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50

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T9911 Tocilizumab

Interleukin Immunology/Inflammation
Tocilizumab 是抗人白细胞介素-6 受体 (IL-6R) 的中和抗体,能够阻碍 IL-6 与 IL-6R 的结合,进而抑制经典和反式信号。它可用于研究类风湿性关节炎,对重症 COVID-19 冠状病毒病方面的研究具有显著效果。
T1421 Aceclofenac

醋氯芬酸,Preservex,Airtal

COX Immunology/Inflammation; Neuroscience
Aceclofenac (Preservex) 是一种可口服的非甾体抗炎药,可用于缓解疼痛、骨关节炎、强直性脊柱炎、类风湿性关节炎的研究。
T11699 J-113863

CCR Immunology/Inflammation; Microbiology/Virology
J-113863 是选择性的 CCR1 (CD18)拮抗剂,有抗炎作用,对人和小鼠 CCR1受体的 IC50值分别为 0.9 和 5.8 nM。它是人 CCR3的强效拮抗剂,还是小鼠 CCR3的弱效拮抗剂,IC50分别为 0.58 和 460 nM。
T0291 Flurbiprofen

氟比洛芬,dl-Flurbiprofen

Apoptosis; COX; MRP Apoptosis; Immunology/Inflammation; Neuroscience
Flurbiprofen (dl-Flurbiprofen) 是一种高效的,具有口服活性的非甾体抗炎化合物,有退热止痛活性, 常用于炎症性疾病的研究。它是一种非选择性的环氧合酶抑制剂,可研究结肠癌。
T4561 Tiaprofenic acid

Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam

Others; COX Immunology/Inflammation; Neuroscience; Others
Tiaprofenic acid (Acido tiaprofenico) 是可口服的非甾体抗炎药,通过抑制环氧化酶抑制前列腺素合成,可用于风湿性疾病的研究。
T60012 HS-243

IRAK; MAPK; CDK Cell Cycle/Checkpoint; Immunology/Inflammation; MAPK; NF-κB
HS-243 是 IRAK-4 和 IRAK-1 的抑制剂,IC50 分别为 20 和 24 nM。 HS-243 显示出抗炎和抗癌活性。
T20168 Aurothiomalate sodium

金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate

Others; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Others
Aurothiomalate sodium (Miochrysin) 是一种选择性的致癌 PKCι信号传导抑制剂,可抑制肿瘤细胞增殖。它是一种硫氧还蛋白还原酶 (TrxR) 抑制剂,也是一种抗风湿剂。
T15253 CCX354

CCR1 antagonist 1,CCX-354,CCX 354

CCR Immunology/Inflammation; Microbiology/Virology
CCX354 (CCR1 antagonist 1) 是一种有效的小分子 CCR1 拮抗剂,具有抗炎活性,可用于治疗类风湿关节炎。
T19641 Epirizole

DA 398,Mepirizole,DA398,Mebron,Methopyrimazole,Dalex,DA-398

Others Others
Epirizole (Mebron) 具有解热、镇痛和抗炎活性,可用于慢性类风湿性关节炎的研究。
T76711 Golimumab

MK-8259,SCH 900259,CNTO-148

TNF Apoptosis
Golimumab (CNTO-148) 是一种有效的人源化抗 TNFα IgG1κ单克隆抗体 。Golimumab 具有抗炎和抗癌活性,对 IL-6 和 IL-1β 的产生有抑制作用,可诱导细胞凋亡。Golimumab 可用来预防炎症发生和软骨或骨骼的破坏,可用于研究类风湿性关节炎和癌症。
T76937 Burfiralimab

hzVSF-v13

HBV Microbiology/Virology
Burfiralimab (hzVSF-v13) 是一种针对波形蛋白的单克隆免疫球蛋白(IgG4),具有抗HBV作用,可用于研究类风湿关节炎。
T27312 Fentiazac

Donorest,Flogene,BR-700

Others Others
Fentiazac(BR-700) 是一种口服活性的非甾体烷酸衍生物,具有显著的镇痛、抗炎和解热活性。Fentiazac 可用于研究类风湿关节炎、骨关节炎、牙周炎和肌腱炎等炎症性疾病。
T0693 Niflumic acid

氟尼酸,Nifluril,Forenol,Landruma

Others; Phospholipase; Chloride channel; COX; Monocarboxylate transporter; UGT Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Niflumic acid (Nifluril) 是钙离子激活的氯离子通道阻断剂,用于治疗类风湿性关节炎的镇痛剂和抗炎剂。
T1432 Phenylbutazone

Butazolidine,保泰松

COX Immunology/Inflammation; Neuroscience
Phenylbutazone (Butazolidine) 是是非甾体类抗炎药,前列腺素 H 合酶过氧化物酶的还原辅助因子,可诱导肌肉盲样蛋白 1 表达,有用于强直性脊柱炎的研究潜力。
T22346 Indomethacin sodium hydrate

Indometacin sodium hydrate

COX Immunology/Inflammation; Neuroscience
Indomethacin sodium hydrate (Indometacin sodium hydrate) 是一种口服活性、竞争性和可逆性的 COX1/2 抑制剂,具有潜在的抗炎活性,可诱发的偏头痛,诱导的胃肠道损伤,可用于研究成人继发于严重创伤性脑损伤的颅内压增高和类风湿性关节。
T20763 Betamethasone disodium phosphate

Vista-Methasone,NSC90616,Betamethasone 21-phosphate disodium salt,NSC-90616

Others Others
Betamethasone disodium phosphate (Betamethasone 21-phosphate disodium salt) 是一种具有抗炎活性的皮质类固醇,通过减少促炎细胞因子的分泌促进 M1 至 M2 巨噬细胞极化,可用于研究瘢痕疙瘩和类风湿性关节炎。
T77093 Theralizumab

TGN1412,TAB-08,TABO8

Others Others
Theralizumab (TGN1412) 是一种抗靶向 CD28 的单克隆抗体,可直接刺激 T 细胞。Theralizumab 具有抗肿瘤活性,用于治疗 B 细胞慢性淋巴细胞白血病和类风湿性关节炎。
T76741 Eldelumab

BMS-936557,MDX-1100

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
Eldelumab (BMS-936557) 是一种人源化抗 IP-10 IgG 1型单克隆抗体,对 CXCL10 具有抑制作用。Eldelumab 具有抗炎活性,可与 CXCL10 结合,可用于研究类风湿性关节炎。
T0855 (R)-Naproxen

COX Immunology/Inflammation; Neuroscience
(R)-Naproxen 是一种抗炎剂,具有解热和镇痛作用。酸及其钠盐都用于治疗急性痛风或痛经、肌肉骨骼疾病、类风湿性关节炎和其他风湿病。
T2513 VX-702

p38 MAPK; Autophagy Autophagy; MAPK
VX702 是一种高度特异性的 p38α MAPK 抑制剂,对 p38α 的选择性比 p38β 高 14 倍。它是一种小分子研究口服抗细胞因子疗法,用于治疗炎症性疾病,如类风湿性关节炎。
T0219 Valdecoxib

伐地考昔,代他考昔,SC 65872

COX Immunology/Inflammation; Neuroscience
Valdecoxib (SC 65872) 是可口服的高选择性 COX-2抑制剂,对 COX-2 和 COX-1 的 IC50值分别为 5 nM 和 140 μM,可用于治疗骨关节炎、类风湿性关节炎以及痛经和经期症状。
T76781 Itolizumab

EQ-001

Others Others
Itolizumab (Anti-Human CD6 Recombinant Antibody) 是一种人源化针对 CD6 的细胞外 SRCR 远端结构域 1的重组 抗 CD6 单克隆抗体。Itolizumab 可减缓 T 细胞增殖并抑制促炎细胞因子的产生。Itolizumab 可用于研究银屑病、类风湿性关节炎 (RA)和 COVID-19 疾病等多种疾病。
T72505 CTP Synthetase-IN-1

Others Others
CTP Synthetase-IN-1 是一种具有口服活性和高效性的胞苷 5'-三磷酸合成酶 (CTPS) 抑制剂,具有潜在的抗肿瘤活性,在炎症动物模型中显示出抗炎活性,抑制人 CTPS1 和人 CTPS2,可用于研究关节炎和类风湿性关节炎。
T63119 NF-κB/MAPK-IN-1

NF-κB; MAPK MAPK; NF-κB
NF-κB/MAPK-IN-1 是一种有效的 NF-κB 和 MAPK 通路双重抑制剂,具有潜在的抗炎活性,抑制 NO 生成,对 LPS 诱导的iNOS,COX-2,ERΚ和P38激活有抑制作用。 NF-κB/MAPK-IN-1 可用于预防和治疗类风湿关节炎 (RA) 。
T25036 Alclofenac sodium

Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.
T69458 Pirprofen

Pirprofen is an anti-inflammatory agent used in therapy of rheumatoid arthritis and a prostaglandin synthetase inhibitor.
T25035 Alclofenac lysinate

Alclofenac is an anti-inflammatory agent used in the treatment of rheumatoid arthritis. It also used as an analgesic and an antipyretic.
T26710 Azapropazone

DuP-141,NSC-102824,AHR-3018,AHR 3018,MI-85

Azapropazone is anti-inflammatory agent. Azapropazone has uricosuric properties used to treat rheumatoid arthritis and ankylosing spondylitis. Azapropazone lowered plasma uric acid but exerted only a modest and variable uricosuric effect without altering
T77116 Plonmarlimab

Plonmarlimab (TJ003234) 是一种抗GM-CSF 单克隆抗体。Plonmarlimab 可用于类风湿性关节炎和 COVID-19 的研究。
T0184L Fenoprofen

Nalgesic,Fenoprofen Calcium,Nalfon

Fenoprofen is a non-steroidal anti-inflammatory drug used to relieve symptoms of rheumatoid arthritis, osteoarthritis, and mild to moderate pain. It can block the enzyme that produces prostaglandin (cyclooxygenase), resulting in a decrease in the concentr
T77025 Gimsilumab

Gimsilumab 是一种人源化的抗 GM-CSF 单克隆抗体。Gimsilumab 具有研究 COVID-19 和 类风湿性关节炎的潜力。
T76898 Adalimumab beta

Adalimumab beta (ABP-501) 是一种抗 TNF-α单克隆抗体。Adalimumab beta 可用于类风湿性关节炎 (RA) 的研究。
T68563 Piroxicam olamine

Piroxicam olamine is a cyclooxygenase inhibiting, non-steroidal anti-inflammatory agent (NSAID) that is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. Its long half-life enables it to be administered once daily.
T78759 VEGFR2-IN-4

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR2-IN-4(化合物25)为一种针对VEGFR2激酶的有效且选择性抑制剂,其GI50为0.7 nM。该化合物表现出抗血管生成活性,可用于类风湿关节炎研究领域。
T62473 Edecesertib

Edecesertib (GS-5718) 是一种选择性的、口服具有活力的 IRAK-4 抑制剂,表现出抗炎活性。Edecessertib 能够用于研究类风湿性关节炎 (RA) 和红斑狼疮 (LE)。
T68211 Piroxicam betadex

Piroxicam betadex is a nonsteroidal anti-inflammatory drug. The mechanism of action of piroxicam is as a cyclooxygenase Inhibitor. It is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. It is used to reduce pain, swelling, and joint stiffness from arthritis. Reducing these symptoms helps you do more of your normal daily activities.
T80744 Zanolimumab

Anti-Human CD4 Recombinant Antibody

Zanolimumab(Anti-HumanCD4Recombinant Antibody)是靶向CD4的人源单克隆抗体,能有效地抑制T细胞受体(TCR)的信号转导。它在类风湿性关节炎、银屑病、黑色素瘤、皮肤及周围T细胞淋巴瘤的研究中有应用。
T72252 RORγt inverse agonist 14

ROR Metabolism
RORγt inverse agonist 14 (8e) 是一种高效、口服活性及选择性 RORγt 反向激动剂(EC50 为 2.5 nM),具有抗炎作用,主要应用于风湿性关节炎和牛皮癣的研究。
T78012 CCP peptide TFA

CCP peptide TFA是一种合成环状瓜氨酸化肽(CCP),在血清学检测中用作抗CCP抗体的底物,是类风湿关节炎(RA)自身抗体的特异性高靶标。
T76935 Briakinumab

Briakinumab (ABT-874) 是一种全人抗 IL-12/23p40单克隆抗体。Briakinumab 靶向并中和 IL-12和 IL-23。Briakinumab 可用于类风湿性关节炎、炎症性肠病和多发性硬化症的研究。
T62969 PDE4-IN-6

PDE4-IN-6 是一种安全的、有效的、中等选择性的 PDE4 抑制剂,作用于 PDE4B (IC50: 0.125 μM) 和 PDE4D (IC50: 0.43 μM)。PDE4-IN-6 能够下调 TNF-α 和 IL-6 的表达水平,表现出抗炎、抗关节炎作用,并具有强大的免疫调节活性。PDE4-IN-6 具有潜力进行抗类风湿性关节炎的研究。
T81403 Priliximab

cM-T412,CEN 000029

Priliximab (CEN 000029) 是一种针对CD4的人源化单克隆抗体。其与T细胞表面CD4的结合作用可引起循环中CD4+T细胞的显著并持久的减少,适用于类风湿性关节炎 (RA) 研究。
T68297 Dilmapimod tosylate

Dilmapimod tosylate is a potent p38 mitogen-activated protein kinase (MAPK) inhibitor. It was investigated for its anti-inflammatory effect in non-head injury trauma patients at risk for developing acute respiratory distress syndrome. IL-1β was identified as a gene regulated by dilmapimod that could influence c-reactive protein levels. Dilmapimod had been in phase III clinical trials by GlaxoSmithKline for the treatment of rheumatoid arthritis, neuropathic pain, coronary artery disease (CAD) and...
T76878 Vobarilizumab

Vobarilizumab (ALX-0061) 是一种抗 IL-6R 单克隆抗体 (mAb) (Kd: 0.19 pM)。Vobarilizumab 由一个抗 IL-6R 结构域和一个抗人血清白蛋白结构域组成。Vobarilizumab 可用于炎症性自身免疫性疾病的研究,如类风湿性关节炎。
TP1409L CCP peptide acetate

CCP peptide acetate(277748-59-1 Free base)

Others Others
CCP peptide acetate 是合成的环状瓜氨酸化肽 (CCP),可以用作血清学检测抗 CCP 抗体的底物。CCP peptide acetate 可作为自身抗体的靶标,对类风湿关节炎 (RA) 具有高度的特异性。
T73666 Proglumetacin

Proglumetacin 是一种口服有效的环加氧酶 (cyclo-oxygenase) 抑制剂。Proglumetacin 可以抑制 SARS-CoVMpro(新冠病毒的主要蛋白酶),其 AC50为 8.9 μM。Proglumetacin 具有抗炎活性,可用于炎症(如类风湿关节炎、过敏性气囊炎)的研究。
T76786 Cabiralizumab

Cabiralizumab (FPA 008) 是一种抗 CSF1R 单克隆抗体 (MAb)。Cabiralizumab 可增强 T 细胞浸润和抗肿瘤 T 细胞免疫反应。Cabiralizumab 抑制破骨细胞的活化并阻止骨质破坏,可用于类风湿性关节炎 (RA) 的研究。Cabiralizumab 可与 Nivolumab 结合用于肺癌研究。
T79260 MCI

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
MCI具有针对性地清除活性氧(ROS)并降低环氧合酶-2(COX-2)表达的功能,COX-2的IC50值为1.23μM。在胶原诱导的关节炎(CIA)模型中展现出的抗炎效果明显,适用于类风湿性关节炎(RA)的研究。
TMIH-0146 Chloroquine-d5

Chloroquine-d5 是 Chloroquine 的氘代化合物。Chloroquine 的 CAS 号为 54-05-7。Chloroquine 是一种自噬和 Toll 样受体抑制剂。 氯喹是一种抗疟疾和抗炎剂,广泛用于治疗疟疾和类风湿性关节炎。它在体外控制 SARS-CoV-2 (COVID-19) 感染方面非常有效,EC50 为 1.13 μM。
T37606 Resolvin D5

7(S),17(S)-diHDHA

Resolvins are a family of potent lipid mediators derived from both eicosapentaenoic acid and docosahexaenoic acid . [1] In addition to being anti-inflammatory, resolvins promote the resolution of the inflammatory response back to a non-inflamed state.[2] Resolvin D5 (RvD5) is a DHA-derived resolvin generated by a double dioxygenation mechanism.[3] RvD5 has been identified in media from ionophore-stimulated trout brain cells, in human synovial fluid from patients with rheumatoid arthritis, and in...

化合物

Tocilizumab
Cat.No: T9911
Synonym:
Target: Interleukin
Aceclofenac
Cat.No: T1421
Synonym: 醋氯芬酸,Preservex,Airtal
Target: COX
J-113863
Cat.No: T11699
Synonym:
Target: CCR
Flurbiprofen
Cat.No: T0291
Synonym: 氟比洛芬,dl-Flurbiprofen
Target: Apoptosis, COX, MRP
Tiaprofenic acid
Cat.No: T4561
Synonym: Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam
Target: Others, COX
HS-243
Cat.No: T60012
Synonym:
Target: IRAK, MAPK, CDK
Aurothiomalate sodium
Cat.No: T20168
Synonym: 金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate
Target: Others, PKC
CCX354
Cat.No: T15253
Synonym: CCR1 antagonist 1,CCX-354,CCX 354
Target: CCR
Epirizole
Cat.No: T19641
Synonym: DA 398,Mepirizole,DA398,Mebron,Methopyrimazole,Dalex,DA-398
Target: Others
Golimumab
Cat.No: T76711
Synonym: MK-8259,SCH 900259,CNTO-148
Target: TNF
Burfiralimab
Cat.No: T76937
Synonym: hzVSF-v13
Target: HBV
Fentiazac
Cat.No: T27312
Synonym: Donorest,Flogene,BR-700
Target: Others
Niflumic acid
Cat.No: T0693
Synonym: 氟尼酸,Nifluril,Forenol,Landruma
Target: Others, Phospholipase, Chloride channel, COX, Monocarboxylate transporter, UGT
Phenylbutazone
Cat.No: T1432
Synonym: Butazolidine,保泰松
Target: COX
Indomethacin sodium hydrate
Cat.No: T22346
Synonym: Indometacin sodium hydrate
Target: COX
Betamethasone disodium phosphate
Cat.No: T20763
Synonym: Vista-Methasone,NSC90616,Betamethasone 21-phosphate disodium salt,NSC-90616
Target: Others
Theralizumab
Cat.No: T77093
Synonym: TGN1412,TAB-08,TABO8
Target: Others
Eldelumab
Cat.No: T76741
Synonym: BMS-936557,MDX-1100
Target: CXCR
(R)-Naproxen
Cat.No: T0855
Synonym:
Target: COX
VX-702
Cat.No: T2513
Synonym:
Target: p38 MAPK, Autophagy
Valdecoxib
Cat.No: T0219
Synonym: 伐地考昔,代他考昔,SC 65872
Target: COX
Itolizumab
Cat.No: T76781
Synonym: EQ-001
Target: Others
CTP Synthetase-IN-1
Cat.No: T72505
Synonym:
Target: Others
NF-κB/MAPK-IN-1
Cat.No: T63119
Synonym:
Target: NF-κB, MAPK
Alclofenac sodium
Cat.No: T25036
Synonym:
Target:
Pirprofen
Cat.No: T69458
Synonym:
Target:
Alclofenac lysinate
Cat.No: T25035
Synonym:
Target:
Azapropazone
Cat.No: T26710
Synonym: DuP-141,NSC-102824,AHR-3018,AHR 3018,MI-85
Target:
Plonmarlimab
Cat.No: T77116
Synonym:
Target:
Fenoprofen
Cat.No: T0184L
Synonym: Nalgesic,Fenoprofen Calcium,Nalfon
Target:
Gimsilumab
Cat.No: T77025
Synonym:
Target:
Adalimumab beta
Cat.No: T76898
Synonym:
Target:
Piroxicam olamine
Cat.No: T68563
Synonym:
Target:
VEGFR2-IN-4
Cat.No: T78759
Synonym:
Target: VEGFR
Edecesertib
Cat.No: T62473
Synonym:
Target:
Piroxicam betadex
Cat.No: T68211
Synonym:
Target:
Zanolimumab
Cat.No: T80744
Synonym: Anti-Human CD4 Recombinant Antibody
Target:
RORγt inverse agonist 14
Cat.No: T72252
Synonym:
Target: ROR
CCP peptide TFA
Cat.No: T78012
Synonym:
Target:
Briakinumab
Cat.No: T76935
Synonym:
Target:
PDE4-IN-6
Cat.No: T62969
Synonym:
Target:
Priliximab
Cat.No: T81403
Synonym: cM-T412,CEN 000029
Target:
Dilmapimod tosylate
Cat.No: T68297
Synonym:
Target:
Vobarilizumab
Cat.No: T76878
Synonym:
Target:
CCP peptide acetate
Cat.No: TP1409L
Synonym: CCP peptide acetate(277748-59-1 Free base)
Target: Others
Proglumetacin
Cat.No: T73666
Synonym:
Target:
Cabiralizumab
Cat.No: T76786
Synonym:
Target:
MCI
Cat.No: T79260
Synonym:
Target: Reactive Oxygen Species
Chloroquine-d5
Cat.No: TMIH-0146
Synonym:
Target:
Resolvin D5
Cat.No: T37606
Synonym: 7(S),17(S)-diHDHA
Target:
Cat. No. Product Name Target Signaling Pathways
T5029 Oxaceprol

奥沙西罗,N-Acetyl-L-hydroxyproline,N-乙酰-L-4-羟基脯氨酸

Others Others
Oxaceprol (N-Acetyl-L-hydroxyproline) 是一种可口服的、具有显著抗炎作用的 L-脯氨酸衍生物,常用于研究骨关节炎和类风湿性关节炎。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T5S1982 Periplocin

Periplocoside,杠柳毒苷

Apoptosis; Others Apoptosis; Others
Periplocin (Periplocoside) 是从黑龙骨中分离出的一种强心类固醇。它可促进肿瘤细胞凋亡并抑制肿瘤生长。它通过激活 Na/K-ATPase 介导的 Src/ERK 和 PI3K/Akt 途径,具有促进伤口愈合的潜力。
T3662 Eleutheroside E

NF-κB NF-κB
Eleutheroside E 是刺五加的重要成分,具有抗炎,保护缺血心脏的功能。
T6S1784 Brazilin

Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素

Apoptosis; Others; AMPK; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Others; PI3K/Akt/mTOR signaling
Brazilin (Braziletto) 是来自几种热带硬木的心材的一种红色染料前体,有软骨保护和抗炎活性。它抑制细胞增殖,促进细胞凋亡并通过 AMPK/mTOR 途径诱导自噬。
T6S1684 8-Gingerol

Antioxidant; Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology; oxidation-reduction
8-Gingerol 分离自姜的根状茎,是口服有效的 TRPV1激活剂,EC50值为5.0 µM。8-Gingerol 抑制 COX-2,还能抑制体外 H. pylori 的生长。
TN3741 Cyclocurcumin

TNF; ROS Apoptosis; Immunology/Inflammation
Cyclocurcumin, a curcumin derivative, exhibits anticancer, anti-inflammatory, and immune-modulating abilities and is a potential compound for the treatment of rheumatoid arthritis as predicted by the MM-PBSA method. It may have a therapeutic potential as
TN3144 6,4'-Dihydroxy-7-methoxyflavanone

檀木

ERK; IL Receptor; Antioxidant; TNF; NF-κB; MAPK; Prostaglandin Receptor; JNK; Autophagy Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; MAPK; NF-κB; oxidation-reduction
6,4'-Dihydroxy-7-methoxyflavanone 是一种从 Dalbergia odorifera T. Chen (Leguminosae) 的心材中分离出来的生物活性化合物,具有抗氧化、抗炎和神经保护作用。 6,4'-二羟基-7-甲氧基黄烷酮可用于治疗破骨性骨病如骨质疏松症、类风湿性关节炎和牙周病的研究。
T83117 Angeloylbinankadsurin A

Angeloylbinankadsurin A(化合物7)是一种从黑虎胡的EtOAc和CH2Cl2提取物中分离出的抗RA试剂,它在RA-FLS细胞上显示出显著的抑制活性(IC50=11.70 μM),同时对人类癌细胞系(Hela和BGC-823)表现出较低的毒性(IC50分别为19.9 μM和21.93 μM)。

天然产物

Oxaceprol
Cat.No: T5029
Synonym: 奥沙西罗,N-Acetyl-L-hydroxyproline,N-乙酰-L-4-羟基脯氨酸
Target: Others
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Periplocin
Cat.No: T5S1982
Synonym: Periplocoside,杠柳毒苷
Target: Apoptosis, Others
Eleutheroside E
Cat.No: T3662
Synonym:
Target: NF-κB
Brazilin
Cat.No: T6S1784
Synonym: Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素
Target: Apoptosis, Others, AMPK, Autophagy
8-Gingerol
Cat.No: T6S1684
Synonym:
Target: Antioxidant, Antibacterial, TRP/TRPV Channel
Cyclocurcumin
Cat.No: TN3741
Synonym:
Target: TNF, ROS
6,4'-Dihydroxy-7-methoxyflavanone
Cat.No: TN3144
Synonym: 檀木
Target: ERK, IL Receptor, Antioxidant, TNF, NF-κB, MAPK, Prostaglandin Receptor, JNK, Autophagy
Angeloylbinankadsurin A
Cat.No: T83117
Synonym:
Target:
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