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94

抑制剂 & 化合物

114

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP2499 Human IgE Pentapeptide HEPP acetate

Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)

Human IgE Pentapeptide HEPP acetate 是一种五肽,在几种不同体系中均不能产生 IgE 抑制作用,可用于治疗结膜炎。
TP2385 Ige decapeptide

Immunoglobulin E decapeptide

Ige decapeptide is a peptide.
TP2386 Ige octapeptide (497-504)

Ige octapeptide (497-504) is a bioactive chemical.
T32139 Igercine

Ige C-terminal nonapeptide

Igercine is the C-terminal nonapeptide in immunoglobulin E.
T81050 Talizumab

TNX 901,Anti-Human IgE Fc Recombinant Antibody

Talizumab(TNX 901)是一种针对IgE的人源化IgG1型单克隆抗体。
T9926 Omalizumab

Others Others
Omalizumab 是针对人免疫球蛋白 E 的重组人源化单克隆抗体(KD:0.393 nM)。它能够结合人 FcγRIIb 受体(KD:6.37 uM)。它对持续性过敏性哮喘具有潜在的研究价值。
T21688L Cytochrome c - pigeon (88-104) Acetate

Cytochrome c - pigeon (88-104) Acetate (86579-06-8 Free base)

Others Others
Cytochrome c - pigeon (88-104) Acetate (Cytochrome c - pigeon ) 对 COOH 末端序列 88-1041 内的肽具有特异性。
TP1286 Carcinoembryonic Antigen CEA

癌胚抗原

Others Others
Carcinoembryonic Antigen CEA 是一种广谱性肿瘤标志物,是大肠癌组织产生的一种糖蛋白,作为抗原可引起患者的免疫反应。
T13926 Tigemonam

Antibacterial; Antibiotic Microbiology/Virology
Tigemonam 是一种单菌霉素,可以抵抗革兰氏阴性需氧细菌病原体。
T19023 Lucigenin

NSC-151912,L-6868,光泽精

Others Others
Lucigenin (NSC-151912) 是化学发光探针,可用于检测内源性产生的超氧阴离子自由基在细胞的存在。
T1569 Tigecycline

替加环素,GAR-936

ribosome; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Tigecycline (GAR-936) 是甘氨酰环素抗生素,对 Acinetobacter baumannii(A. baumannii) 的 MIC50和 MIC90分别为 1 和 2 mg/L。它对 E. coli(MG1655 菌株) 的平均抑制浓度 (MIC) 约 125 ng/ mL。
T36619 Aligeron

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Aligeron 是一种非选择性的prostaglandin (PG)拮抗剂,对PGF2α和PGE2诱导的猫血压下降有抑制作用,可用于抑制PGF2α诱导的小鼠腹泻和PGE2诱导的大鼠爪水肿。Aligeron 对血管并发症具有抗氧化保护作用。
T12452 Digeranyl bisphosphonate

DGBP

Rho; Ras Cell Cycle/Checkpoint; GPCR/G Protein; MAPK
Digeranyl bisphosphonate (DGBP) 是一种有效的香叶基焦磷酸香叶酯 (GGPP) 合酶抑制剂,对 Rac1 的香叶基焦磷酸化有抑制作用。Digeranyl bisphosphonate 诱导细胞发生自噬却不诱导细胞凋亡。
T78289 Ligelizumab

QGE 031,Anti-IGHE Recombinant Antibody

Ligelizumab (QGE 031)为一种针对慢性自发性荨麻疹研究的人源化高亲和性抗IgE单克隆抗体。
T125156 Schidigerasaponin E1

Schidigerasaponin E1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125156,CAS号为 266998-23-6。
T123909 4-O-Methyldavidigenin

4-O-Methyldavidigenin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123909,CAS号为 93435-21-3。
T33670 Nigrescigenin

Canescegenine,Canescegenin,Sarmentosigenin A

Nigrescigenin is a cardenolide from Parquetina nigrescens.
T125131 25-Acetylcimigenol xyloside

25-Acetylcimigenol xyloside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125131,CAS号为 27994-12-3。
T23753 Arctigenin mustard

AgM

Arctigenin mustard is a tumor-growth inhibiting substance.
T23407 surface antigen (208-215) [Hepatitis B Virus]

Others Others
The nucleocapsid of the hepatitis B virus is covered by an envelope of HBV surface antigen (HBsAg), which has the common, group-specific determinant a. The four major subtypes of HBsAg, adw, adr, ayw and ayr, are generated, and they have been proposed to
T81103 SSA antigenic peptide

SSA antigenic peptide为Sjögren综合征相关抗原A(SSA)的成分,具有免疫活性的短肽链。
T73650 Forigerimod

Forigerimod (IPP-201101) 是一种 CD4T 细胞调节剂。Forigerimod 是 U1 小核核糖核蛋白 70 kDa 的 21 个氨基酸片段,在 Ser140 位点被磷酸化。Forigerimod 可以有效抑制自噬。Forigerimod 可用于系统性红斑狼疮 (SLE) 等自身免疫性疾病的研究。
TP2270 MHC class II antigen (45-57) [Homo sapiens]

Others Others
MHC class II antigen (45-57) [Homo sapiens] is a peptide with the sequence H2N-Asp-Leu-Asp-Lys-Lys-Glu-Thr-Val-Trp-His-Leu-Glu- Glu-OH, MW= 1868.07. MHC (major histocompatibility complex) class II molecules are found only on antigen-presenting cells and l
TP1830L SV40 large T antigen NLS acetate

Others Others
SV40 large T antigen NLS acetate 是从大 T 抗原残基 47 到 55,使蛋白质进入细胞核。
T36060 Digoxigenin Monodigitoxoside

Digoxigenin monodigitoxoside是地高辛的一种Na+/K+ ATPase 抑制剂和强心苷代谢物。
T38315 Penigequinolone A

Penigequinolone A 可由 Penicillium sp., No. 410 产生,具有花粉生长抑制剂作用。
T16323 Nigericin

Others Others
Nigericin is an antibiotic derived from Streptomyces hygroscopicus that acts as a K+/H+ ionophore, promoting K+/H+ exchange across mitochondrial membranes. Nigericin can be an NLRP3 activator that causes the release of IL-1β as a NALP3-dependent manner. N
T31842 Folligen

Folligen is a novel gonadotropin-releasing hormone analog against DMBA-induced tumours in the rat.
T29903 Alpinigenine

Alpinigenine is a papaveraceous alkaloid.
T23459 Tigecycline hydrochloride

Others Others
Tigecycline hydrochloride is a first-in-class, broad-spectrum antibiotic. It also has activity against antibiotic-resistant organisms.
T123856 Apigenin 7,4'-di-O-alloside

Apigenin 7,4'-di-O-alloside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T123856。
T125822 3'-O-Demethylarctigenin

3'-O-Demethylarctigenin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125822。
T126101 Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside

Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126101。
T38613 Tigecycline hydrate

GAR-936 hydrate

Tigecycline hydrate (GAR-936 hydrate) is a broad spectrum glycylcycline antibiotic. Tigecycline hydrate is bacteriostatic, that inhibits protein synthesis by binding to the 30S ribosomal subunit of bacteria and thereby blocking entry of Aminoacyl-tRNA into the A site of the ribosome during prokaryotic translation. Tigecycline hydrate is active against resistant strains of Gram-positive and Gram-negative bacteria .
T125155 Schidigerasaponin F1

Schidigerasaponin F1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125155,CAS号为 266998-42-9。
T125158 Schidigerasaponin A3

Schidigerasaponin A3 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125158,CAS号为 266997-31-3。
T77072 Lorigerlimab

Lorigerlimab (MGD019) 为一种IgG4双特异性双亲和力再靶向抗体 (DART)。该化合物通过阻断PD-1与CTLA-4来提升T细胞反应效率,目前正被应用于转移性去势抵抗性前列腺癌 (mCRPC) 研究中。
T76953 Xeligekimab

Xeligekimab (GR 1501)为一种针对人白细胞介素17A (IL-17A) 的人源化单克隆抗体,可抑制促炎级联反应。
T75279 Tigecycline tetramesylate

Tigecycline tetramesylate (GAR-936 tetramesylate)为一款广谱甘氨酰环素类抗生素,对E. coli (MG1655菌株)展现出约125 ng/mL的平均抑制浓度(MIC)。针对Acinetobacter baumannii (A. baumannii)的MIC50与MIC90分别达到1 mg/L与2 mg/L。
T80552 Prostate Specific Antigen Substrate

Prostate Specific Antigen Substrate为前列腺特异性抗原(PSA)的荧光底物,专用于检测PSA的酶活性。
TP1830 SV40 large T antigen NLS

SV40 large T antigen NLS is from Large T antigen residue 47 to 55, enables protein import into cell nucleus. This peptide is generated from Large T antigen residue 47 to 55.
T81883 MAGE-3 Antigen (167-176) (human)

MAGE-3 Antigen (167-176) (human) 是一个由 MAGE-A3 编码并与 HLA-B44 抗原结合的人类抗原决定簇,包含8个氨基酸的多肽序列。
T79849 Igermetostat

Histone Methyltransferase Chromatin/Epigenetic
Igermetostat为EZH2抑制剂,适用于体内外癌症研究。
T37707 14-Anhydrodigitoxigenin

14-Anhydrodigitoxigenin is a cardenolide and a derivative of digitoxin.1 It reduces the activity of guinea pig heart Na+/K+-ATPase by 15% when used at a concentration of 10 μM.2
T29676 Adynerigenine

Adynerigenin

Adynerigenine is a bioactive chemical.
T126160 Apigenin 7-[rhamnosyl-(1->2)-galacturonide]

Apigenin 7-[rhamnosyl-(1->2)-galacturonide] 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126160。
T125629 Schidigerasaponin A1

Schidigerasaponin A1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125629,CAS号为 167221-10-5。
T129680 Hellebrigenin-3-O-?-glucoside

Hellebrigenin-3-O-?-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T129680。
T40184 Cannabigerolic acid

Cannabigerolic acid (CBGA), a dihydroxybenzoic acid, serves as a biosynthetic precursor for Tetrahydrocannabinolic acid (THCA). It is characterized by its ability to exhibit cyclooxygenase (COX) inhibitory effects.
T34829 Tetrazanbigen

TNBG

Tetrazanbigen is an inducer of S phase arrest and apoptosis in hepatocellular carcinoma QGY-7701.

化合物

Human IgE Pentapeptide HEPP acetate
Cat.No: TP2499
Synonym: Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)
Target:
Ige decapeptide
Cat.No: TP2385
Synonym: Immunoglobulin E decapeptide
Target:
Ige octapeptide (497-504)
Cat.No: TP2386
Synonym:
Target:
Igercine
Cat.No: T32139
Synonym: Ige C-terminal nonapeptide
Target:
Talizumab
Cat.No: T81050
Synonym: TNX 901,Anti-Human IgE Fc Recombinant Antibody
Target:
Omalizumab
Cat.No: T9926
Synonym:
Target: Others
Cytochrome c - pigeon (88-104) Acetate
Cat.No: T21688L
Synonym: Cytochrome c - pigeon (88-104) Acetate (86579-06-8 Free base)
Target: Others
Carcinoembryonic Antigen CEA
Cat.No: TP1286
Synonym: 癌胚抗原
Target: Others
Tigemonam
Cat.No: T13926
Synonym:
Target: Antibacterial, Antibiotic
Lucigenin
Cat.No: T19023
Synonym: NSC-151912,L-6868,光泽精
Target: Others
Tigecycline
Cat.No: T1569
Synonym: 替加环素,GAR-936
Target: ribosome, Antibacterial, Antibiotic, Autophagy
Aligeron
Cat.No: T36619
Synonym:
Target: Prostaglandin Receptor
Digeranyl bisphosphonate
Cat.No: T12452
Synonym: DGBP
Target: Rho, Ras
Ligelizumab
Cat.No: T78289
Synonym: QGE 031,Anti-IGHE Recombinant Antibody
Target:
Schidigerasaponin E1
Cat.No: T125156
Synonym:
Target:
4-O-Methyldavidigenin
Cat.No: T123909
Synonym:
Target:
Nigrescigenin
Cat.No: T33670
Synonym: Canescegenine,Canescegenin,Sarmentosigenin A
Target:
25-Acetylcimigenol xyloside
Cat.No: T125131
Synonym:
Target:
Arctigenin mustard
Cat.No: T23753
Synonym: AgM
Target:
surface antigen (208-215) [Hepatitis B Virus]
Cat.No: T23407
Synonym:
Target: Others
SSA antigenic peptide
Cat.No: T81103
Synonym:
Target:
Forigerimod
Cat.No: T73650
Synonym:
Target:
MHC class II antigen (45-57) [Homo sapiens]
Cat.No: TP2270
Synonym:
Target: Others
SV40 large T antigen NLS acetate
Cat.No: TP1830L
Synonym:
Target: Others
Digoxigenin Monodigitoxoside
Cat.No: T36060
Synonym:
Target:
Penigequinolone A
Cat.No: T38315
Synonym:
Target:
Nigericin
Cat.No: T16323
Synonym:
Target: Others
Folligen
Cat.No: T31842
Synonym:
Target:
Alpinigenine
Cat.No: T29903
Synonym:
Target:
Tigecycline hydrochloride
Cat.No: T23459
Synonym:
Target: Others
Apigenin 7,4'-di-O-alloside
Cat.No: T123856
Synonym:
Target:
3'-O-Demethylarctigenin
Cat.No: T125822
Synonym:
Target:
Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside
Cat.No: T126101
Synonym:
Target:
Tigecycline hydrate
Cat.No: T38613
Synonym: GAR-936 hydrate
Target:
Schidigerasaponin F1
Cat.No: T125155
Synonym:
Target:
Schidigerasaponin A3
Cat.No: T125158
Synonym:
Target:
Lorigerlimab
Cat.No: T77072
Synonym:
Target:
Xeligekimab
Cat.No: T76953
Synonym:
Target:
Tigecycline tetramesylate
Cat.No: T75279
Synonym:
Target:
Prostate Specific Antigen Substrate
Cat.No: T80552
Synonym:
Target:
SV40 large T antigen NLS
Cat.No: TP1830
Synonym:
Target:
MAGE-3 Antigen (167-176) (human)
Cat.No: T81883
Synonym:
Target:
Igermetostat
Cat.No: T79849
Synonym:
Target: Histone Methyltransferase
14-Anhydrodigitoxigenin
Cat.No: T37707
Synonym:
Target:
Adynerigenine
Cat.No: T29676
Synonym: Adynerigenin
Target:
Apigenin 7-[rhamnosyl-(1->2)-galacturonide]
Cat.No: T126160
Synonym:
Target:
Schidigerasaponin A1
Cat.No: T125629
Synonym:
Target:
Hellebrigenin-3-O-?-glucoside
Cat.No: T129680
Synonym:
Target:
Cannabigerolic acid
Cat.No: T40184
Synonym:
Target:
Tetrazanbigen
Cat.No: T34829
Synonym: TNBG
Target:
Cat. No. Product Name Target Signaling Pathways
TN2359 Iristectorigenin B

Iristectrigenin B

Liver X Receptor Metabolism
Iristectorigenin B (Iristectrigenin B) 是一种有效的肝脏 X 受体 (LXR) 调节剂,是从 Belamcanda chinensis 中分离的小分子化合物。Iristectrigenin B 可促进巨噬细胞 RAW 1.1 细胞中 ABCA264 和 ABCG7 的表达。
T5S1526 Apigenin-7-O-(2G-rhamnosyl)gentiobioside

Apigenin 7-O-(2G-rhamnosyl)gentiobioside,芹菜素-7-0-(2G-鼠李糖)龙胆糖苷,Apigenin 7-(2-Rhamnosylgentiobioside),金银花

Others Others
Apigenin-7-O-(2G-rhamnosyl)gentiobioside 是一种黄酮类苷化合物,从Lonicera gracilipes var. glandulosa 中提取得到。
TN1260 3-O-beta-D-Glucopyranosylplatycodigenin

Others Others
3-O-Beta-D-Glucopyranosylplatycodigenin 是分离自桔梗根的一种齐墩果烷型三萜类化合物。它具有抗 HSC-T6 细胞增殖活性,IC50为 13.36 μM。
TN2357 Iristectorigenin A

鸢尾黄酮甲素,鸢尾甲黄素A

Others Others
Iristectorigenin A 是从一种天然异黄酮,分离自B. chinensis 根茎中,具有抗氧化作用。
T3488 Tectorigenin

4',5,7-Trihydroxy-6-methoxyisoflavone,Tectorigenine,鸢尾黄酮,鸢尾黄素

Apoptosis Apoptosis
Tectorigenin (4',5,7-Trihydroxy-6-methoxyisoflavone) 是一种从葛根汤干燥的花中分离出来的植物异黄酮。
T5S1026 Apigenin-7-glucuronide

Apigenin 7-O-glucuronide,芹菜素-7-葡萄糖醛酸

MMP Proteases/Proteasome
Apigenin-7-glucuronide (Apigenin 7-O-glucuronide) 能够抑制基质金属蛋白酶的活性,其对 MMP-3 (IC50:12.87 μM),MMP-8 (IC50:22.39 μM),MMP-9 (IC50:17.52 μM),MMP-13 (IC50:0.27 μM)。
T3862 Irigenin

NF-κB; Integrin Cytoskeletal Signaling; NF-κB
Irigenin 可通过特异性和选择性地阻断 Extra Domain A 域的 C-C 环上α9β1和α4β1整合素结合位点,介导其抗转移作用。可通过增强胃癌细胞中促凋亡分子的表达来敏化 TRAIL 诱导的凋亡,具有抗癌作用。
T2957 Arctigenin

牛蒡苷元,牛蒡子苷元,(-)-Arctigenin

Apoptosis; MMP; Influenza Virus; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。
T5690 7,4'-Di-O-methylapigenin

芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE

Amylase Metabolism
7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) 可能具有抗真菌c.zeyheri 的作用,是一种潜在的抗真菌药物。它还能抑制药物流出泵(IC50 = 51.64μg /毫升)。
TN2353 8-Hydroxyapigenin

Isoscutellarein

Antioxidant; Influenza Virus Microbiology/Virology; oxidation-reduction
8-Hydroxyapigenin (Isoscutellarein) 是从植物黄芩中提取的黄铜类化合物,具有抗炎抗氧和抗流感病毒的活性。
T6S1676 Cimigenoside

Others Others
Cimigenoside 是升麻属中的一种成分。
T0725 Isoliquiritigenin

异甘草素,ISL,Isoliquiritigen,GU17

Apoptosis; Influenza Virus; Reductase; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Metabolism; Microbiology/Virology
Isoliquiritigenin (ISL) 是从光果甘草根中分离得到的一种黄酮类天然产物,具有抗肿瘤的活性。它抑制流感病毒复制,EC50为 24.7 μM,还能抑制 aldose reductase 的活性,IC50值为 320 nM。
TN6735 Bigelovin

Apoptosis; Reactive Oxygen Species; Retinoid Receptor; Autophagy; RAR/RXR  Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Bigelovin 是从海百合中分离得到的一种倍半萜内酯,是选择性视黄素 X 受体 α 激动剂。它通过抑制ROS 的生成来调节 mTOR 信号通路。它诱导凋亡和自噬,有抗肿瘤活性。
TMS0943 Platicodigenin

桔梗皂苷元,Platycodigenin

Others Others
Platicodigenin (Platycodigenin) 是从桔梗中分离出的桔梗素,在体外对 HSC-T6 细胞系具有抗增殖活性。
TN4943 Sanguisorbigenin

地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid

Antibacterial Microbiology/Virology
Sanguisorbigenin (Tomentosolic acid) 抑制耐甲氧西林金黄色葡萄球菌,是一种天然抗菌剂。
T3817 Darutigenol

Others Others
Darutigenol 是一种戊二萜,从Siegesbecikia orientalis L.中分离得到。
T4S0295 Apigenin 7-glucoside

波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Apigenin 7-glucoside (Cosmosiin) 是一种 ROS 清除剂,具有抗增殖、抗氧化作用。
TN1217 2'-O-Methylisoliquiritigenin

Dopamine Receptor; 5-HT Receptor; GABA Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
2'-O-Methylisoliquiritigenin 是从洋甘草中分离出来的一种天然产物,是由 NR 中特异性诱导的酶合成的。它上调 5-HT、NE、DA 和 GABA 途径,对 NE 通路有显著影响。
T3232 Higenamine hydrochloride

Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Higenamine hydrochloride (norcoclaurine HCl) 是一种 β2-AR 激动剂,是用于心力衰竭相关研究的中药乌头的关键成分,具有抗凋亡活性。
T3907 Tenuigenin

Senegenin,Senegin,远志皂苷元

NF-κB; Caspase; Antibacterial Apoptosis; Microbiology/Virology; NF-κB; Proteases/Proteasome
Tenuigenin (Senegenin) 是从中草药远志根中分离出来的主要活性成分,用于中药,具有抗氧化和抗炎活性。它抑制 NF-κB 活化,预防金黄色葡萄球菌诱导的肺炎。
TN1465 Cannabigerol

NOS; 5-HT Receptor; ROS GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cannabigerol 是一种植物大麻素,是一种高亲和力 α2-肾上腺素能受体激动剂、中度亲和力 5-HT1A 受体拮抗剂和低亲和力 CB1/CB2受体拮抗剂。它可降低眼压,有潜力治疗青光眼。
TN2262 Tectorigenin 7-​O-​Xylosyl Glucoside

Tectorigenin 7-O-xylosylglucoside,鸢尾黄素-7-O-木糖葡萄糖苷

Others Others
Tectorigenin 7-​O-​Xylosyl Glucoside (Tectorigenin 7-O-xylosylglucoside) 是一种异黄酮糖苷,取自葛根花中。
T3814 Isorhapontigenin

Isorhapotogenin,异丹叶大黄素

Others; Autophagy Autophagy; Others
Isorhapontigenin (Isorhapotogenin) 是一种从中草药闭苞买麻藤中分离出的膳食多酚,诱导自噬并抑制浸润性膀胱癌的形成,有抗炎作用。
TN7233 Pseudobaptigenin

Psi-baptigenin

Others Others
Pseudobaptigenin (Psi-baptigenin) 是一种异黄酮,是一种黄酮类脂质分子,是在Pterocarpus marsupium、Dalbergia spruceana 中发现的一种天然产品。
TN2107 Protoescigenin

Others Others
Protoescigenin 来自七叶树皂甙混合物,可用作用于选择性保护的探索性化学的底物。
T6S0413 Pectolinarigenin

柳穿鱼黄素,Pectolinaringenin

Others; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience; Others
Pectolinarigenin (Pectolinaringenin) 是 COX-2/5-LOX 的双重抑制剂,可抑制炎症病变中类花生酸的形成,具有抗炎活性。
T3325 Liquiritigenin

4',7-Dihydroxyflavanone,甘草素

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Liquiritigenin (4',7-Dihydroxyflavanone) 是一种黄烷酮,从甘草中分离得到,是高度选择性的雌激素受体β 激动剂,用于活化 ERE tk-Luc 的 EC50值为36.5 nM。
T3776 Rhapontigenin

丹叶大黄素,Protigenin

P450; Antibacterial; Antifungal Metabolism; Microbiology/Virology
Rhapontigenin (Protigenin) 是一种基于机制的选择性细胞色素 P450 1A1 (IC50: 400 nM) 灭活剂。它是一种芳烃羟化酶,可激活作为致癌物质的多环芳烃。它是白藜芦醇的天然类似物,具有抗癌,抗氧化剂,抗真菌和抗菌活性。
TN1082 Apigenin 7-O-malonylglucoside

Apigenin 7-O-(6''-O-malonylglucoside)

Apigenin 7-O-malonylglucoside (Apigenin 7-O-(6''-O-malonylglucoside)) 存在于菊花中,是一种黄酮,也是一种糖苷。
T3092 Nigericin sodium salt

尼日利亚菌素,尼日利亚菌素钠盐

Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。
T2175 Apigenin

C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400

P450; Autophagy Autophagy; Metabolism
Apigenin (NSC 83244) 是从韩信草中提取的一种天然产物,是一种竞争性CYP2C9抑制剂,Ki 为 2 μM。它被用作镇静剂、温和的镇痛剂和安眠药。
T4109 Rhapontigenin 3'-O-glucoside

丹叶大黄素 3'-O-葡萄糖苷,丹叶大黄素-3'-O-葡萄糖苷

Others Others
Rhapontigenin 3'-O-glucoside 是一种 Rhapontigenin 的衍生物,是 P450 1A1 抑制剂,可用于预防癌症。
TMS1743 Salvigenin

MAO; Autophagy; ROS Kinase Autophagy; Metabolism; Neuroscience; Tyrosine Kinase/Adaptors
Salvigenin 是从鼠尾草中发现的一种多酚类天然产物,具有神经保护、抗肿瘤、免疫调节和细胞毒作用。
T3212 Digoxigenin

地谷新配基,异羟基洋地黄毒苷元

Others Others
Digoxigenin, a therapeutic drug belonging to the group of cardiac glycosides, is widely used in the management of congestive heart failure and other cardiac diseases
TN1455 Bryodulcosigenin

Immunology/Inflammation related Immunology/Inflammation
Bryodulcosigenin 是一种 Bryoniadioica 根的提取物,具有抗炎活性。
TN5571 16-O-Acetyldarutigenol

16-O-Acetyldarutigenol是一种天然产物,属于菊科豨莶属,其产品编号为 TN5571,CAS号为 1188282-01-0。16-O-Acetyldarutigenol可用作对照参考。
TN2034 Paeoniflorigenone

Others; Caspase Apoptosis; Others; Proteases/Proteasome
Paeoniflorigenone is a depolarizing neuromuscular blocking agent, being similar to succinylcholine.
TN1618 Erigeroside

Others Others
Erigeroside has the protective effects on cerebral ischemia-reperfusion injury in rat, its ability of anti-oxidation and scavenging oxidation free radical may be one of its protective mechanisms.
T83394 25-O-acetyl-7,8-didehydro-cimigenol-3-O-b-Dxylopyaranoside

25-O-acetyl-7,8-didehydro-cimigenol-3-O-β-D-xylopyranoside 是环阿烷三萜类化合物,可从 Cimicifuga acerina 分离得到。
T82987 Apigenin 7-O-sophoroside

Apigenin 7-O-sophoroside, 一种黄酮苷, 可以分离自Lonicera gracilipes var. glandulosa。
T5S0313 Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside

Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷

Others; TNF Apoptosis; Others
Liquiritin apioside has antioxidant property by inducing glutathione (GSH) biosynthesis via the inhibition of cytokines and protected lung epithelial cells against cigarette smoke-mediated oxidative stress, might be as protective agent against epithelial
TN1728 Hellebrigenin

PARP; Akt; CDK Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Hellebrigenin has anti-hepatoma activities, it induces cell cycle arrest and apoptosis in human hepatocellular carcinoma HepG2 cells through inhibition of Akt. Hellebrigenin exhibites moderate to strong activity against human HL-60, SF-295, MDA-MB-435, and HCT-8 cancer cell strains without hemolysis of mouse erythrocytes.
TN1498 Cimigenol

Others Others
Cimigenol is a potential antitumor compound, combination of it with an autophagy inhibitor may be a valuable strategy for the chemoprevention or treatment of colon cancer. It exerted potent cytotoxic activity against SMMC-7721 (7.87μM) and A-549 (12.16 μM
TN2422 6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide

Others Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide is a natural product from Carthamus tinctorius Linn.
TN1497 Cimigenol-3-one

Others Others
Cimigenol-3-one is a natural product from Calophyllum inophyllum.
T10348 Apigenin-7-diglucuronide

Others Others
Apigenin-7-diglucuronide is a flavonoid glycoside that exists in an assortment of medicinal plants with anti-inflammatory or ant-oxidant activities. It protects retinas against bright light-induced photoreceptor degeneration through the inhibition of reti
T25578 Kigelinone

Kigelinone is a quinone used as an antibacterial and antifungal.
T13638 Deacylmetaplexigenin

Others Others
Deacylmetaplexigenin is a pregnane glycoside isolated from Asclepias incarnate.
T83408 2',3'-Dihydro-2'-hydroxyprotoapigenone

2',3'-Dihydro-2'-hydroxyprotoapigenone 是一种蕨类植物中天然存在的原黄酮化合物。
TN3430 Apigenin 4'-O-rhamnoside

Others Others
Apigenin-4'-O-rhamnosylglucoside can strongly inhibit the classical pathway of the complement system.
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天然产物

Iristectorigenin B
Cat.No: TN2359
Synonym: Iristectrigenin B
Target: Liver X Receptor
Apigenin-7-O-(2G-rhamnosyl)gentiobioside
Cat.No: T5S1526
Synonym: Apigenin 7-O-(2G-rhamnosyl)gentiobioside,芹菜素-7-0-(2G-鼠李糖)龙胆糖苷,Apigenin 7-(2-Rhamnosylgentiobioside),金银花
Target: Others
3-O-beta-D-Glucopyranosylplatycodigenin
Cat.No: TN1260
Synonym:
Target: Others
Iristectorigenin A
Cat.No: TN2357
Synonym: 鸢尾黄酮甲素,鸢尾甲黄素A
Target: Others
Tectorigenin
Cat.No: T3488
Synonym: 4',5,7-Trihydroxy-6-methoxyisoflavone,Tectorigenine,鸢尾黄酮,鸢尾黄素
Target: Apoptosis
Apigenin-7-glucuronide
Cat.No: T5S1026
Synonym: Apigenin 7-O-glucuronide,芹菜素-7-葡萄糖醛酸
Target: MMP
Irigenin
Cat.No: T3862
Synonym:
Target: NF-κB, Integrin
Arctigenin
Cat.No: T2957
Synonym: 牛蒡苷元,牛蒡子苷元,(-)-Arctigenin
Target: Apoptosis, MMP, Influenza Virus, Autophagy
7,4'-Di-O-methylapigenin
Cat.No: T5690
Synonym: 芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE
Target: Amylase
8-Hydroxyapigenin
Cat.No: TN2353
Synonym: Isoscutellarein
Target: Antioxidant, Influenza Virus
Cimigenoside
Cat.No: T6S1676
Synonym:
Target: Others
Isoliquiritigenin
Cat.No: T0725
Synonym: 异甘草素,ISL,Isoliquiritigen,GU17
Target: Apoptosis, Influenza Virus, Reductase, Autophagy
Bigelovin
Cat.No: TN6735
Synonym:
Target: Apoptosis, Reactive Oxygen Species, Retinoid Receptor, Autophagy, RAR/RXR 
Platicodigenin
Cat.No: TMS0943
Synonym: 桔梗皂苷元,Platycodigenin
Target: Others
Sanguisorbigenin
Cat.No: TN4943
Synonym: 地榆皂苷元,Tomentosolic acid,3β-Hydroxyurs-12,19-dien-28-oic acid,19-Dehydroursolic acid,Ursa-12,19-dien-28-oic acid
Target: Antibacterial
Darutigenol
Cat.No: T3817
Synonym:
Target: Others
Apigenin 7-glucoside
Cat.No: T4S0295
Synonym: 波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin
Target: Reactive Oxygen Species, HIV Protease
2'-O-Methylisoliquiritigenin
Cat.No: TN1217
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, GABA Receptor
Higenamine hydrochloride
Cat.No: T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Tenuigenin
Cat.No: T3907
Synonym: Senegenin,Senegin,远志皂苷元
Target: NF-κB, Caspase, Antibacterial
Cannabigerol
Cat.No: TN1465
Synonym:
Target: NOS, 5-HT Receptor, ROS
Tectorigenin 7-​O-​Xylosyl Glucoside
Cat.No: TN2262
Synonym: Tectorigenin 7-O-xylosylglucoside,鸢尾黄素-7-O-木糖葡萄糖苷
Target: Others
Isorhapontigenin
Cat.No: T3814
Synonym: Isorhapotogenin,异丹叶大黄素
Target: Others, Autophagy
Pseudobaptigenin
Cat.No: TN7233
Synonym: Psi-baptigenin
Target: Others
Protoescigenin
Cat.No: TN2107
Synonym:
Target: Others
Pectolinarigenin
Cat.No: T6S0413
Synonym: 柳穿鱼黄素,Pectolinaringenin
Target: Others, Lipoxygenase, COX
Liquiritigenin
Cat.No: T3325
Synonym: 4',7-Dihydroxyflavanone,甘草素
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Rhapontigenin
Cat.No: T3776
Synonym: 丹叶大黄素,Protigenin
Target: P450, Antibacterial, Antifungal
Apigenin 7-O-malonylglucoside
Cat.No: TN1082
Synonym: Apigenin 7-O-(6''-O-malonylglucoside)
Target:
Nigericin sodium salt
Cat.No: T3092
Synonym: 尼日利亚菌素,尼日利亚菌素钠盐
Target: Potassium Channel, NOD-like Receptor (NLR), Antibacterial, Antibiotic, NOD
Apigenin
Cat.No: T2175
Synonym: C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400
Target: P450, Autophagy
Rhapontigenin 3'-O-glucoside
Cat.No: T4109
Synonym: 丹叶大黄素 3'-O-葡萄糖苷,丹叶大黄素-3'-O-葡萄糖苷
Target: Others
Salvigenin
Cat.No: TMS1743
Synonym:
Target: MAO, Autophagy, ROS Kinase
Digoxigenin
Cat.No: T3212
Synonym: 地谷新配基,异羟基洋地黄毒苷元
Target: Others
Bryodulcosigenin
Cat.No: TN1455
Synonym:
Target: Immunology/Inflammation related
16-O-Acetyldarutigenol
Cat.No: TN5571
Synonym:
Target:
Paeoniflorigenone
Cat.No: TN2034
Synonym:
Target: Others, Caspase
Erigeroside
Cat.No: TN1618
Synonym:
Target: Others
25-O-acetyl-7,8-didehydro-cimigenol-3-O-b-Dxylopyaranoside
Cat.No: T83394
Synonym:
Target:
Apigenin 7-O-sophoroside
Cat.No: T82987
Synonym:
Target:
Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside
Cat.No: T5S0313
Synonym: Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷
Target: Others, TNF
Hellebrigenin
Cat.No: TN1728
Synonym:
Target: PARP, Akt, CDK
Cimigenol
Cat.No: TN1498
Synonym:
Target: Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide
Cat.No: TN2422
Synonym:
Target: Others
Cimigenol-3-one
Cat.No: TN1497
Synonym:
Target: Others
Apigenin-7-diglucuronide
Cat.No: T10348
Synonym:
Target: Others
Kigelinone
Cat.No: T25578
Synonym:
Target:
Deacylmetaplexigenin
Cat.No: T13638
Synonym:
Target: Others
2',3'-Dihydro-2'-hydroxyprotoapigenone
Cat.No: T83408
Synonym:
Target:
Apigenin 4'-O-rhamnoside
Cat.No: TN3430
Synonym:
Target: Others
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