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60

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8808L LYN-1604 dihydrochloride

LYN-1604 2HCl(2216753-86-3 free base)

Apoptosis; Autophagy Apoptosis; Autophagy
LYN-1604 2HCl 是一种有效的 UNC-51 样激酶 1 激活剂,EC50值为 18.94 nM。LYN-1604 可研究三阴性乳腺癌。
TP2008L Lyn peptide inhibitor acetate

Lyn peptide inhibitor acetate(222018-18-0 free base)

IL Receptor Immunology/Inflammation
Lyn peptide inhibitor acetate(222018-18-0 free base) 是一种有效的细胞渗透性 Lyn 偶联 IL-5 受体信号通路抑制剂,同时保持其他信号完整。它阻断 Lyn 活化并抑制 Lyn 酪氨酸激酶与 IL-3/GM-CSF/IL-5 受体的 βc 亚基的结合。它可用于哮喘、过敏和其他嗜酸性粒细胞疾病的研究。
T11916 Lyn-IN-1

巴非替尼,Bafetinib analog

Bcr-Abl; Src Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Lyn-IN-1 (Bafetinib analog) 是一种高活性 Bcr-Abl 和 Lyn 双重抑制剂。
T39687 LYN-1604 hydrochloride

LYN-1604 hydrochloride, a powerful activator of UNC-51-like kinase 1 (ULK1) with an EC50 value of 18.94 nM, has significant implications in the study of triple-negative breast cancer (TNBC).
T4123 LYN-1604

LYN1604

Apoptosis; Autophagy Apoptosis; Autophagy
LYN-1604 是一种新型 ULK1 激活剂,EC50值为 18.94 nM。它可诱导参与 ATF3、RAD21 和 caspase3 的细胞死亡,并伴有自噬和细胞凋亡,可研究三阴性乳腺癌。
TP2008 Lyn peptide inhibitor

Cell-permeable inhibitor of Lyn-dependent effects of the IL-5 receptor. Blocks binding of Lyn tyrosine kinase to βc subunit of IL-3/GM-CSF/IL-5 receptors, blocking Lyn activation. Inhibits IL-5 receptor-mediated eosinophil differentiation and survival in
T75806 Lyn peptide inhibitor TFA

Lyn peptide inhibitor TFA 是一种有效的,可以细胞渗透的抑制剂,抑制Lyn 偶联的IL-5受体相关信号通路,同时保持其他信号的完整。Lyn peptide inhibitor TFA 可以阻断 Lyn 的激活,抑制 Lyn 酪氨酸激酶与 IL-3/GM-CSF/IL-5 受体的 βc 亚基结合。Lyn peptide inhibitor TFA 可用于哮喘、过敏等嗜酸性疾病的研究。
T13186 TL02-59

Apoptosis; Src; Hck Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
TL02-59 是 Src 家族激酶中 Fgr 的特异性抑制剂 (IC50 = 0.03 nM)。 TL02-59 抑制 Lyn 和 Hck,IC50 分别为 0.1 nM 和 160 nM。 TL02-59 有效抑制急性髓性白血病细胞的生长。
T31011 Coralyne chloride

Topoisomerase DNA Damage/DNA Repair
Coralyne chloride 是一种具有强抗癌活性的原小檗碱。它可用于制备 Coralyne 衍生物,是一种基于荧光 DNA 的分子整流剂,通过位点特异性插入构建成 DNA 双链体。它可作为一种拓扑异构酶 I 毒性分子,诱导拓扑异构酶 I 介导 DNA 裂解。
T1260 Cromolyn sodium

Disodium Cromoglycate,FPL 670 (Cromolyn) Disodium,FPL-670,色甘酸钠,Sodium cromoglycate

Others; Potassium Channel; GSK-3; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others; PI3K/Akt/mTOR signaling; Stem Cells
Cromolyn sodium (FPL-670) 是一种GSK-3β抑制剂,IC50为 2.0 µM,有抗过敏作用。
T31715 Ethynylestradiol mixture with lynestrenol

Ethynylestradiol mixture with lynestrenol is a drug/ therapeutic agent with reproductive effect.
T19656 Pyrazolynate

SW-751,BRN 0860937,Pyrazolate

Pyrazolynate is a herbicide. It is used to evaluate the hydrolyzation to destosyl pyrazolynate (DTP).
T31977 GLYN

NSC 137875,NSC137875,Glycidyl nitrate,NSC-137875

GLYN, a nitric oxide donor, acts by enhancing the therapeutic efficacy of chemotherapy and radiotherapy.
T80275 Lynronne-2

Lynronne-2是抗菌肽,对革兰氏阳性细菌,包含MDR菌株具有活性(耐甲氧西林MRSA菌株MIC: 32-256 μg/mL)。该化合物亦对P. aeruginosa感染展现效用。
T20188 Polynoxylin

Formaldehyde, urea polymer,Gabrite,Hygromull,HSDB 7203

Polynoxylin is an antiseptic. It is used for local treatment of the skin and the mouth.
TP2450 Argipressin, des-glynh2(9)-

9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin

Argipressin, des-glynh2(9)-, can effect on aggregation of blood platelets.
T38326 Cromolyn (sodium salt hydrate)

Cromolyn is a chromone complex that acts as a mast cell stabilizer, preventing the release of histamine. Its mechanism of action is thought to involve an interference with the antigen-stimulated calcium transport across the mast cell membrane, thereby inhibiting mast cell release of histamine, leukotrienes, and other substances that cause hypersensitivity reactions.
T40961 Lynamicin B

Lynamicin B, a promising pesticide, functions as a selective chitinase inhibitor exclusive to lepidoptera. It exhibits a Ki value of 8.76 μM, indicating its potential efficacy.
T33032 Lynestrenol mixture with mestranol

Lynestrenol mixture with mestranol is a bioactive chemical.
T23959 Dactylyne

Dactylyne is a new drug metabolism inhibitor of marine origin. It was isolated from the sea hare Aplysia dactylomela and characterized pharmacologically.
T7974L Lynestrenol acetate

Lynestrenol acetate is a bioactive chemical.
T80274 Lynronne-1

Lynronne-1 是一种具备抗革兰氏阳性细菌能力的抗菌肽,尤其对包括多重耐药(MDR)菌株有效(MRSA菌株的MIC为8-32 μg/mL)。在MRSA感染的伤口小鼠模型中,Lynronne-1能显著降低细菌负荷。此外,Lynronne-1对P. aeruginosa感染也显示出活性。
T33034 Lyngbyatoxin B

Lyngbyatoxin B is an irritant form Lyngbya majuscula.
T80276 Lynronne-3

Lynronne-3 是一种具有抗革兰氏阳性细菌活性的抗菌肽,涵盖 MDR 菌株(对MRSA菌株的 MIC 为 32-128 μg/mL)。此外,Lynronne-3 亦对 P. aeruginosa 感染显示出效力。
TQ0132 A 419259 trihydrochloride

RK 20449 trihydrochloride

Src Angiogenesis; Tyrosine Kinase/Adaptors
A 419259 trihydrochloride (RK 20449 trihydrochloride) 是一种 Src 家族激酶抑制剂,能够抑制 Src (IC50:9 nM)、Lck (IC50:3 nM)、Lyn (IC50:3 nM)。
T6311 Bafetinib

NS-187,巴氟替尼,INNO-406

Bcr-Abl; Src; Autophagy Angiogenesis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Bafetinib (INNO-406) 是一种特异性双重 Bcr-Abl/Lyn 抑制剂,IC50值为5.8和19 nM。
T6997 SU6656

FAK; Akt; Src Angiogenesis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
SU6656 是Src 家族激酶抑制剂,抑制 Src,Yes,Lyn,Fyn 的IC50分别为 280,20,130,170 nM。它还能抑制p-AKT。它可抑制FAK Y576/577、 Y925、Y861位点的磷酸化。
T6078 Saracatinib

AZD0530,塞卡替尼

EGFR; Src; BTK; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Saracatinib (AZD0530) 是一种有效的 Src 抑制剂,抑制 c-Src、Lck、c-YES、Lyn、Fyn、Fgr 和 Blk 的 IC50值在 2.7 到 11 nM 之间,对其他酪氨酸激酶具有选择性。
T17267 XL228

IGF-1R; Bcr-Abl; Src; Aurora Kinase Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
XL228 是一种多靶点酪氨酸激酶抑制剂,对 Bcr-Abl、Aurora A、IGF-1R、Src 和 Lyn 的 IC50 分别为 5、3.1、1.6、6.1和 2 nM。
T6174 R406

R-406 besylate

Apoptosis; FLT; Syk Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
R406 (R-406 besylate) 是一种具有口服活性的 ATP 竞争性 Syk/FLT3抑制剂,Ki 为 30 nM。它有效抑制 Syk 激酶活性,IC50为 41 nM。它还抑制 Lyn 和 Lck,IC50值分别为 63 nM 和 37 nM。它可减轻免疫复合物介导的炎症。
T6115 Fostamatinib

R788,福他替尼

FLT; Syk; Monoamine Transporter; Adenosine Receptor Angiogenesis; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience; Tyrosine Kinase/Adaptors
Fostamatinib (R788) 是一种口服具有活力的 R406 前药。其中R406 是具有口服活性的,有效的,ATP 竞争性的Syk/FLT3抑制剂(Ki:30 nM,IC50:41 nM),也能够抑制 Lyn (IC50:63 nM) 和 Lck (IC50:37 nM)。
T6896 Tolimidone

托利咪酮,NSC 314335,MLR-1023,CP-26154

Src Angiogenesis; Tyrosine Kinase/Adaptors
Tolimidone (NSC 314335) 是选择性的 Lyn kinase 变构激活剂,其 EC50=63 nM。
T2600 AG490

Zinc02557947,Tyrphostin AG 490,AG 490,AG-490,Tyrphostin B42

EGFR; JAK; STAT; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
AG490 (Tyrphostin B42) 是一种 EGFR 抑制剂 ,IC50为 0.1 μM。它对 EGFR 的选择性比 ErbB2 高 135 倍,还抑制 JAK2。
T6093 AZD-7762

AZD7762

Chk Cell Cycle/Checkpoint
AZD-7762 是一种有效的 ATP 竞争性的细胞周期检测点激酶抑制剂,抑制 Chk1的 IC50为 5 nM。
T6318 AZ 628

Apoptosis; Raf Apoptosis; MAPK
AZ 628 是一种泛Raf 激酶抑制剂,抑制B-Raf、B-RafV600E 和c-Raf-1,IC50分别为 105、34和 29 nM。
T2640 Rebastinib

DCC2036,DCC 2036,DCC-2036

Apoptosis; FLT; Bcr-Abl; Src Angiogenesis; Apoptosis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Rebastinib (DCC-2036) 是一种口服有效的,非 ATP 竞争性的 Bcr-Abl 抑制剂,作用于 Abl1WT 和 Abl1T315I,IC50分别为 0.8 nM 和 4 nM,还抑制 LYN、SRC、HCK、FGR、FLT3、KDR 和 Tie-2,对 c-Kit 的活性低。Rebastinib 对 Angiopoietin2-Tie2通路具有抑制作用。
T4263 BAY 61-3606

2-[[7-(3,4-二甲氧基苯基)咪唑并[1,2-C]嘧啶-5-基]氨基]-3-吡啶甲酰胺,Syk inhibitor IV

Apoptosis; Syk Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
BAY 61-3606 (Syk inhibitor IV) 是一种具有口服活性的,ATP 竞争性的可逆选择性Syk 抑制剂。它作用于乳腺癌细胞,通过下调 Mcl-1 促进 TRAIL 诱导的细胞凋亡。它降低神经母细胞瘤细胞中的 ERK1/2 和 Akt 磷酸化,也降低 K-rn 细胞裂解物中 Syk 磷酸化。
T4337 PCI 29732

PCI29732,PCI-29732

Others; BCRP; BTK Angiogenesis; Membrane transporter/Ion channel; Others; Tyrosine Kinase/Adaptors
PCI 29732 是一种有效的可逆BTK 抑制剂,对 BTK、Lck 和 Lyn 的Kiapp 值分别为 8.2、4.6 和 2.5 nM。它通过竞争性结合ABCG2 的 ATP 结合位点来抑制ABCG2的功能。
T2467 R406 free base

R406 (free base)

Apoptosis; FLT; Syk Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
R406 free base (R406(free base)) 是一种具有口服活性的,ATP 竞争性的Syk/FLT3抑制剂,Ki 为 30 nM。它有效抑制 Syk 激酶活性,IC50为 41 nM,可减轻免疫复合物介导的炎症。它还抑制 Lyn 和 Lck,IC50分别为 63 nM 和 37 nM。
T16364 Infigratinib phosphate

NVP-BGJ398 phosphate,BGJ-398 phosphate

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
Infigratinib phosphate (BGJ-398 phosphate) 是 FGFR 抑制剂,对 FGFR1,FGFR2 和 FGFR3 的 IC50 分别为0.9,1.4 和 1 nM,比对 FGFR4 和 VEGFR2 的抑制性高40倍,对 Abl,Fyn,Kit,Lck 和 Lyn 几乎无活性。
T2605 Fostamatinib Disodium

Tamatinib Fosdium,福他替尼二钠盐,R788(Disodium),R788 Disodium,R788 (Fostamatinib) Disodium

FLT; Syk Angiogenesis; Tyrosine Kinase/Adaptors
Fostamatinib Disodium (R788 Disodium) 是一种口服具有活力的 R406 前药。其中R406 是具有口服活性的,有效的,ATP 竞争性的Syk/FLT3抑制剂(Ki:30 nM,IC50:41 nM),也能够抑制 Lyn (IC50:63 nM) 和 Lck (IC50:37 nM)。
T2609 Masitinib

AB1010,马赛替尼

Apoptosis; FAK; c-Fms; FGFR; Bcr-Abl; PDGFR; Src; c-Kit; Hck Angiogenesis; Apoptosis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Masitinib (AB1010) 是生物口服可利用的选择性 c-Kit 抑制剂 (对于人重组c-Kit,IC50=200 nM),它还抑制PDGFRα/β(IC50s=540/800 nM),Lyn(对 LynB 的IC50=510 nM),Lck,较小程度上抑制FGFR3和FAK。它有抗增殖,促凋亡活性,且毒性低。
T10206 A 419259

RK-20449

Src Angiogenesis; Tyrosine Kinase/Adaptors
A 419259 is a pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family (IC50s: 9 nM, <3 nM and <3 nM for Src, Lck and Lyn).
T71819 RK-20448

RK-20448 is an ATP-competitive inhibitor of Lck, Src, KDR/VEGF2R, and Tie-2. It also inhibits BLK, Csk, Fyn, and Lyn. RK-20448 is the cis isomer of A-419259
T15725 Lck inhibitor 2

Others Others
Lck inhibitor 2 is a bis-anilinopyrimidine inhibitor of tyrosine kinases including LCK, BTK, LYN, SYK, and TXK (IC50s: 13nM, 9nM, 3nM, 26nM, and 2nM for Lck, Btk, Lyn, Btk, and Txk respectively).
T13156 TG 100572

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 nM for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src, Yes, respectively).
T22597 Bafetinib (INNO-406)

Others Others
Bafetinib is a potent and selective dual inhibitor of Bcr-Abl/Lyn tyrosine kinase (IC50: 5.8nM and 19nM, respectively).
T16583 Propargyl-PEG1-acid

Others Others
Propargyl-PEG1-acid, a PEG-based PROTAC linker, enables the synthesis of BTK-CRBN PROTACs, specifically Ibrutinib-based PROTAC 4 and PROTAC 5. At a concentration of 10 μM, PROTAC 5 facilitates the degradation of BTK and induces the degradation of CSK, LYN, and LAT2[1].
T13157L TG 100801 Hydrochloride

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a inhibitor of multi-targeted kinase(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.1, 0.4, 1, 0.2 for VEGFR1, VEGFR2, FGFR1, FGFR2, PDGFRβ, Fgr, Fyn, Hck, Lck, Lyn, Src,
T63967 Multi-kinase-IN-2

Multi-kinase-IN-2 是口服具有活力的血管激酶 (angiokinase) 抑制剂。Multi-kinase-IN-2 能够显著抑制血管激酶的活性,如 VEGFR-1/2/3、PDGFRα/β、FGFR-1、LYN 和 c-KIT 激酶。Multi-kinase-IN-2 能够明显减弱 AKT 和 ERK 蛋白的磷酸化,并可诱导细胞凋亡 (apoptosis),具有抗癌作用。

化合物

LYN-1604 dihydrochloride
Cat.No: T8808L
Synonym: LYN-1604 2HCl(2216753-86-3 free base)
Target: Apoptosis, Autophagy
Lyn peptide inhibitor acetate
Cat.No: TP2008L
Synonym: Lyn peptide inhibitor acetate(222018-18-0 free base)
Target: IL Receptor
Lyn-IN-1
Cat.No: T11916
Synonym: 巴非替尼,Bafetinib analog
Target: Bcr-Abl, Src
LYN-1604 hydrochloride
Cat.No: T39687
Synonym:
Target:
LYN-1604
Cat.No: T4123
Synonym: LYN1604
Target: Apoptosis, Autophagy
Lyn peptide inhibitor
Cat.No: TP2008
Synonym:
Target:
Lyn peptide inhibitor TFA
Cat.No: T75806
Synonym:
Target:
TL02-59
Cat.No: T13186
Synonym:
Target: Apoptosis, Src, Hck
Coralyne chloride
Cat.No: T31011
Synonym:
Target: Topoisomerase
Cromolyn sodium
Cat.No: T1260
Synonym: Disodium Cromoglycate,FPL 670 (Cromolyn) Disodium,FPL-670,色甘酸钠,Sodium cromoglycate
Target: Others, Potassium Channel, GSK-3, Calcium Channel
Ethynylestradiol mixture with lynestrenol
Cat.No: T31715
Synonym:
Target:
Pyrazolynate
Cat.No: T19656
Synonym: SW-751,BRN 0860937,Pyrazolate
Target:
GLYN
Cat.No: T31977
Synonym: NSC 137875,NSC137875,Glycidyl nitrate,NSC-137875
Target:
Lynronne-2
Cat.No: T80275
Synonym:
Target:
Polynoxylin
Cat.No: T20188
Synonym: Formaldehyde, urea polymer,Gabrite,Hygromull,HSDB 7203
Target:
Argipressin, des-glynh2(9)-
Cat.No: TP2450
Synonym: 9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin
Target:
Cromolyn (sodium salt hydrate)
Cat.No: T38326
Synonym:
Target:
Lynamicin B
Cat.No: T40961
Synonym:
Target:
Lynestrenol mixture with mestranol
Cat.No: T33032
Synonym:
Target:
Dactylyne
Cat.No: T23959
Synonym:
Target:
Lynestrenol acetate
Cat.No: T7974L
Synonym:
Target:
Lynronne-1
Cat.No: T80274
Synonym:
Target:
Lyngbyatoxin B
Cat.No: T33034
Synonym:
Target:
Lynronne-3
Cat.No: T80276
Synonym:
Target:
A 419259 trihydrochloride
Cat.No: TQ0132
Synonym: RK 20449 trihydrochloride
Target: Src
Bafetinib
Cat.No: T6311
Synonym: NS-187,巴氟替尼,INNO-406
Target: Bcr-Abl, Src, Autophagy
SU6656
Cat.No: T6997
Synonym:
Target: FAK, Akt, Src
Saracatinib
Cat.No: T6078
Synonym: AZD0530,塞卡替尼
Target: EGFR, Src, BTK, Autophagy
XL228
Cat.No: T17267
Synonym:
Target: IGF-1R, Bcr-Abl, Src, Aurora Kinase
R406
Cat.No: T6174
Synonym: R-406 besylate
Target: Apoptosis, FLT, Syk
Fostamatinib
Cat.No: T6115
Synonym: R788,福他替尼
Target: FLT, Syk, Monoamine Transporter, Adenosine Receptor
Tolimidone
Cat.No: T6896
Synonym: 托利咪酮,NSC 314335,MLR-1023,CP-26154
Target: Src
AG490
Cat.No: T2600
Synonym: Zinc02557947,Tyrphostin AG 490,AG 490,AG-490,Tyrphostin B42
Target: EGFR, JAK, STAT, Autophagy
AZD-7762
Cat.No: T6093
Synonym: AZD7762
Target: Chk
AZ 628
Cat.No: T6318
Synonym:
Target: Apoptosis, Raf
Rebastinib
Cat.No: T2640
Synonym: DCC2036,DCC 2036,DCC-2036
Target: Apoptosis, FLT, Bcr-Abl, Src
BAY 61-3606
Cat.No: T4263
Synonym: 2-[[7-(3,4-二甲氧基苯基)咪唑并[1,2-C]嘧啶-5-基]氨基]-3-吡啶甲酰胺,Syk inhibitor IV
Target: Apoptosis, Syk
PCI 29732
Cat.No: T4337
Synonym: PCI29732,PCI-29732
Target: Others, BCRP, BTK
R406 free base
Cat.No: T2467
Synonym: R406 (free base)
Target: Apoptosis, FLT, Syk
Infigratinib phosphate
Cat.No: T16364
Synonym: NVP-BGJ398 phosphate,BGJ-398 phosphate
Target: FGFR
Fostamatinib Disodium
Cat.No: T2605
Synonym: Tamatinib Fosdium,福他替尼二钠盐,R788(Disodium),R788 Disodium,R788 (Fostamatinib) Disodium
Target: FLT, Syk
Masitinib
Cat.No: T2609
Synonym: AB1010,马赛替尼
Target: Apoptosis, FAK, c-Fms, FGFR, Bcr-Abl, PDGFR, Src, c-Kit, Hck
A 419259
Cat.No: T10206
Synonym: RK-20449
Target: Src
RK-20448
Cat.No: T71819
Synonym:
Target:
Lck inhibitor 2
Cat.No: T15725
Synonym:
Target: Others
TG 100572
Cat.No: T13156
Synonym:
Target: VEGFR
Bafetinib (INNO-406)
Cat.No: T22597
Synonym:
Target: Others
Propargyl-PEG1-acid
Cat.No: T16583
Synonym:
Target: Others
TG 100801 Hydrochloride
Cat.No: T13157L
Synonym:
Target: VEGFR
Multi-kinase-IN-2
Cat.No: T63967
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5S1058 Triptonide

雷公藤内酯酮,PG 492,NSC 165677

Apoptosis; Wnt/beta-catenin; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Stem Cells
Triptonide (PG 492) 是从雷公藤中鉴定出的一种天然产物,是一种 Wnt 信号抑制剂,其 IC50约为 0.3 nM。它具有免疫抑制、抗炎、避育、神经保护和抗淋巴瘤作用。
T7974 Lynestrenol

Progesterone Receptor Others
Lynestrenol 是孕烷 X 受体 (PXR) 激动剂,能够作用于 hPXR(EC50:41 µM) 和 zfPXR(EC50:0.23 µM)。它是合成的孕酮,具有免疫刺激作用。
T33033 Lyngbyatoxin A

Lyngbyatoxin A is an indole alkaloid from blue-green alga Lyngbya majuscula Gomont; responsible for dermatitis known as &quot;swimmers' itch&quot; in Hawaii.

天然产物

Triptonide
Cat.No: T5S1058
Synonym: 雷公藤内酯酮,PG 492,NSC 165677
Target: Apoptosis, Wnt/beta-catenin, Autophagy
Lynestrenol
Cat.No: T7974
Synonym:
Target: Progesterone Receptor
Lyngbyatoxin A
Cat.No: T33033
Synonym:
Target:
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