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180

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T20913 Light Green SF Yellowish

Acid Green 5,C.I. Acid Green 5,C.I. 42095

Light Green SF Yellowish (Acid Green 5) 是一种碱性染色剂,可用于动物组织染色,可用于植物组织学中作细胞质和纤维染色。
T22865 immunoglobulin light chain variable region fragment [Homo sapiens]

Others Others
Immunoglobulin light chain variable region fragment [Homo sapiens] is a fragment (Phe-Thr-Leu-Lys-Ile-Ser-Arg) on the variable region of the human immunoglobulin light chain.
TP2259 immunoglobulin light chain variable region fragment [Homo sapiens]/[Mus musculus]

Others Others
Immunoglobulin light chain variable region fragment [Homo sapiens]/[Mus musculus] is a fragment on the variable region of the human and mouse immunoglobulin light chain. Immunoglobulins (Ig) are the antigen recognition molecules of B cells. An Ig molecule
T22856 IgG light chain variable region [Homo sapiens]/IgM/kappa antibody [Mus musculus]

Others Others
IgG has four forms, provides the majority of antibody-based immunity against invading pathogens. The only antibody capable of crossing the placenta to give passive immunity to the fetus. Eliminates pathogens in the early stages of B cell-mediated (humoral
T6617 Optovin

TRP/TRPV Channel Membrane transporter/Ion channel
Optovin 是可逆的光活化 TRPA1配体,可实现光介导的神经元兴奋。它通过与氧化还原敏感的半胱氨酸残基产生结构依赖性光化学反应激活 TRPA1。
T81732 Myosin light chain kinase fragment 11-19 amide

MLCK(11-19) amide

Myosinlight chain kinase fragment 11-19 amide (MLCK(11-19) amide) 为MLCK专一性多肽抑制剂,具抑制低渗透压刺激下Ca2+入细胞的能力,并可应用于人类宫颈癌研究。
T0343 Nimodipine

尼莫地平,BAY-e 9736

Glucocorticoid Receptor; AhR; Calcium Channel; Autophagy Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Nimodipine (BAY-e 9736) 是一种具有口服活性,耐受性良好的光敏二氢吡啶钙拮抗剂。它可研究脑血管疾病。
T3213 Hematoporphyrin dihydrochloride

血卟啉二盐酸盐,Hematoporphyrin IX dihydrochloride

Apoptosis; Others; Endogenous Metabolite Apoptosis; Metabolism; Others
Hematoporphyrin dihydrochloride (Hematoporphyrin IX dihydrochloride) 是一种光敏剂,是血红素结合蛋白亲和色谱底物。它暴露在红光下时,可诱导 U87 胶质瘤细胞凋亡,并降低体内肿瘤的生长。
T21343 PTZ-343

PTZ-343 sodium,PTZ 343,吩噻嗪-10-基-丙基磺酸钠盐

Others Others
PTZ-343 是一种鲁米诺的强效发光增强剂 (enhancer)。它极大的增强了过氧化物酶催化的鲁米诺化学发光氧化反应 (>80%) 的光输出。
T20792 W-7 hydrochloride

N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W 7 HCl,W7 HCl,W-7 HCl

CaMK; Apoptosis; Myosin; PDE Apoptosis; Cytoskeletal Signaling; Metabolism; Neuroscience
W-7 hydrochloride (W-7 HCl) 是一种选择性的钙调蛋白拮抗剂。它抑制Ca2+-钙调蛋白依赖性磷酸二酯酶和肌球蛋白轻链激酶,IC50值分别为 28 μM 和 51 μM。它可诱导细胞凋亡,具有抗癌活性。
T0642 2-Methoxyphenothiazine

Factor Xa Metabolism
2-Methoxyphenothiazine 为淡黄色或淡灰色固体。
T77752 HMBR

4-Thiazolidinone, 5-[(4-hydroxy-3-methylphenyl)methylene]-2-thioxo-, (5Z)-

Others Others
HMBR本身不具有荧光,但当与 Y-FAST 结合时,它们在蓝光激发时会发出黄光。
T0659 Bispyrazolone

NSC 37393,依达拉奉杂质IV

Others Others
Bispyrazolone (NSC-37393) 为淡黄色或白色结晶性粉末。
T9550 Drometrizole Trisiloxane

甲酚曲唑三硅氧烷,Mexoryl XL,Silatrizole

Others Others
Drometrizole Trisiloxane (Mexoryl XL) 是一种光稳定的 UVA 和 UVB 滤光剂。
T24533 Nicotinoyl azide

N-Az,NAz,叠氮烟酸甲酰,N Az

Others Others
Nicotinoyl azide (N-Az) 是一种光活化化学探针。它已被用于测量嘌呤核碱基的溶剂可及性。
T3050 ML-7 hydrochloride

ML-7 HCl,ML-7盐酸盐

Serine/threonin kinase; Myosin; YAP; PKA; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
ML-7 hydrochloride (ML-7 HCl) 是一种可渗透细胞的、可逆的、有效的、ATP 竞争性的肌球蛋白轻链激酶(MLCK) 特异性抑制剂,IC50为300 nM。它还抑制平滑肌肌球蛋白轻链激酶、PKA 和 PKC。
T26078 Rhodblock 6

Rhodblock6,Rhodblock-6

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Rhodblock 6 是一种 Rho 激酶 (ROCK) 抑制剂,可抑制磷酸化 MRLC(肌球蛋白调节轻链)定位,通过特异性抑制 Rho 激酶的活性发挥作用。
T40684 N-Nitrosomorpholine

Others Others
N-Nitrosomorpholine 是一种亚硝胺,具有光敏感性。它对动物有强致癌作用。
T1699 resorufin galactopyranoside

Others Others
resorufin galactopyranoside 是β-半乳糖苷酶的荧光底物,在被β-半乳糖苷酶酶切后,荧光部分间苯二酚被释放,其荧光可用于定量β-半乳糖糖苷酶的活性。它的激发光为570,发射光为580nm。
T21282 Topanol CA

Others Others
Topanol CA 是一种抗氧化剂,可用于树脂和浅色橡胶制品中作稳定剂。
T27931 LY2033298

LY 2033298,LY-2033298

AChR Neuroscience
LY2033298 是毒蕈碱 M4 受体的正变构调节剂,可增强奥昔莫林对仓鼠昼夜节律活动中光诱导的相移的抑制作用,可用于与神经系统相关的疾病。
T0691 Sulisobenzone

舒利苯酮,Benzophenone-4,Sungard

Others Others
Sulisobenzone (Sungard) 是防晒霜的成分,能够保护皮肤,使其免于受UVB 和短波紫外线UVA 的伤害。
T35501 5,6-trans-Vitamin D3

5,6-trans-Colecalciferol,5,6-trans-Cholecalciferol,Cholecalciferol EP Impurity A

Vitamin Metabolism
5,6-trans-Vitamin D3(5,6-trans-Cholecalciferol)是维生素 D3 的异构体,经光照后在皮肤表面由 Vitamin D3 转化而来。
T14994 Coelenterazine h

腔肠素-H,2-Deoxycoelenterazine,CLZN-h

Others Others
Coelenterazine h (CLZN-h) 是一种 Coelenterazine 的衍生物。它对 Ca2+比它的天然复合物更敏感,是一种能够测量 Ca2+浓度的微小变化的有效工具。
T7465 4-Methylbenzylidene camphor

Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC

AChE Neuroscience
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。
T19743 D-Luciferin Sodium

D-萤光素钠盐,D-虫荧光素钠

Others Others
D-Luciferin sodium 是一种萤光素酶底物,能够催化生物发光昆虫产生典型的黄绿光。
T83633 1-N-Methyl-4-mercaptohistidine disulfide

Others Others
1-N-Methyl-4-mercaptohistidine disulfide 是一种潜在的杜氏菌叶绿体偶联因子1氧化还原调节剂,是氧化形式的卵硫醇A,抑制光触发的CF1 ATP酶活性。
T8940 KUN56321

3H-Naphth[1,2-d]imidazole, 2-(4-bromophenyl)-3-phenyl-

Others Others
KUN56321 (3H-Naphth[1,2-d]imidazole, 2-(4-bromophenyl)-3-phenyl-) 是一种发光剂。 KUN56321的应用包括:真空蒸镀将 KUN56321薄膜涂布在 ITO 玻璃的空穴传输层或电子传输层上。将空穴传输层或电子传输层蒸镀在薄膜上,preppg。蒸发金属电极。 KUN56321 展示了提高发光效率和降低 org 驱动电压的能力。发光器件和显示器件。
TP1890L1 MLCK inhibitor peptide 18 acetate

MLCK inhibitor peptide 18 acetate(224579-74-2 free base)

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
MLCK inhibitor peptide 18 acetate(224579-74-2 free base) 是肌球蛋白轻链激酶的选择性竞争性抑制剂 (IC50 = 50 nM)。显示出比 CaM 激酶 II 高 4000 倍的选择性,并且不抑制 PKA。细胞可渗透。
T67886 Girard's Reagent T

Trimethylacetohydrazideammonium Chloride

Others Others
Girard's Reagent T (Trimethylacetohydrazideammonium Chloride) 是生化试剂。Girard's Reagent T 在温和的酸性或碱性条件下,与含有α-二羰基官能团的醛类和酮类反应,生成强吸收紫外线的加成化合物
T16562 Ponceau 4R

Acid Red 18,New Coccine

Others Others
Ponceau 4R (Acid Red 18) 是一种合成草莓红偶氮染料,是一种可用为食品着色剂染料,可用于各种食品。它对光、热和酸都很稳定,但在抗坏血酸存在下会褪色。它通常由芳香烃合成。
T16104 ML-9

Myosin; Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
ML-9 是 Akt 激酶的一种选择性强效抑制剂,可抑制肌球蛋白轻链激酶 (MLCK) 和基质相互作用分子1(STIM1) 活性。它通过刺激自噬小体的形成并抑制其降解来诱导自噬。它抑制 MLCK,PKA 和 PKC 活性,Ki 值分别为 4、32 和 54 μM。
T1433 Ritodrine hydrochloride

DU21220,盐酸利托君,Ritodrine HCl,NSC 291565

Adrenergic Receptor GPCR/G Protein; Neuroscience
Ritodrine hydrochloride (NSC 291565) 是一种 β-2肾上腺素受体激动剂。
T0075 Nicorandil

SG-75,尼可地尔

Potassium Channel Membrane transporter/Ion channel
Nicorandil (SG-75) 是一种有效的钾通道激活剂,靶向血管核苷二磷酸依赖性 K+通道和心脏 ATP 敏感 K+通道 (KATP)。Nicorandil 是一种烟酰胺酯,具有血管舒张和心脏保护作用,并具有治疗心绞痛和缺血性心脏病的潜力。
T9403 1,3,5-tris(pyridin-4-ylethynyl)benzene

Others Others
1,3,5-tris(pyridin-4-ylethynyl)benzene 是一种杂环化合物,具有广泛的性质,如荧光和电化学活性,具有相对较低的毒性。它已被用作合成各种材料的构建块,如聚合物、纳米材料和有机发光二极管(OLED)。它也是开发新型药物递送系统的一种有前途的材料。
T14069 A-3 hydrochloride

CaMK; Casein Kinase; PKA; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Neuroscience; Stem Cells; Tyrosine Kinase/Adaptors
A-3 hydrochloride 是一种细胞可渗透的、可逆的、ATP 竞争性非选择性拮抗剂。它抑制 PKA 、酪蛋白激酶 II 和肌球蛋白轻链激酶,Ki 值分别为4.3 µM、5.1 µM 和7.4 µM。它还抑制 PKC 和酪蛋白激酶 I 的活性,Ki 分别为 47 µM 和 80 µM。
T31144 CycLuc2

CycLuc 2,CycLuc-2

CycLuc2 is a cyclic alkylaminoluciferin substrate for firefly luciferase. CycLuc2 emits 4.7-fold more light than aminoluciferin, and 2.6-fold more light than D-luciferin.
T20096 Octabenzone

Seikalizer E,Rhodialux,Benzophenone 12,P Sanduvor 3035

Octabenzone protects damage against UV light. It also prevents skin cancer.
T31145 CycLuc3

Cyc Luc 3,Cyc-Luc-3

CycLuc3 is a type of mutant firefly luciferase variant with enhanced light emission.
T16145 MS-444

BE-34776

Others Others
MS-444 suppresses the activity of purified smooth muscle myosin light chain kinase (MLCK) (IC50: 10 μM).
T33814 OptoDArG

Opto-DArG,Opto DArG

OptoDArG is a diacylglycerol (DAG) photoswitch, which enables efficient control of TRPC3 by light.
T33451 ML 7

ML7,ML-7

ML 7 is an inhibitor of myosin light chain kinase that protects cardiac function from ischemia/reperfusion (I/R) injury.
T69377 BoNT-IN-33

BoNT-IN-33 is a potent inhibitor of Botulinum neurotoxin/A light chain (BoNT/A LC).
T38229 JF-NP-26

Caged Raseglurant . Releases raseglurant upon exposure to 405 nm (violet) light. Inhibits the effects of Quisqualate in cultured neurons when exposed to 405 nm light. Exhibits analgesic activity in pain models in vivo on photoactivation. Quantum yield = 0.18. Font et al (2017) Optical control of pain in vivo with a photoactive mGlu5 receptor negative allosteric modulator. eLIFE 6 e23545 PMID:28395733
T28287 PA1 2HCl

PA1,PA1 dihydrochloride

PA1 2HCl is a blocker of photoswitchable epithelial sodium channel (ENaC). PA1 2HCl enables the optical control of ENaC channels, in particular the δβγ isoform, by switching between blue and green light, or by turning on and off blue light.
T34777 Talaporfin free acid

Monoaspartyl chlorin,NPe6,Talaporfin,Aspartyl chlorin

Talaporfin, an effective tumor localizer, can produce the selective degradation of tumor tissue following light exposure.
T70626 MS 347a

MS 347a is a myosin light chain kinase (MLCK) inhibitor; an epoxide analog of sydowinin B (MS-347b).
T25818 ML344

ML-344,ML 344

ML344 is a CqsS/LuxQ agonist probe that acts as an inducer of light production without autoinducers.
T31552 DMNP-EDTA

DMNPEDTA,DM-Nitrophen,DM Nitrophen,DMNP EDTA

DMNP-EDTA is a caged Ca2+ chelator which photouncages Cu2+ ions for light-controlled gene expression in yeast.
T25890 NSC-84096

CID 256758,CID-256758,CID256758

NSC-84096 is an endopeptidase activity inhibitor of botulinum neurotoxin type A light chain (rBoNT/A-LC).

化合物

Light Green SF Yellowish
Cat.No: T20913
Synonym: Acid Green 5,C.I. Acid Green 5,C.I. 42095
Target:
immunoglobulin light chain variable region fragment [Homo sapiens]
Cat.No: T22865
Synonym:
Target: Others
immunoglobulin light chain variable region fragment [Homo sapiens]/[Mus musculus]
Cat.No: TP2259
Synonym:
Target: Others
IgG light chain variable region [Homo sapiens]/IgM/kappa antibody [Mus musculus]
Cat.No: T22856
Synonym:
Target: Others
Optovin
Cat.No: T6617
Synonym:
Target: TRP/TRPV Channel
Myosin light chain kinase fragment 11-19 amide
Cat.No: T81732
Synonym: MLCK(11-19) amide
Target:
Nimodipine
Cat.No: T0343
Synonym: 尼莫地平,BAY-e 9736
Target: Glucocorticoid Receptor, AhR, Calcium Channel, Autophagy
Hematoporphyrin dihydrochloride
Cat.No: T3213
Synonym: 血卟啉二盐酸盐,Hematoporphyrin IX dihydrochloride
Target: Apoptosis, Others, Endogenous Metabolite
PTZ-343
Cat.No: T21343
Synonym: PTZ-343 sodium,PTZ 343,吩噻嗪-10-基-丙基磺酸钠盐
Target: Others
W-7 hydrochloride
Cat.No: T20792
Synonym: N-(6-氨基己基)-5-氯-1-萘磺胺盐酸盐,W 7 HCl,W7 HCl,W-7 HCl
Target: CaMK, Apoptosis, Myosin, PDE
2-Methoxyphenothiazine
Cat.No: T0642
Synonym:
Target: Factor Xa
HMBR
Cat.No: T77752
Synonym: 4-Thiazolidinone, 5-[(4-hydroxy-3-methylphenyl)methylene]-2-thioxo-, (5Z)-
Target: Others
Bispyrazolone
Cat.No: T0659
Synonym: NSC 37393,依达拉奉杂质IV
Target: Others
Drometrizole Trisiloxane
Cat.No: T9550
Synonym: 甲酚曲唑三硅氧烷,Mexoryl XL,Silatrizole
Target: Others
Nicotinoyl azide
Cat.No: T24533
Synonym: N-Az,NAz,叠氮烟酸甲酰,N Az
Target: Others
ML-7 hydrochloride
Cat.No: T3050
Synonym: ML-7 HCl,ML-7盐酸盐
Target: Serine/threonin kinase, Myosin, YAP, PKA, PKC
Rhodblock 6
Cat.No: T26078
Synonym: Rhodblock6,Rhodblock-6
Target: ROCK
N-Nitrosomorpholine
Cat.No: T40684
Synonym:
Target: Others
resorufin galactopyranoside
Cat.No: T1699
Synonym:
Target: Others
Topanol CA
Cat.No: T21282
Synonym:
Target: Others
LY2033298
Cat.No: T27931
Synonym: LY 2033298,LY-2033298
Target: AChR
Sulisobenzone
Cat.No: T0691
Synonym: 舒利苯酮,Benzophenone-4,Sungard
Target: Others
5,6-trans-Vitamin D3
Cat.No: T35501
Synonym: 5,6-trans-Colecalciferol,5,6-trans-Cholecalciferol,Cholecalciferol EP Impurity A
Target: Vitamin
Coelenterazine h
Cat.No: T14994
Synonym: 腔肠素-H,2-Deoxycoelenterazine,CLZN-h
Target: Others
4-Methylbenzylidene camphor
Cat.No: T7465
Synonym: Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC
Target: AChE
D-Luciferin Sodium
Cat.No: T19743
Synonym: D-萤光素钠盐,D-虫荧光素钠
Target: Others
1-N-Methyl-4-mercaptohistidine disulfide
Cat.No: T83633
Synonym:
Target: Others
KUN56321
Cat.No: T8940
Synonym: 3H-Naphth[1,2-d]imidazole, 2-(4-bromophenyl)-3-phenyl-
Target: Others
MLCK inhibitor peptide 18 acetate
Cat.No: TP1890L1
Synonym: MLCK inhibitor peptide 18 acetate(224579-74-2 free base)
Target: Serine/threonin kinase
Girard's Reagent T
Cat.No: T67886
Synonym: Trimethylacetohydrazideammonium Chloride
Target: Others
Ponceau 4R
Cat.No: T16562
Synonym: Acid Red 18,New Coccine
Target: Others
ML-9
Cat.No: T16104
Synonym:
Target: Myosin, Akt
Ritodrine hydrochloride
Cat.No: T1433
Synonym: DU21220,盐酸利托君,Ritodrine HCl,NSC 291565
Target: Adrenergic Receptor
Nicorandil
Cat.No: T0075
Synonym: SG-75,尼可地尔
Target: Potassium Channel
1,3,5-tris(pyridin-4-ylethynyl)benzene
Cat.No: T9403
Synonym:
Target: Others
A-3 hydrochloride
Cat.No: T14069
Synonym:
Target: CaMK, Casein Kinase, PKA, PKC
CycLuc2
Cat.No: T31144
Synonym: CycLuc 2,CycLuc-2
Target:
Octabenzone
Cat.No: T20096
Synonym: Seikalizer E,Rhodialux,Benzophenone 12,P Sanduvor 3035
Target:
CycLuc3
Cat.No: T31145
Synonym: Cyc Luc 3,Cyc-Luc-3
Target:
MS-444
Cat.No: T16145
Synonym: BE-34776
Target: Others
OptoDArG
Cat.No: T33814
Synonym: Opto-DArG,Opto DArG
Target:
ML 7
Cat.No: T33451
Synonym: ML7,ML-7
Target:
BoNT-IN-33
Cat.No: T69377
Synonym:
Target:
JF-NP-26
Cat.No: T38229
Synonym:
Target:
PA1 2HCl
Cat.No: T28287
Synonym: PA1,PA1 dihydrochloride
Target:
Talaporfin free acid
Cat.No: T34777
Synonym: Monoaspartyl chlorin,NPe6,Talaporfin,Aspartyl chlorin
Target:
MS 347a
Cat.No: T70626
Synonym:
Target:
ML344
Cat.No: T25818
Synonym: ML-344,ML 344
Target:
DMNP-EDTA
Cat.No: T31552
Synonym: DMNPEDTA,DM-Nitrophen,DM Nitrophen,DMNP EDTA
Target:
NSC-84096
Cat.No: T25890
Synonym: CID 256758,CID-256758,CID256758
Target:
Cat. No. Product Name Target Signaling Pathways
T8024 3-Indoleacetonitrile

Others; Endogenous Metabolite Metabolism; Others
3-Indoleacetonitrile 是内源性代谢产物的一种。
T5682 6-Hydroxyindole

Others Others
6-Hydroxyindole 是白色至浅棕色结晶或结晶性粉末。
T5771 Hypocrellin A

Antibacterial; PKC; Parasite Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
Hypocrellin A 是一种天然的PKC 抑制剂,具有光诱导的抗肿瘤、抗真菌和抗病毒活性,还对 MHC 限制性抗原呈递发挥免疫调节作用。
T1391 4-Methylumbelliferone

Hymecromone,4-MU,胆通

Others Others
4-Methylumbelliferone (Hymecromone) 是透明质酸生物合成抑制剂,显示出抗肿瘤和抗转移活性。
TMA2394 DL-alpha-Tocopherol

DL-α-生育酚,消旋-α-生育酚,DL-α-Tocopherol,Alpha-Tochopherol,Ephanyl

Antioxidant; Ferroptosis Apoptosis; oxidation-reduction
DL-alpha-Tocopherol (Ephanyl) 是一种合成维生素 E,能保护皮肤成纤维细胞免受紫外线的细胞毒性作用,具有抗氧化作用。
TMS2180 Zeaxanthin

Anchovyxanthin,All-Trans-Zeaxanthin,玉米

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
Zeaxanthin (All-Trans-Zeaxanthin) 是食物获得类胡萝卜素,存在于眼睛的黄斑部,具有抗氧化活性。
T1311 4-aminobenzoic acid

PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸

Endogenous Metabolite Metabolism
4-aminobenzoic acid (para-Aminobenzoic acid) 是一种具有紫外线吸收和抗纤维化特性的有机酸。当暴露在光线下时,4-aminobenzoic acid 吸收紫外线并通过光化学反应释放多余的能量,这可能会对DNA造成损害。4-aminobenzoic acid 还可以增加组织水平的摄氧量,并可能增强单胺氧化酶(MAO)活性以促进血清素的降解,过量可能导致纤维化变化。
T2850 Bicuculline

荷包牡丹碱,(+)-Bicuculline,d-Bicuculline

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Bicuculline ((+)-Bicuculline) 是从东北延胡索中提取的一种生物碱,能阻断 Ca2+激活钾 (SK) 通道。它是一种竞争性的神经递质 GABAA 受体拮抗剂,IC50为 2 μM。
TN2286 Tsugaric acid A

NO Synthase Immunology/Inflammation
Tsugaric acid A 能够显著抑制超氧阴离子的形成,还可以保护人类角质形成细胞,使其免受紫外线 B 诱导的损害。
T1301 Guaiacol

O-methylcatechol,2-hydroxyanisole,o-methoxyphenol,2-Methoxyphenol,愈创木酚

NF-κB; COX; Endogenous Metabolite Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Guaiacol (2-Methoxyphenol) 是从小叶栲中提取的一种酚类,可抑制 LPS 刺激的COX-2表达和NF-κB 激活,具有抗炎活性。
T1659 Melatonin

Melatonine,松果体素,N-Acetyl-5-methoxytryptamine,褪黑素

CaMK; Apoptosis; Mitophagy; Estrogen/progestogen Receptor; Melatonin Receptor; Glutathione Peroxidase; Endogenous Metabolite; ROR; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Melatonin (Melatonine) 是一种由松果体制成的激素,可激活褪黑激素受体。它在睡眠中起作用,有抗氧化和抗炎特性。它是新型选择性ATF-6抑制剂,可诱导细胞凋亡。
T3851 Vicenin 2

Vicenin -2,维采宁 2,新西兰牡荆苷

RAAS Endocrinology/Hormones
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。
TN4280 Isodictamnine

Others Others
Isodictamnine is phototoxic to certain bacteria and yeasts in long wave UV light.
T10348 Apigenin-7-diglucuronide

Others Others
Apigenin-7-diglucuronide is a flavonoid glycoside that exists in an assortment of medicinal plants with anti-inflammatory or ant-oxidant activities. It protects retinas against bright light-induced photoreceptor degeneration through the inhibition of reti
T60290 Benzyl salicylate

Benzyl salicylate 是一种水杨酸衍生物,可用作香料添加剂或紫外线吸收剂。
TN3276 8-Epixanthatin

Antifection Microbiology/Virology
8-Epixanthatin, a light-induced growth inhibitor, mediates the phototropic curvature in sunflower (Helianthus annuus) hypocotyls, it can induce germination of O. cumana at nano- to micromolar concentrations. 8-Epixanthatin has antiprotozoal activity.
TN2736 2',6'-Dihydroxy-4'-methoxyacetophenone

Antifection Microbiology/Virology
2',6'-Dihydroxy-4'-methoxyacetophenone is a phytoalexin after fungal inoculation with Botrytis cinerea or UV light irradiation, it has spore germination inhibition on Botrytis cinerea and Phomopsis perniciosa, with ED50 values of 45 and 410 uM, respective
T29607 Acid Red 88

11391 Red,Eniacid Fast Red A,Peony,Red No. 506

Acid red 88 is an anionic dye with potentially useful photocatalytic research applications. Acid red 88 has been used to determine the effect of Au deposition on ZnO photocatalytic activity under visible light. Additionally, the photocatalyst Au-TiO2 was
T75608 Myricetin 3-O-α-L-arabinopyranoside

Myricetin 3-O-α-L-arabinopyranoside 抑制 A2E 光氧化诱导的RPE 细胞死亡。Myricetin 3-O-α-L-arabinopyranoside 对视网膜变性具有保护作用,可保护蓝光 (BL) 诱导对 RPE 细胞和小鼠模型的损伤。
T14047 5-Aminolevulinic acid

5-Amino-4-oxopentanoic acid

Others Others
5-Aminolevulinic acid 是血红素合成的中间体,是卟啉合成途径中的一个化合物。它是一种光敏剂、抗肿瘤剂和前药。它也可以(以盐酸盐的形式)与蓝光照明结合使用,用于治疗面部或头皮的轻度至中度厚的光化性角化病。

天然产物

3-Indoleacetonitrile
Cat.No: T8024
Synonym:
Target: Others, Endogenous Metabolite
6-Hydroxyindole
Cat.No: T5682
Synonym:
Target: Others
Hypocrellin A
Cat.No: T5771
Synonym:
Target: Antibacterial, PKC, Parasite
4-Methylumbelliferone
Cat.No: T1391
Synonym: Hymecromone,4-MU,胆通
Target: Others
DL-alpha-Tocopherol
Cat.No: TMA2394
Synonym: DL-α-生育酚,消旋-α-生育酚,DL-α-Tocopherol,Alpha-Tochopherol,Ephanyl
Target: Antioxidant, Ferroptosis
Zeaxanthin
Cat.No: TMS2180
Synonym: Anchovyxanthin,All-Trans-Zeaxanthin,玉米
Target: Antioxidant, Endogenous Metabolite
4-aminobenzoic acid
Cat.No: T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸
Target: Endogenous Metabolite
Bicuculline
Cat.No: T2850
Synonym: 荷包牡丹碱,(+)-Bicuculline,d-Bicuculline
Target: GABA Receptor
Tsugaric acid A
Cat.No: TN2286
Synonym:
Target: NO Synthase
Guaiacol
Cat.No: T1301
Synonym: O-methylcatechol,2-hydroxyanisole,o-methoxyphenol,2-Methoxyphenol,愈创木酚
Target: NF-κB, COX, Endogenous Metabolite
Melatonin
Cat.No: T1659
Synonym: Melatonine,松果体素,N-Acetyl-5-methoxytryptamine,褪黑素
Target: CaMK, Apoptosis, Mitophagy, Estrogen/progestogen Receptor, Melatonin Receptor, Glutathione Peroxidase, Endogenous Metabolite, ROR, Autophagy
Vicenin 2
Cat.No: T3851
Synonym: Vicenin -2,维采宁 2,新西兰牡荆苷
Target: RAAS
Isodictamnine
Cat.No: TN4280
Synonym:
Target: Others
Apigenin-7-diglucuronide
Cat.No: T10348
Synonym:
Target: Others
Benzyl salicylate
Cat.No: T60290
Synonym:
Target:
8-Epixanthatin
Cat.No: TN3276
Synonym:
Target: Antifection
2',6'-Dihydroxy-4'-methoxyacetophenone
Cat.No: TN2736
Synonym:
Target: Antifection
Acid Red 88
Cat.No: T29607
Synonym: 11391 Red,Eniacid Fast Red A,Peony,Red No. 506
Target:
Myricetin 3-O-α-L-arabinopyranoside
Cat.No: T75608
Synonym:
Target:
5-Aminolevulinic acid
Cat.No: T14047
Synonym: 5-Amino-4-oxopentanoic acid
Target: Others
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