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680

抑制剂 & 化合物

339

天然产物

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Cat. No. Product Name Target Signaling Pathways
T9612 Antibacterial agent 27 

Anti-infection Microbiology/Virology
Antibacterial agent 27 是抗菌化合物,显示出有效的抗念珠菌活性。
T11427 Antibacterial compound 2

Antifungal Microbiology/Virology
Antibacterial compound 2 是一种有效的抗菌剂,对许多人类兽医病原体有效,对多重耐药葡萄球菌、肠球菌和链球菌,以及厌氧菌有抑制作用。
T72047 Antibacterial agent 125

Antibacterial Microbiology/Virology
Antibacterial agent 125 是一种抗菌剂。Antibacterial agent 125 对临床相关的革兰氏阳性病原体具有有效的抗菌活性,MIC50值范围为 0.25 - 8 μM。Antibacterial agent 125 可用于抗菌药物耐药性研究。
T38877 Antibacterial agent 52

Antibacterial agent 52 (example 18) is a antibacterial agent.
T40338 Antibacterial agent 31

Antibacterial agent 31 exhibits (shows) efficacy (activity) in combating (against) rice bacterial leaf streak.
T61159 Antibacterial agent 26

Antibacterial Microbiology/Virology
Antibacterial agent 26 是一种抗菌化合物,是有效的DHFR 抑制剂(金黄色葡萄球菌DHFR Ki 为0.020 nM)。
T38886 Antibacterial agent 61

Antibacterial agent 61 (example 27) is a antibacterial agent.
T38874 Antibacterial agent 35

Antibacterial Agent 35 (AA35) is a potent antibacterial agent that effectively reduces the minimum inhibitory concentration (MIC) of Ceftazidime, another antibacterial agent.
T38866 Antibacterial agent 39

Antibacterial agent 39 is a potent compound that exhibits antibacterial properties. It effectively reduces the minimum inhibitory concentration (MIC) of Ceftazidime, another antibacterial agent.
T38939 Antibacterial agent 38

Antibacterial agent 38 is an effective antibacterial agent. It can be utilized in the scientific investigation of bacterial infections.
T40301 Antibacterial agent 28

Antibacterial agent 28, with a minimum inhibitory concentration (MIC) range of 0.5-2 μg/mL, exhibits promising potential as an antibacterial candidate targeting MRSA infections.
T38916 Antibacterial agent 51

Antibacterial agent 51 (example 45) is a potent antibacterial compound effective against E. coli strains NCTC 13351, M 50, and 7 MP, with MIC values of 4, 8, and 8 mcg/mL, respectively (WO2013030733A1).
T38883 Antibacterial agent 59

Antibacterial agent 59 (example 24) is a antibacterial agent.
T38878 Antibacterial agent 53

Antibacterial agent 53 (example 19) is a antibacterial agent.
T38873 Antibacterial agent 49

Antibacterial agent 49 (example 12) is a antibacterial agent.
T38882 Antibacterial agent 58

Antibacterial Agent 58 (AA58) is a potent antibacterial compound that effectively reduces the minimum inhibitory concentration (MIC) value of Ceftazidime, another antibacterial agent.
T38869 Antibacterial agent 44

Antibacterial agent 44 is a novel antibacterial compound (WO2013030735A1, example 7). It exhibits potent antibacterial activity and is suitable for research purposes related to the study of bacterial infections.
T38885 Antibacterial agent 60

Antibacterial agent 60 is a potent compound that effectively reduces the minimum inhibitory concentration (MIC) of Ceftazidime, an antibacterial agent.
T38875 Antibacterial agent 34

Antibacterial agent 35 is a compound that effectively reduces the minimum inhibitory concentration (MIC) of Ceftazidime, enhancing its antibacterial activity.
T38868 Antibacterial agent 43

Antibacterial agent 43, is a potent antibacterial compound. It exhibits promising activity against bacterial infections and offers great potential for research purposes.
T38872 Antibacterial agent 47

Antibacterial Agent 47 demonstrates potent antibacterial activity as an adjunct therapy to parenteral antibiotic Ceftazidime. By effectively reducing the minimum inhibitory concentration (MIC) of Ceftazidime, Antibacterial Agent 47 acts as a highly promising antimicrobial agent, thereby enhancing the overall efficacy of the treatment.
T36657 Antibacterial agent 18

Antibacterial agent 18, a multi-arm AIE molecule, demonstrates efficacy against both Gram-positive and Gram-negative bacteria. Antibacterial agent 18 functions by conjugating with the cell wall of bacteria with rigid arm configuration, thereby interfering with the sugar and peptide processes essential for cell wall turning. This mechanism inhibits or eradicates bacterial growth[1].
T72309 Antibacterial agent 131

Antibacterial Microbiology/Virology
Antibacterial agent 131 是一种具有抗菌作用的化合物。
T72310 Antibacterial agent 132

Antifungal Microbiology/Virology
Antibacterial agent 132 对 C. parapsilosis (ATCC 22019) 和 C. krusei (ATCC 6258) 实验中显示出抗菌作用,MIC90 值分别为 <0.06 μg/mL 和 62.50 μg/mL。Antibacterial agent 132 对芳香化酶 (aromatase enzyme)具有抑制作用,IC50 为 0.047μM。
T39249 Antibacterial agent 40

Antibacterial agent 40 is an antibacterial agent.
T38881 Antibacterial agent 56

Antibacterial agent 56 (example 22) is a antibacterial agent.
T38879 Antibacterial agent 54

Antibacterial agent 54 (example 20) is a antibacterial agent.
T38865 Antibacterial agent 41

Antibacterial agent 41 (example 3) is a antibacterial agent.
T38870 Antibacterial agent 45

Antibacterial Agent 45 (AA45) exemplifies a potent antibacterial compound that effectively reduces the minimal inhibitory concentration (MIC) value of Ceftazidime, another antibacterial agent.
T38917 Antibacterial agent 50

Antibacterial agent 50 (example 47) is a compound that exhibits antibacterial activity. It shows minimum inhibitory concentration (MIC) values of 32, 64, and 128 mcg/mL against three strains of E. coli, namely NCTC 13351, M 50, and 7 MP, respectively (WO2013030733A1).
T38876 Antibacterial agent 33

Antibacterial Agent 33, a potent antibacterial compound, effectively decreases the minimum inhibitory concentration (MIC) of Ceftazidime, another antibacterial agent.
T38884 Antibacterial agent 57

Antibacterial agent 57 (example 25) is a antibacterial agent.
T38880 Antibacterial agent 55

Antibacterial agent 55 (example 21) is a antibacterial agent.
T38867 Antibacterial agent 42

Antibacterial Agent 42 demonstrates potent antibacterial activity by effectively reducing the Minimum Inhibitory Concentration (MIC) of the broad-spectrum antibacterial agent Ceftazidime.
T38871 Antibacterial agent 46

Antibacterial agent 46, serves as a potent antibacterial compound. With its versatile properties, this agent demonstrates considerable potential for supporting research on bacterial infections.
T38938 Antibacterial agent 37

Antibacterial agent 37 is an effective antimicrobial compound. It holds potential as a valuable tool for researching bacterial infections.
T40316 Antibacterial agent 30

Antibacterial agent 30 exhibits remarkable in vitro activity against Xoo, as evidenced by its EC50 value of 1.9 μg/mL.
T38915 Antibacterial agent 32

Antibacterial agent 32 exhibits potent antimicrobial activity against E. coli strains NCTC 13351, M 50, and 7 MP, with minimum inhibitory concentration (MIC) values of 1 mcg/mL, 2 mcg/mL, and 8 mcg/mL, respectively (WO2013030733A1, example 43).
T10500 Antibacterial compound 1

Antibacterial Microbiology/Virology
Antibacterial compound 1 is an antibacterial compound.
T62880 Antibacterial agent 99

Antibacterial agent 99 (compound 7b) 是一种有效的抗菌剂。Antibacterial agent 99 具有显著的抗菌和抗真菌作用,且没有溶血活性。
T62120 Antibacterial agent 79

Antibacterial agent 79 是一种抗菌剂。
T63224 Antibacterial agent 104

Antibacterial agent 104 是有效的抗细菌 (antibacterial) 剂,体外具有显著的抗细菌作用,体内表现出良好的抗 MRSA 效果。
T63252 Antibacterial agent 113

Antibacterial agent 113 是有效的抗菌剂 (antibacterial),对P.aeruginosa、S.mutans、B.subtilis、E.coli、E.faecalis、S.typhimuriumand 和S.aureus microorganisms 表现出抗菌作用,MIC 值均为 15625 μM。
T61123 Antibacterial agent 111

Antibacterial agent 111 (Compound 3) exhibits potent antibacterial activity against B. cereus and K. pneumonia, with MIC values of 3.90 μg/mL and 0.49 μg/mL, respectively. It achieves this antibacterial effect by strongly binding to specific residues of tyrosyl-tRNA synthetase [1].
T61170 Antibacterial agent 96

Antibacterial agent 96 (compound 4k) 是一种有效的抗菌剂。Antibacterial agent 96 对药物敏感和耐多药的结核分枝杆菌 (M.tuberculosis)显示出抗结核活性。Antibacterial agent 96 对 HepG2 和 Vero 细胞有毒性。
T60455 Antibacterial agent 65

Antibacterial agent 65 是潜在的抗菌剂和抗氧化剂。
T73911 Antibacterial agent 12

Antibacterial agent 12 是一种联芳基恶唑烷酮类似物,是一种针对抗生素敏感和耐药革兰氏阳性菌的抗菌剂。
T62627 Antibacterial agent 69

Antibacterial agent 69 是一种新型结构抗菌调节剂,并被用来对抗致命的耐多药细菌感染 (MICs: 2.978 μM)。
T78976 Antibacterial agent 141

Antibacterialagent 141(Compound B14)针对四种植物病原体Xoo、Xac、Psa与Cmm展现出了抗菌效果,其EC50值为1.28 μM。该化合物能够抑制细胞膜形成并改变细胞透性。
T72303 Antibacterial agent 124

Antibacterial agent 124 是一种有效的细菌脯氨酸-tRNA 合成酶 (ProRS) 抑制剂,对 Staphylococcus aureusProRS (SaProRS) 的 IC50为 0.18 μM。

化合物

Antibacterial agent 27 
Cat.No: T9612
Synonym:
Target: Anti-infection
Antibacterial compound 2
Cat.No: T11427
Synonym:
Target: Antifungal
Antibacterial agent 125
Cat.No: T72047
Synonym:
Target: Antibacterial
Antibacterial agent 52
Cat.No: T38877
Synonym:
Target:
Antibacterial agent 31
Cat.No: T40338
Synonym:
Target:
Antibacterial agent 26
Cat.No: T61159
Synonym:
Target: Antibacterial
Antibacterial agent 61
Cat.No: T38886
Synonym:
Target:
Antibacterial agent 35
Cat.No: T38874
Synonym:
Target:
Antibacterial agent 39
Cat.No: T38866
Synonym:
Target:
Antibacterial agent 38
Cat.No: T38939
Synonym:
Target:
Antibacterial agent 28
Cat.No: T40301
Synonym:
Target:
Antibacterial agent 51
Cat.No: T38916
Synonym:
Target:
Antibacterial agent 59
Cat.No: T38883
Synonym:
Target:
Antibacterial agent 53
Cat.No: T38878
Synonym:
Target:
Antibacterial agent 49
Cat.No: T38873
Synonym:
Target:
Antibacterial agent 58
Cat.No: T38882
Synonym:
Target:
Antibacterial agent 44
Cat.No: T38869
Synonym:
Target:
Antibacterial agent 60
Cat.No: T38885
Synonym:
Target:
Antibacterial agent 34
Cat.No: T38875
Synonym:
Target:
Antibacterial agent 43
Cat.No: T38868
Synonym:
Target:
Antibacterial agent 47
Cat.No: T38872
Synonym:
Target:
Antibacterial agent 18
Cat.No: T36657
Synonym:
Target:
Antibacterial agent 131
Cat.No: T72309
Synonym:
Target: Antibacterial
Antibacterial agent 132
Cat.No: T72310
Synonym:
Target: Antifungal
Antibacterial agent 40
Cat.No: T39249
Synonym:
Target:
Antibacterial agent 56
Cat.No: T38881
Synonym:
Target:
Antibacterial agent 54
Cat.No: T38879
Synonym:
Target:
Antibacterial agent 41
Cat.No: T38865
Synonym:
Target:
Antibacterial agent 45
Cat.No: T38870
Synonym:
Target:
Antibacterial agent 50
Cat.No: T38917
Synonym:
Target:
Antibacterial agent 33
Cat.No: T38876
Synonym:
Target:
Antibacterial agent 57
Cat.No: T38884
Synonym:
Target:
Antibacterial agent 55
Cat.No: T38880
Synonym:
Target:
Antibacterial agent 42
Cat.No: T38867
Synonym:
Target:
Antibacterial agent 46
Cat.No: T38871
Synonym:
Target:
Antibacterial agent 37
Cat.No: T38938
Synonym:
Target:
Antibacterial agent 30
Cat.No: T40316
Synonym:
Target:
Antibacterial agent 32
Cat.No: T38915
Synonym:
Target:
Antibacterial compound 1
Cat.No: T10500
Synonym:
Target: Antibacterial
Antibacterial agent 99
Cat.No: T62880
Synonym:
Target:
Antibacterial agent 79
Cat.No: T62120
Synonym:
Target:
Antibacterial agent 104
Cat.No: T63224
Synonym:
Target:
Antibacterial agent 113
Cat.No: T63252
Synonym:
Target:
Antibacterial agent 111
Cat.No: T61123
Synonym:
Target:
Antibacterial agent 96
Cat.No: T61170
Synonym:
Target:
Antibacterial agent 65
Cat.No: T60455
Synonym:
Target:
Antibacterial agent 12
Cat.No: T73911
Synonym:
Target:
Antibacterial agent 69
Cat.No: T62627
Synonym:
Target:
Antibacterial agent 141
Cat.No: T78976
Synonym:
Target:
Antibacterial agent 124
Cat.No: T72303
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T72235 Antibacterial synergist 2

Antibacterial synergist 2 是菌膜抑制剂。Antibacterial synergist 2 对肠球菌、金色葡萄球菌、铜绿假单胞菌和白色假单胞菌具有抑制效应。Antibacterial synergist 2 可用于与形成菌膜的病原体的相关研究。
TN1774 Isobavachromene

Others; Antibacterial Microbiology/Virology; Others
Isobavachromene 是一种抗菌剂。
TN1148 Isopsoralenoside

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Antibacterial Endocrinology/Hormones; Microbiology/Virology
Isopsoralenoside 是补骨脂多糖中的一种苯并呋喃苷。它在消化道内容物中可迅速代谢为补骨脂素。它具有雌激素样活性、促进成骨细胞增殖活性、抗肿瘤活性和抗菌活性。
T37345 5,7-Dihydroxycoumarin

Antibacterial Microbiology/Virology
5,7-Dihydroxycoumarin 是分离自Macaranga triloba 花序的香豆素,具有抗菌活性。
T8249 Hexahydrofarnesyl acetone

植酮,Phytone

Others; Antibacterial Microbiology/Virology; Others
Hexahydrofarnesyl acetone (Phytone) 是从Launaea mucronata 中分离得到的倍半萜,具有抗菌和抗炎活性,可研究缓解疼痛。
T10668 Camalexin

Reactive Oxygen Species; ROS; Antibacterial; Antifungal Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Camalexin 是从Camelina sativa 和Arabidopsis 中分离出来的一种植物抗毒素,可诱导活性氧的产生,具有抗菌、抗真菌、抗增殖和抗癌活性。
T3S0970 Thermopsine

Thermospine,黄华碱

Antibacterial Microbiology/Virology
Thermopsine (Thermospine) 是从槐豆亚种的果实,豆荚和茎皮中分离出来的一种喹诺酮类生物碱,具有抗菌活性。
T3S1088 Isoforsythiaside

异连翘脂苷,异连翘酯苷

Anti-infection; Antibacterial Microbiology/Virology
Isoforsythiaside 有抗氧化和抗菌活性。
TN2085 Piperlonguminine

Anti-infection; Antibacterial; Antifungal Microbiology/Virology
Piperlonguminine 是一种从 Piper 中分离出的生物碱酰胺。它具有多种生物活性,如神经保护、抗炎、抗肿瘤、抗血小板、抗黑素生成、抗真菌和抗菌活性。
T5802 Stearyl glycyrrhetinate

Antiviral; Antibacterial Immunology/Inflammation; Microbiology/Virology
Stearyl glycyrrhetinate 是甘草提取物中的主要成分之一,具有抗菌作用,对金黄色葡萄球菌菌株的 MIC 大于 256 mg/L。
T3947 Nonanoic acid

pelargonic acid,Nonoic acid,壬酸

Others; Antibacterial Microbiology/Virology; Others
Nonanoic acid (Nonoic acid) 是一种天然存在的具有九个碳原子的饱和脂肪酸。它减少细菌易位,增强抗菌活性,并增加猪 β-防御素 1 (pBD-1) 和 pBD-2 的分泌。
TN2010 Ombuin

商陆黄素,商陆素

Antibacterial Microbiology/Virology
Ombuin 是一种从花椒中分离出的广谱抗菌剂,MIC 为 125 至 500 μg/mL。
T3S2381 Perillene

3-Isohexenylfuran,紫苏烯,Perillen

Others; Antibacterial Microbiology/Virology; Others
Perillene (3-Isohexenylfuran) 是促进肠蠕动的药物中的活性成分,它对金黄色葡萄球菌和大肠杆菌具有很强的抗药性。
T3332 Isosteviol

异甜菊醇,(-)-Isosteviol

IL Receptor; Potassium Channel; TNF; NF-κB; Reactive Oxygen Species; COX; Topoisomerase Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Isosteviol ((-)-Isosteviol) 是一种常见的天然甜味剂,属于四环二萜糖苷,是甜菊糖苷通过酸催化水解产生的。它抑制 DNA 聚合酶和 DNA 拓扑异构酶,具有抗菌、抗癌和抗结核作用。
T1134 Clofoctol

叔辛酚氯,氯福克酚

Antibacterial; Antibiotic Microbiology/Virology
Clofoctol 是一种抗生素,,可研究革兰氏阳性菌感染。它仅对革兰氏阳性菌起作用, 可渗透入人类肺组织。
TN1403 Arjunolic acid

IL Receptor; TNF; Reactive Oxygen Species; JNK; AChE Apoptosis; Immunology/Inflammation; MAPK; Metabolism; Neuroscience; NF-κB
Arjunolic acid 是分离自蓝莓的皂苷,具有抗氧化、抗菌和抗炎症等多种生物活性,在保护细胞和组织免受活性氧的有害作用中发挥重要作用。
T10933 D-Cysteine

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-Cysteine 是一种大肠杆菌生长的有力抑制剂,是半胱氨酸的 D 型异构体。它由 D-氨基酸氧化酶介导产生 H2S,是一种对抗小脑共济失调的神经保护剂。 D-半胱氨酸可以抑制由变形链球菌和链球菌血红蛋白形成的两种生物膜的生长和致龋性。
TN1733 Hesperetin 7-O-glucoside

Anti-infection; Antibacterial; HMG-CoA Reductase Metabolism; Microbiology/Virology
Hesperetin 7-O-glucoside 是通过 Hesperidin 的酶促转化产生的一种人 HMG-CoA 还原酶抑制剂,具有降压作用,可抑制幽门螺杆菌的生长。
TN1008 Psoralenoside

CaMK; Calcium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T8211 (±)-Decursinol

紫花前胡醇,3',4'-dihydro-3'-hydroxy-Xanthyletin

Others; Antibacterial Microbiology/Virology; Others
(±)-Decursinol (3',4'-dihydro-3'-hydroxy-Xanthyletin) 是来自当归的一种 FtsZ 抑制剂,抑制 B. anthracis 的 FtsZ 聚合,IC50为 102 μM。
TN1019 Beta-mangostin

β-Mangostin,beta-倒捻子素

Apoptosis; Antibacterial; Parasite Apoptosis; Microbiology/Virology
Beta-mangostin (β-Mangostin) 是存在 Cratoxylum arborescens 中的一种氧杂蒽酮类天然产物,有抗癌和抗菌活性,对结核分枝杆菌的 MIC 值为 6.25 μg/mL。它在体外有抗疟活性,对恶性疟原虫的 IC50值为 3.00 μg/mL。
TN2158 Robinetin

3,3',4',5',7-Pentahydroxyflavone,洋槐黄素

Anti-infection; HIV Protease; Antibacterial Microbiology/Virology; Proteases/Proteasome
Robinetin (3,3',4',5',7-Pentahydroxyflavone) 是一种天然黄酮,具有显著的“两种颜色”固有荧光特性。它具有抗真菌、抗病毒、抗菌、抗突变、抗氧化和抗自由基活性,高效抑制 EYPC 膜脂质过氧化和 HbA 糖基化。
T2S0961 Chalcone

benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮

EGFR; Antibacterial Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Chalcone (Cinnamophenone) 是从甘草中分离得到的一种芳香酮,可合成查耳酮衍生物。它具有多种生物和药理的活性,如抗炎、抗菌、抗癌、抗氧化、抗寄生虫等活性。
T1687 Doxycycline

Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素

MMP; ribosome; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。
T6702 Terbinafine

Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine (TDT 067) 是念珠菌属的角鲨烯环氧化酶有效的非竞争性抑制剂,Ki 值为 30 nM。它具有抗真菌感染活性。
TN3920 Effusanin A

Raf; Antifection MAPK; Microbiology/Virology
Effusanin A 是一种存在于Isodon rugosus 之中的天然产物。 它具有 DNA 损伤和抗菌作用。
TN6722 Terminolic acid

2α,6β,23-trihydroxyl oleanolic acid

Antibacterial Microbiology/Virology
Terminolic acid (2α,6β,23-trihydroxyl oleanolic acid) 是一种从 Combretum racemosum 中分离得到的五环三萜糖苷,可通过与 IL-1β 和 IL-6 的受体活性位点结合抑制促炎细胞因子,并通过与 IL-4 受体结合位点结合增强抗炎细胞因子。它还表现出适度的抗菌活性。
T4S1173 Agrimol B

仙鹤草酚B,仙鹤草酚 B

Sirtuin; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物,可抑制脂肪形成,降低PPARγ的表达,诱导SIRT1易位和表达。
T3008 Lawsone methyl ether

2-Methoxy-1,4-naphthoquinone,2-Methoxy-p-naphthoquinone,2-Methoxynaphthoquinone,2-甲氧基-1,4-萘并醌

Apoptosis; Antibacterial; Antifungal Apoptosis; Microbiology/Virology
Lawsone methyl ether (2-Methoxy-1,4-naphthoquinone) 是从凤仙花和Swertia calycina 中分离出的,有抗真菌和抗菌活性。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
T2S0493 Isoeugenol

4-Propenylguaiacol,2-Methoxy-4-propenylphenol,异丁香酚,异丁香酚;4-丙烯基-2-甲氧基苯酚、对丙烯基邻甲氧基本酚、异丁子香酚

Antibacterial Microbiology/Virology
Isoeugenol (4-Propenylguaiacol) 是肉豆蔻,丁香和肉桂的精油成分,具有抗菌活性。它抑制Escherichia coli 和Listeria innocua,MIC 值分别为 0.6 mg/mL 和 1 mg/mL。
T3417 Amentoflavone

Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin

Apoptosis; P450; Phospholipase; Reactive Oxygen Species; Opioid Receptor; COX; Antibacterial; RSV; Antifungal Apoptosis; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
Amentoflavone (3',8''-Biapigenin) 是一种具有很多生物活性的双黄酮类天然产物,有抗炎、抗氧化和神经保护等作用。
T1411 Terbinafine hydrochloride

KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。
TN4893 Rapanone

拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌

Apoptosis; Phospholipase; Antibacterial; Parasite Apoptosis; Metabolism; Microbiology/Virology
Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) 是一种具有广泛生物活性的天然苯醌,如抗肿瘤、抗氧化、抗炎、抗菌和抗寄生虫活性。它还是选择性人滑膜 PLA2抑制剂,IC50值为 2.6 μM。
T3208 Brevianamide F

Cyclo-L-tryptophyl-L-proline,cyclo-(L-Trp-L-Pro),Cyclo(L-Pro-L-Trp)

BCRP; PI3K; Antibacterial Membrane transporter/Ion channel; Microbiology/Virology; PI3K/Akt/mTOR signaling
Brevianamide F (Cyclo(L-Pro-L-Trp)) 是一种从Colletotrichum gloeosporioides 中分离得到的真菌毒素,属于天然存在的 2,5-二酮哌嗪类,具有抗菌活性。它具有PI3Kα抑制活性,IC50值为 4.8 µM。
T3739 2,6-Dimethoxyquinone

2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌

Others Others
2,6-Dimethoxyquinone (2,6-Dimethoxy-p-benzoquinone) 是一种植物中提取吸脂诱导因子。它具有抗脂肪、抗癌、抗菌、抗疟疾和抗炎的作用。
T1100 Polymyxin B Sulfate

Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B Sulfate (Poly-RX) 是一个阳离子型表面活性剂抗生素剂,能够提高细胞膜的渗透性。
TN4943 Sanguisorbigenin

地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid

Antibacterial Microbiology/Virology
Sanguisorbigenin (Tomentosolic acid) 抑制耐甲氧西林金黄色葡萄球菌,是一种天然抗菌剂。
T3376 Cynaroside

朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside

Others; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。
T2S2104 Sinigrin hydrate

黑芥子苷,Sinigrin monohydrate,芥子甙单水合物,Allylglucosinolate monohydrate

Antibacterial Microbiology/Virology
Sinigrin hydrate (Allylglucosinolate monohydrate) 是一种天然脂肪族芥子油苷,存在于十字花科植物中。它具有消炎、抗癌、抗真菌、抗菌、抗氧化作用。
T4984 Cefozopran hydrochloride

SCE-2787 hydrochloride

Antifungal Microbiology/Virology
Cefozopran hydrochloride (SCE-2787 hydrochloride) 是一种半合成的非肠道头孢菌素。它是一种广谱抗菌抗生素,能抑制大多数革兰氏阴性和革兰氏阳性菌。
T3827 Rhein-8-glucoside calcium

大黄酸-8-O-β-D-葡萄糖苷,Rhein-8-O-β-D-glucopyranoside,Rhein-8-glucoside calcium salt

Phosphatase; Antibacterial Metabolism; Microbiology/Virology
Rhein-8-glucoside calcium (Rhein-8-glucoside calcium salt) salt 是一种从 Saussurea lappa 根的 EtOH 提取物中,分离得到的蒽醌类 hPTP1B 抑制剂,IC50值为11.5 μM,具有抗菌作用。
T20345 Benzoylacetone

AI3 10572,苯甲酰丙酮,AI3-10572,AI310572

Antibacterial Microbiology/Virology
Benzoylacetone (AI3 10572) 具有抗菌活性。
TN6780 Carvacrol methyl ether

Methyl carvacrol,Methyl carvacryl ether

Antibacterial Microbiology/Virology
Carvacrol methyl ether 来源于植物挥发油,具有抗菌活性。
T4S0528 Rhodojaponin V

闹羊花素 V,闹羊花毒素V

Others; Antibacterial Microbiology/Virology; Others
Rhodojaponin V 是一种从Rhododendron molle 叶子中获得的二萜类化合物,具有抗炎作用。
T12014 Methyl carnosate

Others Others
Methyl camosate, a diterpene sourced from Salvia officinalis or Rosmarinus officinalis, exhibits pronounced antioxidant and antibacterial properties.
T0144 Ftaxilide

Histanorm,安息香酸,伏保克西里

Antibacterial Microbiology/Virology
Ftaxilide (Histanorm) 是新型抗结核剂。
T20446 Creosol

Endogenous Metabolite Metabolism
Creosol 是内源性代谢产物的一种。
T20550 Thiobarbituric acid

NSC4733,NSC 4733,4,6-二羟基-2-巯基嘧啶,NSC-4733

Antibacterial Microbiology/Virology
Thiobarbituric acid (NSC-4733) 具有抗菌活性。
T5757 Loganetin

Antibacterial Microbiology/Virology
Loganetin 是无毒的天然产物,来源于Cornus officinalis Sieb. et Zucc.,可用于耐多药革兰氏阴性菌感染的研究。
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天然产物

Antibacterial synergist 2
Cat.No: T72235
Synonym:
Target:
Isobavachromene
Cat.No: TN1774
Synonym:
Target: Others, Antibacterial
Isopsoralenoside
Cat.No: TN1148
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Antibacterial
5,7-Dihydroxycoumarin
Cat.No: T37345
Synonym:
Target: Antibacterial
Hexahydrofarnesyl acetone
Cat.No: T8249
Synonym: 植酮,Phytone
Target: Others, Antibacterial
Camalexin
Cat.No: T10668
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antifungal
Thermopsine
Cat.No: T3S0970
Synonym: Thermospine,黄华碱
Target: Antibacterial
Isoforsythiaside
Cat.No: T3S1088
Synonym: 异连翘脂苷,异连翘酯苷
Target: Anti-infection, Antibacterial
Piperlonguminine
Cat.No: TN2085
Synonym:
Target: Anti-infection, Antibacterial, Antifungal
Stearyl glycyrrhetinate
Cat.No: T5802
Synonym:
Target: Antiviral, Antibacterial
Nonanoic acid
Cat.No: T3947
Synonym: pelargonic acid,Nonoic acid,壬酸
Target: Others, Antibacterial
Ombuin
Cat.No: TN2010
Synonym: 商陆黄素,商陆素
Target: Antibacterial
Perillene
Cat.No: T3S2381
Synonym: 3-Isohexenylfuran,紫苏烯,Perillen
Target: Others, Antibacterial
Isosteviol
Cat.No: T3332
Synonym: 异甜菊醇,(-)-Isosteviol
Target: IL Receptor, Potassium Channel, TNF, NF-κB, Reactive Oxygen Species, COX, Topoisomerase
Clofoctol
Cat.No: T1134
Synonym: 叔辛酚氯,氯福克酚
Target: Antibacterial, Antibiotic
Arjunolic acid
Cat.No: TN1403
Synonym:
Target: IL Receptor, TNF, Reactive Oxygen Species, JNK, AChE
D-Cysteine
Cat.No: T10933
Synonym:
Target: Endogenous Metabolite, Antibacterial
Hesperetin 7-O-glucoside
Cat.No: TN1733
Synonym:
Target: Anti-infection, Antibacterial, HMG-CoA Reductase
Psoralenoside
Cat.No: TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
(±)-Decursinol
Cat.No: T8211
Synonym: 紫花前胡醇,3',4'-dihydro-3'-hydroxy-Xanthyletin
Target: Others, Antibacterial
Beta-mangostin
Cat.No: TN1019
Synonym: β-Mangostin,beta-倒捻子素
Target: Apoptosis, Antibacterial, Parasite
Robinetin
Cat.No: TN2158
Synonym: 3,3',4',5',7-Pentahydroxyflavone,洋槐黄素
Target: Anti-infection, HIV Protease, Antibacterial
Chalcone
Cat.No: T2S0961
Synonym: benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮
Target: EGFR, Antibacterial
Doxycycline
Cat.No: T1687
Synonym: Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
Terbinafine
Cat.No: T6702
Synonym: Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067
Target: Antibacterial, Antibiotic, Antifungal
Effusanin A
Cat.No: TN3920
Synonym:
Target: Raf, Antifection
Terminolic acid
Cat.No: TN6722
Synonym: 2α,6β,23-trihydroxyl oleanolic acid
Target: Antibacterial
Agrimol B
Cat.No: T4S1173
Synonym: 仙鹤草酚B,仙鹤草酚 B
Target: Sirtuin, PPAR
Lawsone methyl ether
Cat.No: T3008
Synonym: 2-Methoxy-1,4-naphthoquinone,2-Methoxy-p-naphthoquinone,2-Methoxynaphthoquinone,2-甲氧基-1,4-萘并醌
Target: Apoptosis, Antibacterial, Antifungal
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Isoeugenol
Cat.No: T2S0493
Synonym: 4-Propenylguaiacol,2-Methoxy-4-propenylphenol,异丁香酚,异丁香酚;4-丙烯基-2-甲氧基苯酚、对丙烯基邻甲氧基本酚、异丁子香酚
Target: Antibacterial
Amentoflavone
Cat.No: T3417
Synonym: Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin
Target: Apoptosis, P450, Phospholipase, Reactive Oxygen Species, Opioid Receptor, COX, Antibacterial, RSV, Antifungal
Terbinafine hydrochloride
Cat.No: T1411
Synonym: KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride
Target: Antibacterial, Antibiotic, Antifungal
Rapanone
Cat.No: TN4893
Synonym: 拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌
Target: Apoptosis, Phospholipase, Antibacterial, Parasite
Brevianamide F
Cat.No: T3208
Synonym: Cyclo-L-tryptophyl-L-proline,cyclo-(L-Trp-L-Pro),Cyclo(L-Pro-L-Trp)
Target: BCRP, PI3K, Antibacterial
2,6-Dimethoxyquinone
Cat.No: T3739
Synonym: 2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌
Target: Others
Polymyxin B Sulfate
Cat.No: T1100
Synonym: Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX
Target: Antibacterial, Antibiotic
Sanguisorbigenin
Cat.No: TN4943
Synonym: 地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid
Target: Antibacterial
Cynaroside
Cat.No: T3376
Synonym: 朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside
Target: Others, Influenza Virus, DNA/RNA Synthesis
Sinigrin hydrate
Cat.No: T2S2104
Synonym: 黑芥子苷,Sinigrin monohydrate,芥子甙单水合物,Allylglucosinolate monohydrate
Target: Antibacterial
Cefozopran hydrochloride
Cat.No: T4984
Synonym: SCE-2787 hydrochloride
Target: Antifungal
Rhein-8-glucoside calcium
Cat.No: T3827
Synonym: 大黄酸-8-O-β-D-葡萄糖苷,Rhein-8-O-β-D-glucopyranoside,Rhein-8-glucoside calcium salt
Target: Phosphatase, Antibacterial
Benzoylacetone
Cat.No: T20345
Synonym: AI3 10572,苯甲酰丙酮,AI3-10572,AI310572
Target: Antibacterial
Carvacrol methyl ether
Cat.No: TN6780
Synonym: Methyl carvacrol,Methyl carvacryl ether
Target: Antibacterial
Rhodojaponin V
Cat.No: T4S0528
Synonym: 闹羊花素 V,闹羊花毒素V
Target: Others, Antibacterial
Methyl carnosate
Cat.No: T12014
Synonym:
Target: Others
Ftaxilide
Cat.No: T0144
Synonym: Histanorm,安息香酸,伏保克西里
Target: Antibacterial
Creosol
Cat.No: T20446
Synonym:
Target: Endogenous Metabolite
Thiobarbituric acid
Cat.No: T20550
Synonym: NSC4733,NSC 4733,4,6-二羟基-2-巯基嘧啶,NSC-4733
Target: Antibacterial
Loganetin
Cat.No: T5757
Synonym:
Target: Antibacterial
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