首页 工具
登录
购物车

搜索结果

Search Results for " applications "

530

抑制剂 & 化合物

57

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T7460 α-Cyano-4-hydroxycinnamic acid

α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基

Monocarboxylate transporter Membrane transporter/Ion channel
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) 是非竞争性单羧酸盐转运蛋白 (MCTs) 抑制剂,可抑制线粒体丙酮酸转运蛋白,Ki 值为 6.3 μM。它可作为基质辅助激光解吸电离-飞行时间质谱 (MALDI-TOF) 分析的基质,可以促进肽离子化。
T31786 Ferumoxytol

Magnetic Black,Black Iron BM,Magnetic oxide,Black Gold F 89,11557 Black

Others Others
Ferumoxytol (Magnetic Black) 是一种非钆基造影剂,可用于磁共振成像应用,可用于治疗缺铁性贫血和慢性肾病。
T77704 N-Isopropylacrylamide

Others Others
N-Isopropylacrylamide 具有热响应效应,被生物医学领域广泛应用。
T3225 16,17-Epoxy-21-acetoxypregnenolone

Others Others
16,17-Epoxy-21-acetoxypregnenolone 用作药物中间体。
T40645 PIPES

1,4-Piperazinediethanesulfonic acid,1,4-piperazine bis(ethanesulfonic acid),1,4-Piperazinebis(ethanesulfonic acid),PIPES

Others Others
PIPES (1,4-Piperazinediethanesulfonic acid) 作为PIPES缓冲液的关键成分,广泛应用于生化领域作为试剂。
T61148 Flutrimazole

Antifungal Microbiology/Virology
Flutrimazole is a dual-action imidazole antifungal compound, exhibiting both anti-inflammatory and antifungal properties. Notably, flutrimazole demonstrates limited transdermal penetration, making it particularly advantageous for topical applications in the treatment of fungal infections, especially those accompanied by inflammation.
T8415 4-Benzyl-2-carboxymorpholine hydrochloride

Others Others
4-Benzyl-2-carboxymorpholine hydrochloride 是一种用于蛋白质组学研究应用的专业产品,来自 Santa Cruz。
T19734 Triethoxyoctylsilane

Oleth-30,正辛基三乙氧基硅烷,NSC 42964,Triethoxycaprylylsilane

Others Others
Triethoxyoctylsilane (NSC 42964) 是用于塑料应用的化合物。
T12649 Ibafloxacine

S25930,Ibafloxacin,R835

Antifungal Microbiology/Virology
Ibafloxacine (R835) 是一种氟喹诺酮类抗生素,专门用于兽类,对巴氏杆菌显示出良好的抑菌效果。
T60226 CT52923

PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
CT52923 is a selective, orally active antagonist of platelet-derived growth factor receptor (PDGFR), functioning as an ATP-competitive inhibitor. It has versatile applications for researching an array of pathological diseases such as atherosclerosis, glomerulonephritis, liver cirrhosis, pulmonary fibrosis, and cancer.
T19521 PLGA

poly(lactic-co-glycolic acid),聚乳酸-羟基乙酸共聚物

Others Others
PLGA (poly(lactic-co-glycolic acid)) 是一种聚乳酸和聚乙醇酸的共聚物,能够制造用于药物递送和组织工程应用的装置。
T9981 RDR03785

Others Others
RDR 03785 可以控制 MIF 的生物活性,是 MIF 的拮抗剂。这种小分子/抑制剂主要用于细胞结构应用。
T4178 NSC 80538

Others Others
NSC 80538 是多重 HTS 检测中 MEK Kinase PB1 Domains 的抑制剂。
T6071 Parbendazole

SKF 29044,帕苯咪唑

Microtubule Associated; Parasite Cytoskeletal Signaling; Microbiology/Virology
Parbendazole (SKF 29044) 是一种有效的 microtubule 重组抑制剂,能够破坏微管蛋白,EC50值为 530 nM,也是广谱驱虫剂。
T76673 Bemarituzumab

FPA144

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
Bemarituzumab是一种新型人源化IgG1单抗,靶向xGFR2b。Bemarituzumab可防止FGFR2b与 FGF的结合并活化。Bemarituzumab在癌症研究中的潜在应用。
T18898 5(6)-TAMRA SE

5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯

Others Others
5(6)-TAMRA SE (5(6)-Carboxytetramethylrhodamine N-succinimidyl ester) 是荧光染料,能够结合寡聚核苷酸,并用于DNA 测序。
T22115 SM-7368

NF-κB NF-κB
NF-κB Activation Inhibitor III 是一种NF-kB 抑制剂,抑制 TNF-α 诱导的MMP-9上调,靶向抑制下游的MAPK p38,可用于靶向 TNF-α 介导的肿瘤侵袭和转移的化疗研究。
Fr14534 Pyrazinamine

Pyrazinamine 是一种合成中间体,可以用于各种科学研究应用,包括作为合成试剂以及作为生化和生理试剂。
T82236 HBED-CC-tris(tert-butyl ester)

HBED-CC-tris(tert-butyl ester)为HBED-CC的衍生物,具有双功能螯合性能,主要应用于农业研究和放射性药物领域。
T14527 Benfluralin

Benfluralin 是一种除草剂,是一种农用化学品,可用作芽前除草剂。 用于控制一系列粮食和非粮食作物中的草和其他杂草。
T35862 Cucurbit[8]uril

Others Others
Cucurbit[8]uril is a highly effective and safe supramolecular compound that promotes protein heterodimerization. It selectively induces the heterodimerization of methylviologen and naphthalene functionalized proteins, demonstrating its specificity and versatility. Additionally, Cucurbit[8]uril shows exceptional oral activity and low toxicity, making it a promising candidate for various pharmaceutical and biotechnological applications.
T7528 3,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate

Others Others
3,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate 是一种有用的研究化合物,适用于许多研究应用,包括化学领域和生命科学领域等。
T27710 K6PC-5

K6PC5,K6PC 5

S1P Receptor GPCR/G Protein
K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels. With its potential applications in skin diseases associated with abnormal keratinocyte function, as well as in studies on neurodegeneration and virus infection, K6PC-5 presents a promising compound for research purposes.
T72026 p53-MDM2-IN-1

Mdm2; p53 Apoptosis
p53-MDM2-IN-1 (Example 30) 是一种 p53-MDM2/X 蛋白相互作用的抑制剂,Ki 值为 23.35 µM。p53-MDM2-IN-1 能用于抗肿瘤研究。
T1477 AICAR

NSC105823,AICA Riboside,Acadesine,阿卡地新,AICAR (Acadesine)

Mitophagy; YAP; AMPK; Autophagy Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
AICAR (NSC105823) 是一种腺苷类似物,是一种 AMP 激活的蛋白激酶激活剂,可用于治疗急性淋巴细胞白血病和糖尿病。
T9404 2,5-DIBROMO-3,4-DINITROTHIOPHENE

Others Others
2,5-DIBROMO-3,4-DINITROTHIOPHENE 又称2,5-DBT,是一种有机溴化合物,在生物学研究、化学合成的中具有广泛应用。
T5363 Tempo

2,2,6,6-四甲基哌啶氧化物,2,2,6,6-Tetramethylpiperidinooxy

Free radical scavengers; Reactive Oxygen Species; DNA/RNA Synthesis; Mitochondrial Metabolism Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Tempo (2,2,6,6-Tetramethylpiperidinooxy) 可用作自由基清除剂、有机合成中的试剂和电子自旋共振光谱中的结构探针。它可在催化循环中使超氧化物歧化,也可诱导DNA 链断裂。
T72023 JB002

Myosin Cytoskeletal Signaling
JB002为一种肌球蛋白 II 抑制剂,IC50值不大于10 μM。适用于研究肌肉痉挛、慢性肌肉骨骼疼痛及肥厚型心肌病。
TP1125 Insulin(cattle)

牛胰岛素,Insulin from bovine pancreas,胰岛素

IGF-1R Tyrosine Kinase/Adaptors
Insulin cattle (Insulin from bovine pancreas) 是一种在胰腺 β 细胞中产生的两链多肽激素,在很多哺乳动物细胞培养体系中用作生长因子。
T17881 (S,R,S)-AHPC-C10-NH2

VH032-C10-NH2

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC-C10-NH2 (VH032-C10-NH2) 包含基于 (S,R,S)-AHPC 的VHL 配体和 1 个 linker,是一种合成的 E3 连接酶配体-linker 偶联物 (E3 ligase ligand-linker conjugate)。用于 BET 的靶向 PROTAC 的合成。
T50089 2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine

Others Others
2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine 是一种吲哚胺类化合物,在结构上与血清素相似。它是5-HT2A 受体的选择性激动剂,在神经科学领域具有潜在的应用。
T72031 BI 1015550

PDE Metabolism
BI 1015550 是一种具有口服活性的PDE4B 抑制剂,IC50值为 7.2 nM。BI 1015550 具有良好的安全性,在炎症、过敏疾病、肺纤维化和慢性阻塞性肺疾病 (COPD) 中有潜在应用。
T64321 Octyl-beta-D-glucopyranoside

Octyl glucoside,11β-HSD1-IN-11

Others Others
Octyl-beta-D-glucopyranoside (11β-HSD1-IN-11) 是一种非离子洗涤剂,广泛应用于生物技术,生化应用,膜蛋白的增溶和结晶的研究中。
T9523 TGFβRI-IN-3

TGF-beta/Smad Stem Cells
TGFβRI-IN-3 抑制TGFβR1,IC50为 0.79 nM,是对 MAP4K4 的选择性2000 倍。TGFβRI-IN-3 是一种高选择性的 TGFβR1 抑制剂,在免疫肿瘤中具有潜在的应用。
T76937 Burfiralimab

Burfiralimab (hzVSF-v13) 是一种针对病毒感染细胞表面表达的波形蛋白的单克隆IgG4抗体,具有广谱抗病毒活性和对病毒引起的炎症的抗炎作用。Burfiralimab 可用于重症 COVID-19 研究。
TP1809 TAT

HIV Protease Microbiology/Virology; Proteases/Proteasome
TAT 源自人免疫缺陷病毒的转录反式激活因子,是一种细胞穿透肽。它可以增加异源蛋白质的产量和溶解度。
T22168 Vialinin A

Terrestrin A

DUB Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
Vialinin A (Terrestrin A) (Terrestrin A) 是一种具有抗氧化性质的对三苯化合物。Vialinin A (Terrestrin A) 是 TNF-α,USP4, USP5 和 SENP1 特异性蛋白酶 1 的有效抑制剂。Vialinin A (Terrestrin A) 可用于自身免疫疾病和癌症研究。
T33639 Neotame

NC 00723,HSDB 7965,NC-00723,NC00723,纽甜

Others Others
Neotame (HSDB 7965) 是阿斯巴甜的衍生物,是低热量、高效的人造甜味剂,非营养性甜味剂和增味剂,其甜度是糖的 7000-13,000 倍,可用于多种食品。
T21142 Bupirimate

Nimrod

Antifungal Microbiology/Virology
Bupirimate (Nimrod) 是植物保护产品中的一种活性成分,常用作全身杀菌剂,可用于控制玫瑰和苹果种植园中的白粉病。Bupirimate 属于嘧啶类。
T38715 MSDC-0602K

MSDC-0602K,Azemiglitazone potassium

PPAR DNA Damage/DNA Repair; Metabolism
MSDC-0602K (Azemiglitazone potassium) (Azemiglitazone potassium) is a PPARγ-sparing thiazolidinedione (Ps-TZD) compound that binds to PPARγ with an IC50 of 18.25 μM. It also modulates the mitochondrial pyruvate carrier (MPC). This compound, MSDC-0602K, has potential applications in researching fatty liver conditions, including dysfunctional lipid metabolism, inflammation, and insulin resistance. MSDC-0602K acts as an insulin sensitizer, improving insulinemia and fatty liver disease in mice both ...
T50021 3-(3,6-dichloro-9H-carbazol-9-yl)propanoic acid

Others Others
3-(3,6-dichloro-9H-carbazol-9-yl)propanoic acid (DCPPA)是一种ASIC3抑制剂,可以有效阻断ASIC3介导的疼痛和炎症,已被证明在治疗中风、癫痫和癌症等其他疾病方面具有潜在应用。
T36958 BODIPY 505/515

BODIPY 505/515 是一种亲脂性荧光探针,可定位到细胞内的脂质体,已被用于标记脂滴。BODIPY 505/515 已被用于电子显微镜、外荧光显微镜、共聚焦显微镜以及各种藻类物种的流式细胞仪应用中。
T19027 Methyl Blue

Others Others
Methyl blue 是一种三氨基三苯甲烷染料。它在多色染色法中被广泛用作抗菌染料,并能够应用于组织学和微生物学染色溶液。它已被用作研究各种催化剂对染料光降解影响的模型。
T36957 BODIPY 493/503

BDP 493/503 lipid stain,Pyrromethene 546

Others Others
BODIPY 493/503 (Pyrromethene 546) 是一种亲脂性荧光探针,Ex/Em 为 493/503 nm。 BODIPY 493/503 定位于极性脂质,可用于标记细胞中性脂质含量以及活细胞和固定细胞应用。
T72083 Octadecyl Rhodamine B chloride

Octadecyl Rhodamine B chloride 也被叫做RBOE, 是一种极性敏感染料,常作为一种发色基团与其他化合物一起使用,可用于给细胞膜染色,在有机分子组装、膜结构及蛋白质结构域中的电子能量转移中都有应用。
T27794 λ-Cyhalothrin

lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon

Sodium Channel; Parasite Membrane transporter/Ion channel; Microbiology/Virology
λ-Cyhalothrin (Icon) 是广谱的 II 型合成除虫菊酯杀虫剂,含有 α-氰基,用于防治多种害虫。它是一种钠通道神经毒素,靶向中枢神经系统中神经元膜。
TD1006 4-Hydroxyindole

4-Hydroxyindole 是一种芳香杂环化合物,在科学研究和实验室实验中都有广泛的研究。4-Hydroxyindole 以其抗氧化特性而闻名,并已被用于从癌症治疗到神经退行性疾病预防的各种应用中。
T50046 2-(2-amino-3-methylbutanamido)-3-phenylpropanoic acid hydrochloride

Others Others
2-(2-amino-3-methylbutanamido)-3-phenylpropanoic acid hydrochloride 是一种氨基酸类化合物,是谷氨酸的合成类似物,谷氨酸是中枢神经系统中的一种重要神经递质。它已被研究其在各种神经疾病中的潜在治疗应用,包括阿尔茨海默病、帕金森病和癫痫。
T72025 PCSK9-IN-10

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
PCSK9-IN-10 是一种有效的,具有口服活性的PCSK9抑制剂,IC50值为 6.4 µM。PCSK9-IN-10 增加LDLR 蛋白的表达并降低 PCSK9 的表达。PCSK9-IN-10 可减缓动脉粥样硬化进展。PCSK9-IN-10 具有研究高脂血症的潜力。
T9492 3-METHOXY-DL-TYROSINE

Others Others
3-METHOXY-DL-TYROSINE 是一种在人体和许多其他生物体中发现的天然氨基酸,是一种非必需氨基酸。它是神经递质多巴胺的前体,参与大脑中多巴胺水平的调节,在多种疾病中有潜在治疗应用,包括帕金森病、抑郁症和肥胖症。

化合物

α-Cyano-4-hydroxycinnamic acid
Cat.No: T7460
Synonym: α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基
Target: Monocarboxylate transporter
Ferumoxytol
Cat.No: T31786
Synonym: Magnetic Black,Black Iron BM,Magnetic oxide,Black Gold F 89,11557 Black
Target: Others
N-Isopropylacrylamide
Cat.No: T77704
Synonym:
Target: Others
16,17-Epoxy-21-acetoxypregnenolone
Cat.No: T3225
Synonym:
Target: Others
PIPES
Cat.No: T40645
Synonym: 1,4-Piperazinediethanesulfonic acid,1,4-piperazine bis(ethanesulfonic acid),1,4-Piperazinebis(ethanesulfonic acid),PIPES
Target: Others
Flutrimazole
Cat.No: T61148
Synonym:
Target: Antifungal
4-Benzyl-2-carboxymorpholine hydrochloride
Cat.No: T8415
Synonym:
Target: Others
Triethoxyoctylsilane
Cat.No: T19734
Synonym: Oleth-30,正辛基三乙氧基硅烷,NSC 42964,Triethoxycaprylylsilane
Target: Others
Ibafloxacine
Cat.No: T12649
Synonym: S25930,Ibafloxacin,R835
Target: Antifungal
CT52923
Cat.No: T60226
Synonym:
Target: PDGFR
PLGA
Cat.No: T19521
Synonym: poly(lactic-co-glycolic acid),聚乳酸-羟基乙酸共聚物
Target: Others
RDR03785
Cat.No: T9981
Synonym:
Target: Others
NSC 80538
Cat.No: T4178
Synonym:
Target: Others
Parbendazole
Cat.No: T6071
Synonym: SKF 29044,帕苯咪唑
Target: Microtubule Associated, Parasite
Bemarituzumab
Cat.No: T76673
Synonym: FPA144
Target: FGFR
5(6)-TAMRA SE
Cat.No: T18898
Synonym: 5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯
Target: Others
SM-7368
Cat.No: T22115
Synonym:
Target: NF-κB
Pyrazinamine
Cat.No: Fr14534
Synonym:
Target:
HBED-CC-tris(tert-butyl ester)
Cat.No: T82236
Synonym:
Target:
Benfluralin
Cat.No: T14527
Synonym:
Target:
Cucurbit[8]uril
Cat.No: T35862
Synonym:
Target: Others
3,7-dimethylocta-2,6-dienyl 5,9,13-trimethyltetradeca-4,8,12-enoate
Cat.No: T7528
Synonym:
Target: Others
K6PC-5
Cat.No: T27710
Synonym: K6PC5,K6PC 5
Target: S1P Receptor
p53-MDM2-IN-1
Cat.No: T72026
Synonym:
Target: Mdm2, p53
AICAR
Cat.No: T1477
Synonym: NSC105823,AICA Riboside,Acadesine,阿卡地新,AICAR (Acadesine)
Target: Mitophagy, YAP, AMPK, Autophagy
2,5-DIBROMO-3,4-DINITROTHIOPHENE
Cat.No: T9404
Synonym:
Target: Others
Tempo
Cat.No: T5363
Synonym: 2,2,6,6-四甲基哌啶氧化物,2,2,6,6-Tetramethylpiperidinooxy
Target: Free radical scavengers, Reactive Oxygen Species, DNA/RNA Synthesis, Mitochondrial Metabolism
JB002
Cat.No: T72023
Synonym:
Target: Myosin
Insulin(cattle)
Cat.No: TP1125
Synonym: 牛胰岛素,Insulin from bovine pancreas,胰岛素
Target: IGF-1R
(S,R,S)-AHPC-C10-NH2
Cat.No: T17881
Synonym: VH032-C10-NH2
Target: Others, Ligand for E3 Ligase
2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine
Cat.No: T50089
Synonym:
Target: Others
BI 1015550
Cat.No: T72031
Synonym:
Target: PDE
Octyl-beta-D-glucopyranoside
Cat.No: T64321
Synonym: Octyl glucoside,11β-HSD1-IN-11
Target: Others
TGFβRI-IN-3
Cat.No: T9523
Synonym:
Target: TGF-beta/Smad
Burfiralimab
Cat.No: T76937
Synonym:
Target:
TAT
Cat.No: TP1809
Synonym:
Target: HIV Protease
Vialinin A
Cat.No: T22168
Synonym: Terrestrin A
Target: DUB
Neotame
Cat.No: T33639
Synonym: NC 00723,HSDB 7965,NC-00723,NC00723,纽甜
Target: Others
Bupirimate
Cat.No: T21142
Synonym: Nimrod
Target: Antifungal
MSDC-0602K
Cat.No: T38715
Synonym: MSDC-0602K,Azemiglitazone potassium
Target: PPAR
3-(3,6-dichloro-9H-carbazol-9-yl)propanoic acid
Cat.No: T50021
Synonym:
Target: Others
BODIPY 505/515
Cat.No: T36958
Synonym:
Target:
Methyl Blue
Cat.No: T19027
Synonym:
Target: Others
BODIPY 493/503
Cat.No: T36957
Synonym: BDP 493/503 lipid stain,Pyrromethene 546
Target: Others
Octadecyl Rhodamine B chloride
Cat.No: T72083
Synonym:
Target:
λ-Cyhalothrin
Cat.No: T27794
Synonym: lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon
Target: Sodium Channel, Parasite
4-Hydroxyindole
Cat.No: TD1006
Synonym:
Target:
2-(2-amino-3-methylbutanamido)-3-phenylpropanoic acid hydrochloride
Cat.No: T50046
Synonym:
Target: Others
PCSK9-IN-10
Cat.No: T72025
Synonym:
Target: Serine/threonin kinase
3-METHOXY-DL-TYROSINE
Cat.No: T9492
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T4741 N-Formylglycine

Others; Endogenous Metabolite Metabolism; Others
N-Formylglycine 是内源性代谢产物的一种。
T2P2898 Neodiosmin

新地奥斯明,Diosmetin-7-neohesperidoside,新地奥司明,Diosmetin-7-O-neohesperidoside

Antioxidant oxidation-reduction
Neodiosmin (Diosmetin-7-O-neohesperidoside) 是一种黄酮苷,分离自柑桔叶中。
T3018 Protocatechualdehyde

Protocatechuic aldehyde,3,4-Dihydroxybenzaldehyde,Rancinamycin IV,Catechaldehyde,原儿茶醛

Reactive Oxygen Species; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Protocatechualdehyde (3,4-Dihydroxybenzaldehyde), a natural polyphenol compound derived from radix Salviae Miltiorrhizae roots, exhibits diverse biological activities and finds extensive medicinal applications as an antioxidant, anti-aging, antibacterial, and anti-inflammatory agent.
T9780 3,4, 5-trimethoxyphenylacetic acid

Endogenous Metabolite Metabolism
3,4, 5-trimethoxyphenylacetic acid 是有机合成中常见的中间体,其主要用途是将其羧基转化为相应的用途。
T5664 Bovine Serum Albumin

牛血清白蛋白,BSA,Bovine albumin,Albumin bovine serum,白蛋白

Others Others
Bovine Serum Albumin (BSA) 是一种由三个同源全 α 结构域组成的 583 个氨基酸的蛋白质,是一种球状蛋白,可用于多种生物化学实验中。
T3313 D-Luciferin

Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin

Others Others
D-Luciferin (D-(-)-Luciferin) 是一种萤光素酶的底物,能够催化生物发光昆虫产生典型的黄绿光。
T7520 Deoxycytidine triphosphate

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Deoxycytidine triphosphate 是一种核苷三磷酸,是合成 DNA 的原料,可用于实时荧光定量 PCR、cDNA 合成和 DNA 测序。
TN7029 (2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol

Others Others
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol 是一种有用的研究化合物,适用于许多研究应用,包括化学领域和生命科学领域等。
T4842 1H-pyrazole

1,2-Diazole,Pyrazole,吡唑

Others; Endogenous Metabolite Metabolism; Others
1H-pyrazole (1,2-Diazole) 是内源性代谢产物的一种。
T7916 4-Acetamidobenzenesulfonyl azide

Others Others
4-Acetamidobenzenesulfonyl azide 用于各种科学研究应用,包括药物、肽和其他生物活性分子的合成,也被用作聚合反应和聚合物合成中的催化剂。
T4781 N-Acetyl-L-phenylalanine

N-Ac-Phenylalanine,N-乙酰-L-苯丙氨酸

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-phenylalanine (N-Ac-Phenylalanine) 是一种大肠杆菌中的主要酰基氨基酸,由 L-苯丙氨酸和乙酰辅酶 A 合成。
T8279 Isobornyl acetate

Others Others
Isobornyl acetate 是一种从柠檬草植物精油中提取的天然产物,属于双环单萜。它被用于多种应用,包括作为调味剂、香料成分和药物成分。
T4840 3-Hydroxybenzoic acid

Others; Endogenous Metabolite Metabolism; Others
3-Hydroxybenzoic acid 是内源性代谢产物的一种。
T16223 N-Dodecyl-β-D-maltoside

十二烷基-β-D-麦芽糖苷,Lauryl Maltoside

Others Others
N-Dodecyl-β-D-maltoside (Lauryl Maltoside) 是一种芘 (Py) 的衍生物。它可用作烷基吡喃麦芽糖苷清洁剂,尤其是在转运蛋白和呼吸复合物中。它已用于诸如 RNA 聚合酶的纯化和稳定化,以及蛋白质-脂质相互作用的检测的应用中。
T0332 D-Sorbitol

山梨醇,Glucitol,Sorbitol,D-Glucitol

Others; Endogenous Metabolite Metabolism; Others
D-Sorbitol (Sorbitol) 是一种六碳糖醇,能够用作糖的替代品。D-Sorbitol 能够用作稳定的赋形剂和/或等渗剂,保湿剂,增稠剂,甜味剂和膳食补充剂。
T5619 (±)-1,2-Propanediol

1,2-Propanediol,Propylene glycol,1,2-Dihydroxypropane,Methyl ethyl glycol,丙二醇

Others Others
(±)-1,2-Propanediol 是一种脂肪族醇,具有多种作用,可作为防腐剂和防冻剂,在食品工业和护肤品行业应用广泛。 (±)-1,2-Propanediol 是一种天然抑菌剂,能够在一定程度上抑制细菌的生长和繁殖
T4429 Rauwolscine hydrochloride

Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。
TN1448 (-)-Bornyl acetate

L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯

p38 MAPK; NF-κB; JNK; Antifungal MAPK; Microbiology/Virology; NF-κB
(-)-Bornyl acetate (L-(-)-Bornyl acetate) 是存在于牛膝草油中的一种具有抗真菌活性的 (+)-Bornyl acetate 低活性异构体。
TMM2618 Gibberllin A7

Gibberellin A7,Gibberllin 7,赤霉素GA7

Others Others
Gibberllin A7 (Gibberllin 7) 是重要的植物生长激素,可促进植物细胞生长和伸长。它可促进茎和根的快速生长,诱导有丝分裂并启动(打破休眠)并提高种子发芽率。它还参与诸如作为向地力、张力和花卉展示。Gibberellin A3(G1025, G7645) 和 A4 (G7276) 可用作植物生长培养基如 Murashige 和 Skoog 培养基的补充剂。 A3 和 A4 或 Gebberellins 组合的具体作用应在具体的植物应用中确定。
T6S1559 Aurantio-obtusin

Others Others
Aurantio-obtusin 是从决明子中分离出的蒽醌类化合物,具有抗炎、抗凝血、抗氧化、抗高血压的活性。它能抑制 IgE 介导的肥大细胞和过敏模型中的过敏反应,具有研究过敏相关疾病的潜力。在大鼠中,它通过内皮细胞 PI3K/AKT/ eNOS 依赖信号通路放松全身动脉,是潜在的新型血管扩张剂。
T5136 Kongensin A

Kongensin A is an effective heat shock protein 90 (HSP90) inhibitor that has potential anti-necroptosis and anti-inflammation applications.
T40733 Kakkanin

Kakkanin, a compound extracted from the roots of O. henryi, holds potential for anti-inflammatory research applications.
T21027 Guar gum

Guaran,Gum cyamopsis,Gum guar,Guar flour

Guar gum is a galactomannan polysaccharide extracted from guar beans, it has stabilizing and thickening properties useful in food, feed, and industrial applications.
T81248 Rubriflorin B

Rubriflorin B为木脂素类化合物,原自Schisandra rubriflora分离得到。
T82001 Justin C

Justin C (compound 14),一种从Justicia procumbens分离得到的天然产物,主要应用于癌症研究领域。
T82301 Gluconapin potassium

Gluconapin potassium为萝卜硫素前体,后者为一抗癌效能显著的异硫氰酸酯。
T80688 β-Patchoulene

β-Patchoulene, 一种三环倍半萜类化合物,源自广藿香油,主要应用于炎症性疾病治疗。
T40578 β-Bisabolene

β-Bisabolene is a sesquiterpene isolated from opoponax ( Commiphora guidotti ). β-Bisabolene, an anti-cancer agent , can be used for the study of breast cancer.
TN3285 8-Hydroxypinoresinol

AChR Neuroscience
8-Hydroxypinoresinol has antioxidant activity,it and phillygenin significantly reduce the cell injury by 3-morpholinosydnonimine (SIN-1), a ONOO- generator, may be useful for the therapeutic or preventive applications in treating ONOO--related diseases.
T81975 Kopsininic acid

Kopsininic acid, 源自Kopsia hainanensis的天然产物,主要用于类风湿性关节炎、咽炎、扁桃体炎和水肿的研究。
T79968 Coumarinic acid

Coumarinic acid为具有脑穿透性的双重功能抑制剂,能够抑制AChE和β-amyloid,适用于开发治疗阿尔茨海默病的药物研究。
T78501 Glucoamylase

葡萄糖淀粉酶(Glucoamylase)是源于植物、动物和微生物的工业用酶,主要应用于淀粉糖化、酿酒及蒸馏产业。
T81701 Nardoguaianone K

10-epi-Nardoguaianone J

Nardoguaianone K,一种从Nardostachys chinensis根中分离得到的愈创木脂类化合物,用于胰腺癌研究。
T80702 α-Thevetin B

α-Thevetin B(Compound 24), 一种从Thevetia peruviana分离得到的心脏苷,用于肺癌、胃癌和胰腺癌的研究。
T80680 γ-Isofagarine

Iso-γ-fagarine

Isofagarine (Iso-γ-fagarine) 为一生物碱,源自Dictamnus angustifolius根皮。该化合物参与风湿、出血、瘙痒、黄疸、慢性肝炎和皮肤病等病态研究。
T81584 Oxyresveratrol 4-O-β-D-glucopyranoside

Oxyresveratrol 4-O-β-D-glucopyranoside (化合物 3),一种从Morus atropurpurea根皮分离的天然产物,具有研究治疗糖尿病、关节炎、风湿、咳嗽及头痛的潜力。
TN3882 Dodoviscin A

cAMP; Tyrosinase; transporter GPCR/G Protein; Metabolism; Proteases/Proteasome
Dodoviscin A may be a new promising pigmentation-altering agent for cosmetic and therapeutic applications, it can inhibit melanin biosynthesis induced by 3-isobutyl-1-methylxanthine and PD98059.Dodoviscin A can promote adipocyte differentiation as charact
T79933 (−)-N-Hydroxyapiosporamide

NHAP

NF-κB NF-κB
(−)-N-Hydroxyapiosporamide (NHAP)为生物碱类NF-κB抑制剂,表现出体外及体内抗肿瘤活性,常用于结直肠癌(CRC)研究。
T75622 β-Apopicropodophyllin

β-Apopicropodophyllin 是一种天然产物,可以从Hyptis wticillata 中分离得到。β-Apopicropodophyllin 通过诱导微管破坏、DNA 损伤、细胞周期停滞和 ER 应激来诱导细胞凋亡。β-Apopicropodophyllin 可用于癌症研究。
T80008 Stevisaliosides D

Phosphatase Metabolism
Stevisaliosides D (Compound 5) 是从甜叶菊根中提取的化合物,具有抑制PTP1B的活性(IC50:31.8 μM),应用于抗糖尿病研究。
T75514 Blestrin D

Blestrin D,作为一种丁酰胆碱酯酶(BChE)的有效混合型抑制剂,具有8.1 μM的IC50值,可从白芨(Bletilla striata)中分离提取,适用于阿尔兹海默症(AD)研究。
T75425 Synephrine hemitartrate

Synephrine (Oxedrine) hemitartrate,一种生物碱,是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂。Synephrine hemitartrate 是一种拟交感神经化合物,可用于减肥。
T4735 2'-Deoxyuridine 5'-monophosphate disodium

2'-脱氧尿苷-5'-单磷酸二钠,2'-dUMP⋅2Na,2-脱氧尿嘧啶核苷-5'-单磷酸二钠盐,2'-Deoxyuridine 5'-monophosphate disodium salt

Others; Endogenous Metabolite Metabolism; Others
2'-Deoxyuridine 5'-monophosphate disodium (2'-dUMP⋅2Na) salt 能够被双底物酶胸苷酸合酶(TS) 还原甲基化为 dTMP (2'-deoxythymidine 5'-monophosphate)。其中 dTMP 是 DNA 合成所需的核苷酸。
T83411 2,3,4,6,8-Pentahydroxy-1-methylxanthone

2,3,4,6,8-Pentahydroxy-1-methylxanthone,一种源自Wardomyces anomalus的山酮衍生物,展示了显著的抗氧化活性,并作为p56lck酪氨酸激酶的抑制剂发挥作用。它在心血管疾病治疗研究中具备潜在应用价值。
T75704 Isoharringtonine

Isoharringtonine,一种从Cephalotaxus koreanaNakai 纯化得到的天然生物碱,具有抑制癌细胞增殖和迁移的能力,同时能诱导癌细胞(apoptosis)。该化合物在癌症研究中应用。
T82754 Celangulatin D

Celangulatin D (Compound 2),一种从南蛇藤根皮中分离出的倍半萜多元醇酯类化合物,具备对粘虫的显著杀虫活性。该化合物亦适用于杀虫剂和抗肿瘤研究领域。
T29607 Acid Red 88

11391 Red,Eniacid Fast Red A,Peony,Red No. 506

Acid red 88 is an anionic dye with potentially useful photocatalytic research applications. Acid red 88 has been used to determine the effect of Au deposition on ZnO photocatalytic activity under visible light. Additionally, the photocatalyst Au-TiO2 was
T83323 4-Chloro-3-methoxy-5-methylphenyl 6-O-(6-deoxy-β-L-mannopyranosyl)-β-D-glucopyranoside

化合物3(4-Chloro-3-methoxy-5-methylphenyl 6-O-(6-deoxy-β-L-mannopyranosyl)-β-D-glucopyranoside)是一种从Lilium regale提取的抗癌天然产物,具有显著抑制肺癌A549细胞增殖的活性,显示出其研究癌症治疗潜力。
T79948 Kadsurenin B

Kadsurenin B为PAF(platelet-activating factor)拮抗剂,展现出神经保护作用。该化合物在药理学领域显示出广泛的研究潜力,包括抗菌、抗炎、神经保护、抗氧化、抗血小板聚集、细胞毒性和抗寄生虫等效能。
T82764 Cd1a

β-TRTX-cd1a,β-Theraphotoxin-cd1a

Cd1a是从非洲蜘蛛Ceratogyrus darlingi中提取的β-毒素,具有调节钙离子通道的功能。它能够抑制人类的钙离子通道(Cav2.2)(IC50 2.6 μM)以及小鼠的钠离子通道(Nav1.7),有望用于开发治疗外周疼痛的药物。
------------------------ 更多 ------------------------

天然产物

N-Formylglycine
Cat.No: T4741
Synonym:
Target: Others, Endogenous Metabolite
Neodiosmin
Cat.No: T2P2898
Synonym: 新地奥斯明,Diosmetin-7-neohesperidoside,新地奥司明,Diosmetin-7-O-neohesperidoside
Target: Antioxidant
Protocatechualdehyde
Cat.No: T3018
Synonym: Protocatechuic aldehyde,3,4-Dihydroxybenzaldehyde,Rancinamycin IV,Catechaldehyde,原儿茶醛
Target: Reactive Oxygen Species, Antibacterial
3,4, 5-trimethoxyphenylacetic acid
Cat.No: T9780
Synonym:
Target: Endogenous Metabolite
Bovine Serum Albumin
Cat.No: T5664
Synonym: 牛血清白蛋白,BSA,Bovine albumin,Albumin bovine serum,白蛋白
Target: Others
D-Luciferin
Cat.No: T3313
Synonym: Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin
Target: Others
Deoxycytidine triphosphate
Cat.No: T7520
Synonym:
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, Endogenous Metabolite
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol
Cat.No: TN7029
Synonym:
Target: Others
1H-pyrazole
Cat.No: T4842
Synonym: 1,2-Diazole,Pyrazole,吡唑
Target: Others, Endogenous Metabolite
4-Acetamidobenzenesulfonyl azide
Cat.No: T7916
Synonym:
Target: Others
N-Acetyl-L-phenylalanine
Cat.No: T4781
Synonym: N-Ac-Phenylalanine,N-乙酰-L-苯丙氨酸
Target: Others, Endogenous Metabolite
Isobornyl acetate
Cat.No: T8279
Synonym:
Target: Others
3-Hydroxybenzoic acid
Cat.No: T4840
Synonym:
Target: Others, Endogenous Metabolite
N-Dodecyl-β-D-maltoside
Cat.No: T16223
Synonym: 十二烷基-β-D-麦芽糖苷,Lauryl Maltoside
Target: Others
D-Sorbitol
Cat.No: T0332
Synonym: 山梨醇,Glucitol,Sorbitol,D-Glucitol
Target: Others, Endogenous Metabolite
(±)-1,2-Propanediol
Cat.No: T5619
Synonym: 1,2-Propanediol,Propylene glycol,1,2-Dihydroxypropane,Methyl ethyl glycol,丙二醇
Target: Others
Rauwolscine hydrochloride
Cat.No: T4429
Synonym: Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
(-)-Bornyl acetate
Cat.No: TN1448
Synonym: L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯
Target: p38 MAPK, NF-κB, JNK, Antifungal
Gibberllin A7
Cat.No: TMM2618
Synonym: Gibberellin A7,Gibberllin 7,赤霉素GA7
Target: Others
Aurantio-obtusin
Cat.No: T6S1559
Synonym:
Target: Others
Kongensin A
Cat.No: T5136
Synonym:
Target:
Kakkanin
Cat.No: T40733
Synonym:
Target:
Guar gum
Cat.No: T21027
Synonym: Guaran,Gum cyamopsis,Gum guar,Guar flour
Target:
Rubriflorin B
Cat.No: T81248
Synonym:
Target:
Justin C
Cat.No: T82001
Synonym:
Target:
Gluconapin potassium
Cat.No: T82301
Synonym:
Target:
β-Patchoulene
Cat.No: T80688
Synonym:
Target:
β-Bisabolene
Cat.No: T40578
Synonym:
Target:
8-Hydroxypinoresinol
Cat.No: TN3285
Synonym:
Target: AChR
Kopsininic acid
Cat.No: T81975
Synonym:
Target:
Coumarinic acid
Cat.No: T79968
Synonym:
Target:
Glucoamylase
Cat.No: T78501
Synonym:
Target:
Nardoguaianone K
Cat.No: T81701
Synonym: 10-epi-Nardoguaianone J
Target:
α-Thevetin B
Cat.No: T80702
Synonym:
Target:
γ-Isofagarine
Cat.No: T80680
Synonym: Iso-γ-fagarine
Target:
Oxyresveratrol 4-O-β-D-glucopyranoside
Cat.No: T81584
Synonym:
Target:
Dodoviscin A
Cat.No: TN3882
Synonym:
Target: cAMP, Tyrosinase, transporter
(−)-N-Hydroxyapiosporamide
Cat.No: T79933
Synonym: NHAP
Target: NF-κB
β-Apopicropodophyllin
Cat.No: T75622
Synonym:
Target:
Stevisaliosides D
Cat.No: T80008
Synonym:
Target: Phosphatase
Blestrin D
Cat.No: T75514
Synonym:
Target:
Synephrine hemitartrate
Cat.No: T75425
Synonym:
Target:
2'-Deoxyuridine 5'-monophosphate disodium
Cat.No: T4735
Synonym: 2'-脱氧尿苷-5'-单磷酸二钠,2'-dUMP⋅2Na,2-脱氧尿嘧啶核苷-5'-单磷酸二钠盐,2'-Deoxyuridine 5'-monophosphate disodium salt
Target: Others, Endogenous Metabolite
2,3,4,6,8-Pentahydroxy-1-methylxanthone
Cat.No: T83411
Synonym:
Target:
Isoharringtonine
Cat.No: T75704
Synonym:
Target:
Celangulatin D
Cat.No: T82754
Synonym:
Target:
Acid Red 88
Cat.No: T29607
Synonym: 11391 Red,Eniacid Fast Red A,Peony,Red No. 506
Target:
4-Chloro-3-methoxy-5-methylphenyl 6-O-(6-deoxy-β-L-mannopyranosyl)-β-D-glucopyranoside
Cat.No: T83323
Synonym:
Target:
Kadsurenin B
Cat.No: T79948
Synonym:
Target:
Cd1a
Cat.No: T82764
Synonym: β-TRTX-cd1a,β-Theraphotoxin-cd1a
Target:
--------- 更多 ---------
共530条,每页50条 1 2 3 4 5 6 7 8 9 10 11
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼