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Search Results for " enantiomer "

300

抑制剂 & 化合物

19

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T12064	Niraparib (R-enantiomer) MK 4827 (R-enantiomer),Niraparib R-enantiomer	PARP	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Niraparib R-enantiomer (MK 4827 R-enantiomer) 是一种 PARP1抑制剂，IC50为 2.4 nM。
T12697	Refametinib R enantiomer RDEA119 R enantiomer,Refametinib R enantiomer,BAY 869766 R enantiomer	MEK	MAPK
	Refametinib R enantiomer (RDEA119 R enantiomer) 是一种 MEK 抑制剂，EC50为 2.0-15 nM。Refametinib R enantiomer 具有抗癌活性，可用于研究癌症。
T15263	Selisistat R-enantiomer EX-527 (R-enantiomer)	Sirtuin	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Selisistat R-enantiomer (EX-527 (R-enantiomer)) 是 Selisistat R 型对映体。Selisistat 是SIRT1的选择性抑制剂，IC50为98 nM。
T13140	Umbralisib R-enantiomer TGR-1202 R-enantiomer,RP5264 R-enantiomer	PI3K	PI3K/Akt/mTOR signaling
	Umbralisib R-enantiomer (RP5264 R-enantiomer) 是 PI3K 的δ型抑制剂，是 TGR-1202 活性较低的对映体。Umbralisib R-enantiomer 对δ型 pi3激酶的 IC50，至少比抑制剂对其他 PI3K 亚型(A， β和γ)的 IC50低20倍。
T17102	Tipifarnib (S enantiomer) Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer	Transferase	Metabolism
	Tipifarnib S enantiomer ((S)-(-)-R-115777) 是Tipifarnib 的 S 型对映体，它比 Tipifarnib 特性低。其中 Tipifarnib 是farnesyltransferase 高效特异性抑制剂，IC50=0.6 nM。
T7058	Selisistat S-enantiomer EX-527 S-enantiomer,(1S)-6-氯-2,3,4,9-四氢-1H-咔唑-1-甲酰胺,EX-527 (S-enantiomer)	Sirtuin	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Selisistat S-enantiomer (EX-527 S-enantiomer) 是一种选择性的SIRT1抑制剂，IC50值为 98 nM。
T11129L	Duvelisib (R enantiomer) hydrochloride IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl	PI3K	PI3K/Akt/mTOR signaling
	Duvelisib (R enantiomer) hydrochloride (INK1197 R enantiomer HCl) 是 PI3K 抑制剂。Duvelisib (R enantiomer) hydrochloride 是 Duvelisib 的活性较低的对映体。
T12831	SAR405 R enantiomer	Others	Others
	SAR405 R enantiomer 是一种 PIK3C3/Vps34 抑制剂，也是活性低于 SAR405 的对映体。
T6156	Ruxolitinib (S enantiomer) S-Ruxolitinib,环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯,Ruxolitinib S enantiomer,INCB018424,INCB18424	Tyrosine Kinases; JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
	Ruxolitinib S enantiomer (INCB18424) 是 Ruxolitinib 的 S 型对映体，是一种JAK 抑制剂。
T9825	CORT-108297 Enantiomer	Others	Others
	CORT-108297 Enantiomer 是 CORT-108297 的对映体，CORT-108297是糖皮质激素受体的拮抗剂。
T19618	(R)-(-)-JQ1 Enantiomer (R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯	Epigenetic Reader Domain	Chromatin/Epigenetic
	(R)-(-)-JQ1 Enantiomer 是 (+)-JQ1 的立体异构体。 (+)-JQ1 是一种 BET 溴结构域抑制剂，对BRD4(1/2)的IC50 为 77 和 33 nM。
T10819	Cipropride S enantiomer	Others	Others
	Cipropride S enantiomer 是止吐药环普必利的S 对映体。
T7695	PNU-282987 S enantiomer free base	AChR	Neuroscience
	PNU-282987 S enantiomer free base 是 PNU-282987 的 S 型对映体，是 α7 烟碱乙酰胆碱受体的激动剂。
T67881	Acalabrutinib enantiomer R-Acalabrutinib	BTK	Angiogenesis; Tyrosine Kinase/Adaptors
	Acalabrutinib enantiomer (R-Acalabrutinib) 是一类属于布鲁顿酪氨酸激酶(BTK)抑制剂的化合物。Acalabrutinib enantiomer 可用于癌症、自身免疫性疾病和慢性炎症等领域的研究。
T19112L	Sacubitril Enantiomer 2R,4S-Sacubitril,LCZ 696杂质A,ahu377 isomer 2	Others	Others
	Sacubitril Enantiomer (ahu377 isomer 2) 是 Sacubitril 的对映体，它是一种脑啡肽酶抑制剂。
T80678	(S)-AK-242 (-)-Resatorvid,(S)-Resatorvid,AK-242 (S enantiomer),(-)-AK-242	Others	Others
	(S)-AK-242 ((S)-Resatorvid) 是一种细胞因子抑制剂，可用于治疗心脏病、自身免疫性疾病、炎症性疾病。
T22450	Tyrphostin B44, (+) enantiomer 酪氨酸磷酸化抑制剂AG 835	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Tyrphostin B44, (+) enantiomer 是一种表皮生长因子受体 (EGFR) 激酶抑制剂，IC50 为 0.86 μM，活性低于 (-) 对映体。
T12274	Siremadlin (R Enantiomer) Siremadlin R Enantiomer,HDM201 R Enantiomer,NVP-HDM201 R Enantiomer	Others	Others
	Siremadlin R Enantiomer is the R enantiomer of Siremadlin. Siremadlin is a potent and highly specific inhibitor of MDM-2/p53.
T12200	Firsocostat S enantiomer ND-630 S enantiomer,NDI-010976 S enantiomer,GS-0976 S enantiomer	Others	Others
	Firsocostat S enantiomer is the less active S enantiomer of Firsocostat.
T11129	Duvelisib (R enantiomer) Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer	PI3K	PI3K/Akt/mTOR signaling
	Duvelisib R enantiomer (IPI-145 R enantiomer) 是一种 Duvelisib 的对映异构体，活性较低。它是一种 PI3K 抑制剂。
T11334	Fulvestrant (R enantiomer) ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer	Others	Others
	Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T11335	Fulvestrant (S enantiomer) ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer	Others	Others
	Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T10552	Bitopertin (R enantiomer) RO4917838 (R enantiomer),RG1678 (R enantiomer),Bitopertin R enantiomer	GlyT	Neuroscience
	Bitopertin R enantiomer (RG1678 R enantiomer) is the R-enantiomer of Bitopertin. Bitopertin is a noncompetitive glycine reuptake inhibitor and inhibits glycine uptake at human GlyT1 (IC50: 25 nM).
T11391	Gepotidacin S enantiomer GSK2140944 S enantiomer	Others	Others
	Gepotidacin S enantiomer is an S enantionmer of gepotidacin.
T11173	Elacestrant S enantiomer RAD1901 S enantiomer	Others	Others
	Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
T13120	Tenalisib R Enantiomer RP6530 R Enantiomer	Others	Others
	Tenalisib R Enantiomer is an R enantiomer of Tenalisib .
T11410	GLPG0492 (R enantiomer) GLPG0492 R enantiomer	Others	Others
	GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.
T12775	RSV604 (R enantiomer) RSV604 R enantiomer	Others	Others
	RSV604 R enantiomer is the R-enantiomer of RSV604. RSV604 is a respiratory syncytial virus (RSV) replication inhibitor.
T13312	Seviteronel R enantiomer VT-464 (R enantiomer)	Others	Others
	Seviteronel R enantiomer is the R enantiomer of Seviteronel and is a potent inhibitor of CYP17 lyase (IC50: 69 nM for h-Lyase).
T13422L	Talarozole (R enantiomer) (R)-Talarozole,Talarozole R enantiomer	Others	Others
	Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.
T11156	Nazartinib S-enantiomer EGF816 (S-enantiomer)	Others	Others
	Nazartinib is an EGFR inhibitor. Nazartinib S-enantiomer is the less active S-enantiomer of Nazartinib.
T10465	Atuveciclib S-Enantiomer BAY-1143572 S-Enantiomer	CDK	Cell Cycle/Checkpoint
	Atuveciclib S-Enantiomer (BAY-1143572 S-Enantiomer) 是 BAY-1143572的 S-对映异构体，是一种有效的选择性 CDK9抑制剂，抑制 CDK9/CycT1，IC50为 16 nM。
T10856	Cobimetinib (R-enantiomer) 考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer	Others	Others
	Cobimetinib R-enantiomer is the less active R-enantiomer of Cobimetinib which is a selective MEK inhibitor.
T11173L	Elacestrant S enantiomer dihydrochloride RAD1901 S enantiomer dihydrochloride,RAD-1901 S enantiomer dihydrochloride,RAD 1901 S enantiomer dihydrochloride	Others	Others
	Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively. Elacestrant S enantiomer dihydrochloride is an low activity enantiomer of elacestrant dihydrochloride.
T11627	IACS-8968 R-enantiomer IDO/TDO Inhibitor (R-enantiomer)	IDO	Metabolism
	IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T11662	INT-777 R-enantiomer S-EMCA R enantiomer	Others	Others
	INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5.
T10252L	ADU-S100 enantiomer ammonium salt MIW815 enantiomer ammonium salt,ML RR-S2 CDA enantiomer ammonium salt	Others	Others
	ADU-S100 (MIW815) enantiomer ammonium salt is the less active enantiomer of ADU-S100. ADU-S100 is an activator of the stimulator of interferon genes (STING).
T11628	IACS-8968 S-enantiomer IDO/TDO Inhibitor (S-enantiomer)	IDO	Metabolism
	IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T67880	NITD-609 Enantiomer	Others	Others
	NITD-609 Enantiomer 是 NITD-609 的对映体，NITD-609 是一种具有抗疟活性的螺酮类药物。
T9848	GSK2850163 (S enantiomer)	IRE1	Cell Cycle/Checkpoint
	GSK2850163 (S enantiomer) 是 GSK2850163 的无活性对映体。GSK2850163 是一种新型的肌醇需求酶-1α (IRE1a) 抑制剂。
T39541	THK5351 (R enantiomer)
	THK5351 R enantiomer is an R enantiomer of THK5351.
T41114	LIN28 inhibitor LI71 enantiomer
	LIN28 inhibitor LI71 enantiomer, the enantiomer of LIN28 inhibitor LI71，exhibits reduced activity compared to its parent compound. LIN28 inhibitor LI71 is a highly potent and cell-permeable inhibitor of LIN28, effectively blocking LIN28-mediated oligouridylation with an IC50 of 7 uM.
T10757	Cenobamate S-Enantiomer	Others	Others
	Cenobamate S-Enantiomer is a Cenobamate's S-enantiomer.
T12915	Silvestrol aglycone (enantiomer)	Others	Others
	Silvestrol aglycone (enantiomer) is a cyclopenta benzofuran core phenol.
T11195	Enantiomer of Sofosbuvir	Others	Others
	Enantiomer of Sofosbuvir 是Sofosbuvir 的对映异构体，Sofosbuvir 是一种治疗慢性丙型肝炎的处方药，目前尚无enantiomer of Sofosbuvir 的生物活性报道。
T22401	PNU-282987 S enantiomer hydrochloride (S)-PNU-282987 HCl	Others	Others
	(S)-PNU-282987 is the absolute stereochemistry form of PNU-282987. PNU 282987, a potent agonist of α7-containing neuronal nicotinic acetylcholine receptors (nAChRs) with Ki of 26 nM for the rat receptor, has negligible activity against α1β1γδ and α3β4 nAC
T12067	MK-7246 S enantiomer	Others	Others
	MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.
T12723	Ribocil-C R enantiomer	Others	Others
	Ribocil-C R enantiomer is the R enantiomer of Ribocil-C. Ribocil-C is a highly selective bacterial riboflavin riboswitches inhibitor.
T11841	Leu-AMS R enantiomer	Others	Others
	Leu-AMS R enantiomer 是 Leu-AMS 的 R 对映体。 Leu-AMS 是一种有效的亮氨酰-tRNA 合成酶 (LRS) 抑制剂，可抑制细菌的生长。
T12203	Necrostatin 2 S enantiomer	Others	Others
	Necrostatin 2 S enantiomer is the S enantiomer of Necrostatin 2

化合物

Niraparib (R-enantiomer)

Cat.No: T12064

Synonym: MK 4827 (R-enantiomer),Niraparib R-enantiomer

Target: PARP

Refametinib R enantiomer

Cat.No: T12697

Synonym: RDEA119 R enantiomer,Refametinib R enantiomer,BAY 869766 R enantiomer

Target: MEK

Selisistat R-enantiomer

Cat.No: T15263

Synonym: EX-527 (R-enantiomer)

Target: Sirtuin

Umbralisib R-enantiomer

Cat.No: T13140

Synonym: TGR-1202 R-enantiomer,RP5264 R-enantiomer

Target: PI3K

Tipifarnib (S enantiomer)

Cat.No: T17102

Synonym: Tipifarnib S enantiomer,(S)-(-)-R-115777,(S)-Tipifarnib,IND-58359 S enantiomer

Target: Transferase

Selisistat S-enantiomer

Cat.No: T7058

Synonym: EX-527 S-enantiomer,(1S)-6-氯-2,3,4,9-四氢-1H-咔唑-1-甲酰胺,EX-527 (S-enantiomer)

Target: Sirtuin

Duvelisib (R enantiomer) hydrochloride

Cat.No: T11129L

Synonym: IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl

Target: PI3K

SAR405 R enantiomer

Cat.No: T12831

Target: Others

Ruxolitinib (S enantiomer)

Cat.No: T6156

Synonym: S-Ruxolitinib,环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯,Ruxolitinib S enantiomer,INCB018424,INCB18424

Target: Tyrosine Kinases, JAK

CORT-108297 Enantiomer

Cat.No: T9825

Target: Others

(R)-(-)-JQ1 Enantiomer

Cat.No: T19618

Synonym: (R)-(-)2-(4-(4-氯苯基)-2,3,9-三甲基-6H-噻吩并[3,2-F][1,2,4]三唑并[4,3-A][1,4]二氮杂环庚烷-6-基)乙酸叔丁酯

Target: Epigenetic Reader Domain

Cipropride S enantiomer

Cat.No: T10819

Target: Others

PNU-282987 S enantiomer free base

Cat.No: T7695

Target: AChR

Acalabrutinib enantiomer

Cat.No: T67881

Synonym: R-Acalabrutinib

Target: BTK

Sacubitril Enantiomer

Cat.No: T19112L

Synonym: 2R,4S-Sacubitril,LCZ 696杂质A,ahu377 isomer 2

Target: Others

Cat.No: T80678

Synonym: (-)-Resatorvid,(S)-Resatorvid,AK-242 (S enantiomer),(-)-AK-242

Target: Others

Tyrphostin B44, (+) enantiomer

Cat.No: T22450

Synonym: 酪氨酸磷酸化抑制剂AG 835

Target: EGFR

Siremadlin (R Enantiomer)

Cat.No: T12274

Synonym: Siremadlin R Enantiomer,HDM201 R Enantiomer,NVP-HDM201 R Enantiomer

Target: Others

Firsocostat S enantiomer

Cat.No: T12200

Synonym: ND-630 S enantiomer,NDI-010976 S enantiomer,GS-0976 S enantiomer

Target: Others

Duvelisib (R enantiomer)

Cat.No: T11129

Synonym: Duvelisib R enantiomer,IPI-145 R enantiomer,INK1197 R enantiomer

Target: PI3K

Fulvestrant (R enantiomer)

Cat.No: T11334

Synonym: ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer

Target: Others

Fulvestrant (S enantiomer)

Cat.No: T11335

Synonym: ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer

Target: Others

Bitopertin (R enantiomer)

Cat.No: T10552

Synonym: RO4917838 (R enantiomer),RG1678 (R enantiomer),Bitopertin R enantiomer

Target: GlyT

Gepotidacin S enantiomer

Cat.No: T11391

Synonym: GSK2140944 S enantiomer

Target: Others

Elacestrant S enantiomer

Cat.No: T11173

Synonym: RAD1901 S enantiomer

Target: Others

Tenalisib R Enantiomer

Cat.No: T13120

Synonym: RP6530 R Enantiomer

Target: Others

GLPG0492 (R enantiomer)

Cat.No: T11410

Synonym: GLPG0492 R enantiomer

Target: Others

RSV604 (R enantiomer)

Cat.No: T12775

Synonym: RSV604 R enantiomer

Target: Others

Seviteronel R enantiomer

Cat.No: T13312

Synonym: VT-464 (R enantiomer)

Target: Others

Talarozole (R enantiomer)

Cat.No: T13422L

Synonym: (R)-Talarozole,Talarozole R enantiomer

Target: Others

Nazartinib S-enantiomer

Cat.No: T11156

Synonym: EGF816 (S-enantiomer)

Target: Others

Atuveciclib S-Enantiomer

Cat.No: T10465

Synonym: BAY-1143572 S-Enantiomer

Target: CDK

Cobimetinib (R-enantiomer)

Cat.No: T10856

Synonym: 考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer

Target: Others

Elacestrant S enantiomer dihydrochloride

Cat.No: T11173L

Synonym: RAD1901 S enantiomer dihydrochloride,RAD-1901 S enantiomer dihydrochloride,RAD 1901 S enantiomer dihydrochloride

Target: Others

IACS-8968 R-enantiomer

Cat.No: T11627

Synonym: IDO/TDO Inhibitor (R-enantiomer)

Target: IDO

INT-777 R-enantiomer

Cat.No: T11662

Synonym: S-EMCA R enantiomer

Target: Others

ADU-S100 enantiomer ammonium salt

Cat.No: T10252L

Synonym: MIW815 enantiomer ammonium salt,ML RR-S2 CDA enantiomer ammonium salt

Target: Others

IACS-8968 S-enantiomer

Cat.No: T11628

Synonym: IDO/TDO Inhibitor (S-enantiomer)

Target: IDO

NITD-609 Enantiomer

Cat.No: T67880

Target: Others

GSK2850163 (S enantiomer)

Cat.No: T9848

Target: IRE1

THK5351 (R enantiomer)

Cat.No: T39541

LIN28 inhibitor LI71 enantiomer

Cat.No: T41114

Cenobamate S-Enantiomer

Cat.No: T10757

Target: Others

Silvestrol aglycone (enantiomer)

Cat.No: T12915

Target: Others

Enantiomer of Sofosbuvir

Cat.No: T11195

Target: Others

PNU-282987 S enantiomer hydrochloride

Cat.No: T22401

Synonym: (S)-PNU-282987 HCl

Target: Others

MK-7246 S enantiomer

Cat.No: T12067

Target: Others

Ribocil-C R enantiomer

Cat.No: T12723

Target: Others

Leu-AMS R enantiomer

Cat.No: T11841

Target: Others

Necrostatin 2 S enantiomer

Cat.No: T12203

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T5113	L-GLUCOSE L-葡萄糖,L-(-)-Glucose	Others	Others
	L-Glucose (L-(-)-Glucose) 是一种 D-glucose 的对映体，可促进食物的摄取。
T0185	Escitalopram Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体，是一种选择性 5-羟色胺再摄取抑制剂，Ki=0.89 nM，比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性，是一种研究抑郁症的抗抑郁药。
T5218	DL-Threitol	Others	Others
	DL-Threitol 是苏糖醇的 D-对映异构体。它具有作为人体代谢物的作用。它是 L-苏糖醇的对映异构体。
T20191	(-)-Camphoric acid (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-	GluR	Neuroscience
	(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体，樟脑酸可诱导 GluR 表达。
T10935	D-Glutamic acid (R)-Glutamic acid,D-谷氨酸	Endogenous Metabolite	Metabolism
	D-Glutamic acid ((R)-Glutamic acid) 是一种广泛用于药物和食品中的L-glutamic acid 对映异构体。
T12796	S-Dihydrodaidzein S-二氢大豆苷元,(3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one	Others	Others
	S-Dihydrodaidzein ((3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one) 是一种 dihydrodaidzein 的 (S) 型对映体。其中 dihydrodaidzein 是一种可食用性植物雌激素。
T1317	Cinchonidine 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine	5-HT Receptor; Serotonin Transporter; Parasite	GPCR/G Protein; Microbiology/Virology; Neuroscience
	Cinchonidine (L-Cinchonidine) 是在金鸡纳和角蒿中发现的一种生物碱，有抗疟活性。它是用于有机化学中不对称合成的砌块，是血清素转运蛋白的弱抑制剂。
T38251	L-Uridine	Nucleoside Antimetabolite/Analog; Antibiotic	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	L-Uridine 是从Polyporaceae fungus Poria cocos (Schw.)分离得到的正常 RNA 成分中的 D-尿苷的对映异构体，属于一种核苷，可充当核苷磷酸转移酶的磷酸受体。L-Uridine 具有潜在的抗病毒活性。
TN1448	(-)-Bornyl acetate L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯	p38 MAPK; NF-κB; JNK; Antifungal	MAPK; Microbiology/Virology; NF-κB
	(-)-Bornyl acetate (L-(-)-Bornyl acetate) 是存在于牛膝草油中的一种具有抗真菌活性的 (+)-Bornyl acetate 低活性异构体。
T4000	(±)-Equol Equol,(±)-雌马酚,(R,S)-Equol	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Drug Metabolite	Endocrinology/Hormones; Metabolism
	(±)-Equol ((R,S)-Equol) 是 equol 的外消旋体。它对 ERα 和 ERβ 的 EC50s of 分别为 200 和 74 nM。Equol 是大豆异黄酮黄豆苷和大豆黄素的代谢产物。
T6491	(-)-(S)-Equol (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	(-)-(S)-Equol (4',7-Dihydroxyisoflavan) 是雌激素受体β的高亲和力配体。
TQ0109	Cephaeline dihydrochloride (-)-Cephaeline dihydrochloride,盐酸吐根酚碱,NSC 32944	P450	Metabolism
	(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM).
T13464L	(-)-Ketoconazole (-)-R 41400,(-)-Ketoconazol	Others	Others
	(-)-Ketoconazole is one of the enantiomer of Ketoconazole. Ketoconazole is a racemic mixture of two enantiomers.
T40529	(R)-(-)-1,2-Propanediol
	(R)-(-)-1,2-Propanediol is the (R)-enantiomer of 1,2-Propanediol, which is derived from glucose through the expression of NADH-linked glycerol dehydrogenase genes in Escherichia coli.
T72509	Apoptosis inducer 5
	Apoptosisinducer 5 是一种木脂素对映异构体，存在于Crataegus pinnatifida 中。Apoptosisinducer 5 通过 Hep3B 细胞中的凋亡和自噬表现出细胞毒性作用。
T38497	(-)-Taxifolin (-)-二氢槲皮素,(-)-Dihydroquercetin
	(-)-Taxifolin is the less active enantiomer of Taxifolin, demonstrating vital anti-tyrosinase activity and notable inhibition against collagenase (IC50 = 193.3 μM). It is valued as an essential natural compound showing antifibrotic potential, while also acting as a capable free radical scavenger and possessing antioxidant capacity.
T40576	(S)-Salsolidine
	(S)-Salsolidine, a chemical compound, functions as a weak inhibitor of monoamine oxidase (MAO), exhibiting an inhibition constant (K i ) of 63 μM. R enantiomer demonstrating a greater efficacy than (S)-Salsolidine, boasting a K i value of 26 μM compared to the S form.
T83138	Aloinoside A
	Aloinoside A，一种可自黄芪分离的芦荟素，为Aloinoside B的对映异构体，应用于代谢研究的生物标志物。其通过大鼠肠道细菌代谢生成物包括芦荟苷、异芦荟苷及羟基代谢物。
TN4469	Lyoniresinol
	Lyoniresinol 是一种从 Tarenna attenuata 分离出来的木质素，具有清除自由基的活性（IC50为82.4μM）和 DPPH 的抗氧化活性，显示出抗黑色素生成活性。Lyoniresinol 有强烈的苦味，而其对映体(-)-Lyoniresinol 是无味的。

天然产物

Cat.No: T5113

Synonym: L-葡萄糖,L-(-)-Glucose

Target: Others

Cat.No: T0185

Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor

Cat.No: T5218

Target: Others

(-)-Camphoric acid

Cat.No: T20191

Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

Target: GluR

D-Glutamic acid

Cat.No: T10935

Synonym: (R)-Glutamic acid,D-谷氨酸

Target: Endogenous Metabolite

S-Dihydrodaidzein

Cat.No: T12796

Synonym: S-二氢大豆苷元,(3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one

Target: Others

Cat.No: T1317

Synonym: 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine

Target: 5-HT Receptor, Serotonin Transporter, Parasite

Cat.No: T38251

Target: Nucleoside Antimetabolite/Analog, Antibiotic

(-)-Bornyl acetate

Cat.No: TN1448

Synonym: L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯

Target: p38 MAPK, NF-κB, JNK, Antifungal

Cat.No: T4000

Synonym: Equol,(±)-雌马酚,(R,S)-Equol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite

Cat.No: T6491

Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite

Cephaeline dihydrochloride

Cat.No: TQ0109

Synonym: (-)-Cephaeline dihydrochloride,盐酸吐根酚碱,NSC 32944

Target: P450

(-)-Ketoconazole

Cat.No: T13464L

Synonym: (-)-R 41400,(-)-Ketoconazol

Target: Others

(R)-(-)-1,2-Propanediol

Cat.No: T40529

Apoptosis inducer 5

Cat.No: T72509

Cat.No: T38497

Synonym: (-)-二氢槲皮素,(-)-Dihydroquercetin

(S)-Salsolidine

Cat.No: T40576

Cat.No: T83138

Cat.No: TN4469

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