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Targets Recommended: HIF

360

抑制剂 & 化合物

10

天然产物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T19832 Acriflavine Hydrochloride

盐酸吖啶黄,Acriflavine HCl

HIF Angiogenesis; Chromatin/Epigenetic
Acriflavine Hydrochloride (Acriflavine HCl) 是一种 HIF-1α 抑制剂。它通过靶向 HIF-1α 介导的途径并在体外和体内降低 PGK1、VEGF 和 HIF-1α 的水平发挥作用。
T60124 1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea

TNF Apoptosis
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea 是一种能够激动 TNF-α的化合物,可以诱导细胞分泌 TNF-α。
T60231 N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine

Others Others
N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine 是一种生物活性化合物,属于哌嗪类。它是一种重要的合成中间体,用于制备多种药物、农用化学品和其他化学品。它被认为是参与药物代谢的某些酶的抑制剂,例如细胞色素P450酶,也已被证明具有抗炎和抗肿瘤作用。
T0705 Triflusal

三氟柳,三氟醋柳酸,UR1501

COX; PDE; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience
Triflusal (UR1501) 能够利用乙酰化COX-1途径,不可逆地减少血小板中血栓素B2的生成。
T8832 Eledoisin trifluoroacetate (69-25-0 free base)

Eledoisin trifluoroacetate

Others Others
Eledoisin trifluoroacetate (69-25-0 free base) 是从某些小章鱼(Eledone spp.,Mollusca)的后唾液腺中提取或合成获得的肽。它的作用类似于 P 物质的作用;它是一种有效的血管扩张剂,可增加毛细血管的通透性。
T9323 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide

Carbonic Anhydrase Metabolism
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) 是一种碳酸酐酶抑制剂,用作潜在的抗肿瘤和抗青光眼药物。
T77702 4-Chloro-3-(trifluoromethyl)phenyl isocyanate

Others Others
4-Chloro-3-(trifluoromethyl)phenyl isocyanate 是一种生化试剂,可被邻氯三氟甲苯与醋酐通过一系列反应生成。
T9438 2,3,4-Trifluoro-5-Nitro-Benzoic Acid

Others Others
2,3,4-Trifluoro-5-Nitro-Benzoic Acid 是有机合成中有用的中间体。它已被用于研究氟取代对有机分子反应性的影响,还被用于研究硝基取代对有机分子反应性的影响。
T7750 N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea

N-[3,5-双(三氟甲基)苯基]-N′-[(9R)-6′-甲氧基-9-金鸡宁]硫脲

Others Others
N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea 是金鸡纳生物碱衍生的双功能催化剂。
TP1315 c-Myc Peptide Trifluoroacetate

Others Others
c-Myc Peptide Trifluoroacetate (145646-22-6 free base) 是一种合成肽,对应于人类 c-myc 蛋白的 C 末端氨基酸 (410-419),参与调控生长相关基因的转录。
T6813 Cyclo(RGDyK) trifluoroacetate

Cyclo(RGDyK)

Integrin Cytoskeletal Signaling
Cyclo(RGDyK) trifluoroacetate 是一种选择性αVβ3整联蛋白抑制剂,IC50为 20 nM。
T1428 Trifluridine

曲氟尿苷,NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,曲氟胸苷,Viroptic,Trifluridina

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Trifluridine (NSC-75520) 是一种氟化胸苷类似物,具有潜在的抗肿瘤活性,还具有抗病毒活性。它掺入 DNA 并抑制胸苷酸合酶,从而抑制 DNA 合成、抑制蛋白质合成和细胞凋亡。
T1360 4-Nitro-3-trifluoromethyl aniline

Others Others
4-Nitro-3-trifluoromethyl aniline 也被称为5-Amino-2-nitrobenzotrifluoride。
T22424 1-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea

Apoptosis; STAT Apoptosis; JAK/STAT signaling; Stem Cells
SC-1 是一种 Sorafenib 的衍生物,可抑制 STAT3磷酸化,通过依赖 SHP-1 的 STAT3失活诱导细胞凋亡,具有抗癌作用。
T60186 (S)-4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide

Discoidin Domain Receptor (DDR) Tyrosine Kinase/Adaptors
MitoBloCK-6 是一种有效的 Erv1/ALR 抑制剂,IC50 分别为 900 nM 和 700 nM。MitoBloCK-6 还抑制 Erv2 (IC50=1.4 μM)。MitoBloCK-6 可通过细胞色素 c 的释放诱导 hESCs 细胞凋亡。
T9042 Teriflunomide impurity 3

4-Amino-N-(4-trifluoromethylphenyl)benzamide

COX Immunology/Inflammation; Neuroscience
Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) 是一种选择性COX-1抑制剂,IC50为 30 µM。
T3044 (E/Z)-Teriflunomide

Aubagio,HMR-1726,Flucyamide,A77 1726,特立氟胺

Dehydrogenase Metabolism
(E/Z)-Teriflunomide (Aubagio) 是一种可口服的嘧啶合成抑制剂,用于治疗复发性多发性硬化症。
T8389 Trifluoperazine

三氟拉嗪,trifluoroperazine

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine (trifluoroperazine) 是一种多巴胺 D2 受体抑制剂,可治疗精神分裂症。它是NUPR1抑制剂,具有抗癌活性。它是α1-adrenergic 受体拮抗剂,是流感病毒形态发生的可逆抑制剂。
T11486 GSK2807 Trifluoroacetate

Histone Methyltransferase Chromatin/Epigenetic
GSK2807 Trifluoroacetate 是一种选择性和 SAM 竞争性的 SMYD3 抑制剂,IC50为 130 nM,Ki 值为 14 nM。
T0302 Triflupromazine hydrochloride

Neoprin,盐酸三氟丙嗪,Fluopromazine hydrochloride,Fluorofen,Flumazin

Dopamine Receptor; 5-HT Receptor; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Triflupromazine hydrochloride (Fluopromazine hydrochloride) 是一种抗精神病药物,是多巴胺 D1/D2 受体拮抗剂。
T3658 Trifluridine/tipiracil hydrochloride mixture

Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Trifluridine/tipiracil hydrochloride mixture (TAS-102) 是一种新型口服组合药物,含有摩尔比为 2:1 的曲氟尿苷(TFT) 和盐酸替吡嘧啶 (TTP)。它主要通过抑制胸苷酸合酶 (TS) 和掺入 DNA 来显示抗肿瘤活性。
T1222 Trifluoperazine dihydrochloride

Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox

CaMK; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; P-gp; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Trifluoperazine dihydrochloride (SKF5019) 是一种抗精神病药物,靶向中枢多巴胺受体。它是流感病毒形态发生的可逆抑制剂,是NUPR1抑制剂,具有抗癌活性。它是钙调蛋白抑制剂,还可抑制 P-糖蛋白,可研究精神分裂症。
T7455 4-Chloro-2-(trifluoroacetyl)aniline hydrochloride

HIV Protease Microbiology/Virology; Proteases/Proteasome
4-Chloro-2-(trifluoroacetyl)aniline hydrochloride 是 HIV-1 RT(HIV 逆转录酶)的抑制剂。
T4303 4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid

Others Others
4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid 用作医药中间体。
T9367 3-(Trifluoromethyl)benzaldehyde

3-三氟甲基苯甲醛,3-Trifluoromethylbenzaldehyde

Others Others
3-(Trifluoromethyl)benzaldehyde (3-Trifluoromethylbenzaldehyde) 有强烈的甜味,被用作调味剂,香水和化妆品的生产,以及作为中间体合成各种化合物。
T5819 Rapastinel Trifluoroacetate

Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) 是一种 NMDA 受体调节剂,具有甘氨酸位点部分激动剂性质,有研究抑郁症的潜力。
T50107 ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate

Others Others
ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate 是一种合成化合物,属于姜黄素家族。它通过抑制NF-κB 信号通路参与免疫反应和炎症的调节,通过激活Nrf2信号通路参与抗氧化反应的调节,通过抑制Akt 信号通路参与细胞存活和增殖的调节。
T22624L Carcinine ditrifluoroacetate Acetate

β-Alanylhistamine dihydrochloride,Carcinine ditrifluoroacetate Acetate (56897-53-1 Free base),Carcinine dihydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) 是一种 H3 受体拮抗剂。
T10397 ATN-161 trifluoroacetate salt

ATN-161 TFA salt

Integrin Cytoskeletal Signaling
ATN-161 trifluoroacetate salt (ATN-161 TFA salt) 是一种新型整合素 α5β1 拮抗剂,可在小鼠模型中抑制血管生成和肝转移瘤的生长。
T67753 Trifluoromethyl-tubercidin

Influenza Virus Microbiology/Virology
Trifluoromethyl-tubercidin (TFMT)可抑制宿主Mtr1并抑制病毒复制。TFMT 通过其S-adenosyl-l-methionine 结合袋相互作用抑制Mtr1,限制流感病毒复制。TFMT 能有效抑制病毒在小鼠体内的复制,毒性很小。
T5637 Triflumuron

Others Others
Triflumuron 是一种杀虫剂,属于所谓的昆虫生长调节剂。它抑制昆虫幼虫合成甲壳素,导致死亡。
T12851 SB290157 trifluoroacetate

Complement System Immunology/Inflammation
SB290157 trifluoroacetate 是一种选择性 C3a 受体拮抗剂,IC50值为200 nM。
T0309 Ipriflavone

Osteofix,依普黄酮

advanced glycation end products Others
Ipriflavone (Osteofix) 是一种合成异黄酮衍生物,可用于抑制骨吸收。
T9191 XMD-17-51 Trifluoroacetate

XMD-17-51 Trifluoroacetate (1628614-50-5 free base)

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
XMD-17-51 Trifluoroacetate 是可调控蛋白激酶的嘧啶-安定酮化合物。
T67966 Triflubazam

Triflubazam 具有广泛的生物活性,可影响睡眠,可用于治疗焦虑综合征和心理疾病。
T7783 2-(4-TRIFLUOROMETHYL-PHENYL)-ETHYLAMINE

Others Others
2-(4-TRIFLUOROMETHYL-PHENYL)-ETHYLAMINE 是一种单胺类神经递质,已被研究其调节各种神经递质活性的潜力,包括血清素、多巴胺和去甲肾上腺素,还研究了其作为5-HT2A 受体激动剂的潜力。
T9894 2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate

Others Others
2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate 是一种天然产物,可作为参考标准。
T50011 (2-methylpropyl)({[3-(trifluoromethyl)phenyl]methyl})amine

Others Others
(2-methylpropyl)({[3-(trifluoromethyl)phenyl]methyl})amine 是一种选择性血清素受体激动剂,特异性靶向5-HT2A 和5-HT2C 受体,已被用于研究血清素在各种生理和病理条件下的作用。
T1361 2-Trifluoromethyl thioxanthone

Others Others
2-Trifluoromethyl thioxanthone 是一种淡黄色晶体,分子式 C14H7F3OS。
T7272 2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE

2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T7272,CAS号为 675602-93-4。
Fr12535 2-(Trifluoromethyl)benzimidazole

Compound Fr12535 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12535,CAS号为 312-73-2。
T7534 Teriflunomide

A 77-1726,特立氟胺

Others Others
Teriflunomide (A 77-1726) 是一种来氟米特的活性代谢产物,能够抑制嘧啶合成,有效降低T 细胞和B 细胞增殖,可用于研究类风湿性关节炎。
T50071 5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile

Others Others
5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile 是一种用作分子结构单元的化合物,被认为是 COX-2、5-LOX 等酶的抑制剂,具有多种生化和生理作用,包括抗肿瘤活性、抗炎作用和抗氧化活性。
T7592 Trifloxystrobin

CGA 279202,肟菌酯

Antifungal Microbiology/Virology
Trifloxystrobin (CGA 279202) 是一种杀菌剂,可抑制从甜菜作物中分离出的立枯病菌的生长。对大型水蚤新生儿和胚胎的 EC50 分别为 23.0 μg/L 和 1.7 μg/L。
T64860 3-(Trifluoromethyl)cinnamic acid

3-(3-(Trifluoromethyl)phenyl)acrylic acid

Antibiotic Microbiology/Virology
3-(Trifluoromethyl)cinnamic acid (3-(3-(Trifluoromethyl)phenyl)acrylic acid) 可用于研究耐药性细菌感染。
T50023 ethyl 1-(4-aminophenyl)-5-(trifluoromethyl)-1H-pyrazole-4-carboxylate

Others Others
ethyl 1-(4-aminophenyl)-5-(trifluoromethyl)-1H-pyrazole-4-carboxylate 又称 EAPT,是一种有效的选择性 PDE4抑制剂,调节细胞内环腺苷酸(cAMP)水平。它已被用于多种科研应用,包括 cAMP 介导的信号转导通路的研究,并有潜力作为治疗炎症和免疫相关疾病的药物。
T9728 1-(3,5-Dichloro-4-fluorophenyl)-2,2,2-trifluoroethanone

sarolaner,沙罗拉纳

Others Others
1-(3,5-Dichloro-4-fluorophenyl)-2,2,2-trifluoroethanone (sarolaner) 是 Sarolaner 的中间体。
T18911 Acriflavine

Acriflavinium chloride 3,6-Acridinediamine mix

SARS-CoV; Antibacterial Microbiology/Virology
Acriflavine (Acriflavinium chloride 3,6-Acridinediamine mix) 是木瓜蛋白酶样蛋白酶(PL(pro))抑制剂,是一种用于标记高分子量 RNA 的荧光染料,具有抗菌抗癌活性,抑制 SARS-CoV-2 和其他 β 冠状病毒,可用于研究白血病。
T11991 Mefentrifluconazole

P450; Antifungal Metabolism; Microbiology/Virology
Mefentrifluconazole 是一种有效的、选择性的和具有口服活性的真菌 CYP51 (Kd= 0.5 nM) 抑制剂,但对人芳香酶的抑制活性较低,IC50值为0.92 μM。它是一种新型唑类衍生物,用作农用广谱抗真菌剂。
T1608 ADH-1 trifluoroacetate

Exherin trifluoroacetate

Dehydrogenase Metabolism
ADH-1 trifluoroacetate (Exherin trifluoroacetate) 是一种选择性的、竞争性N-钙粘蛋白拮抗剂,具有潜在抗肿瘤和抗血管生成作用。

化合物

Acriflavine Hydrochloride
Cat.No: T19832
Synonym: 盐酸吖啶黄,Acriflavine HCl
Target: HIF
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea
Cat.No: T60124
Synonym:
Target: TNF
N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine
Cat.No: T60231
Synonym:
Target: Others
Triflusal
Cat.No: T0705
Synonym: 三氟柳,三氟醋柳酸,UR1501
Target: COX, PDE, PPAR
Eledoisin trifluoroacetate (69-25-0 free base)
Cat.No: T8832
Synonym: Eledoisin trifluoroacetate
Target: Others
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
Cat.No: T9323
Synonym: 4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide
Target: Carbonic Anhydrase
4-Chloro-3-(trifluoromethyl)phenyl isocyanate
Cat.No: T77702
Synonym:
Target: Others
2,3,4-Trifluoro-5-Nitro-Benzoic Acid
Cat.No: T9438
Synonym:
Target: Others
N-[3,5-bis(trifluoroMethyl)phenyl]-N'-[(9R)-6'-Methoxycinchonan-9-yl]- Thiourea
Cat.No: T7750
Synonym: N-[3,5-双(三氟甲基)苯基]-N′-[(9R)-6′-甲氧基-9-金鸡宁]硫脲
Target: Others
c-Myc Peptide Trifluoroacetate
Cat.No: TP1315
Synonym:
Target: Others
Cyclo(RGDyK) trifluoroacetate
Cat.No: T6813
Synonym: Cyclo(RGDyK)
Target: Integrin
Trifluridine
Cat.No: T1428
Synonym: 曲氟尿苷,NSC 529182,Trifluorothymidine,5-Trifluorothymidine,NSC 75520,曲氟胸苷,Viroptic,Trifluridina
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis, HSV
4-Nitro-3-trifluoromethyl aniline
Cat.No: T1360
Synonym:
Target: Others
1-(4-Chloro-3-(trifluoromethyl)phenyl)-3-(4-(4-cyanophenoxy)phenyl)urea
Cat.No: T22424
Synonym:
Target: Apoptosis, STAT
(S)-4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide
Cat.No: T60186
Synonym:
Target: Discoidin Domain Receptor (DDR)
Teriflunomide impurity 3
Cat.No: T9042
Synonym: 4-Amino-N-(4-trifluoromethylphenyl)benzamide
Target: COX
(E/Z)-Teriflunomide
Cat.No: T3044
Synonym: Aubagio,HMR-1726,Flucyamide,A77 1726,特立氟胺
Target: Dehydrogenase
Trifluoperazine
Cat.No: T8389
Synonym: 三氟拉嗪,trifluoroperazine
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
GSK2807 Trifluoroacetate
Cat.No: T11486
Synonym:
Target: Histone Methyltransferase
Triflupromazine hydrochloride
Cat.No: T0302
Synonym: Neoprin,盐酸三氟丙嗪,Fluopromazine hydrochloride,Fluorofen,Flumazin
Target: Dopamine Receptor, 5-HT Receptor, AChR, Autophagy
Trifluridine/tipiracil hydrochloride mixture
Cat.No: T3658
Synonym: Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Trifluoperazine dihydrochloride
Cat.No: T1222
Synonym: Trifluoperazine 2HCl,盐酸三氟拉嗪,SKF5019,Urinox
Target: CaMK, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, P-gp, Autophagy
4-Chloro-2-(trifluoroacetyl)aniline hydrochloride
Cat.No: T7455
Synonym:
Target: HIV Protease
4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxylic acid
Cat.No: T4303
Synonym:
Target: Others
3-(Trifluoromethyl)benzaldehyde
Cat.No: T9367
Synonym: 3-三氟甲基苯甲醛,3-Trifluoromethylbenzaldehyde
Target: Others
Rapastinel Trifluoroacetate
Cat.No: T5819
Synonym: Thr-Pro-Pro-Thr-NH2 Trifluoroacetate,GLYX-13 Trifluoroacetate
Target: NMDAR, iGluR
ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate
Cat.No: T50107
Synonym:
Target: Others
Carcinine ditrifluoroacetate Acetate
Cat.No: T22624L
Synonym: β-Alanylhistamine dihydrochloride,Carcinine ditrifluoroacetate Acetate (56897-53-1 Free base),Carcinine dihydrochloride
Target: Histamine Receptor
ATN-161 trifluoroacetate salt
Cat.No: T10397
Synonym: ATN-161 TFA salt
Target: Integrin
Trifluoromethyl-tubercidin
Cat.No: T67753
Synonym:
Target: Influenza Virus
Triflumuron
Cat.No: T5637
Synonym:
Target: Others
SB290157 trifluoroacetate
Cat.No: T12851
Synonym:
Target: Complement System
Ipriflavone
Cat.No: T0309
Synonym: Osteofix,依普黄酮
Target: advanced glycation end products
XMD-17-51 Trifluoroacetate
Cat.No: T9191
Synonym: XMD-17-51 Trifluoroacetate (1628614-50-5 free base)
Target: AMPK
Triflubazam
Cat.No: T67966
Synonym:
Target:
2-(4-TRIFLUOROMETHYL-PHENYL)-ETHYLAMINE
Cat.No: T7783
Synonym:
Target: Others
2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl methanesulfonate
Cat.No: T9894
Synonym:
Target: Others
(2-methylpropyl)({[3-(trifluoromethyl)phenyl]methyl})amine
Cat.No: T50011
Synonym:
Target: Others
2-Trifluoromethyl thioxanthone
Cat.No: T1361
Synonym:
Target: Others
2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE
Cat.No: T7272
Synonym:
Target:
2-(Trifluoromethyl)benzimidazole
Cat.No: Fr12535
Synonym:
Target:
Teriflunomide
Cat.No: T7534
Synonym: A 77-1726,特立氟胺
Target: Others
5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile
Cat.No: T50071
Synonym:
Target: Others
Trifloxystrobin
Cat.No: T7592
Synonym: CGA 279202,肟菌酯
Target: Antifungal
3-(Trifluoromethyl)cinnamic acid
Cat.No: T64860
Synonym: 3-(3-(Trifluoromethyl)phenyl)acrylic acid
Target: Antibiotic
ethyl 1-(4-aminophenyl)-5-(trifluoromethyl)-1H-pyrazole-4-carboxylate
Cat.No: T50023
Synonym:
Target: Others
1-(3,5-Dichloro-4-fluorophenyl)-2,2,2-trifluoroethanone
Cat.No: T9728
Synonym: sarolaner,沙罗拉纳
Target: Others
Acriflavine
Cat.No: T18911
Synonym: Acriflavinium chloride 3,6-Acridinediamine mix
Target: SARS-CoV, Antibacterial
Mefentrifluconazole
Cat.No: T11991
Synonym:
Target: P450, Antifungal
ADH-1 trifluoroacetate
Cat.No: T1608
Synonym: Exherin trifluoroacetate
Target: Dehydrogenase
Cat. No. Product Name Target Signaling Pathways
TN1768 Iriflophenone

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Iriflophenone 是从 Aquilaria sinensis 中分离得到,能诱导 MCF-7 和 T-47D 人乳腺癌细胞增殖。
TJS0341 7-Amino-4-(trifluoromethyl)coumarin

香豆素151,Coumarin 151,AFC,7-氨基-4-(三氟甲基)香豆素

5-HT Receptor GPCR/G Protein; Neuroscience
7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) 是一种荧光标记物,其激发和发射波长分别为400和500 nm,可用来灵敏的检测蛋白酶。
T11676 Iriflophenone 3-C-glucoside

Iriflophenone 3-C-β-D-glucopyranoside

Others Others
Iriflophenone 3-C-glucoside (Iriflophenone 3-C-β-D-glucopyranoside) 是一种从Cyclopia genistoides 中分离出来的物质,具有抗氧化作用。
T75705 Pepstatin Trifluoroacetate

Pepstatin (Pepstatin A) Trifluoroacetate 是一种由放线菌产生的特异性天冬氨酸蛋白酶(aspartic proteases)抑制剂,口服活性强。该化合物能有效抑制hemoglobin-pepsin、hemoglobin-proctase、casein-pepsin、casein-proctase、casein-acid protease和hemoglobin-acid protease的活性,其IC50值分别为4.5 nM、6.2 nM、150 nM、290 nM、520 nM和260 nM。此外,对HIV protease也有抑制作用。
TN5176 Trifloroside

Others Others
Trifloroside is a bitter iridoid glycoside.
TN6663 trans-4-(Trifluoromethyl)cinnamic acid

trans-4-(Trifluoromethyl)cinnamic acid 是一种光敏化合物。它被用作合成各种化合物的试剂,如杂环化合物和药物。它也被用作有机反应的催化剂,例如赫克反应和铃木-宫浦反应。它还被用作生物学研究中的荧光探针,以检测和监测各种生物分子。
T81248 Rubriflorin B

Rubriflorin B为木脂素类化合物,原自Schisandra rubriflora分离得到。
T62258 Bestatin trifluoroacetate

Bestatin trifluoroacetate (Ubenimex trifluoroacetate) 是一种 CD13 (Aminopeptidase N)/APN 和 leukotriene A4 hydrolase 抑制剂,经常用于研究癌症。
TN2006 Odoriflavene

Others Others
Odoriflavene has antioxidant activity, and it also shows inhibition effects on the decrease of glutathione level of rat lens induced by UV irradiation. Odoriflavene shows cytotoxic activity against a SH-SY5Y cell line in vitro.
TN3870 Iriflophenone 2-O-Rhamnoside

Dimethylmatairesinol

Others Others
Dimethylmatairesinol can reduce the amount of Immunoglobulin E (IgE) secreted by human myeloma U266 cells, it has potential as an anti-allergic agent. Dimethylmatairesinol also exhibits significant cytotoxicity against three human tumor cells(A-549 lung c

天然产物

Iriflophenone
Cat.No: TN1768
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
7-Amino-4-(trifluoromethyl)coumarin
Cat.No: TJS0341
Synonym: 香豆素151,Coumarin 151,AFC,7-氨基-4-(三氟甲基)香豆素
Target: 5-HT Receptor
Iriflophenone 3-C-glucoside
Cat.No: T11676
Synonym: Iriflophenone 3-C-β-D-glucopyranoside
Target: Others
Pepstatin Trifluoroacetate
Cat.No: T75705
Synonym:
Target:
Trifloroside
Cat.No: TN5176
Synonym:
Target: Others
trans-4-(Trifluoromethyl)cinnamic acid
Cat.No: TN6663
Synonym:
Target:
Rubriflorin B
Cat.No: T81248
Synonym:
Target:
Bestatin trifluoroacetate
Cat.No: T62258
Synonym:
Target:
Odoriflavene
Cat.No: TN2006
Synonym:
Target: Others
Iriflophenone 2-O-Rhamnoside
Cat.No: TN3870
Synonym: Dimethylmatairesinol
Target: Others
Cat. No. Product Name Species Expression System
TMPH-02509 ANGPTL8 Protein, Mouse, Recombinant (E. coli, His)

Angiopoietin-like protein 8,Lipasin,Gm6484,Refeeding-induced...

Mouse E. coli
Hormone that acts as a blood lipid regulator by regulating serum triglyceride levels. May be involved in the metabolic transition between fasting and refeeding: required to direct fatty acids to adipose tissue for storage in the fed state. According to a report, may act by promoting ANGPTL3 cleavage. According to another study, not required for cleavage of ANGPTL3.
TMPH-02510 ANGPTL8 Protein, Mouse, Recombinant (His)

Rifl,Refeeding-induced fat and liver protein,Betatr...

Mouse P. pastoris (Yeast)
Hormone that acts as a blood lipid regulator by regulating serum triglyceride levels. May be involved in the metabolic transition between fasting and refeeding: required to direct fatty acids to adipose tissue for storage in the fed state. According to a report, may act by promoting ANGPTL3 cleavage. According to another study, not required for cleavage of ANGPTL3. ANGPTL8 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 22.5 kDa and the...

重组蛋白

ANGPTL8 Protein, Mouse, Recombinant (E. coli, His)
Cat.No: TMPH-02509
Species: Mouse
Expression System: E. coli
ANGPTL8 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02510
Species: Mouse
Expression System: P. pastoris (Yeast)
TargetMol Loading
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