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74

抑制剂 & 化合物

10

天然产物

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Cat. No. Product Name Target Signaling Pathways
T32419 KRAS4b-PDEδ stabilizer C19

KRAS4b-PDEδ stabilizer C19 is a stabilizer of the KRAS4b-PDEδ complex which decreases the proliferation of colorectal cancer cells, and increases apoptosis via decreased activation of oncogenic KRAS4b signaling.
T32500 L6Y

TTR stabilizer L6

L6Y is a transthyretin (TTR) stabilizer which binds to the T4 binding pocket of TTR and prevents the dissociation of TTR to monomer.
T33261 MDK-5432

AMPA stabilizer (R,R)-2a,MDK 5432

MDK-5432, also known as AMPA stabilizer (R,R)-2a, is the most potent AMPA stabilizer.
T72286 LC kinetic stabilizer-2

LC kinetic stability-2 是一种有效的淀粉样免疫球蛋白轻链 (LC) 动力学稳定剂,EC50为 24 nM。
T72285 LC kinetic stabilizer-1

LC kinetic stabilizer-1 为一种高效、选择性的淀粉样免疫球蛋白轻链动力学稳定剂,对 WIL-FL* 与 WIL-FL*T46L/F49Y 的EC50值分别为140 nM与74.1 nM。其中,WIL-FL 为一种淀粉样变FL-LC二聚体。
T79736 14-3-3σ/ERα stabilizer-1

Estrogen Receptor/ERR Endocrinology/Hormones
14-3-3σ/ERα stabilizer-1 (Compound 181) 是一种针对14-3-3σ/ERα的共价稳定剂,主要应用于分子胶研究领域。
T8239 Cromoglicic acid

Others Others
Cromoglicic acid 可防止肥大细胞释放炎性化学物质,例如组胺。
T60028 MM41

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
MM41 是一种人类端粒和基因启动子 DNA 四链体稳定剂,对 MIA PaCa-2 胰腺癌细胞系的 IC50 <10 nM。
T22891 KL001

KL 001,KL-001

Others Others
KL001 是一流的隐花色素蛋白 (CRY)稳定剂,可与 CRY1 和 CRY2 特异性相互作用。其中CRY 是一种对蓝光敏感的黄素蛋白,参与调节动植物的昼夜节律。KL001能够防止泛素依赖性 CRY 降解,从而延长了昼夜节律周期,具有控制空腹激素诱导的糖异生的潜力。
T12678 (Rac)-Telmesteine

替美司坦,3-(Ethoxycarbonyl)thiazolidine-4-carboxylic acid,3-ethoxycarbonyl-1,3-thiazolidine-4-carboxylic acid,3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester

Protease Proteases/Proteasome
(Rac)-Telmesteine (3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester) 是蛋白酶抑制剂,可用作含蛋白酶的洗涤剂和清洗剂中的酶稳定剂。
T31614 Elpetrigine

GW-273293,JZP 4,JZP4,GW273293,JZP-4,GW 273293

Elpetrigine( GW 273293, JZP-4) is effective calcium and sodium channel blocker and is currently being evaluated in patients as an anticonvulsant and mood stabilizer.
T35044 Velaresol

BW 12C79,BW 12C,BW-12C79,BW12C79,BW-12C

Velaresol (BW12C, BW12C79) is an oxygenated hemoglobin stabilizer that, in addition to stabilizing oxygenated hemoglobin, protects sickle cells from calcium-mediated dehydration.
T4457 Pyridostatin Trihydrochloride

Pyridostatin Trihydrochloride(free base 1085412-37-8 ),RR-82 Trihydrochloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Pyridostatin Trihydrochloride (RR-82 Trihydrochloride) 是一种 G-四链体稳定剂,Kd 为 490 nM。
T21282 Topanol CA

Others Others
Topanol CA 是一种抗氧化剂,可用于树脂和浅色橡胶制品中作稳定剂。
T7582 tafamidis meglumine

Fx-1006A,他发米帝司甲葡胺

Others Others
Tafamidis meglumine (Fx-1006A) 是transthyretin (TTR)的选择性稳定剂,对野生型 WT-TTR 和突变型同源四聚体 V30M-TTR,V122I-TTR 的活性相当,EC50值为 2.7-3.2 μM。它能够阻碍淀粉样蛋白的生成。
T0211 Azelastine

Azelastina,Astelin,Azelastinum,氮卓斯汀

SARS-CoV; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。
T4566 Lodoxamide

Lodoxamidum,洛草氨酸

GPR; Histamine Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Lodoxamide (Lodoxamidum) 是一种抗过敏药物,作为肥大细胞稳定剂,对治疗哮喘和过敏性结膜炎有效。
T15772 Lodoxamide tromethamine

U-42585E

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Lodoxamide tromethamine 是一种的肥大细胞稳定剂,具有抗过敏特性,可用于治疗哮喘和过敏性结膜炎的研究。
T9608 KL201

Others Others
KL201 是一种昼夜节律调制器,是 CRY1选择性的 稳定剂, 对 CRY2 没有稳定作用。KL201 延长了细胞和组织中的昼夜节律周期。
T33816 Ordopidine

ACR-325,ACR 325,ACR325

Dopamine Receptor GPCR/G Protein; Neuroscience
Ordopidine (ACR325) 是一种多巴胺能稳定剂,可抑制精神刺激剂引起的多动症,并在不活动时刺激行为。Ordopidine 在体外作为多巴胺 D2 受体拮抗剂起作用,尽管亲和力低,但其依赖于特定状态的行为效应特征是 D2 受体拮抗剂所不具备的。
T0008 Phenytoin sodium

5,5-Diphenylhydantoin sodium salt,Diphantoine,苯妥英钠,Dilantin sodium,Diphenylhydantoin Sodium

Virus Protease; Sodium Channel Membrane transporter/Ion channel; Microbiology/Virology
Phenytoin sodium (Diphantoine) 是一种有效的电压门控钠离子通道阻滞剂,可减少小鼠乳腺肿瘤的生长和转移,具有抗癫痫活性。
T0404 8-Hydroxyquinoline

Hydroxyquinoline,8-Quinolinol,羟基喹啉,Oxine,8-羟基喹啉,8-Oxychinolin

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
8-Hydroxyquinoline (8-Quinolinol) 是单质子二齿螯合剂, 也是转录抑制剂,防腐剂,消毒剂和杀虫剂。
T7352 Pridopidine

ACR16,ASP2314,FR310826,4-[3-(甲磺酰基)苯基]-1-丙基哌啶

Dopamine Receptor GPCR/G Protein; Neuroscience
Pridopidine (FR310826) 是多巴胺稳定剂,是一种低亲和力的多巴胺 D2 受体拮抗剂。它高亲和力作用于 sigma 1受体,Ki=70-80 nM,比其对 D2R 的亲和力高约 100 倍。
T26955 Cavosonstat

N91115,N 91115,N-91115

GSNOR; CFTR Membrane transporter/Ion channel; Metabolism
Cavosonstat (N91115) 是一种口服活性 S-亚硝基谷胱甘肽还原酶(GSNOR)抑制剂,可促进囊性纤维化跨膜传导调节器(CFTR)成熟和质膜稳定。
T9526 Polysorbate 20

Tween-20,吐温 20

Others Others
Polysorbate 20 (Tween-20) 是聚氧乙烯型非离子表面活性剂。
T6488 Epinastine hydrochloride

Alesion,Epinastine HCl,WAL-801CL HCl,依匹斯汀盐酸盐,Elestat

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Epinastine hydrochloride (WAL-801CL HCl) 是抗组胺剂和肥大细胞稳定剂,是一种可口服的选择性组胺 H1 受体拮抗剂,可抑制 IL-8 释放,具有抗过敏作用。
T17217 Vamorolone

地塞米松EP杂质E,VBP15

Glucocorticoid Receptor; NF-κB Endocrinology/Hormones; NF-κB
Vamorolone (VBP15) 是一种首创的,具有口服活性的解离性类固醇 (dissociative steroidal) 抗炎药和膜稳定剂。它抑制 (NF-κB) 抑制作用,并降低了激素的影响。它改善肌营养不良,无副作用。
T21648 CP-31398 dihydrochloride

CP 31398 dihydrochloride

p53 Apoptosis
CP-31398 dihydrochloride 是一种 p53 稳定剂,可稳定 p53 的活性构象并促进具有突变型或野生型 p53 的癌细胞系中的 p53 活性。
T4470 Pyridostatin TFA

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Pyridostatin TFA 是一种 G-四链体稳定剂,靶向原癌基因 Src,降低人乳腺癌细胞 SRC 蛋白水平和 SRC 依赖的细胞运动。它通过诱导复制和转录依赖的 DNA 损伤促进人类癌细胞生长停滞。
T9447 AG-10

Acoramidis

Others Others
AG-10 (Acoramidis) 是选择性的、口服有效的甲状腺素转运蛋白 (TTR (transthyretin)) 的稳定剂,显示出对野生型和 V1221 突变型均有效。
T0680 Lamotrigine

LTG,BW430C,拉莫三嗪

5-HT Receptor; Sodium Channel; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Lamotrigine (BW430C) 是一种抗癫痫剂和情绪稳定剂,可研究癫痫、局灶性癫痫等。。它选择性地阻断电压门控钠离子通道,稳定突触前神经元膜,抑制谷氨酸释放。
T39740 Acoramidis hydrochloride

AG10 hydrochloride,Alxn2060 hydrochloride

Others Others
Acoramidis hydrochloride (Alxn2060 hydrochloride) 是具有口服活性的、选择性的甲状腺素转运蛋白 (TTR (transthyretin)) 的稳定剂,对野生型和 V1221 突变型均有效。Acoramidis hydrochloride 可用于转体甲状腺素淀粉样变性的研究。
T19820 MOPS sodium salt

MOPS-Na,3-(N-morpholino)propanesulfonic acid sodium salt,3-吗啉丙磺酸钠盐,Sodium 3-Morpholinopropanesulfonate,4-Morpholinepropanesulfonic acid, sodium salt

Others Others
MOPS sodium salt (MOPS-Na) 在生物学中常用作缓冲剂。其中MOPS 缓冲液能使哺乳动物细胞培养基的 pH 值保持稳定。
T21300 Trientine-2HCl

Triethylenetetramine,Trientine HCl,Trientine,盐酸三乙烯四胺,Triethylene tetramine,TETA,Trien

Others Others
Trientine-2HCl (Trien) 是一种螯合剂,通过结合和去除体内的铜来治疗威尔逊氏病。曲恩汀还可用作肝豆状核变性中铜的螯合剂,环氧树脂的稳定剂,等电聚焦的两性电解质。
TF0106 Cholesteryl Hemisuccinate Tris Salt

Apoptosis Apoptosis
Cholesteryl Hemisuccinate Tris Salt 是一种具有保肝和抗癌活性的酸性胆固醇酯,是一种含有柴胡皂苷-d的二棕榈酰磷脂酰胆碱脂质体中的膜稳定剂,可增强顺铂的抗癌功效。Cholesteryl hemisuccinate 具有抗肿瘤活性,抑制肿瘤生长,抑制对乙酰氨基酚 (AAP) 的肝毒性,预防 AAP 诱导的肝细胞凋亡。Cholesteryl hemisuccinate 可保护啮齿动物免受对乙酰氨基酚、阿霉素、四氯化碳、氯仿和半乳糖胺的毒性作用。
T4565 Tafamidis

他发米帝司甲葡胺,氯苯唑酸,Fx-1006A

Others Others
Tafamidis (Fx-1006A) 是选择性的transthyretin (TTR)稳定剂,对野生型 WT-TTR 、突变型同源四聚体 V30M-TTR、V122I-TTR 的活性相当,它们的EC50值为2.7-3.2 μM。它对淀粉样蛋白的生成具有抑制作用。
T35841 5-Benzyloxygramine

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
5-Benzyloxygramine 是一种 N 蛋白、蛋白互作的原位稳定剂,具有抗病毒和稳定 N-NTD 蛋白的作用。它能够阻断多巴胺受体,可拮抗 5-HT 对大鼠子宫和兔耳的作用。
T20780 Dibutyltin maleate

Stavinor Sn 1300,Stavinor 1300SN

Dibutyltin maleate is used as a condensation catalyst and pvc Stabilizer.
T34759 Synstab A

Synstab-A

Synstab A is a microtubule stabilizer.
T23114 OSU 6162 hydrochloride

Others Others
Dopamine stabilizer
T30587 Brl 22321

Brl22321,Brl-22321

Brl 22321 is a mast cell stabilizer.
T19212 BMVC2

o-BMVC

Others Others
BMVC2 (o-BMVC), a carbazole derivative of BMVC, is a G-quadruplex (G4) stabilizer.
T26872 BMVC4

BMVC 4,BMVC-4

BMVC4 is a G-quadruplex stabilizer. BMVC4 induces senescence by activation of pathways of response to DNA damage that was independent of its telomerase inhibitory activity.
T19837 O4

O 4,O-4

O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.
T19472 Nedocromil sodium

Nedocromil disodium salt,FPL 59002KP

Others Others
Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.
T13504 360A iodide

360 A iodide

Telomerase DNA Damage/DNA Repair
360A iodide is a selective stabilizer of G-quadruplex and inhibits telomerase activity (IC50: 300 nM in TRAP-G4 assay).
T31364 Dehydelone

KOS1584,SK-10088,KOS-1584,R-1645,SK10088,R1645

Dehydelone(KOS-1584, R-1645, SK-10088) is a microtubule stabilizer that may be used in the treatment of non-small cell lung cancer.
T35319 Zy 15109

N-Acetyl-aspartyl magnesium glutamate,Zy15109,Magnesium N-acetyl-aspartylglutamate

Zy 15109 can be used as inhaled mast cell stabilizer.
T69584 GMC-1111 dihydrochloride

GMC-1111 dihydrochloride is a dopamine partial agonist and stabilizer.
T69585 GMC-1111 free base

GMC-1111 free base is a dopamine partial agonist and stabilizer.

化合物

KRAS4b-PDEδ stabilizer C19
Cat.No: T32419
Synonym:
Target:
L6Y
Cat.No: T32500
Synonym: TTR stabilizer L6
Target:
MDK-5432
Cat.No: T33261
Synonym: AMPA stabilizer (R,R)-2a,MDK 5432
Target:
LC kinetic stabilizer-2
Cat.No: T72286
Synonym:
Target:
LC kinetic stabilizer-1
Cat.No: T72285
Synonym:
Target:
14-3-3σ/ERα stabilizer-1
Cat.No: T79736
Synonym:
Target: Estrogen Receptor/ERR
Cromoglicic acid
Cat.No: T8239
Synonym:
Target: Others
MM41
Cat.No: T60028
Synonym:
Target: DNA/RNA Synthesis
KL001
Cat.No: T22891
Synonym: KL 001,KL-001
Target: Others
(Rac)-Telmesteine
Cat.No: T12678
Synonym: 替美司坦,3-(Ethoxycarbonyl)thiazolidine-4-carboxylic acid,3-ethoxycarbonyl-1,3-thiazolidine-4-carboxylic acid,3,4-Thiazolidinedicarboxylic Acid 3-Ethyl Ester
Target: Protease
Elpetrigine
Cat.No: T31614
Synonym: GW-273293,JZP 4,JZP4,GW273293,JZP-4,GW 273293
Target:
Velaresol
Cat.No: T35044
Synonym: BW 12C79,BW 12C,BW-12C79,BW12C79,BW-12C
Target:
Pyridostatin Trihydrochloride
Cat.No: T4457
Synonym: Pyridostatin Trihydrochloride(free base 1085412-37-8 ),RR-82 Trihydrochloride
Target: DNA/RNA Synthesis
Topanol CA
Cat.No: T21282
Synonym:
Target: Others
tafamidis meglumine
Cat.No: T7582
Synonym: Fx-1006A,他发米帝司甲葡胺
Target: Others
Azelastine
Cat.No: T0211
Synonym: Azelastina,Astelin,Azelastinum,氮卓斯汀
Target: SARS-CoV, Histamine Receptor
Lodoxamide
Cat.No: T4566
Synonym: Lodoxamidum,洛草氨酸
Target: GPR, Histamine Receptor
Lodoxamide tromethamine
Cat.No: T15772
Synonym: U-42585E
Target: Histamine Receptor
KL201
Cat.No: T9608
Synonym:
Target: Others
Ordopidine
Cat.No: T33816
Synonym: ACR-325,ACR 325,ACR325
Target: Dopamine Receptor
Phenytoin sodium
Cat.No: T0008
Synonym: 5,5-Diphenylhydantoin sodium salt,Diphantoine,苯妥英钠,Dilantin sodium,Diphenylhydantoin Sodium
Target: Virus Protease, Sodium Channel
8-Hydroxyquinoline
Cat.No: T0404
Synonym: Hydroxyquinoline,8-Quinolinol,羟基喹啉,Oxine,8-羟基喹啉,8-Oxychinolin
Target: Others, Antibacterial, Antibiotic
Pridopidine
Cat.No: T7352
Synonym: ACR16,ASP2314,FR310826,4-[3-(甲磺酰基)苯基]-1-丙基哌啶
Target: Dopamine Receptor
Cavosonstat
Cat.No: T26955
Synonym: N91115,N 91115,N-91115
Target: GSNOR, CFTR
Polysorbate 20
Cat.No: T9526
Synonym: Tween-20,吐温 20
Target: Others
Epinastine hydrochloride
Cat.No: T6488
Synonym: Alesion,Epinastine HCl,WAL-801CL HCl,依匹斯汀盐酸盐,Elestat
Target: 5-HT Receptor, Histamine Receptor
Vamorolone
Cat.No: T17217
Synonym: 地塞米松EP杂质E,VBP15
Target: Glucocorticoid Receptor, NF-κB
CP-31398 dihydrochloride
Cat.No: T21648
Synonym: CP 31398 dihydrochloride
Target: p53
Pyridostatin TFA
Cat.No: T4470
Synonym:
Target: DNA/RNA Synthesis
AG-10
Cat.No: T9447
Synonym: Acoramidis
Target: Others
Lamotrigine
Cat.No: T0680
Synonym: LTG,BW430C,拉莫三嗪
Target: 5-HT Receptor, Sodium Channel, Autophagy
Acoramidis hydrochloride
Cat.No: T39740
Synonym: AG10 hydrochloride,Alxn2060 hydrochloride
Target: Others
MOPS sodium salt
Cat.No: T19820
Synonym: MOPS-Na,3-(N-morpholino)propanesulfonic acid sodium salt,3-吗啉丙磺酸钠盐,Sodium 3-Morpholinopropanesulfonate,4-Morpholinepropanesulfonic acid, sodium salt
Target: Others
Trientine-2HCl
Cat.No: T21300
Synonym: Triethylenetetramine,Trientine HCl,Trientine,盐酸三乙烯四胺,Triethylene tetramine,TETA,Trien
Target: Others
Cholesteryl Hemisuccinate Tris Salt
Cat.No: TF0106
Synonym:
Target: Apoptosis
Tafamidis
Cat.No: T4565
Synonym: 他发米帝司甲葡胺,氯苯唑酸,Fx-1006A
Target: Others
5-Benzyloxygramine
Cat.No: T35841
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Dibutyltin maleate
Cat.No: T20780
Synonym: Stavinor Sn 1300,Stavinor 1300SN
Target:
Synstab A
Cat.No: T34759
Synonym: Synstab-A
Target:
OSU 6162 hydrochloride
Cat.No: T23114
Synonym:
Target: Others
Brl 22321
Cat.No: T30587
Synonym: Brl22321,Brl-22321
Target:
BMVC2
Cat.No: T19212
Synonym: o-BMVC
Target: Others
BMVC4
Cat.No: T26872
Synonym: BMVC 4,BMVC-4
Target:
O4
Cat.No: T19837
Synonym: O 4,O-4
Target:
Nedocromil sodium
Cat.No: T19472
Synonym: Nedocromil disodium salt,FPL 59002KP
Target: Others
360A iodide
Cat.No: T13504
Synonym: 360 A iodide
Target: Telomerase
Dehydelone
Cat.No: T31364
Synonym: KOS1584,SK-10088,KOS-1584,R-1645,SK10088,R1645
Target:
Zy 15109
Cat.No: T35319
Synonym: N-Acetyl-aspartyl magnesium glutamate,Zy15109,Magnesium N-acetyl-aspartylglutamate
Target:
GMC-1111 dihydrochloride
Cat.No: T69584
Synonym:
Target:
GMC-1111 free base
Cat.No: T69585
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2S1865 Octyl gallate

Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯

Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。
T8064 Lactobionic acid

Others; Antibacterial Microbiology/Virology; Others
Lactobionic acid 是在里海酸奶中的一种仿生酸,化学上由与半乳糖键合的葡萄糖酸组成。它是具有抗氧化、抗菌和保湿特性的乳糖酸。
T8704 4-hydroxyphenyl acetate

Nrf2 Immunology/Inflammation
4-hydroxyphenyl acetate 通过作为 NRF2 稳定剂防止 RPE 氧化应激诱导的坏死。
T0968 Paclitaxel

Taxol,紫杉醇,NSC 125973

Apoptosis; Microtubule Associated; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling
Paclitaxel (Taxol) 属于天然产物,是一种微管聚合物稳定剂。Paclitaxel 具有抗肿瘤活性;通过诱导有丝分裂停滞、细胞凋亡、细胞自噬等,导致细胞死亡。
T5247 Trimethylamine N-oxide dihydrate

二水氧化三甲胺,TMANO Dihydrate

Others; Endogenous Metabolite Metabolism; Others
Trimethylamine N-oxide dihydrate (TMANO Dihydrate) 是内源性代谢产物的一种。
T2S0157 Methyl palmitate

Methyl hexadecanoate,软脂酸甲酯,十六烷酸甲酯,Palmitic acid methyl ester,十六酸甲酯

Others Others
Methyl palmitate (Palmitic acid methyl ester) 是存在于绿色核桃壳中的杀螨化合物,具有抗炎和抗纤维化作用,可抑制吞噬活性和免疫应答。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
TQ0202 Epothilone D

KOS 862,埃博霉素

Microtubule Associated Cytoskeletal Signaling
Epothilone D (KOS 862) is an effective microtubule stabilizer.
T75573 Taccalonolide E

Taccalonolide E 是一种微管稳定剂,诱导癌细胞凋亡 (apoptosis)。
TN2255 Taccalonolide AJ

Others Others
Taccalonolide AJ is a microtubule stabilizer; it has excellent and highly persistent antitumor efficacy when administered directly to the tumor, suggesting that the lack of antitumor efficacy seen with systemic administration of AJ is likely due to its sh

天然产物

Octyl gallate
Cat.No: T2S1865
Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯
Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV
Lactobionic acid
Cat.No: T8064
Synonym:
Target: Others, Antibacterial
4-hydroxyphenyl acetate
Cat.No: T8704
Synonym:
Target: Nrf2
Paclitaxel
Cat.No: T0968
Synonym: Taxol,紫杉醇,NSC 125973
Target: Apoptosis, Microtubule Associated, Autophagy
Trimethylamine N-oxide dihydrate
Cat.No: T5247
Synonym: 二水氧化三甲胺,TMANO Dihydrate
Target: Others, Endogenous Metabolite
Methyl palmitate
Cat.No: T2S0157
Synonym: Methyl hexadecanoate,软脂酸甲酯,十六烷酸甲酯,Palmitic acid methyl ester,十六酸甲酯
Target: Others
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Epothilone D
Cat.No: TQ0202
Synonym: KOS 862,埃博霉素
Target: Microtubule Associated
Taccalonolide E
Cat.No: T75573
Synonym:
Target:
Taccalonolide AJ
Cat.No: TN2255
Synonym:
Target: Others
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