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133

抑制剂 & 化合物

27

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22595 B2

Linazolamide intermediate B impurity 2,CPNQ,5-[4-(4-Chlorobenzoyl)-1-piperazinyl]-8-nitroquinoline,奥司他韦杂质B(2-叠氮杂合物)

Others; Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
B2 (Linazolamide intermediate B impurity 2) 促进亨廷顿病和帕金森病细胞模型中的包涵体形成。
T35519 Aflatoxin B2-13C17

Aflatoxin B2-13C17

Aflatoxin B2-13C17(AFB2-13C17) is intended for use as an internal standard for the quantification of AFB2by GC- or LC-MS. AFB2is a mycotoxin that has been found inA. terricola.1It induces hepatic autophagy and apoptosis in broiler chickens when administered at doses of 0.2, 0.4, and 0.8 mg/kg.2AFB2(0.5 and 1 mg/animal) also induces parenchymal cell hyperplasia in rats.3 1.Moubasher, A.H., el-Kady, I.A., and Shoriet, A.Toxigenic Aspergilli isolated from different sources in EgyptAnn. Nutr. Alimen...
T36543 Prostaglandin B2

PGB2

Prostaglandin B2 (PGB2) is a non-enzymatic dehydration product resulting from the treatment of PGE2 or PGA2 with strong base. It has weak agonist activity on TP receptors and can increase pulmonary blood pressure in the rabbit at relatively high doses (5 ug/kg). [1]
T35771 Destruxin B2

Destruxin B2 is a cyclic hexadepsipeptide mycotoxin that has been found in M. anisopliae and has antiviral, insecticidal, and phytotoxic activities.1,2,3 It inhibits secretion of hepatitis B virus surface antigen (HBsAg) by Hep3B cells expressing hepatitis B virus (HBV) DNA (IC50 = 1.3 μM).1 Destruxin B2 is toxic to Sf9 insect cells in an electric cell-substrate impedance sensing (ECIS) test with a 50% inhibitory concentration (ECIS50) value of 92 μM.4 It is also phytotoxic to B. napus leaves.3 ...
T41246 Thromboxane B2

Thromboxane B2 是一种在过敏反应期间释放的前列腺素衍生物。Thromboxane B2 诱导动脉收缩和血小板聚集。
T30988 Clostomycin B2

Lipiarmycin B3,Tiacumicin C

Clostomycin B2 is a bioactive chemical.
T25515 I5B2

I5 B2,I5-B2

I5B2 is a novel phosphorus-containing angiotensin I converting enzyme inhibitor. Angiotensin I converting enzyme is produced by Actinomadura sp.
T126496 Plipastatin B2

Plipastatin B2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126496,CAS号为 103955-74-4。
T126111 Calystegine B2

Calystegine B2 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126111。
T125453 Dracoflavan B2

Dracoflavan B2 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125453。
T124249 Madurastatin B2

Madurastatin B2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124249,CAS号为 768384-52-7。
T126123 Wistariasaponin B2

Wistariasaponin B2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126123,CAS号为 126594-46-5。
T80389 Adenoregulin

Dermaseptin b2

Antibiotic Microbiology/Virology
Adenoregulin (Dermaseptin b2) 是一种具有广谱活性的抗菌肽类抗生素,能够对革兰氏阴性及阳性细菌、酵母和真菌表现出抗生效果。此外,Adenoregulin 也能增强激动剂与 A1 腺苷受体之间的结合。
T82345 Galanin-B2

NAX-5055

Galanin-B2 在癫痫模型中表现出活性,并能穿透血脑屏障。
T30941 Cinerubine A

MA144A2,MA 144A2,MA-144A2,Ryemycin B2,Rhodirubin C

Cinerubine A is an anthracycline.
T32319 Julimycin B-II

NSC 248605,Julimycin B2, calcium salt,BRN 2688327,NSC-248605,NSC248605

Julimycin B-II is a type of bioacive chemical.
T9230 KM 91104

ATPase Membrane transporter/Ion channel
KM 91104 是一种细胞通透性 V-ATPase 抑制剂,选择性作用于 V-ATPase 的 a3-b2 亚单位。
T16856 SB228357

5-HT Receptor GPCR/G Protein; Neuroscience
SB228357 是一种有效且的选择性 5-HT 受体拮抗剂,对 5-HT2A、5-HT2B 和 5-HT2C 的 pKis 分别为 6.9、8.0 和 9.0。
T10922 CYP11B2-IN-1

P450 Metabolism
CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。
T7678 SJB2-043

2-苯基萘并[2,3-D]恶唑-4,9-二酮

DUB Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
SJB2-043 是一种 USP1-UAF1 的抑制剂 ,IC50值 544 nM。
T9194 UMB298

Epigenetic Reader Domain Chromatin/Epigenetic
UMB298 是一种有效的选择性 CBP/P300 溴结构域抑制剂,抑制 BRD4,IC50 为 5193nM。
T67745 CB2R/FAAH modulator-2

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-2 (compound 26) 是一种双重靶点的调节剂,是 CB2R 的激动剂,也是 FAAH 的抑制剂,作用于 CB2R 和 CB1R 的 Ki 值分别是 10.8 和 152.9 nM,作用于FAAH 的 IC50 值为 6.2 μM。CB2R/FAAH modulator-2 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。
T10696 CB2 modulator 1

Cannabinoid Receptor GPCR/G Protein
CB2 modulator 1 是一种有效的 CB2 调节剂。 可用于免疫疾病、骨质疏松症、炎症、肾缺血的研究。
T10445 B220

HSV Microbiology/Virology
B220 是一种能抑制 HSV-1,HSV-2 和人巨细胞病毒 (CMV) 生长的抗病毒剂。
T1955 SB225002

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
SB225002 是一种有效的选择性 CXCR2 拮抗剂,抑制白介素 IL-8 与 CXCR2 的结合,IC50为 22 nM。
T22009 CB2 receptor agonist 2

ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist,CB2受体拮抗剂2

Cannabinoid Receptor GPCR/G Protein
CB2 receptor agonist 2 (ZINC72105556) 是有效和选择性的 CB2 受体激动剂。对 CB2 的 Ki 为 8.5 nM。CB2 receptor agonist 2 对 CB2 具有高亲和力和选择性。
T67747 CB2R/FAAH modulator-3

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-3 (compound 27) 是一种双重靶点的调节剂,是 CB2R 的激动剂, 也是FAAH 的抑制剂, 作用于 CB2R 和 CB1R 的 Ki 值分别是 20.1 和 67.6 nM,作用于 FAAH 的IC50值为 3.4 μM。CB2R/FAAH modulator-3 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。
T8839 ICCB280

Apoptosis; Others Apoptosis; Others
ICCB280 是一种 C/EBPα诱导剂,通过激活 C/EBPα 并影响其下游靶点,具有终末分化、增殖停滞和凋亡的抗白血病特性。
T77340L AB21 HCl

Sigma receptor GPCR/G Protein
AB21 HCl 是 σ1 受体的选择性拮抗剂,σ1 受体的 Ki 为 13 nM,σ2 受体的 Ki 为 102 nM。 AB21 HCl 具有降低机械过敏的能力。
T25209 CB29

CB-29,CB 29

Dehydrogenase Metabolism
CB29 是醛脱氢酶 3A1 (ALDH3A1) 的特异性抑制剂。
T9707 DB2313

Carboximidamide

Apoptosis Apoptosis
DB2313 (Carboximidamide) 是一种有效的转录因子 PU.1 抑制剂,IC50 为 14 nM。DB2313 破坏了 PU.1 与靶基因启动子的相互作用。DB2313 可诱导急性髓细胞性白血病 (AML) 细胞凋亡 (apoptosis),并具有抗癌作用。
T11728 JR-AB2-011

mTOR PI3K/Akt/mTOR signaling
JR-AB2-011 是一种选择性 mTORC2抑制剂,IC50值为 0.36 μM。JR-AB2-011 通过阻断 Rictor-mTOR 联合体 (Ki: 0.19 μM) 抑制 mTORC2 活性,并且具有抗多形性胶质母细胞瘤 (GBM) 的活性。
T77766 (Z)-Nexinhib20

Others Others
(Z)-Nexinhib20 是一种生化试剂,可用于生物实验。
T7138 FB23-2

Apoptosis; Others Apoptosis; Others
FB23-2 是一种 mRNA N6- 甲基腺嘌呤脱甲基酶 FTO 选择性抑制剂,IC50值为 2.6 μM。它具有抗增殖作用,可研究急性髓系白血病。
T12851 SB290157 trifluoroacetate

Complement System Immunology/Inflammation
SB290157 trifluoroacetate 是一种选择性 C3a 受体拮抗剂,IC50值为200 nM。
T4674 SB297006

SB 297006

CCR Immunology/Inflammation; Microbiology/Virology
SB297006 是一种CCR3拮抗剂,IC50为39 nM。它能够显著抑制 CCL11 处理的神经祖细胞的增殖和神经球形成。
T37075 CB2R PAM

Ec2la

Cannabinoid Receptor GPCR/G Protein
CB2R PAM 是一种口服活性大麻素 2 型受体(CB2Rs)阳性突变调节剂,它能增强 CP 55940 和 2-Arachidonylglycerol 刺激的 [35S]GTPγS 与 CB2 受体的结合,但在没有激动剂的情况下没有作用。CB2R PAM 在神经病理性疼痛小鼠模型中显示出抗损伤活性。
T8874 FB23

Others Others
FB23 是FTO 去甲基化酶选择性抑制剂(IC50:60 nM)。它能够直接与FTO 结合,选择性的抑制FTO 的 mRNA N6-甲基腺嘌呤脱甲基酶活性。
T67896 CB2R/FAAH modulator-1

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-1是一种大麻素2型受体(CB2R)激动剂,同时也是脂肪酸酰胺水解酶(FAAH)抑制剂(IC50=4 μM),可减少促炎和增加抗炎细胞因子的产生,常用于炎症研究。对 CB2R 和 CB1R 的Kis 分别为14.8 nM 和241.3 nM。
T23709 alphaSYN-IN-NAB2

alphaSYN inhibitor NAB2,alphaSYNINNAB2,alphaSYN-IN-NAB2,NAB2,alphaSYN inhibitor-NAB2

alphaSYN-IN-NAB2 是一种神经元保护剂,是一种由 NAB2基因编码的蛋白质。NAB2 高效且具有选择性地保护多种细胞免受 α-syn 毒性。NAB2 对依赖于 E3 泛素连接酶 Rsp5/Nedd4 的内体转运具有促进作用。NAB2 确定 α-syn 生物学中的一个可活性分子节点,该节点可以纠正其潜在病理学的多个方面,包括功能失调的内体和内质网到高尔基体囊泡的运输。NAB2参与细胞分化、凋亡和应激反应等细胞过程,可用来研究癌症、神经发育和神经元活动。
T82605 DB21, Galectin-1 Antagonist

Galectin Immunology/Inflammation
DB21, Galectin-1 Antagonist 是一种用于抑制galectin-1 (GAL1)与细胞表面聚糖结合的二苯并呋喃缀合肽模拟物。在黑色素瘤、肺腺癌和卵巢癌模型中,该化合物能增强血管生成和肿瘤生长的抑制效果。
TP1534 HSV-gB2 (498-505)

HSV-gB2 498-505

This is the immunodominant epitope gB-8p from herpes simplex virus (HSV) glycoprotein B (gB), amino acids 498 to 505.
T74604 CB2R probe 1

CB2R probe 1 是一种安全绿色的 CB2R (2 型大麻素受体)荧光探针,Ki 为 130 nM。CB2R probe 1 在癌细胞中显示出低细胞毒性。
T35889 PB2

PB2, a tris(2-carboxyethyl)phosphine (TCEP) analogue, enhances the survival of retinal ganglion cells (RGCs) following axotomy in vitro. Even at nanomolar and picomolar concentrations, PB2 demonstrates pronounced efficacy in promoting RGC survival. Notably, PB2 exhibits superior permeability compared to TCEP. Serving as a potent reducing agent, PB2 provides robust neuroprotection for RGCs[1].
T24432 MB21

MB-21,MB 21

MB21 is a dengue type 2 protease inhibitor that acts by inhibiting each one of the four serotypes of dengue viruses in infected cells in culture.
T10697 CB2R-IN-1

Others Others
CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
T75013 SB26019

SB26019 是一种有效的抗神经炎症剂。SB26019 通过诱导单体 α-微管蛋白 (α-tubulin) 形成来调节 NF-κB 激活。SB26019 诱导的 α-微管蛋白单体抑制 p65 易位。
T82771 CB2-H

CB2-H为一种高特异性双通道荧光探针,专门设计用于HOCl和ONOO-的同时检测。该探针在两个分离的通道中对HOCl和ONOO-无交叉干扰的检测能力使其适用于对活细胞和斑马鱼样本内HOCl及ONOO-的内源性水平进行双通道荧光成像分析,即使在不同生物刺激下也能保持准确性。
T24397 ZTB23(R)

ZTB 23(R),ZTB-23(R)

ZTB23(R) is the first potent and selective inhibitor of Mycobacterium tuberculosis Zmp1.
T19270 DTPA-DAB2

Others Others
DAB2-DTPA is a conjugate of DTPA and two DABs used in the photooxidation experiment.

化合物

B2
Cat.No: T22595
Synonym: Linazolamide intermediate B impurity 2,CPNQ,5-[4-(4-Chlorobenzoyl)-1-piperazinyl]-8-nitroquinoline,奥司他韦杂质B(2-叠氮杂合物)
Target: Others, Sirtuin
Aflatoxin B2-13C17
Cat.No: T35519
Synonym: Aflatoxin B2-13C17
Target:
Prostaglandin B2
Cat.No: T36543
Synonym: PGB2
Target:
Destruxin B2
Cat.No: T35771
Synonym:
Target:
Thromboxane B2
Cat.No: T41246
Synonym:
Target:
Clostomycin B2
Cat.No: T30988
Synonym: Lipiarmycin B3,Tiacumicin C
Target:
I5B2
Cat.No: T25515
Synonym: I5 B2,I5-B2
Target:
Plipastatin B2
Cat.No: T126496
Synonym:
Target:
Calystegine B2
Cat.No: T126111
Synonym:
Target:
Dracoflavan B2
Cat.No: T125453
Synonym:
Target:
Madurastatin B2
Cat.No: T124249
Synonym:
Target:
Wistariasaponin B2
Cat.No: T126123
Synonym:
Target:
Adenoregulin
Cat.No: T80389
Synonym: Dermaseptin b2
Target: Antibiotic
Galanin-B2
Cat.No: T82345
Synonym: NAX-5055
Target:
Cinerubine A
Cat.No: T30941
Synonym: MA144A2,MA 144A2,MA-144A2,Ryemycin B2,Rhodirubin C
Target:
Julimycin B-II
Cat.No: T32319
Synonym: NSC 248605,Julimycin B2, calcium salt,BRN 2688327,NSC-248605,NSC248605
Target:
KM 91104
Cat.No: T9230
Synonym:
Target: ATPase
SB228357
Cat.No: T16856
Synonym:
Target: 5-HT Receptor
CYP11B2-IN-1
Cat.No: T10922
Synonym:
Target: P450
SJB2-043
Cat.No: T7678
Synonym: 2-苯基萘并[2,3-D]恶唑-4,9-二酮
Target: DUB
UMB298
Cat.No: T9194
Synonym:
Target: Epigenetic Reader Domain
CB2R/FAAH modulator-2
Cat.No: T67745
Synonym:
Target: Cannabinoid Receptor, FAAH
CB2 modulator 1
Cat.No: T10696
Synonym:
Target: Cannabinoid Receptor
B220
Cat.No: T10445
Synonym:
Target: HSV
SB225002
Cat.No: T1955
Synonym:
Target: CXCR
CB2 receptor agonist 2
Cat.No: T22009
Synonym: ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist,CB2受体拮抗剂2
Target: Cannabinoid Receptor
CB2R/FAAH modulator-3
Cat.No: T67747
Synonym:
Target: Cannabinoid Receptor, FAAH
ICCB280
Cat.No: T8839
Synonym:
Target: Apoptosis, Others
AB21 HCl
Cat.No: T77340L
Synonym:
Target: Sigma receptor
CB29
Cat.No: T25209
Synonym: CB-29,CB 29
Target: Dehydrogenase
DB2313
Cat.No: T9707
Synonym: Carboximidamide
Target: Apoptosis
JR-AB2-011
Cat.No: T11728
Synonym:
Target: mTOR
(Z)-Nexinhib20
Cat.No: T77766
Synonym:
Target: Others
FB23-2
Cat.No: T7138
Synonym:
Target: Apoptosis, Others
SB290157 trifluoroacetate
Cat.No: T12851
Synonym:
Target: Complement System
SB297006
Cat.No: T4674
Synonym: SB 297006
Target: CCR
CB2R PAM
Cat.No: T37075
Synonym: Ec2la
Target: Cannabinoid Receptor
FB23
Cat.No: T8874
Synonym:
Target: Others
CB2R/FAAH modulator-1
Cat.No: T67896
Synonym:
Target: Cannabinoid Receptor, FAAH
alphaSYN-IN-NAB2
Cat.No: T23709
Synonym: alphaSYN inhibitor NAB2,alphaSYNINNAB2,alphaSYN-IN-NAB2,NAB2,alphaSYN inhibitor-NAB2
Target:
DB21, Galectin-1 Antagonist
Cat.No: T82605
Synonym:
Target: Galectin
HSV-gB2 (498-505)
Cat.No: TP1534
Synonym: HSV-gB2 498-505
Target:
CB2R probe 1
Cat.No: T74604
Synonym:
Target:
PB2
Cat.No: T35889
Synonym:
Target:
MB21
Cat.No: T24432
Synonym: MB-21,MB 21
Target:
CB2R-IN-1
Cat.No: T10697
Synonym:
Target: Others
SB26019
Cat.No: T75013
Synonym:
Target:
CB2-H
Cat.No: T82771
Synonym:
Target:
ZTB23(R)
Cat.No: T24397
Synonym: ZTB 23(R),ZTB-23(R)
Target:
DTPA-DAB2
Cat.No: T19270
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T6S1367 Procyanidin B2

原花青素 B2,Proanthocyanidin B2

Reactive Oxygen Species; NOD Immunology/Inflammation; Metabolism; NF-κB
Procyanidin B2 (Proanthocyanidin B2) 是天然黄酮类物质,具有抗肿瘤,抗氧化等活性。
TN1470 Cassiaside B2

决明子苷B2

Phosphatase; MAO; 5-HT Receptor GPCR/G Protein; Metabolism; Neuroscience
Cassiaside B2 是蛋白酪氨酸磷酸酶1B (PTP1B) 和人单胺氧化酶A (hMAO-A) 的抑制剂。Cassiaside B2是 5-HT2C 受体的激动剂, 具有抗过敏活性。Cassiaside B2 是萘吡喃酮参比提取物(NRE)的有效成分之一。
T3810 Saikosaponin B2

柴胡皂苷 B2,柴胡皂甙 B2

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。
TJS0502 Ilexsaponin B2

Ilexsaponin B2 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TJS0502,CAS号为 108906-69-0。
T0937 Riboflavin

Vitamin B2,维生素B2,E101

Endogenous Metabolite Metabolism
Riboflavin (E101),一种人内源性代谢物, 是极易吸收的微量营养素。
T15357 Fumonisin B2

伏马菌素B2

Others Others
Fumonisin B2 is a mycotoxin produced by Fusarium moniliforme in various grains. It also is a potent inhibitor of sphingosine N-acyltransferase (ceramide synthase). Which disrupts de novo sphingolipid biosynthesis.
T25971 Polymyxin B2

Polymyxin-B2,PolymyxinB2

Polymyxin B2 is an antibiotic primarily utilized for resistant Gram-negative infections. It is derived from the bacterium Bacillus polymyxa.
T19359 Hydrolyzed Fumonisin B2

Others Others
Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.
TN5492 Procyanidin B2 3''-O-gallate

Epicatechin-(4β→8)-epicatechin 3''-O-gallate,原花青素B2-3"-O-没食子酸

Procyanidin B2 3''-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5492,CAS号为 73086-04-1。
TN5497 Procyanidin B2 3,3'-di-O-gallate

Procyanidin B-2 3,3'-di-O-gallate,原花青素B2-3,3'-二-O-没食子酸酯

Procyanidin B2 3,3'-di-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5497,CAS号为 79907-44-1。
T1331 Riboflavin phosphate sodium

Riboflavin 5'-phosphate sodium,核黄素磷酸钠(维生素B2),Vitamin B2 Phosphate Sodium Salt,Flavin mononucleotide,FMN,核黄素磷酸钠,FMN-Na,riboflavin-5'-phosphate

Endogenous Metabolite Metabolism
Riboflavin phosphate sodium (FMN) 是 riboflavin 的磷酸钠盐形式,riboflavin 是一种水溶性和必需的微量营养素,是自然产生的维生素B复合物的主要生长促进因子。Riboflavin phosphate sodium 转化为2种辅酶,黄素单核苷酸(FMN)和黄素腺嘌呤二核苷酸(FAD),这两种辅酶通过帮助脂肪、碳水化合物和蛋白质的代谢来产生能量,并且是红细胞形成和呼吸、抗体产生以及调节人体生长和繁殖所必需的。
T2872 Ginsenoside Re

人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re

Beta Amyloid; NF-κB; Endogenous Metabolite; JNK MAPK; Metabolism; Neuroscience; NF-κB
Ginsenoside Re (Ginsenoside B2) 是一种人参提取物,可降低 β-淀粉样蛋白 (Aβ),还通过抑制 JNK 和 NF-κB 发挥抗炎作用。
T82721 Cinnamtannin B2

Cinnamtannin B2(化合物12)为肉桂单宁类化合物,可自越橘(Vaccinium vitis-idaea L.)中提取。
T83133 Alternaphenol B2

Isocitrate Dehydrogenase (IDH) Metabolism
IDH1 Inhibitor 是一种化学化合物,其通过选择性抑制异柠檬酸脱氢酶1 (IDH1) 酶的活性来起作用。这种抑制剂对R132突变的IDH1酶特别有效,因此在某些类型的癌症治疗中具有潜在的应用价值。IDH1 Inhibitor能够阻断异常的代谢途径和纠正肿瘤细胞增殖的代谢异常。在药物研发和临床试验中,研究人员评估其对特定肿瘤生长的抑制效果及其安全性和耐受性。
T2932 Ginsenoside Rh1

Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1

IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。
TN1804 Isosilybin A

异水飞蓟素 A,异水飞蓟宾A,水飞蓟素 B2

Apoptosis; Tyrosinase; PPAR; ABC Apoptosis; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome
Isosilybin A 是从水飞蓟中分离出来的一种黄酮木脂素,可抑制癌细胞增殖并诱导 G1 期停滞和凋亡,通过靶向 Akt-NF-κB-雄激素受体轴激活前列腺癌细胞的凋亡机制,具有抗前列腺癌活性。
T83903 Polymyxin B2 sulfate

Polymyxin B2是一种抗生素,并且是从B. polymyxa分离出的阳离子脂肽抗生素polymyxin B的主要成分。该化合物对P. aeruginosa、A. baumannii、K. pneumoniae和E. cloacae菌株具有活性(MICs分别为1-2、0.5-1、0.25-0.5和0.25-1 µg/ml)。在体内实验中,以4 mg/kg剂量的Polymyxin B2能显著降低P. aeruginosa血液感染小鼠模型中的血液集落形成单位(CFUs)数量。
T3919 Ginsenoside Rb2

Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2

GPR; Others; Influenza Virus; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Others
Ginsenoside Rb2 (Ginsenoside C) 是人参提取物中的一种主要生物活性成分,具有抗病毒活性,可上调 GPR120 基因表达。
T2964 2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside

芪多酚,2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside,2,3,5,4'-Tetrahydroxystilbene-2-O-b-D-glucopyranoside,Astragalus polyphenols

Others Others
2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside (Astragalus polyphenols) 是分离自蓼属植物物种的根中,对5-HETE、HHT、thromboxane B2的形成具有抑制作用。
T7053 p-Hydroxycinnamic acid

p-Coumaric acid,p-Cumaric acid,p-Hydroxy-cinnamic acid,对羟基肉桂酸,NSC 59260

Thrombin; Endogenous Metabolite; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Proteases/Proteasome
p-Hydroxycinnamic acid (NSC-59260) 是常见的食用酚,可抑制血小板活性,对血栓素 B2 和前列腺素 E2 的 IC50值分别为 371 和 126 μM。
TN1957 Mulberrofuran Q

MulberrofuranQ

Mulberrofuran Q是一种有活性的化合物,可抑制12-羟基-5,8,10-十七碳三烯酸(HHT)和血栓烷B2(环加氧酶产物)的形成 ,可保护神经细胞免受缺氧-缺糖(OGD)诱导的氧化应激的影响。
T36831 9-Oxononanoic Acid

9-ONA

Phospholipase; CPT Metabolism
9-Oxononanoic Acid是一种氧化脂肪酸,由亚油酸自氧化形成,它能提高磷脂酶 A2(PLA2)的活性,并增加离体人体血浆中血栓素 B2 的生成。9-Oxononanoic Acid 能减少肝脏新脂肪酸的合成,并提高大鼠肝脏肉碱棕榈酰转移酶(β-氧化的标志物)的活性。
T1100 Polymyxin B Sulfate

Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B Sulfate (Poly-RX) 是一个阳离子型表面活性剂抗生素剂,能够提高细胞膜的渗透性。
T6480 D-Pantothenic acid

vitamin B5,pantothenate,D-泛酸

Others Others
D-Pantothenic acid (vitamin B5) 是必需的微量营养素,是辅酶 A 的前体,在很多生物过程中发挥关键作用,如调节碳水化合物,脂质,蛋白和核酸代谢。
TN5939 Glutinone

赤杨酮,5-Glutinen-3-one

Glutinone (IC50=24 microM) shows a significant effect on thromboxane B2 (TXB2)-release induced by calcium ionophore in human platelets.
TN4586 Mulberrofuran A

COX Immunology/Inflammation; Neuroscience
Mulberrofuran A can inhibit the formations of 12-hydroxy-, 8, 10-heptadecatrienoic acid (HHT) and thromboxane B2, but it can increase the formation of 12-hydroxy-5, 8, 10, 14-eicosatetraenoic acid (12-HETE).
T13534 Aflatoxin M1

黄曲霉毒素 M1

Others Others
Aflatoxin M1, a significant metabolite of Aflatoxin B1, is a mycotoxin synthesized by Aspergillus flavus and Aspergillus parasiticus fungi. Toxicity levels of Aflatoxins follow the order: Aflatoxin B1 > Aflatoxin M1 > Aflatoxin G1 > Aflatoxin B2 > Aflatoxin M2 > Aflatoxin G2.

天然产物

Procyanidin B2
Cat.No: T6S1367
Synonym: 原花青素 B2,Proanthocyanidin B2
Target: Reactive Oxygen Species, NOD
Cassiaside B2
Cat.No: TN1470
Synonym: 决明子苷B2
Target: Phosphatase, MAO, 5-HT Receptor
Saikosaponin B2
Cat.No: T3810
Synonym: 柴胡皂苷 B2,柴胡皂甙 B2
Target: Others, HCV Protease
Ilexsaponin B2
Cat.No: TJS0502
Synonym:
Target:
Riboflavin
Cat.No: T0937
Synonym: Vitamin B2,维生素B2,E101
Target: Endogenous Metabolite
Fumonisin B2
Cat.No: T15357
Synonym: 伏马菌素B2
Target: Others
Polymyxin B2
Cat.No: T25971
Synonym: Polymyxin-B2,PolymyxinB2
Target:
Hydrolyzed Fumonisin B2
Cat.No: T19359
Synonym:
Target: Others
Procyanidin B2 3''-O-gallate
Cat.No: TN5492
Synonym: Epicatechin-(4β→8)-epicatechin 3''-O-gallate,原花青素B2-3"-O-没食子酸
Target:
Procyanidin B2 3,3'-di-O-gallate
Cat.No: TN5497
Synonym: Procyanidin B-2 3,3'-di-O-gallate,原花青素B2-3,3'-二-O-没食子酸酯
Target:
Riboflavin phosphate sodium
Cat.No: T1331
Synonym: Riboflavin 5'-phosphate sodium,核黄素磷酸钠(维生素B2),Vitamin B2 Phosphate Sodium Salt,Flavin mononucleotide,FMN,核黄素磷酸钠,FMN-Na,riboflavin-5'-phosphate
Target: Endogenous Metabolite
Ginsenoside Re
Cat.No: T2872
Synonym: 人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re
Target: Beta Amyloid, NF-κB, Endogenous Metabolite, JNK
Cinnamtannin B2
Cat.No: T82721
Synonym:
Target:
Alternaphenol B2
Cat.No: T83133
Synonym:
Target: Isocitrate Dehydrogenase (IDH)
Ginsenoside Rh1
Cat.No: T2932
Synonym: Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1
Target: IL Receptor, TNF, Endogenous Metabolite, PPAR, Interleukin
Isosilybin A
Cat.No: TN1804
Synonym: 异水飞蓟素 A,异水飞蓟宾A,水飞蓟素 B2
Target: Apoptosis, Tyrosinase, PPAR, ABC
Polymyxin B2 sulfate
Cat.No: T83903
Synonym:
Target:
Ginsenoside Rb2
Cat.No: T3919
Synonym: Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2
Target: GPR, Others, Influenza Virus, Endogenous Metabolite
2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside
Cat.No: T2964
Synonym: 芪多酚,2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside,2,3,5,4'-Tetrahydroxystilbene-2-O-b-D-glucopyranoside,Astragalus polyphenols
Target: Others
p-Hydroxycinnamic acid
Cat.No: T7053
Synonym: p-Coumaric acid,p-Cumaric acid,p-Hydroxy-cinnamic acid,对羟基肉桂酸,NSC 59260
Target: Thrombin, Endogenous Metabolite, Prostaglandin Receptor
Mulberrofuran Q
Cat.No: TN1957
Synonym: MulberrofuranQ
Target:
9-Oxononanoic Acid
Cat.No: T36831
Synonym: 9-ONA
Target: Phospholipase, CPT
Polymyxin B Sulfate
Cat.No: T1100
Synonym: Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX
Target: Antibacterial, Antibiotic
D-Pantothenic acid
Cat.No: T6480
Synonym: vitamin B5,pantothenate,D-泛酸
Target: Others
Glutinone
Cat.No: TN5939
Synonym: 赤杨酮,5-Glutinen-3-one
Target:
Mulberrofuran A
Cat.No: TN4586
Synonym:
Target: COX
Aflatoxin M1
Cat.No: T13534
Synonym: 黄曲霉毒素 M1
Target: Others
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