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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T72785 PRMT5:MEP50 PPI

PRMT5:MEP50 PPI是一款新型的抑制剂,专门针对PRMT5:MEP50蛋白-蛋白相互作用,展现了抗肿瘤活性,并对肺癌及前列腺癌细胞具有显著的抗增殖效果。
T9962 Mepolizumab

美泊利单抗,SB 240563

IL Receptor Immunology/Inflammation
Mepolizumab (SB 240563) 是一种中和 IL-5 的人源化单克隆抗体。 美泊利单抗可用于严重嗜酸性哮喘和嗜酸性肉芽肿伴多血管炎的研究。
T21425 Mephenytoin

Mesantoin,Methoin,Insulton,Phenantoin,美芬妥因,Methylphenetoin

P450 Metabolism
Mephenytoin (Phenantoin) 是 CYP2C19 及 CYP2B6 的底物,是一种抗惊厥剂。
T24449 Mepacrine

Haffkinine,Erion

Others Others
Mepacrine (Erion) 是一种吖啶衍生物,以前广泛用作抗疟药。它在细胞生物学实验中用作磷脂酶A2的抑制剂。
T2686 Esomeprazole Magnesium

(S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium

ATPase; Proton pump Membrane transporter/Ion channel
Esomeprazole Magnesium (NEXIUM) 是一种口服有效的 H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病中具有研究价值。Esomeprazole magnesium 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T6580 Meprednisone

SCH 4358,Methylprednisone,NSC 527579,Betanisona,Betapar,泼尼松

Glucocorticoid Receptor; Autophagy Autophagy; Endocrinology/Hormones
Meprednisone (Betapar) 是糖皮质激素,用于糖皮质激素受体,是泼尼松的甲基化衍生物。
T2687 Omeprazole sulfide

Omeprazole metabolite Omeprazole sulfide,Ufiprazole,奥美拉唑硫醚

Proton pump; Drug Metabolite Membrane transporter/Ion channel; Metabolism
Omeprazole sulfide (Ufiprazole) 是 Omeprazole 的代谢物。
T10138 4-Desmethoxy Omeprazole

Drug Metabolite Metabolism
4-Desmethoxy Omeprazole 是 Omeprazole 的活性代谢物。Omeprazole 是质子泵抑制剂。Omeprazole 竞争性抑制 CYP2C19 活性,Ki=2 - 6 μM。Omeprazole 还抑制革兰氏阴性菌和革兰氏阳性菌生长。
T64332 Glimepiride sulfonamide

Immunology/Inflammation related Immunology/Inflammation
Glimepiride sulfonamide 是一种抗炎活性化合物。
T71704 Navamepent

RX-10045

Others Others
Navamepent (RX-10045) 是 resolvin E1 (一种膳食-3多不饱和脂肪酸代谢物)的类似物,具有强大的抗炎活性,可减少角膜炎症、上皮损伤,加速角膜组织修复。Navamepent 可抑制角膜上皮细胞释放几种关键促炎介质。Navamepent 对干眼和杯状细胞损失非常有效,可加速泪液的产生。
T0257 Mepiroxol

Mepyroxol,Lysateril,3-吡啶基甲醇氮氧化物

Others Others
Mepiroxol (Lysateril) 是一种抗高血脂药,也称为 3-PYRIDINEMETHANOL N-OXIDE。
T0201 Meptazinol hydrochloride

Meptazinol HCl,盐酸美普他酚

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Meptazinol hydrochloride (Meptazinol HCl) 是一种独特的中枢opioid 类镇痛剂,用作具有镇痛特性的麻醉拮抗剂。
T22391 Omeprazole Sodium

P450; Proton pump; Antibacterial; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。
T2686L Esomeprazole Sodium

埃索美拉唑钠,(S)-Omeprazole sodium

ATPase; Proton pump Membrane transporter/Ion channel
Esomeprazole Sodium ((S)-Omeprazole sodium) 是一种口服有效的活性质子泵抑制剂。Esomeprazole sodium 通过抑制胃壁细胞中的 H+, K+-ATPase 来降低酸分泌,在胃食管反流疾病中有研究价值。Esomeprazole 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T2078 Fimepinostat

CUDC-907,PI3K/HDAC Inhibitor,CUDC 907

Apoptosis; PI3K; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Fimepinostat (CUDC 907) 是一种 I 型PI3K 及 I 和 II 型HDAC 酶抑制剂,作用于 PI3Kα/PI3Kβ/PI3Kδ 和 HDAC1/HDAC2/HDAC3/HDAC10 ,IC50分别为 19/54/39 nM 和 1.7/5.0/1.8/2.8 nM。
T22361 Mepivacaine

Carbocaine

Sodium Channel Membrane transporter/Ion channel
Mepivacaine (Carbocaine) 是一种可用于局部麻醉的酰胺类化合物,可使人或动物短暂的失去自知觉。Mepivacaine 通过与神经细胞膜上特定的电压门控钠离子通道结合,抑制钠离子内流和膜去极化来发挥作用。Mepivacaine 适用于神经阻滞和硬膜外麻醉。
T36839 (R)-Mephenytoin

R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin

Others Others
(R)-Mephenytoin ((–)-Mephenytoin) 是 Mephenytoin 的 R-对映体,Mephenytoin 是一种抗惊厥药。
T0997 Temephos

双硫磷,Temefos

AChR; Parasite Microbiology/Virology; Neuroscience
Temephos (Temefos) 是一种胆碱酯酶抑制剂,是一种有机硫代磷酸盐杀虫剂,用于治疗被携带疾病的昆虫侵染的水。
T21529 (S)-Mephenytoin

Others Others
(S)-Mephenytoin 是一种抗惊厥剂。(S)-Mephenytoin 作为细胞色素 P450 (CYP) 同种型 CYP2C19 的底物,可用于分析细胞色素 P450 代谢。
T8386 Esomeprazole Magnesium trihydrate

埃索美拉唑镁三水合物,埃索美拉唑镁(三水),(S)-Omeprazole magnesium trihydrate

Proton pump Membrane transporter/Ion channel
Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) 是一种口服有效的H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病的研究中具有价值。它是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。
T24451 Mepyramine

NSC-13136,NSC13136,NSC 13136

Mepyramine is a histamine H1 antagonist. It has mild hypnotic properties and some local anesthetic action and is used for allergies both parenterally and locally.
T1860 Imepitoin

AWD 131-138,ELB-138,伊匹妥英

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Imepitoin (AWD 131-138) 是一种新型的低亲和力部分苯二氮卓受体激动剂,有抗惊厥和抗焦虑作用。
T0015 Mephenesin

Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Mephenesin (Cresoxydiol) 是 NMDA 受体拮抗剂,也是中枢性肌松弛剂。
T40922 Fluroxypyr-meptyl

氟草烟-1-甲基庚基酯,Fluroxypyr-1-methylheptyl ester

Others Others
Fluroxypyr-meptyl (Fluroxypyr-1-methylheptyl ester) 是一种麦田除草剂。
T3444 Merimepodib

美泊地布,VX-497,VI-21497

Dehydrogenase; Antiviral; HCV Protease; HBV Immunology/Inflammation; Metabolism; Microbiology/Virology; Proteases/Proteasome
Merimepodib (VX-497) 是一种新型非竞争性肌苷一磷酸脱氢酶抑制剂,具有广谱抗病毒活性。
T0127 Glimepiride

Glimperide,HOE-490,格列美脲

Potassium Channel Membrane transporter/Ion channel
Glimepiride (HOE-490) 是一种中长效的磺酰脲类抗糖尿病化合物,其 ED50=182 μg/k。
T20626 Esomeprazole

Proton pump; Cysteine Protease Membrane transporter/Ion channel; Proteases/Proteasome
Esomeprazole 是奥美拉唑(omeprazole) 的S-异构体,抑制溶酶体半胱氨酸蛋白酶legumain,防止癌症转移。它是一种质子泵抑制剂(PPI)。
T0264 Zomepirac sodium salt

Zomepirac Sodium,佐美酸钠,McN-2783-21-98

PGE Synthase; PDE Immunology/Inflammation; Metabolism
Zomepirac sodium salt (McN-2783-21-98) 是前列腺素合成酶抑制剂。它是一种非甾体抗炎药,但能够导致免疫介导的肝损伤。
T7574 Meptyldinocap

敌螨普,2,4-DNOPC

Antibacterial Microbiology/Virology
Meptyldinocap (2,4-DNOPC) 是一种新型白粉病杀菌剂。
T16040 Mepazine

甲哌啶嗪,Pecazine

Apoptosis; MALT Apoptosis; Immunology/Inflammation
Mepazine (Pecazine) 是一种有效的特异性 MALT1 抑制剂。 Mepazine 抑制 GSTMALT1 全长和 GSTMALT1 325-760,IC50 为 0.83 μM 和 0.42 μM。 Mepazine 增强细胞凋亡并影响细胞活力。
T0946 Mepivacaine hydrochloride

Mepivacaine HCl,盐酸甲哌卡因

Sodium Channel Membrane transporter/Ion channel
Mepivacaine hydrochloride (Mepivacaine HCl) 是具有局部麻醉特性的酰胺衍生物。Mepivacaine hydrochloride 与神经元细胞膜上特定的电压门控钠离子通道结合,抑制钠离子内流和膜去极化。
T5333 Rimeporide hydrochloride

盐酸Rimeporide,EMD-87580 hydrochloride

Sodium Channel Membrane transporter/Ion channel
Rimeporide hydrochloride (EMD-87580 hydrochloride) 是一种有效的 Na+/H+交换泵(NHE-1) 选择性抑制剂。
T21746 Terameprocol

tetramethyl Nordihydroguaiaretic Acid,EM-1421

HIV Protease Microbiology/Virology; Proteases/Proteasome
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。
T12309 Omeprazole metabolite Omeprazole sulfone

Omeprazole sulphone,Omeprazole sulfone

Others Others
Omeprazole metabolite Omeprazole sulfone 是Omeprazole 的代谢物,能够抑制质子泵。
T5319 Rimeporide

EMD-87580

Sodium Channel Membrane transporter/Ion channel
Rimeporide (EMD-87580) 是有效的 Na+/H+交换泵 (NHE-1) 选择性抑制剂。
T0757 Omeprazole

Losec,Prilosec,奥美拉唑,奥美拉挫,H 16868,Antra

Proton pump; Phospholipase; Antibacterial; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Omeprazole (Losec) 是一种质子泵抑制剂,有研究胃肠道疾病的潜力。它竞争性抑制 CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阳性菌和革兰氏阴性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。
T1232 Mepyramine maleate

马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mepyramine maleate (Pyrilamine maleate) 是一种组胺 H1 拮抗剂,对 H1、H2 和 H3 受体的 Kd 值分别为 0.8、5200 和大于 3000 nM,对 H1 受体的 pKd 值为 9.4。它是感冒药的常见成分,具有温和的催眠特性和局部麻醉作用,可用于胃肠外和局部过敏。
T0765 Fomepizole

Antizol-Vet,4-甲基吡唑,甲吡唑,4-Methylpyrazole,Antizol

P450; CAT; AChR Metabolism; Neuroscience; oxidation-reduction
Fomepizole (4-Methylpyrazole) 是细胞色素 P450 (CYP2E1) 抑制剂。它是乙醇脱氢酶 (alcohol dehydrogenase) 竞争性抑制剂。它能够阻断甲醇和乙二醇进一步转化为有毒代谢产物。它具有成为乙二醇或甲醇中毒的解毒剂的潜力。
T4686 Simeprevir

TMC435,西咪匹韦,TMC-435350,Olysio

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Simeprevir (TMC435) 是一种有效的 HCV NS3/4A 蛋白酶抑制剂,抑制 HCV 复制,EC50 为 7.8 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。
T33288 Mepramidil

PF26,PF-26,PF 26

Mepramidil is a potential bioactive agent.
T69424 Zomepirac free acid

Zomepirac is a prostaglandin synthetase inhibitor. Zomepirac is an orally effective nonsteroidal anti-inflammatory drug (NSAID) that has antipyretic actions.
T71160 Levomepromazine HCl

Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS SYSTEM effects resembling those of chlorpromazine.
T20855 Gemeprost

SC-37681,SC 37681,Carprost,Gemeprostum,Cervagem,Preglandin

Gemeprost, an analog of prostaglandin E1, is used for the treatment of obstetric bleeding. It is used to terminate pregnancy up to 24 weeks gestation together with mifepristone.
T29410 3-Hydroxymephenytoin

3-Hydroxymephenytoin is a bioactive chemical.
T61740 Esomeprazole hemistrontium

Esomeprazole hemistrontium, also known as (S)-Omeprazole, is a potent and orally active proton pump inhibitor that effectively reduces acid secretion by inhibiting the H+, K+-ATPase in gastric parietal cells. This compound exhibits promising potential for research in symptomatic gastroesophageal reflux disease [1] [2] [3].
T16041 Mepixanox

甲哌呫诺,Pimexone

Others Others
Mepixanox is an analeptic drug. It is used for treating respiratory and cardiorespiratory insufficiency.
T39063 Azilsartan mepixetil

Azilsartan mepixetil is a potent angiotensin II receptor antagonist with enhanced efficacy and prolonged duration of action. It exhibits more prominent and sustained effects in lowering blood pressure and heart rate, while maintaining a high level of safety. Furthermore, Azilsartan mepixetil demonstrates optimal protective efficacy for cardiovascular and renal functions. Hence, it holds promise for the research and treatment of hypertension, chronic heart failure, and diabetic nephropathy.
T68994 Mepazine hydrochloride monohydrate

Mepazine hydrochloride monohydrate is a MALT1 inhibitor.
T37659 5-hydroxy Omeprazole

5-hydroxy Omeprazole is a major metabolite of omeprazole , an inhibitor of the gastric H+/K+-ATPase pump.[1] 5-hydroxy Omeprazole is produced from omeprazole by the action of cytochrome P450 (CYP) isoform 2C19, a monooxygenase. [2][3] CYP2C19 polymorphisms significantly influence the metabolism of omeprazole, and individuals may be classified as homozygous extensive metabolizers, heterozygous extensive metabolizers, and poor metabolizers.[1]
T9931 meplazumab

Others Others
meplazumab 是一种人源化抗 CD147 抗体,作为 COVID-19 肺炎患者的附加疗法。

化合物

PRMT5:MEP50 PPI
Cat.No: T72785
Synonym:
Target:
Mepolizumab
Cat.No: T9962
Synonym: 美泊利单抗,SB 240563
Target: IL Receptor
Mephenytoin
Cat.No: T21425
Synonym: Mesantoin,Methoin,Insulton,Phenantoin,美芬妥因,Methylphenetoin
Target: P450
Mepacrine
Cat.No: T24449
Synonym: Haffkinine,Erion
Target: Others
Esomeprazole Magnesium
Cat.No: T2686
Synonym: (S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium
Target: ATPase, Proton pump
Meprednisone
Cat.No: T6580
Synonym: SCH 4358,Methylprednisone,NSC 527579,Betanisona,Betapar,泼尼松
Target: Glucocorticoid Receptor, Autophagy
Omeprazole sulfide
Cat.No: T2687
Synonym: Omeprazole metabolite Omeprazole sulfide,Ufiprazole,奥美拉唑硫醚
Target: Proton pump, Drug Metabolite
4-Desmethoxy Omeprazole
Cat.No: T10138
Synonym:
Target: Drug Metabolite
Glimepiride sulfonamide
Cat.No: T64332
Synonym:
Target: Immunology/Inflammation related
Navamepent
Cat.No: T71704
Synonym: RX-10045
Target: Others
Mepiroxol
Cat.No: T0257
Synonym: Mepyroxol,Lysateril,3-吡啶基甲醇氮氧化物
Target: Others
Meptazinol hydrochloride
Cat.No: T0201
Synonym: Meptazinol HCl,盐酸美普他酚
Target: Opioid Receptor
Omeprazole Sodium
Cat.No: T22391
Synonym:
Target: P450, Proton pump, Antibacterial, Autophagy
Esomeprazole Sodium
Cat.No: T2686L
Synonym: 埃索美拉唑钠,(S)-Omeprazole sodium
Target: ATPase, Proton pump
Fimepinostat
Cat.No: T2078
Synonym: CUDC-907,PI3K/HDAC Inhibitor,CUDC 907
Target: Apoptosis, PI3K, HDAC
Mepivacaine
Cat.No: T22361
Synonym: Carbocaine
Target: Sodium Channel
(R)-Mephenytoin
Cat.No: T36839
Synonym: R-Mephenytoin,(R)-Mephenytoin,(–)-Mephenytoin
Target: Others
Temephos
Cat.No: T0997
Synonym: 双硫磷,Temefos
Target: AChR, Parasite
(S)-Mephenytoin
Cat.No: T21529
Synonym:
Target: Others
Esomeprazole Magnesium trihydrate
Cat.No: T8386
Synonym: 埃索美拉唑镁三水合物,埃索美拉唑镁(三水),(S)-Omeprazole magnesium trihydrate
Target: Proton pump
Mepyramine
Cat.No: T24451
Synonym: NSC-13136,NSC13136,NSC 13136
Target:
Imepitoin
Cat.No: T1860
Synonym: AWD 131-138,ELB-138,伊匹妥英
Target: GABA Receptor
Mephenesin
Cat.No: T0015
Synonym: Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl
Target: NMDAR, iGluR
Fluroxypyr-meptyl
Cat.No: T40922
Synonym: 氟草烟-1-甲基庚基酯,Fluroxypyr-1-methylheptyl ester
Target: Others
Merimepodib
Cat.No: T3444
Synonym: 美泊地布,VX-497,VI-21497
Target: Dehydrogenase, Antiviral, HCV Protease, HBV
Glimepiride
Cat.No: T0127
Synonym: Glimperide,HOE-490,格列美脲
Target: Potassium Channel
Esomeprazole
Cat.No: T20626
Synonym:
Target: Proton pump, Cysteine Protease
Zomepirac sodium salt
Cat.No: T0264
Synonym: Zomepirac Sodium,佐美酸钠,McN-2783-21-98
Target: PGE Synthase, PDE
Meptyldinocap
Cat.No: T7574
Synonym: 敌螨普,2,4-DNOPC
Target: Antibacterial
Mepazine
Cat.No: T16040
Synonym: 甲哌啶嗪,Pecazine
Target: Apoptosis, MALT
Mepivacaine hydrochloride
Cat.No: T0946
Synonym: Mepivacaine HCl,盐酸甲哌卡因
Target: Sodium Channel
Rimeporide hydrochloride
Cat.No: T5333
Synonym: 盐酸Rimeporide,EMD-87580 hydrochloride
Target: Sodium Channel
Terameprocol
Cat.No: T21746
Synonym: tetramethyl Nordihydroguaiaretic Acid,EM-1421
Target: HIV Protease
Omeprazole metabolite Omeprazole sulfone
Cat.No: T12309
Synonym: Omeprazole sulphone,Omeprazole sulfone
Target: Others
Rimeporide
Cat.No: T5319
Synonym: EMD-87580
Target: Sodium Channel
Omeprazole
Cat.No: T0757
Synonym: Losec,Prilosec,奥美拉唑,奥美拉挫,H 16868,Antra
Target: Proton pump, Phospholipase, Antibacterial, Autophagy
Mepyramine maleate
Cat.No: T1232
Synonym: 马来酸吡纳明,Pyrilamine maleate,吡拉明马来酸盐
Target: Histamine Receptor
Fomepizole
Cat.No: T0765
Synonym: Antizol-Vet,4-甲基吡唑,甲吡唑,4-Methylpyrazole,Antizol
Target: P450, CAT, AChR
Simeprevir
Cat.No: T4686
Synonym: TMC435,西咪匹韦,TMC-435350,Olysio
Target: HCV Protease, SARS-CoV
Mepramidil
Cat.No: T33288
Synonym: PF26,PF-26,PF 26
Target:
Zomepirac free acid
Cat.No: T69424
Synonym:
Target:
Levomepromazine HCl
Cat.No: T71160
Synonym:
Target:
Gemeprost
Cat.No: T20855
Synonym: SC-37681,SC 37681,Carprost,Gemeprostum,Cervagem,Preglandin
Target:
3-Hydroxymephenytoin
Cat.No: T29410
Synonym:
Target:
Esomeprazole hemistrontium
Cat.No: T61740
Synonym:
Target:
Mepixanox
Cat.No: T16041
Synonym: 甲哌呫诺,Pimexone
Target: Others
Azilsartan mepixetil
Cat.No: T39063
Synonym:
Target:
Mepazine hydrochloride monohydrate
Cat.No: T68994
Synonym:
Target:
5-hydroxy Omeprazole
Cat.No: T37659
Synonym:
Target:
meplazumab
Cat.No: T9931
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T10147 4-Hydroxymephenytoin

(+/-)-4'-Hydroxymephenytoin

Others; Drug Metabolite Metabolism; Others
4-Hydroxymephenytoin ((+/-)-4'-Hydroxymephenytoin) 是抗癫痫药 mephenytoin 的代谢产物。Mephenytoin 是 CYP2C19的配体。
TN4664 Norarmepavine

Others Others
N-norarmepavine shows significant cytotoxic activities against HL-60 carcinoma cell line with inhibitory ratios of 51.43% at concentration of 1 x 10(-5) M. Norarmepavine shows inhibition against Trypanosoma cruzi. D-(+)- N-norarmepavine exhibits significa
T3775 Armepavine

亚美罂粟碱,R-Armepavine,(-)-Armepavine

IκB/IKK; NF-κB NF-κB
Armepavine (R-Armepavine) 是来自Nelumbo nucifera 的活性化合物,能够抑制 TNF-α 诱导的MAPK 和NF-κB 信号级联反应。它不仅对人外周血单核细胞具有抗炎作用,且对 T 淋巴细胞和狼疮肾炎小鼠也具有免疫抑制作用。

天然产物

4-Hydroxymephenytoin
Cat.No: T10147
Synonym: (+/-)-4'-Hydroxymephenytoin
Target: Others, Drug Metabolite
Norarmepavine
Cat.No: TN4664
Synonym:
Target: Others
Armepavine
Cat.No: T3775
Synonym: 亚美罂粟碱,R-Armepavine,(-)-Armepavine
Target: IκB/IKK, NF-κB
Cat. No. Product Name Species Expression System
TMPY-01318 Meprin alpha/MEP1A Protein, Mouse, Recombinant (His)

meprin A, alpha (PABA peptide hydrolase),AW107200,<...

Mouse HEK293 Cells
Meprin alpha/MEP1A Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69 kDa and the accession number is A0A0R4J043.
TMPY-00504 EphB6 Protein, Mouse, Recombinant (His)

EPH receptor B6,Mep,Cekl

Mouse HEK293 Cells
EphB6 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 61.1 kDa and the accession number is O08644-1.
TMPY-02171 Cathepsin L Protein, Mouse, Recombinant (His)

Ctsl1,1190035F06Rik,nkt,cathepsin L,MEP,fs

Mouse HEK293 Cells
Cathepsin L Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.3 kDa and the accession number is P06797.
TMPJ-00508 CTSL Protein, Human, Recombinant (His)

CTSL,CTSL1,Cathepsin L1,Major Excreted Protein,MEP

Human HEK293 Cells
Cathepsin L is an enzyme. Cathepsin L, a lysosomal endopeptidase expressed in most eukaryotic cells, is a member of the papain-like family of cysteine proteinases. Cathepsin L plays a major role in antigen processing, tumor invasion and metastasis, bone resorption, and turnover of intracellular and secreted proteins involved in growth regulation. Unlike the precursor forms of other papain family members, the 43 kDa pro-cathepsin L itself is secreted from various cells. Pro-cathepsin L is the maj...
TMPY-00734 Cathepsin L Protein, Human, Recombinant (His)

MEP,CTSL1,CTSL,cathepsin L,FLJ31037,CATL

Human HEK293 Cells
Cathepsin L Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.3 kDa and the accession number is A0A024R276.
TMPY-03916 Neurolysin Protein, Human, Recombinant (His)

NLN,EP24.16,KIAA1226,MEP,neurolysin (metallopeptida...

Human E. coli
Neurolysin Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 78.7 kDa and the accession number is Q9BYT8.
TMPY-01737 Meprin alpha/MEP1A Protein, Human, Recombinant (His)

meprin A, α (PABA peptide hydrolase),mepri...

Human HEK293 Cells
Meprin alpha/MEP1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 67.7 kDa and the accession number is Q16819.
TMPK-01095 MEPE Protein, Mouse, Recombinant (His)

Osteoregulin,MEPE,OF45

Mouse HEK293 Cells
Matrix extracellular phosphoglycoprotein (MEPE) is expressed in bone and teeth where it has multiple functions. The C-terminus of MEPE contains a mineral-binding, acidic serine- and aspartate-rich motif (ASARM) that is also present in other noncollagenous proteins of mineralized tissues.MEPE-derived ASARM peptides function in phosphate homeostasis and direct inhibition of bone mineralization in a phosphorylation-dependent manner.
TMPY-00261 Meprin beta Protein, Human, Recombinant (His)

meprin A, β,Meprin β,meprin A, be...

Human HEK293 Cells
MEP1B (Meprin A Subunit Beta) is a Protein Coding gene. This gene encodes the beta subunit. Targeted disruption of this gene in mice affects embryonic viability, renal gene expression profiles, and distribution of the membrane-associated alpha subunit in the kidney and intestine. Meprins are cell membrane, oligomeric metalloendopeptidases composed of two distinct but evolutionarily related subunits, alpha, and beta. MEP1A is mapped to the short arm of chromosome 6 by the use of radiation and som...
TMPH-03140 Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His)

Plasmodium falciparum E. coli
During the asexual blood stage, catalyzes the initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation; specifically cleaves between Phe-33 and Leu-34 of Hb alpha-chain. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 41.0 k...
TMPH-03142 Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc)

Plasmodium falciparum E. coli
During the asexual blood stage, participates in initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation. May cleave preferentially denatured hemoglobin that has been cleaved by PMI. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. T...
TMPH-03141 Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc)

Plasmodium falciparum Baculovirus Insect Cells
During the asexual blood stage, participates in initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation. May cleave preferentially denatured hemoglobin that has been cleaved by PMI. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predict...
TMPH-00557 DXP reductoisomerase Protein, E. coli, Recombinant (His & Myc)

1-deoxy-D-xylulose 5-phosphate reductoisomerase,DXP reductoi...

E. coli E. coli
Catalyzes the NADP-dependent rearrangement and reduction of 1-deoxy-D-xylulose-5-phosphate (DXP) to 2-C-methyl-D-erythritol 4-phosphate (MEP).

重组蛋白

Meprin alpha/MEP1A Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01318
Species: Mouse
Expression System: HEK293 Cells
EphB6 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00504
Species: Mouse
Expression System: HEK293 Cells
Cathepsin L Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02171
Species: Mouse
Expression System: HEK293 Cells
CTSL Protein, Human, Recombinant (His)
Cat.No: TMPJ-00508
Species: Human
Expression System: HEK293 Cells
Cathepsin L Protein, Human, Recombinant (His)
Cat.No: TMPY-00734
Species: Human
Expression System: HEK293 Cells
Neurolysin Protein, Human, Recombinant (His)
Cat.No: TMPY-03916
Species: Human
Expression System: E. coli
Meprin alpha/MEP1A Protein, Human, Recombinant (His)
Cat.No: TMPY-01737
Species: Human
Expression System: HEK293 Cells
MEPE Protein, Mouse, Recombinant (His)
Cat.No: TMPK-01095
Species: Mouse
Expression System: HEK293 Cells
Meprin beta Protein, Human, Recombinant (His)
Cat.No: TMPY-00261
Species: Human
Expression System: HEK293 Cells
Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His)
Cat.No: TMPH-03140
Species: Plasmodium falciparum
Expression System: E. coli
Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc)
Cat.No: TMPH-03142
Species: Plasmodium falciparum
Expression System: E. coli
Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc)
Cat.No: TMPH-03141
Species: Plasmodium falciparum
Expression System: Baculovirus Insect Cells
DXP reductoisomerase Protein, E. coli, Recombinant (His & Myc)
Cat.No: TMPH-00557
Species: E. coli
Expression System: E. coli
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