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221

抑制剂 & 化合物

48

天然产物

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Cat. No. Product Name Target Signaling Pathways
T29668 ADP-2341

ADP 2341

ADP-2341 is a soluble analog of FiVe1.
T29669 ADP-Ribosylarginine

alpha-ADP-ribosylarginine

ADP-Ribosylarginine can regulate cell proliferation and tumorigenesis.
T37118 ADP-Glucose (sodium salt)

ADPG,Adenosine-5'-diphosphoglucose,ADP-Glucose (sodium salt)

ADP-Glucose (ADPG) is an immediate precursor used in the biosynthesis, by glucose addition, of storage polysaccharides in plants, green algae, and cyanobacteria, as well as structural polysaccharides in certain bacteria.[1],[2] It is used by amylose synthases or starch synthases in plastids in the production of amylose, amylopectins, starch, and other polysaccharides. ADPG is normally generated within plastids, although it can be biosynthesized in the cytoplasm of certain grasses and imported in...
T37475 Cyclic ADP-Ribose (ammonium salt)

cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)

Cyclic ADP-ribose (cADP-ribose) is an endogenous metabolite of NAD+ that mobilizes the release of stored Ca2+ in the endoplasmic reticulum via ryanodine receptors in various cell types.[1],[2],[3],[4],[5] This second messenger is generated via the cADP-ribose synthases CD38 and CD157.[6],[5],[7] cADP-Ribose may also trigger the cell surface Ca2+ influx channel TRPM2 in a temperature-dependent manner.[8] In vitro, cADP-ribose modulates Ca2+ signaling in rat and mouse cardiomyocytes treated with i...
T10247 Adenosine 5'-diphosphoribose sodium

Adenosine 5'-diphosphoribose sodium,ADP ribose sodium

Endogenous Metabolite; TRP/TRPV Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Adenosine 5'-diphosphoribose sodium (ADP ribose sodium) 是一种烟酰胺腺嘌呤核苷酸 (NAD+) 的代谢产物,广泛存在于生物体内。Adenosine 5'-diphosphoribose sodium (ADP ribose sodium) 是一种高效的细胞内 Ca2+ 渗透性阳离子 TRPM2 通道激活剂,还可以诱导自噬 (autophagy)。
T29348 2-Fluoro-ADP

2-Fluoro-ADP is a bioactive chemical.
T37803 8-bromo-Cyclic ADP-Ribose (sodium salt)

Cyclic ADP-ribose (cADP-ribose) is a calcium mobilizing nucleotide that is biosynthesized from NAD+ by cADP-ribose synthases, including CD38. cADP-Ribose appears to activate calcium channels in intracellular membranes, which in turn activate ryanodine receptors. 8-bromo-cADP-Ribose is a stable, cell-permeable analog that blocks calcium release evoked by cADP-ribose in sea urchin egg homogenates with an IC50 value of 1.7 μM. It is commonly used to investigate intracellular signaling through cADP-...
T23581 2-Methylthioadenosine diphosphate trisodium

2 Methylthio ADP,2MeSADP,2-Methylthio-ADP,2 MeS ADP,2-MeS-ADP

2-MeS-ADP is a purinergic agonist that acts by displaying selectivity for P2Y1, P2Y12, and P2Y13 receptors and inhibiting cAMP accumulation.
T78401 pNP-ADPr disodium

ADP-ribose-pNP disodium

pNP-ADPr 二钠是一种用于检测Poly(ADP-ribose) glycohydrolase (PARG)和ADP-ribosyl hydrolase 3 (ARH3)活性的比色底物。它也适用于poly(ADP-ribose)polymerase (PARP)酶相关研究。
T50098 TIQ-A

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
TIQ-A 是一种 PARP1 抑制剂,通过碱基切除修复途径参与 DNA 单链断裂修复。 PARP1 由 DNA 损伤触发,其过度激活已被认为是许多病理状况的致病因素,包括缺血和再灌注损伤、哮喘相关炎症和动脉粥样硬化形成。
T63538 8-Azido-ADP disodium

8-Azido-ADP (disodium) 是一种线粒体腺嘌呤核苷酸易位的共价结合抑制剂,对ADP 诱导的线粒体呼吸的 4 到 3 正常转变表现出抑制作用。在光依赖反应中,8-Azido-ADP (disodium) 不可逆的抑制腺嘌呤核苷酸交换。
T41083 pNP-ADPr

pNP-ADPr,ADP-ribose-pNP

pNP-ADPr is a colorimetric substrate employed in the first continuous activity assays for Poly(ADP-ribose) glycohydrolase (PARG) and ADP-ribosyl hydrolase 3 (ARH3). Its utilization facilitates research on poly(ADP-ribose) polymerase (PARP) enzymes.
T83785 2-Chloroadenosine-5'-O-diphosphate sodium

2-chloro ADP

2-Chloroadenosine-5'-O-diphosphate是一种腺苷5'二磷酸(ADP)的衍生物。它在浓度依赖性的方式下,促进了人类富含血小板的血浆中的聚集,并抑制了由前列腺素E2(PGE2)诱导的环磷酸腺苷(cAMP)的产生。2-Chloroadenosine-5'-O-diphosphate引起预收缩的孤立的豚鼠taenia coli条带放松(pD2 = 6.74),降低大鼠的动脉血压。此外,它还抑制了热休克蛋白70(Hsp70)家族成员mortalin的ATP酶活性(人类酶的表观Ki = 45.05 µM)。
T32764 Linear-benzoadenosine diphosphate

Lin-benzo-ADP

Linear-benzoadenosine diphosphate is a nucleotide analog.
T83806 Sp-Adenosine-5'-O-(1-thiodiphosphate) sodium

Sp-ADP-α-S

Sp-Adenosine-5’-O-(1-thiodiphosphate) (Sp-ADP-α-S) 是硫含量核苷酸衍生物ADP-α-S的一种异构体。它是磷酸化酶激酶的抑制剂(Ki = 0.53 µM)。Sp-ADP-α-S能引起人类孤立血小板聚集(EC50 = 20 µM),并能使羧胺胆碱预收缩的豚鼠taenia coli松弛(EC50 = 58.9 µM)。
T83805 Rp-Adenosine-5'-O-(1-thiodiphosphate) sodium

Rp-ADP-α-S

Rp-Adenosine-5'-O-(1-thiodiphosphate)(Rp-ADP-α-S)是ADP-α-S的含硫异构体,是磷酸化酶激酶的抑制剂(Ki = 0.53 µM)。此化合物能诱导分离的人类血小板聚集(EC50 = 20 µM),并能引发经卡巴胆碱预收缩的豚鼠乙状结肠松弛(EC50 = 58.9 µM)。
T22749 DR2313

DR 2313

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
DR2313 是一种选择性,竞争性的和可透过血脑屏障的PARP 抑制剂,对PARP-1和PARP-2的IC50值分别为 0.20 和 0.24 μM。它在体内外均有对缺血性损伤的神经保护作用。
T16761 RK-287107

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
RK-287107 是一种有效且特异性的 tankyrase 抑制剂,可阻断结直肠癌细胞生长,对 tankyrase-1和 tankyrase-2的 IC50分别为 14.3 和 10.6 nM。
T6181 UPF 1069

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
UPF 1069 是一种特异性PARP 抑制剂,对 PARP-1 和 PARP-2 的IC50值分别为 8 和 0.3 μM。
T83813 8-Azidoadenosine-5'-O-diphosphate sodium

8-azido-ADP,Click Tag™ 8-Azidoadenosine-5'-O-diphosphate

8-Azidoadenosine-5'-O-diphosphate(8-azido-ADP)是ATP前体和嘌呤受体配体ADP的可点击形式。8-azido-ADP的放射性标记形式已被用作各种蛋白质的光亲和标签,包括从牛脑中分离的谷氨酸脱氢酶(GDH)同工酶,以及从兔网织红细胞中分离的真核翻译起始因子2(eIF2)和鸟苷核苷酸交换因子(GEF)。
T2484 AZD-2461

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
AZD-2461 是一种 PARP 抑制剂,可抑制 PARP1、PARP2 和 PARP3 的活性,IC50值分别为 5、2 和 200 nM。
T21524 4-amino-1,8-Naphthalimide

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
4-amino-1,8-Naphthalimide 是PARP 抑制剂,可增强癌细胞对 γ 辐射诱导的细胞毒性的敏感度。
T15639 K-756

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
K-756 是一种直接的 tankyrase(TNKS) 选择性抑制剂,对 TNKS1和 TNKS2的 ADP-核糖基化活性有抑制作用,IC50分别为 31 和 36 nM。
T6578 ME0328

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
ME0328 是一种有效的选择性 PARP 抑制剂,对 PARP3 的 IC50 为 0.89 μM。
T6197 PJ34

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
PJ34 是一种PARP1/2的特异性有效抑制剂,IC50分别为 110 nM 和 86 nM。
T6768 AZ6102

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
AZ6102 是TNKS1和TNKS2双重抑制剂,IC50值分别为 3 和 1 nM,选择性是对 PARP 家族其他蛋白的 100 多倍,对 PARP1、PARP2 和 PARP6 的IC50值分别为 2.0、0.5 和大于 3 μM。
T4022 QS11

QS 11

GTPase GPCR/G Protein
QS11 是一种ARFGAP1抑制剂(EC50:1.5 µM)。QS 11 能抑制 ARFGAP 过表达的乳腺癌细胞迁移。QS 11 通过影响蛋白质运输来增强 Wnt/β-catenin 信号。
T6842 G007-LK

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
G007-LK 是 TNKS1 和 TNKS2 的选择性抑制剂,IC50 分别为 46 nM 和 25 nM。
T8964 G244-LM

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
G244-LM 是一种特异性有效的tankyrase 1/2抑制剂,可抑制Wnt 信号传导。
T39785L TH5427

NUDIX hydrolase Metabolism
TH5427 在 NUDT5 活性和 ADP-核糖代谢中有研究的价值。它阻断孕激素依赖性、PAR 衍生的核 ATP 合成以及随后的乳腺癌细胞染色质重塑、基因调控和增殖。NUDT5是乳腺癌细胞激素依赖性基因调控和增殖的变阻器。
T9165 AZD5305

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
AZD5305 是一种强效、选择性和口服活性 PARP 抑制剂,可用于肿瘤异体移植模型研究。
T3168 MN-64

MN64

Others; PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Others; Stem Cells
MN-64 是一种有效的tankyrase 1抑制剂,对TNKS1、TNKS2、ARTD1 和 ARTD2 的IC50值分别为 6、72、19.1 和 39.4 μM。
T1807 JW 55

JW55

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
JW 55 (JW55) 是一种有效且选择性的 β-catenin 信号通路抑制剂,通过抑制 tankyrase 1 和 tankyrase 2 (TNKS1/2) 的 PARP 结构域起作用。
T22264 AZ9482

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
AZ9482 是一种选择性 PARP1/2/6的三重抑制剂,IC50值分别为 1 、1 和640 nM。
T4471 E7449

Stenoparib,UNII-9X5A2QIA7C

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
E7449 (UNII-9X5A2QIA7C) 是一种有效的 PARP1 和 PARP2 抑制剂,也抑制 TNKS1 和 TNKS2,使用 32P-NAD+ 作为底物,对 PARP1、PARP2、TNKS1 和 TNKS2 的 IC50 分别为 2.0、1.0、约 50 和约 50 nM。
T7042 1,5-Isoquinolinediol

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
1,5-Isoquinolinediol 是一种多聚(ADP-核糖)合成酶抑制剂,对PARP1的IC50值为 0.39 µM。它用于研究 PARP1 在 DNA 修复和氧化应激诱导的细胞死亡中的作用。
T3062 WIKI4

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
WIKI4 是tankyrase 有效抑制剂,其对TNKS2的IC50值为 26 nM。它有效抑制Wnt/β-catenin 信号传导,其EC50值为 75 nM。它通过抑制TNKS2的酶活性来介导其对Wnt/β-catenin 信号传导的影响。它对 SCLC 细胞具有细胞毒性,其IC50值为 0.02 μM。
T6339 AG14361

AG 14361,AG-14361

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
AG14361 是一种 PARP-1抑制剂,Ki 值小于 5 nM,在通透的 SW620 细胞和完整的 SW620 细胞中,抑制 PARP-1的活性,IC50值分别为 29 和 14 nM。
T5058 Pamiparib

BGB-290

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Pamiparib (BGB-290) 是一种具有口服活性、强效、高选择性的 PARP 抑制剂,对PARP1和PARP2的IC50值分别为 0.9 nM 和 0.5 nM。它具有强大的 PARP 捕获能力,具有穿透大脑的能力,可用于研究癌症。
T5399 GeA-69

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
GeA-69 是一种选择性变构 PARP14 大结构域 2 (MD2) 抑制剂,Kd 值为 2.1 µM。
T4472 NMS-P118

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
NMS-P118是可口服的高选择性PARP-1抑制剂,用于癌症治疗,在HeLa 细胞中的IC50值为0.04 μM。
T22414 RBN012759

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
RBN012759 是选择性和具有口服活性的 PARP14抑制剂,IC50值小于3 nM,可降低促肿瘤巨噬细胞功能并在肿瘤外植体中引发炎症反应,比对 monoPARPs 的选择性高 300 倍,比对 polyPARPs 的选择性高 1000 倍。
T9593 Senaparib

IMP4297

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Senaparib (IMP4297) 是一种选择性和口服有效的PARP1/2抑制剂,具有强效的抗肿瘤活性。
T3649 BGP-15

BGP15,BGP-15 2HCl

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
BGP-15 (BGP-15 2HCl) 是一种PARP 抑制剂,IC50和Ki 值分别为 120 和 57 μM,在缺血再灌注损伤后具有保护作用。
T7896 BYK204165

RT-017290

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
BYK204165 (RT-017290) 是一种选择性PARP1抑制剂,对重组人 PARP1的pIC50值为 7.35,pKi 值为7.05。它对鼠 PARP-2的pIC50值为 5.38 ,其对 PARP1 的选择性比对 PARP2 高 100 倍。
T9430 Venadaparib

NOV140101,IDX-1197

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Venadaparib (NOV140101) 是一种选择性和具有口服活性的 PARP 抑制剂,对 PARP1和 PARP2的 IC50分别为 1.4 和 1.0 nM。它可防止 DNA 单链断裂 (SSB) 的修复,可研究实体瘤。
T12695 RBN-2397

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
RBN-2397 是一种有效的、选择性的、具有口服活性的跨物种 NAD+ 竞争性 PARP7 抑制剂,IC50 小于 3 nM。它选择性结合 PARP7 ,Kd 为0.001 μM,可恢复干扰素 I 型信号转导,有用于晚期或转移性实体肿瘤的研究潜力。
T1878 XAV-939

XAV939,NVP-XAV939

PARP; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Stem Cells
XAV-939 (NVP-XAV939) 是一种 Tankyrase (TNKS) 抑制剂,抑制 TNKS1 和 TNKS2 (IC50=11/4 nM)。XAV-939 可以选择性抑制 Wnt/β-catenin 介导的转录。
T9497 Niraparib tosylate monohyrate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Niraparib tosylate monohyrate 也称为 MK-4827,是一种聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂,具有潜在的抗肿瘤活性。 MK4827 抑制 PARP 活性,增强 DNA 链断裂的积累,促进基因组不稳定性和细胞凋亡。 PARP 蛋白家族通过碱基切除修复 (BER) 途径检测和修复单链 DNA 断裂。
T2591 Veliparib

ABT-888,NSC 737664,维利帕尼

PARP; Autophagy Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair
Veliparib (ABT-888) 是一种可口服的 PARP 抑制剂,抑制PARP1和PARP2的Ki 分别为 5.2 和 2.9 nM。它增强细胞凋亡和自噬。

化合物

ADP-2341
Cat.No: T29668
Synonym: ADP 2341
Target:
ADP-Ribosylarginine
Cat.No: T29669
Synonym: alpha-ADP-ribosylarginine
Target:
ADP-Glucose (sodium salt)
Cat.No: T37118
Synonym: ADPG,Adenosine-5'-diphosphoglucose,ADP-Glucose (sodium salt)
Target:
Cyclic ADP-Ribose (ammonium salt)
Cat.No: T37475
Synonym: cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)
Target:
Adenosine 5'-diphosphoribose sodium
Cat.No: T10247
Synonym: Adenosine 5'-diphosphoribose sodium,ADP ribose sodium
Target: Endogenous Metabolite, TRP/TRPV Channel, Autophagy
2-Fluoro-ADP
Cat.No: T29348
Synonym:
Target:
8-bromo-Cyclic ADP-Ribose (sodium salt)
Cat.No: T37803
Synonym:
Target:
2-Methylthioadenosine diphosphate trisodium
Cat.No: T23581
Synonym: 2 Methylthio ADP,2MeSADP,2-Methylthio-ADP,2 MeS ADP,2-MeS-ADP
Target:
pNP-ADPr disodium
Cat.No: T78401
Synonym: ADP-ribose-pNP disodium
Target:
TIQ-A
Cat.No: T50098
Synonym:
Target: PARP
8-Azido-ADP disodium
Cat.No: T63538
Synonym:
Target:
pNP-ADPr
Cat.No: T41083
Synonym: pNP-ADPr,ADP-ribose-pNP
Target:
2-Chloroadenosine-5'-O-diphosphate sodium
Cat.No: T83785
Synonym: 2-chloro ADP
Target:
Linear-benzoadenosine diphosphate
Cat.No: T32764
Synonym: Lin-benzo-ADP
Target:
Sp-Adenosine-5'-O-(1-thiodiphosphate) sodium
Cat.No: T83806
Synonym: Sp-ADP-α-S
Target:
Rp-Adenosine-5'-O-(1-thiodiphosphate) sodium
Cat.No: T83805
Synonym: Rp-ADP-α-S
Target:
DR2313
Cat.No: T22749
Synonym: DR 2313
Target: PARP
RK-287107
Cat.No: T16761
Synonym:
Target: Others, PARP
UPF 1069
Cat.No: T6181
Synonym:
Target: PARP
8-Azidoadenosine-5'-O-diphosphate sodium
Cat.No: T83813
Synonym: 8-azido-ADP,Click Tag™ 8-Azidoadenosine-5'-O-diphosphate
Target:
AZD-2461
Cat.No: T2484
Synonym:
Target: PARP
4-amino-1,8-Naphthalimide
Cat.No: T21524
Synonym:
Target: PARP
K-756
Cat.No: T15639
Synonym:
Target: PARP, Wnt/beta-catenin
ME0328
Cat.No: T6578
Synonym:
Target: PARP
PJ34
Cat.No: T6197
Synonym:
Target: PARP
AZ6102
Cat.No: T6768
Synonym:
Target: PARP, Wnt/beta-catenin
QS11
Cat.No: T4022
Synonym: QS 11
Target: GTPase
G007-LK
Cat.No: T6842
Synonym:
Target: PARP, Wnt/beta-catenin
G244-LM
Cat.No: T8964
Synonym:
Target: Others, PARP
TH5427
Cat.No: T39785L
Synonym:
Target: NUDIX hydrolase
AZD5305
Cat.No: T9165
Synonym:
Target: PARP
MN-64
Cat.No: T3168
Synonym: MN64
Target: Others, PARP, Wnt/beta-catenin
JW 55
Cat.No: T1807
Synonym: JW55
Target: PARP, Wnt/beta-catenin
AZ9482
Cat.No: T22264
Synonym:
Target: PARP
E7449
Cat.No: T4471
Synonym: Stenoparib,UNII-9X5A2QIA7C
Target: Others, PARP
1,5-Isoquinolinediol
Cat.No: T7042
Synonym:
Target: PARP
WIKI4
Cat.No: T3062
Synonym:
Target: PARP, Wnt/beta-catenin
AG14361
Cat.No: T6339
Synonym: AG 14361,AG-14361
Target: PARP
Pamiparib
Cat.No: T5058
Synonym: BGB-290
Target: PARP
GeA-69
Cat.No: T5399
Synonym:
Target: PARP
NMS-P118
Cat.No: T4472
Synonym:
Target: PARP
RBN012759
Cat.No: T22414
Synonym:
Target: PARP
Senaparib
Cat.No: T9593
Synonym: IMP4297
Target: PARP
BGP-15
Cat.No: T3649
Synonym: BGP15,BGP-15 2HCl
Target: PARP
BYK204165
Cat.No: T7896
Synonym: RT-017290
Target: PARP
Venadaparib
Cat.No: T9430
Synonym: NOV140101,IDX-1197
Target: PARP
RBN-2397
Cat.No: T12695
Synonym:
Target: PARP
XAV-939
Cat.No: T1878
Synonym: XAV939,NVP-XAV939
Target: PARP, Wnt/beta-catenin
Niraparib tosylate monohyrate
Cat.No: T9497
Synonym:
Target: PARP
Veliparib
Cat.No: T2591
Synonym: ABT-888,NSC 737664,维利帕尼
Target: PARP, Autophagy
Cat. No. Product Name Target Signaling Pathways
T19253 Cyclic ADP-​ribose

cADPR

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cyclic ADP-ribose (cADPR) is an effective calcium mobilization second messenger, which is synthesized from NAD + by ADP-ribosyl cyclase. Cyclic ADP-ribose mainly increases cytosolic calcium through Ryanodine receptor-mediated endoplasmic reticulum release
T37687 Cyclic ADP-ribose ammonium

Cyclic ADP-ribose ammonium (cADPR ammonium) is a powerful calcium mobilization second messenger synthesized from NAD+ by an ADP-ribosyl cyclase. It primarily raises cytosolic calcium levels through Ryanodine receptor-mediated release from the endoplasmic reticulum, while also facilitating extracellular influx through the opening of TRPM2 channels [1][2][3].
T1723 Adenosine 5'-diphosphate

腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP

Endogenous Metabolite Metabolism
Adenosine 5'-diphosphate (ADP) 是一种嘌呤核糖核苷5'-二磷酸,是 ATP 在 ATP 酶作用下去磷酸化的产物。Adenosine 5'-diphosphate (adenosine pyrophosphate) 可诱导人血小板聚集并通过作用于P2T-嘌呤受体抑制受刺激的腺苷酸环化酶。
T5079 Adenosine 5'-diphosphate sodium salt

腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt

Others; Endogenous Metabolite Metabolism; Others
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。
T83789 7-Deazaadenosine-5'-O-diphosphate sodium

7-CH-ADP,Tubercidin 5’-diphosphate,TuDP

7-Deazaadenosine-5'-O-diphosphate是一种修饰过的核苷酸和tubercidin的代谢物。该化合物通过磷酸化tubercidin形成,并进一步磷酸化生成活性代谢物7-deazaadenosine-5'-O-triphosphate。
T8184 Fucosterol

岩皂甾醇,岩藻甾醇

PARP; Endogenous Metabolite; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Fucosterol 是从藻类、海藻或硅藻中分离的一种甾醇,具有抗氧化、抗脂肪、降低血液胆固醇、抗糖尿病和抗癌活性。它通过抑制 PPARα和C/EBPα的表达调控脂肪生成,可用于抗肥胖试剂开发研究。
T7443 4'-Methoxychalcone

4'-甲氧基查耳酮,4'-甲氧基查尔酮

PARP; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
4'-Methoxychalcone 通过PPARγ活化调节脂肪细胞分化,并调节参与胰岛素敏感性的脂肪组织中各种脂肪因子的表达和分泌,具抗肿瘤和抗炎活性。
T8150 Nudifloramide

1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide,1-甲基-6-氧代吡啶-3-甲酰胺

PARP; Endogenous Metabolite Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Nudifloramide (1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide) 是烟酰胺-腺嘌呤二核苷酸(NAD) 降解的一种最终产物,可显著抑制PARP-1活性。
T3S0156 Atractyloside potassium salt

Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐

Others Others
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。
T5S2358 Dehydrocorydaline

Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T6780 Benzamide

Amid kyseliny benzoove,苯甲酰胺,Phenylcarboxyamide,Benzoylamide

PARP; Endogenous Metabolite Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Benzamide (Amid kyseliny benzoove) 是聚(ADP-核糖)聚合酶的抑制剂,是苯甲酸的衍生物。
T10990 Dehydrocorydaline chloride

盐酸脱氢紫堇碱,13-Methylpalmatine chloride

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。
T5S1805 5,7-Dihydroxychromone

5,7-Dihydroxy-4H-Chromen-4-One,5,7-二羟基色酮,5,7-二羟基色原酮

Others; Virus Protease; PARP; Caspase; Nrf2 Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology; Others; Proteases/Proteasome
5,7-Dihydroxychromone (5,7-Dihydroxy-4H-Chromen-4-One) 是一种Cudrania tricuspidata 的提取物,通过激活 Nrf2/ARE 信号对 6-OHDA 诱导的氧化应激和细胞凋亡发挥神经保护作用。它抑制 6-OHDA 诱导的 SH-SY5Y 细胞中活化的caspase-3,caspase-9以及切割的PARP 表达。
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
T8296 5,​7,​4'-​Trimethoxyflavone

5,7,4'-三甲氧基黄酮,芹菜素三甲醚,4',5,7-三甲氧基黄酮,4',5,7-Trimethoxyflavone

Apoptosis; PARP; Caspase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
5,​7,​4'-​Trimethoxyflavone (4',5,7-Trimethoxyflavone) 是从泰国著名的药用植物 Kaempferia parviflora 中分离出来的一种天然产物。它以浓度依赖性方式显著有效抑制 SNU-16 人胃癌细胞的增殖,诱导细胞凋亡。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
T4085 Paris saponin VII

重楼皂苷 VII,Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII

Apoptosis; BCL; Others; PARP; p38 MAPK; Akt; Caspase; P-gp; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; MAPK; Membrane transporter/Ion channel; Neuroscience; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Paris saponin VII (Dioscini) 是从延龄草的根和根茎中分离的一种甾体皂苷。它减弱线粒体膜电位,增加凋亡相关蛋白的表达,并降低Bcl-2、caspase-9、caspase-3、PARP-1和p-Akt 的蛋白表达水平。它在 K562/ADR 细胞中诱导强烈的自噬,可研究白血病。
TN6732 Oenothein B

Apoptosis; HCV Protease; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Proteases/Proteasome
Oenothein B 是一种聚(ADP-核糖)糖水解酶的特异性抑制剂。 Oenothein B 具有抗氧化、抗炎、抗真菌、抗 HCV 和抗肿瘤特性。
T22446 NADP disodium salt

Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐

Others Others
NADP disodium salt (Disodium NADP) 是一种氧化还原辅助因子,是一种烟酰胺腺嘌呤二核苷酸。它是代谢中电子转移的关键辅因子,可以被交替氧化 (NADP+) 和还原 (NADPH)。
T4448 NADP

NADP,也称为烟酰胺腺嘌呤二核苷酸磷酸,是各种代谢过程中电子转移所必需的重要氧化还原辅因子。 它在促进细胞能量产生和维持细胞内氧化还原平衡方面发挥着关键作用。
T8170 Carboxyatractyloside

羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt

Others Others
Carboxyatractyloside (Carboxyatractyloside tripotassium salt) tripotassium salt 是一种 ADP/ATP 载体蛋白 (ADP/ATP carrier) 抑制剂,抑制线粒体 ADP/ATP 的转运。它是一种具有毒性的天然产物,
T6942 Picolinamide

2-Pyridinecarboxamide,2-Carbamoylpyridine,2-吡啶甲酰胺,2-Picolinamide,Picolinoylamide

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Picolinamide (Picolinoylamide) 被发现是大鼠胰岛细胞核聚 (ADP-核糖) 合成酶的强抑制剂。
T4888 Phosphocreatine disodium hydrate

磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium hydrate 是内源性代谢产物的一种。
T3781 Jujuboside B

酸枣仁皂苷 B,酸枣仁皂苷B

Others Others
Jujuboside B 是一种提取自Zizyphus jujuba 中的活性成分,对血小板聚集具有抑制作用。
T40834 5-Hydroxymethyl-2'-deoxycytidine

5hmdC,2'-脱氧-5-(羟甲基)胞啶

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
5-Hydroxymethyl-2'-deoxycytidine 是 DNA 中 5-methyl-2'-deoxycytidine (5-mdC) 的氧化衍生物,引起DNA损伤反应,染色体畸变,复制叉损伤和细胞活力丧失。5-Hydroxymethyl-2’-deoxycytidine 复制叉不稳定性与染色质上聚(ADP-核糖)聚合酶1(PARP1)的存在有关。
T5S0896 Loureirin A

龙血素 A,龙血素A

Akt; PI3K Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Loureirin A 是一种黄酮类物质,从龙血树中分离得到,能够降低Akt 的磷酸化,具有抗血小板聚集作用。
T4786 D-Ribose(mixture of isomers)

D-Ribose,D-(-)-Ribose,D-(-)-核糖

Others; Endogenous Metabolite Metabolism; Others
D-Ribose(mixture of isomers) (D-(-)-Ribose) 是 ATP 的糖部分,可作为能量增强剂,被广泛用作慢性疲劳综合症和心肌能量代谢的代谢疗法补充剂。它在蛋白质糖化中具有特性,能够 RAGE 依赖的方式诱导 NF-Κb 炎症。
T2860 Vanillyl Alcohol

4-Hydroxy-3-methoxybenzenemethanol,3-Methoxy-4-hydroxybenzyl alcohol,4-Hydroxy-3-methoxybenzyl alcohol,香兰醇,Vanillin alcohol,Vanillic alcohol

Apoptosis; Others Apoptosis; Others
Vanillyl Alcohol (3-Methoxy-4-hydroxybenzyl alcohol) 是一种酚类醇,具有抗血管生成、抗惊厥、抗炎、抗氧化、神经保护和抗伤害活性。它由香兰素衍生而来,在食品和饮料中用作调味剂。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T7982 3,6-Dihydroxyflavone

Others Others
3,6-Dihydroxyflavone 是一种抗癌剂。它能够提高细胞内氧化应激和脂质过氧化。它是能够根据剂量和时间依赖性地降低细胞活力,并活化半胱天冬酶级联、切割聚 (ADP-核糖) 聚合酶 (PARP) 诱导细胞凋亡。
T7032 Eupatorin

Others; P450 Metabolism; Others
Eupatorin 是天然存在的黄酮,可捕获 G2-M 细胞周期,激活多个 caspase、细胞色素 C 的释放、多聚 (ADP-核糖) 聚合酶的裂解,促使凋亡细胞死亡。
T15721 Latrunculin A

LAT-A

Others Others
Latrunculin A is a toxin isolated from the red sea sponge Latrunculia magnifica. Latrunculin A binds to actin monomers and it also inhibits polymerization of actin (Kds: 0.1, 0.4, 4.7 μM, and 0.19 μM for ATP-actin, ADP-Pi-actin, ADP-actin, and G-actin, re
TN3069 4beta-Carboxy-19-nortotarol

NADPH-oxidase Immunology/Inflammation
4 beta-Carboxy-19-nortotarol can inhibit microsomal lipid peroxidation induced by Fe(III)-ADP/NADPH and mitochondrial lipid peroxidation induced by Fe(III)-ADP/ NADH, it inhibits linoleic acid autoxidation but not generation of superoxide anion.
T25211 CC 1014

CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885

CC 1014 is a polypeptide antibiotic isolated from Penicillium lilacinum that inhibits phosphorylation of ADP, Mg ATPase.
T17273 YM-254890

Others Others
YM-254890 inhibits platelet aggregation induced by ADP by blocking the P2Y1 signal transduction pathway (IC50: below 0.6 μM). YM-254890 is a selective Gαq/11 protein inhibitor. YM-254890 displays no inhibition of other G protein subtypes.
T37714 Fuscin

Fuscin is a quinonoid fungal metabolite originally isolated from O. fuscum that has diverse biological activities. It inhibits binding of the ADP/ATP translocase inhibitor atractyloside to rat liver mitochondria in an ADP-dependent manner when used at a concentration of 50 μM in a radioligand binding assay. Fuscin (20 μM) reduces the glutathione content of rat liver mitochondria to 28% of controls and inhibits NADH oxidation in sonicated pigeon heart mitochondria preparations in a concentration-...
T83460 11-O-β-D-glucopyranosyl thamnosmonin

11-O-β-D-glucopyranosyl thamnosmonin是一种香豆素苷,能够从Angelica apaensis根部提取。该化合物对PAF、AA和ADP诱发的兔血小板聚集表现出轻度的抑制效果。
TN1309 6-Hydroxykaempferol-3,6,7-triglucoside

Others Others
6-Hydroxykaempferol 3,6,7-tri-O-glucoside and 6-hydroxykaempferol 3,6-di-O-glucoside can inhibit platelet aggregation induced by collagen, they also show weak inhibitory effects on the adenosine 5'-diphosphate (ADP)- induced platelet aggregation.
TN1310 6-Hydroxykaempferol 3,6-diglucoside

Others Others
6-Hydroxykaempferol 3,6-di-O-glucoside and 6-hydroxykaempferol 3,6,7-tri-O-glucoside can inhibit platelet aggregation induced by collagen, they also show weak inhibitory effects on the adenosine 5'-diphosphate (ADP)- induced platelet aggregation.
T38015 Herquline A

Herquline A is an alkaloid fungal metabolite originally isolated from P. herquei. It inhibits cell death induced by influenza A strain A/PR/8/34 in MDCK cells with an IC50 value of 10 μg/ml and inhibits viral replication in a plaque assay in a concentration-dependent manner. Herquline A also inhibits platelet aggregation induced by ADP and platelet-activating factor (PAF) in vitro (IC50s = 180 and 240 μM, respectively).
TN6014 Norcepharadione B

鱼腥草

Norcepharadione B shows good inhibitory activity against the replication of HSV-1, it also shows antimalarial activity with EC50 values of 7.5mug/ml. Norcepharadione B exhibits significant cytotoxicity against five human tumor cell lines (A-549, SK-OV-3,
TN6924 Anhydrosafflor yellow B

(2S,3S)-6,7-dihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-2-[(1S,2R,3R)-1,2,3,4-tetrahydroxybutyl]-3-{2,3,4-trihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-6-oxo-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]cyclohexa-1,4-dien-1,脱水红花黄色素B,AHSYB

Others Others
Anhydrosafflor yellow B ((2S,3S)-6,7-dihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-2-[(1S,2R,3R)-1,2,3,4-tetrahydroxybutyl]-3-{2,3,4-trihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-6-oxo-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]cyclohexa-1,4-dien-1) 是从红花中分离出来的,可抑制 ADP 诱导的血小板聚集,在体外表现出显着的抗氧化作用,并对 H2O2 诱导的细胞毒性具有一定的活性。
TN4046 Excisanin A

MMP; FAK; PARP; GSK-3; NF-κB; Wnt/beta-catenin; Akt; Caspase; PI3K; Prostaglandin Receptor; JNK Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; MAPK; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
ExcisaninA may be a potent inhibitor of AKT signaling pathway in tumor cells, it can inhibit invasion by suppressing MMP-2 and MMP-9 expression, it may be a potential anti-metastatic chemotherapeutic agent for the treatment of breast cancer. Excisanin A shows comparable inhibitory effects on the LPS-induced production of NO and PGE2, and activation of NF-kappaB without affecting cell viability.Excisanin A induces apoptosis in colon cancer cell line SW620 as determined by Annexin V staining, the ...
TN4664 Norarmepavine

Others Others
N-norarmepavine shows significant cytotoxic activities against HL-60 carcinoma cell line with inhibitory ratios of 51.43% at concentration of 1 x 10(-5) M. Norarmepavine shows inhibition against Trypanosoma cruzi. D-(+)- N-norarmepavine exhibits significa
T73403 Aviculin

Aviculin 是一种木聚糖苷,是一种有效的抗癌剂 (anticanceragent)。Aviculin 可降低 MCF-7 细胞代谢活性到 50% 以下,IC50为 75.47 μM。Aviculin 通过内在凋亡途径诱导乳腺癌细胞凋亡 (apoptosis)。Aviculin 增加了 caspase-9、caspase-7和 PARP 的表达。Aviculin 使 Bax/Bcl-2 的比值升高。
T4883 Creatine

Methylguanidoacetic acid,肌酸

Endogenous Metabolite Metabolism
Creatine (Methylguanidoacetic acid) 是一种内源性氨基酸代谢物,在细胞能量中发挥重要作用,尤其是在肌肉和大脑中。
T35624 Ajoene

Ajoene is a disulfide that has been found inA. sativumand has diverse biological activities, including antibacterial, anticancer, antiplatelet, and antioxidant properties.1,2,3,4It is active against Gram-positive (MICs = 5-160 &#181g/ml) and Gram-negative bacteria (MICs = 136-200 &#181g/ml), as well as yeasts (MICs = 10-20 &#181g/ml).1Ajoene is cytotoxic to mouse melanoma cells (IC50= 18 &#181M), as well as human colon, lung, mammary, and pancreatic cancer cells (IC50s = 7-41 &#181M).2It reduces...

天然产物

Cyclic ADP-​ribose
Cat.No: T19253
Synonym: cADPR
Target: Calcium Channel
Cyclic ADP-ribose ammonium
Cat.No: T37687
Synonym:
Target:
Adenosine 5'-diphosphate
Cat.No: T1723
Synonym: 腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP
Target: Endogenous Metabolite
Adenosine 5'-diphosphate sodium salt
Cat.No: T5079
Synonym: 腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt
Target: Others, Endogenous Metabolite
7-Deazaadenosine-5'-O-diphosphate sodium
Cat.No: T83789
Synonym: 7-CH-ADP,Tubercidin 5’-diphosphate,TuDP
Target:
Fucosterol
Cat.No: T8184
Synonym: 岩皂甾醇,岩藻甾醇
Target: PARP, Endogenous Metabolite, PPAR
4'-Methoxychalcone
Cat.No: T7443
Synonym: 4'-甲氧基查耳酮,4'-甲氧基查尔酮
Target: PARP, PPAR
Nudifloramide
Cat.No: T8150
Synonym: 1-Methyl-6-oxo-1,6-dihydropyridine-3-carboxamide,1-甲基-6-氧代吡啶-3-甲酰胺
Target: PARP, Endogenous Metabolite
Atractyloside potassium salt
Cat.No: T3S0156
Synonym: Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐
Target: Others
Dehydrocorydaline
Cat.No: T5S2358
Synonym: Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Benzamide
Cat.No: T6780
Synonym: Amid kyseliny benzoove,苯甲酰胺,Phenylcarboxyamide,Benzoylamide
Target: PARP, Endogenous Metabolite
Dehydrocorydaline chloride
Cat.No: T10990
Synonym: 盐酸脱氢紫堇碱,13-Methylpalmatine chloride
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
5,7-Dihydroxychromone
Cat.No: T5S1805
Synonym: 5,7-Dihydroxy-4H-Chromen-4-One,5,7-二羟基色酮,5,7-二羟基色原酮
Target: Others, Virus Protease, PARP, Caspase, Nrf2
3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
5,​7,​4'-​Trimethoxyflavone
Cat.No: T8296
Synonym: 5,7,4'-三甲氧基黄酮,芹菜素三甲醚,4',5,7-三甲氧基黄酮,4',5,7-Trimethoxyflavone
Target: Apoptosis, PARP, Caspase
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
Paris saponin VII
Cat.No: T4085
Synonym: 重楼皂苷 VII,Chonglou Saponin VII,Polyphyllin-VII,Dioscinin,Paris saponin-VII
Target: Apoptosis, BCL, Others, PARP, p38 MAPK, Akt, Caspase, P-gp, Autophagy
Oenothein B
Cat.No: TN6732
Synonym:
Target: Apoptosis, HCV Protease, Antibacterial, Antifungal
NADP disodium salt
Cat.No: T22446
Synonym: Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐
Target: Others
NADP
Cat.No: T4448
Synonym:
Target:
Carboxyatractyloside
Cat.No: T8170
Synonym: 羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt
Target: Others
Picolinamide
Cat.No: T6942
Synonym: 2-Pyridinecarboxamide,2-Carbamoylpyridine,2-吡啶甲酰胺,2-Picolinamide,Picolinoylamide
Target: PARP
Phosphocreatine disodium hydrate
Cat.No: T4888
Synonym: 磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate
Target: Others, Endogenous Metabolite
Jujuboside B
Cat.No: T3781
Synonym: 酸枣仁皂苷 B,酸枣仁皂苷B
Target: Others
5-Hydroxymethyl-2'-deoxycytidine
Cat.No: T40834
Synonym: 5hmdC,2'-脱氧-5-(羟甲基)胞啶
Target: PARP
Loureirin A
Cat.No: T5S0896
Synonym: 龙血素 A,龙血素A
Target: Akt, PI3K
D-Ribose(mixture of isomers)
Cat.No: T4786
Synonym: D-Ribose,D-(-)-Ribose,D-(-)-核糖
Target: Others, Endogenous Metabolite
Vanillyl Alcohol
Cat.No: T2860
Synonym: 4-Hydroxy-3-methoxybenzenemethanol,3-Methoxy-4-hydroxybenzyl alcohol,4-Hydroxy-3-methoxybenzyl alcohol,香兰醇,Vanillin alcohol,Vanillic alcohol
Target: Apoptosis, Others
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
3,6-Dihydroxyflavone
Cat.No: T7982
Synonym:
Target: Others
Eupatorin
Cat.No: T7032
Synonym:
Target: Others, P450
Latrunculin A
Cat.No: T15721
Synonym: LAT-A
Target: Others
4beta-Carboxy-19-nortotarol
Cat.No: TN3069
Synonym:
Target: NADPH-oxidase
CC 1014
Cat.No: T25211
Synonym: CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885
Target:
YM-254890
Cat.No: T17273
Synonym:
Target: Others
Fuscin
Cat.No: T37714
Synonym:
Target:
11-O-β-D-glucopyranosyl thamnosmonin
Cat.No: T83460
Synonym:
Target:
6-Hydroxykaempferol-3,6,7-triglucoside
Cat.No: TN1309
Synonym:
Target: Others
6-Hydroxykaempferol 3,6-diglucoside
Cat.No: TN1310
Synonym:
Target: Others
Herquline A
Cat.No: T38015
Synonym:
Target:
Norcepharadione B
Cat.No: TN6014
Synonym: 鱼腥草
Target:
Anhydrosafflor yellow B
Cat.No: TN6924
Synonym: (2S,3S)-6,7-dihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-2-[(1S,2R,3R)-1,2,3,4-tetrahydroxybutyl]-3-{2,3,4-trihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-6-oxo-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]cyclohexa-1,4-dien-1,脱水红花黄色素B,AHSYB
Target: Others
Excisanin A
Cat.No: TN4046
Synonym:
Target: MMP, FAK, PARP, GSK-3, NF-κB, Wnt/beta-catenin, Akt, Caspase, PI3K, Prostaglandin Receptor, JNK
Norarmepavine
Cat.No: TN4664
Synonym:
Target: Others
Aviculin
Cat.No: T73403
Synonym:
Target:
Creatine
Cat.No: T4883
Synonym: Methylguanidoacetic acid,肌酸
Target: Endogenous Metabolite
Ajoene
Cat.No: T35624
Synonym:
Target:
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