 激动剂,EC50为 4 nM。
T1394 Ibuprofen

Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil

COX Immunology/Inflammation; Neuroscience
Ibuprofen (Advil) 是一种丙酸衍生物和非甾体抗炎药 (NSAID),具有抗炎、镇痛和解热作用。它是COX-1和COX-2的抑制剂,IC50值分别为 13 和 370 μM,导致前列腺素和血栓素前体的形成减少。
T0463L Loxoprofen sodium

CS-600,CS600,Loxoprofen,CS 600

COX Immunology/Inflammation; Neuroscience
Loxoprofen sodium (CS-600) 是一种有效的和具有口服活性的非选择性 COX 抑制剂,对 COX-1 和 COX-2具有抑制作用, IC50 分别为 6.5 和 13.5 μM。 Loxoprofen sodium 通过减少花生四烯酸合成前列腺素而起作用。Loxoprofen sodium 具有抗炎和抗肿瘤活性,可用来治疗动脉粥样硬化。
T0448 (S)-(+)-Ibuprofen

左旋布洛芬,Dexibuprofen,(S)-Ibuprofen,(S)-(+)-布洛芬

BCL; Thrombin; Cysteine Protease; COX; PPAR Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; Proteases/Proteasome
(S)-(+)-Ibuprofen (Dexibuprofen) 是 Ibuprofen 的 S(+)-对映异构体,能够有效的抑制COX-1(IC50:2.1 μM)和COX-2(IC50:1.6 μM),。它具有抗癌、退热、止痛,抗炎的效果。
T6498 Fenoprofen calcium hydrate

Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate,非诺洛芬钙二水合物

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Fenoprofen calcium hydrate (Progesic dihydrate) 是一非甾体类抗炎症化合物。
T11854 Lipofermata

Others; Antibacterial Microbiology/Virology; Others
Lipofermata 是一种脂肪酸转运蛋白 2抑制剂,可阻止脂质转运至黑色素瘤细胞并减少黑色素瘤的生长和侵袭。
T15773 Lofepramine

Gamanil,洛非帕明,Amplit,Leo 640,Lopramine

5-HT Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Lofepramine (Leo 640) 是一种有效的三环抗抑郁药,广泛地代谢为 Desipramine。它能够抑制摄取促进去甲肾上腺素能神经传递,以及抑制神经元摄取 5-羟色胺和色氨酸吡咯酶,增强 5-羟色胺能神经传递,进而发挥其抗抑郁作用。它还具有显著的抗焦虑效果。

化合物

(R)-baclofen
Cat.No: T6355
Synonym: STX209,Arbaclofen,(R)-巴氯芬
Target: GABA Receptor
(S)-Flurbiprofen
Cat.No: T5843L
Synonym: esflurbiprofen,(S)-氟比洛芬
Target: COX, PGE Synthase
Dofequidar fumarate
Cat.No: T11071
Synonym: MS-209
Target: P-gp
Piketoprofen
Cat.No: T25956
Synonym: Calmatel
Target: Others
Halofenozide
Cat.No: T4384
Synonym:
Target: Others
Arhalofenate
Cat.No: T16022
Synonym: JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102
Target: PPAR
Pitofenone hydrochloride
Cat.No: T4466
Synonym: Baralgin Ketone Hydrochloride,Pitophenone hydrochloride,吡托非农盐酸盐
Target: AChE
Ketoprofen
Cat.No: T0839
Synonym: 酮基布洛芬,RP-19583,酮洛芬
Target: Apoptosis, COX, MRP
Saclofen
Cat.No: T4440
Synonym:
Target: GABA Receptor
Flurbiprofen
Cat.No: T0291
Synonym: 氟比洛芬,dl-Flurbiprofen
Target: Apoptosis, COX, MRP
Dofetilide
Cat.No: T6476
Synonym: UK 68789,UK-68798,Tikosyn,多非利特
Target: Potassium Channel
Diclofenac Potassium
Cat.No: T6470
Synonym: 双氯芬酸钾,CGP-45840B,Cataflam,Voltfast
Target: Apoptosis, Others, COX
Zofenopril calcium
Cat.No: T5030
Synonym: SQ26991,佐芬普利钙,Zofenopril (calcium)
Target: RAAS, Reactive Oxygen Species
Tocofersolan
Cat.No: T4994
Synonym: Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯
Target: Others
Vedaprofen
Cat.No: T36683
Synonym: Quadrisol,PM 150,维达洛芬,CERM 10202
Target: COX, Antibacterial, Prostaglandin Receptor
Indoprofen
Cat.No: T0321
Synonym: 吲哚洛芬,(±)-Indoprofe,茚酮苯丙酸
Target: COX
Fenoprofen calcium dihydrate
Cat.No: T0184
Synonym:
Target: COX
Lofemizole
Cat.No: T50053
Synonym:
Target: P450
Baclofen
Cat.No: T1065
Synonym: 巴氯芬,Lioresal
Target: GABA Receptor
Ibuprofen Lysine
Cat.No: T6540
Synonym: 布洛芬赖氨酸盐,Neoprofen
Target: COX
Spirodiclofen
Cat.No: T12987
Synonym: BAJ-2740,螺螨酯
Target: Parasite
Mebrofenin
Cat.No: T8364
Synonym: N-(3-溴-2,4,6-三甲基苯基甲酰甲基)乙酰乙酸,SQ 26962
Target: Others
Licofelone
Cat.No: T6568
Synonym: 利克飞龙,ML-3000
Target: Apoptosis, Lipoxygenase, COX
Diclofenac Amide
Cat.No: T0643
Synonym:
Target: Others
Fluorofenidone
Cat.No: T15300
Synonym: AKF-PD
Target: Others
Diclofenac methyl ester
Cat.No: T37482
Synonym:
Target: Others
Nitroflurbiprofen
Cat.No: T16329
Synonym: NO-flurbiprofen,Nitroxybutyl flurbiprofen,硝基氟比洛芬,HCT 1206
Target: COX
Rofecoxib
Cat.No: T1185
Synonym: MK 966,罗非昔布,罗非考昔,MK-0966
Target: COX
Mofezolac
Cat.No: T5460
Synonym: 莫苯唑酸,莫非佐酸
Target: COX
Etofenamate
Cat.No: T2553
Synonym:
Target: COX
Loxoprofen
Cat.No: T0463
Synonym: Loxoprofene,洛索洛芬,Loxoprofeno,Koloxo
Target: COX
Pranoprofen
Cat.No: T0159
Synonym: 普拉洛芬,Pyranoprofen
Target: Apoptosis, COX, PGE Synthase, Prostaglandin Receptor
Diclofenac
Cat.No: T0196
Synonym: 双氯芬酸,奥尔芬,Diclofenacum,Voltaren
Target: Apoptosis, COX
Suprofen
Cat.No: T6687
Synonym: Maldocil,Suprol,TN-762,舒洛芬,Profenal
Target: COX, PGE Synthase
Ibuprofen Piconol
Cat.No: T7363
Synonym: U75630,匹美诺芬,布洛芬吡啶甲醇
Target: Others
Fenoprofen Calcium
Cat.No: T6497
Synonym:
Target: Others, COX
Raxofelast
Cat.No: T34268
Synonym: IRFI016,IRFI-016,IRFI 016
Target:
Ibuprofen diethylaminoethyl ester
Cat.No: T27572
Synonym: Brufen diethylaminoethyl ester,BF-DEAE,BF DEAE
Target: Others
Buprofezin
Cat.No: T3496
Synonym: 噻嗪酮,NNI 750,Applaud,Buprofezine
Target: Reactive Oxygen Species
Benoxaprofen
Cat.No: T19679
Synonym: 氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459
Target: COX
Nitrofen
Cat.No: T39280
Synonym:
Target: Others
Rebamipide mofetil
Cat.No: T9472
Synonym:
Target: COX
Diclofenac sodium
Cat.No: T1555
Synonym: GP 45840,双氯芬酸钠
Target: Apoptosis, COX
Turofexorate Isopropyl
Cat.No: T6053
Synonym: XL335,FXR-450,WAY-362450,妥芬异丙酯
Target: FXR, Autophagy
Ibuprofen
Cat.No: T1394
Synonym: Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil
Target: COX
Loxoprofen sodium
Cat.No: T0463L
Synonym: CS-600,CS600,Loxoprofen,CS 600
Target: COX
(S)-(+)-Ibuprofen
Cat.No: T0448
Synonym: 左旋布洛芬,Dexibuprofen,(S)-Ibuprofen,(S)-(+)-布洛芬
Target: BCL, Thrombin, Cysteine Protease, COX, PPAR
Fenoprofen calcium hydrate
Cat.No: T6498
Synonym: Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate,非诺洛芬钙二水合物
Target: Apoptosis, Others, COX
Lipofermata
Cat.No: T11854
Synonym:
Target: Others, Antibacterial
Lofepramine
Cat.No: T15773
Synonym: Gamanil,洛非帕明,Amplit,Leo 640,Lopramine
Target: 5-HT Receptor, Norepinephrine
Cat. No. Product Name Target Signaling Pathways
T6293 Mycophenolate Mofetil

TM-MMF,吗替麦考酚酯,RS 61443

Apoptosis; Dehydrogenase; Drug Metabolite Apoptosis; Metabolism
Mycophenolate Mofetil (TM-MMF) 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。
T4394 Methyl Isoferulate

Others Others
Methyl Isoferulate 从毛竹叶中分离纯化。
T0558 Dihydroferulic acid

Dihydroconiferylic acid,氢化阿魏酸,Hydroferulic acid

Others Others
Dihydroferulic acid 是一种姜黄素的主要代谢产物,具有抗氧化/清除自由基的活性,其IC50=19.5 μM。它是香草酸的前体物质,也是人类肠道菌群的代谢产物。
TN1145 Isofebrifugine

Parasite Microbiology/Virology
Isofebrifugine 是一种来自虎耳草科植物常山的生物碱,具有抗疟抗感染活性。
T2889 Isoferulic acid

Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate,异阿魏酸

Influenza Virus; Adrenergic Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience
Isoferulic acid (Hesperetate) 是一种肉桂酸衍生物,有抗糖尿病活性和抗流感病毒活性。它能结合并激活 α1-肾上腺素能受体,增强 β-内啡肽的分泌并增加体外葡萄糖的使用。
T9790 Lactoferrin

Lactoferrin (Bovine)

Endogenous Metabolite Metabolism
Lactoferrin 由哺乳动物分泌,具有广泛的生物学作用,包括提高应用良好的益生菌菌株的耐寒性。
T81099 Staphyloferrin A

Staphyloferrin A,一种铁载体蛋白,与抗生素结合对抗抗药性细菌性皮肤病进行研究。
TN3662 Cinnamyl isoferulate

Others Others
Cinnamyl isoferulate是一种天然产物,属于杨柳科杨属,其产品编号为 TN3662,CAS号为 115610-31-6。Cinnamyl isoferulate可用作对照参考。
T40988 (+)-Norlirioferine

(+)-Norlirioferine is an alkaloid compound that exhibits cell growth inhibitory effects on macrophages and VERO cells.
T10072 2-Hydroxy Ibuprofen

2-羟基布洛芬,(±)-2-Hydroxy Ibuprofen

Others Others
2-Hydroxy Ibuprofen is a metabolite of Ibuprofen. Ibuprofen is an anti-inflammatory inhibitor targeting COX-1/COX-2 (IC50s: 13 μM/370 μM).

天然产物

Mycophenolate Mofetil
Cat.No: T6293
Synonym: TM-MMF,吗替麦考酚酯,RS 61443
Target: Apoptosis, Dehydrogenase, Drug Metabolite
Methyl Isoferulate
Cat.No: T4394
Synonym:
Target: Others
Dihydroferulic acid
Cat.No: T0558
Synonym: Dihydroconiferylic acid,氢化阿魏酸,Hydroferulic acid
Target: Others
Isofebrifugine
Cat.No: TN1145
Synonym:
Target: Parasite
Isoferulic acid
Cat.No: T2889
Synonym: Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate,异阿魏酸
Target: Influenza Virus, Adrenergic Receptor
Lactoferrin
Cat.No: T9790
Synonym: Lactoferrin (Bovine)
Target: Endogenous Metabolite
Staphyloferrin A
Cat.No: T81099
Synonym:
Target:
Cinnamyl isoferulate
Cat.No: TN3662
Synonym:
Target: Others
(+)-Norlirioferine
Cat.No: T40988
Synonym:
Target:
2-Hydroxy Ibuprofen
Cat.No: T10072
Synonym: 2-羟基布洛芬,(±)-2-Hydroxy Ibuprofen
Target: Others
Cat. No. Product Name Species Expression System
TMPY-04142 RANK/TNFRSF11A Protein, Human, Recombinant (hFc)

OPTB7,OFE,OSTS,LOH18CR1,FEO,TRANCER,tumor necrosis ...

Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small intestine and adrenal gland. It is an essential mediator for osteoclast and lymph node development. TNFRSF11A and its ligand are important regulators of the interaction between T cells and dendritic cells. It can interact with various TRAF family proteins, through which this recep...
TMPY-05514 RANK/TNFRSF11A Protein, Human, Recombinant (mFc)

OFE,RANK,OPTB7,FEO,tumor necrosis factor receptor s...

Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small intestine and adrenal gland. It is an essential mediator for osteoclast and lymph node development. TNFRSF11A and its ligand are important regulators of the interaction between T cells and dendritic cells. It can interact with various TRAF family proteins, through which this recep...
TMPY-04157 RANK/TNFRSF11A Protein, Human, Recombinant (His)

ODFR,OFE,CD265,PDB2,RANK,tumor necrosis factor rece...

Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small intestine and adrenal gland. It is an essential mediator for osteoclast and lymph node development. TNFRSF11A and its ligand are important regulators of the interaction between T cells and dendritic cells. It can interact with various TRAF family proteins, through which this recep...
TMPJ-00349 RANK/TNFRSF11A Protein, Human, Recombinant (aa 30-212, His)

CD265 antigen,FEO,TRANCER,ODFR,ODFROSTS,TRANCE R,TNFRSF11A,<...

Human Human Cells
Receptor Activator of Nuclear Factor κ B (RANK), also known as CD265, TRANCE Receptor or TNFRSF11A, is member of the tumor necrosis factor receptor (TNFR) molecular superfamily. RANK is the receptor for RANK-Ligand (RANKL) and part of the RANK/RANKL/OPG signaling pathway that regulates osteoclast differentiation and activation. It plays a vital role in bone remodeling and repair, immune cell function, lymph node development, thermal regulation, and mammary gland development. RANK is constitutive...
TMPY-02728 Lactoferrin/LTF Protein, Mouse, Recombinant (His)

MMS10R,Lf,Csp82,lactotransferrin,Ms10r

Mouse HEK293
Lactotransferrin, also known as Lactoferrin, Talalactoferrin, and LTF, is a secreted protein that belongs to the transferrin family. Transferrins are iron binding transport proteins that can bind two Fe3+ions in association with the binding of an anion, usually bicarbonate. Lactotransferrin has antimicrobial activity which depends on the extracellular cation concentration. Lactoferroxins A, B, and C have opioid antagonist activity. Lactoferrin A shows a preference for mu-receptors, while lactofe...
TMPY-02188 Lactoferrin/LTF Protein, Human, Recombinant (His)

HEL110,LF,HLF2,GIG12,lactotransferrin

Human HEK293
Lactotransferrin, also known as Lactoferrin, Talalactoferrin, and LTF, is a secreted protein that belongs to the transferrin family. Transferrins are iron binding transport proteins that can bind two Fe3+ions in association with the binding of an anion, usually bicarbonate. Lactotransferrin has antimicrobial activity which depends on the extracellular cation concentration. Lactoferroxins A, B, and C have opioid antagonist activity. Lactoferrin A shows a preference for mu-receptors, while lactofe...
TMPH-02646 Erythroferrone Protein, Mouse, Recombinant (His)

Mouse Yeast
Iron-regulatory hormone that acts as an erythroid regulator after hemorrhage: produced by erythroblasts following blood loss and mediates suppression of hepcidin (HAMP) expression in the liver, thereby promoting increased iron absorption and mobilization from stores. Promotes lipid uptake into adipocytes and hepatocytes via transcriptional up-regulation of genes involved in fatty acid uptake.
TMPH-01301 Erythroferrone Protein, Human, Recombinant (His & SUMO)

Human E. coli
Iron-regulatory hormone that acts as an erythroid regulator after hemorrhage: produced by erythroblasts following blood loss and mediates suppression of hepcidin (HAMP) expression in the liver, thereby promoting increased iron absorption and mobilization from stores. Promotes lipid uptake into adipocytes and hepatocytes via transcriptional up-regulation of genes involved in fatty acid uptake.

重组蛋白

RANK/TNFRSF11A Protein, Human, Recombinant (hFc)
Cat.No: TMPY-04142
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (mFc)
Cat.No: TMPY-05514
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (His)
Cat.No: TMPY-04157
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (aa 30-212, His)
Cat.No: TMPJ-00349
Species: Human
Expression System: Human Cells
Lactoferrin/LTF Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02728
Species: Mouse
Expression System: HEK293
Lactoferrin/LTF Protein, Human, Recombinant (His)
Cat.No: TMPY-02188
Species: Human
Expression System: HEK293
Erythroferrone Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02646
Species: Mouse
Expression System: Yeast
Erythroferrone Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01301
Species: Human
Expression System: E. coli
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