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62

抑制剂 & 化合物

13

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1837 Acyl Carrier Protein (ACP) (65-74)

Acyl Carrier Protein (ACP) 65-74

Acyl Carrier Protein (ACP) (65-74) is an active acyl carrier protein (ACP) fragment.Acyl Carrier Protein (ACP) is a component of plastid-located plant fatty acid synthetase. It binds acyl groups covalently via the prosthetic group, 4-phosphopantetheine, d
T8732 CTPI-2

Others; Mitochondrial Metabolism Metabolism; Others
CTPI-2 是一种特异性线粒体柠檬酸盐载体SLC25A1抑制剂,KD=3.5 μM,具有抗肿瘤作用。它能够抑制糖酵解、PPARγ 及其下游靶点葡萄糖转运蛋白 GLUT4。它阻断非酒精性脂肪性肝炎逆转脂肪变性的显著改变,防止演变为脂肪性肝炎,减少肝脏和脂肪组织中炎性巨噬细胞的浸润,并显著减轻由高脂肪饮食引起的肥胖。
T2607 MSDC 0160

CAY10415,Mitoglitazone,MSDC0160,MSDC-0160

Others; IGF-1R; Mitochondrial Metabolism Metabolism; Others; Tyrosine Kinase/Adaptors
MSDC 0160 (CAY10415) 是一种线粒体丙酮酸载体(MPC) 的调节剂,也是调节噻唑烷二酮的线粒体靶标 (mTOT) 的胰岛素增敏剂。它是一种噻唑烷二酮 (TZD),具有抗糖尿病和神经保护活性作用。它具有用于阿尔茨海默氏病的潜力。
T19507 Perfluamine

FTPA,Tris(perfluoropropyl)amine,Perfluorotripropylamine

Others Others
Perfluamine (FTPA) 是一种疏水性载液,可用作血液替代品。
T83656 DLIN-MC4-DMA

Others Others
DLIN-MC4-DMA 是一种脂质膜,是一种潜在的核酸载体。
T19642 Nilofabicin

CG 0549,CG-0549,CG-400549,CG 400549,CG0549,CG400549

Antibacterial Microbiology/Virology
Nilofabicin (CG-400549) 是一种有效的烯酰-(酰基-载体-蛋白)还原酶下降(FabI)抑制剂,可用于治疗复杂急性疾病的研究。
T83655 DLIN-MC2-DMA

DLin-M-C2-DMA

Others Others
DLIN-MC2-DMA (DLin-M-C2-DMA) 是一种脂质膜,是一种潜在的核酸载体。
TP1798 Pep-1 (uncapped)

Pep-1 uncapped

Others Others
Pep-1 (uncapped) 是一种能够透过细胞的多肽。
T74233 Dlin-MeOH

Others Others
Dlin-MeOH 是一种脂质膜,是一种潜在的核酸载体,可用于合成 DLin-MC3-DMA。
T83654 Dilinoleyl Ketone

Bis(linoleyl) ketone

Others Others
Dilinoleyl Ketone (Bis(linoleyl) ketone) 是一种脂质膜,是一种潜在的核酸载体。
T6834 FCCP

Carbonyl cyanide 4-(trifluoromethoxy)phenylhydrazone,Trifluoromethoxy carbonylcyanide phenylhydrazone

ATPase; Mitochondrial Metabolism Membrane transporter/Ion channel; Metabolism
FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) 是一种氧化磷酸化 (OXPHOS) 抑制剂,线粒体质子载体解偶联剂。FCCP 常被用作细胞凋亡诱导剂。
T11938L Macropa-NH2

Others Others
Macropa-NH2 是 macropa 双功能类似物,是一种常与抗体偶联的载体分子,常作为螯合剂使用,参与癌症研究。
T41324 L319

Di((Z)-Non-2-en-1-yl) 9-((4-(dimethylamino)butanoyl)oxy)heptadecanedioate

Others Others
L319 (Di((Z)-Non-2-en-1-yl) 9-((4-(dimethylamino)butanoyl)oxy)heptadecanedioate) 是一种脂质膜,是一种潜在的核酸载体。
T9807 CPDS

Others Others
CPDS 是一种非渗透性硫醇剂,可影响多种线粒体功能。在大鼠肝线粒体中,它仅抑制 Pi/OH- 载体。它和丙二酸正丁酯都是完全抑制 Pi 进入所必需的。
T4105 AFN-1252

Debio 1452,API-1252

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
AFN-1252 (Debio 1452)是一种FabI 的高效抑制剂,能抑制金黄色葡萄球菌。
T38715 MSDC-0602K

MSDC-0602K,Azemiglitazone potassium

PPAR DNA Damage/DNA Repair; Metabolism
MSDC-0602K (Azemiglitazone potassium) (Azemiglitazone potassium) is a PPARγ-sparing thiazolidinedione (Ps-TZD) compound that binds to PPARγ with an IC50 of 18.25 μM. It also modulates the mitochondrial pyruvate carrier (MPC). This compound, MSDC-0602K, has potential applications in researching fatty liver conditions, including dysfunctional lipid metabolism, inflammation, and insulin resistance. MSDC-0602K acts as an insulin sensitizer, improving insulinemia and fatty liver disease in mice both ...
T7081 CCCP

Carbonyl Cyanide m-Chlorophenylhydrazone,Carbonyl cyanide 3-chlorophenylhydrazone,羰基氰化氯苯腙

Apoptosis; IκB/IKK; COX; Mitochondrial Metabolism; STING; IFNAR; Antibacterial Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
CCCP (Carbonyl Cyanide m-Chlorophenylhydrazone) 是一种氧化磷酸化 (OXPHOS) 抑制剂,线粒体质子载体解偶联剂。CCCP 抑制 STING 及其下游信号分子 TBK1 和 IRF3 的激活。
T4441 UK-5099

UK 5099,PF-1005023,UK5099

Others; Mitochondrial Metabolism Metabolism; Others
UK-5099 (PF-1005023) 是一种有效的线粒体丙酮酸转运蛋白(MPC) 抑制剂, 抑制丙酮酸依赖性 O2消耗的 IC50值为50 nM。
T72968 ZINC00640089

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
ZINC00640089 是一种选择性的脂质运载蛋白-2 (LCN2) 抑制剂。ZINC00640089 对细胞增殖、细胞活力有抑制作用,可减少 SUM149 细胞的 AKT 磷酸化水平。ZINC00640089 可用于研究炎症性乳腺癌 (IBC) 。
T9405 1,4-Dipierazino-2,3,5,6-tetrafluorobenzene

Others Others
1,4-Dipierazino-2,3,5,6-tetrafluorobenzene 是一种四氟苯衍生物,它的独特结构使其能够作为药物的载体,药物可以以可控的方式释放,使其能够用于开发靶向药物递送系统。
T6170 Elesclomol

伊利司莫,STA-4783

Apoptosis; HSP; Reactive Oxygen Species Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB
Elesclomol (STA-4783) 是一种氧化应激诱导剂,也是一种高度亲脂性的铜离子载体。Elesclomol 可以诱导肿瘤细胞凋亡,用于铜死亡相关研究。Elesclomol 还可以抑制 FDX1 介导的 Fe-S 簇生物合成。
T6120 Pralatrexate

Folotyn,10-炔丙基-10-去氮杂氨基蝶呤,10-Propargyl-10-deazaaminopterin,普拉曲沙

Apoptosis; DHFR; Antifolate; TAM Receptor Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Tyrosine Kinase/Adaptors
Pralatrexate (10-Propargyl-10-deazaaminopterin) 是一种抗叶酸剂,也是二氢叶酸还原酶抑制剂,Ki 值为 13.4 pM。它具有抗肿瘤活性,可研究复发/难治性 T 细胞淋巴瘤。它是叶酰聚谷氨酸合成酶的底物,具有改善的细胞摄取和保留能力。
T67727 MCT1-IN-3

Monocarboxylate transporter Membrane transporter/Ion channel
MCT1-IN-3是一种单羧酸转运蛋白1 (MCT1)抑制剂。溶质载体(SLC)单羧酸转运蛋白1 (MCT1);SLC16A1)是治疗癌症的一个有希望的靶点。MCT1-IN-3(化合物24)对MCT1转运抑制作用强,IC50值为81.0 nM。MCT1-IN-3对多药转运体ABCB1也有明显的抑制作用。
T72054 SLC26A3-IN-1

transporter Metabolism
SLC26A3-IN-1 是一种阴离子交换蛋白 SLC26A3 的抑制剂 ,IC50值为340 nM。SLC26A3 属于溶质载体 (SLC) 蛋白,是 SLC26 家族成员之一。SLC26 家族对氯化物、碳酸氢盐、硫酸盐和草酸盐具有广泛的阴离子特异性。SLC26A3 在腺瘤 (DRA) 中下调,参与氯化物和草酸盐的肠道吸收且与氯离子丢失性腹泻有关。
T8637 DMNB

6-Nitroveratraldehyde,6-硝基藜芦醛

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
DMNB (6-Nitroveratraldehyde) 可用于合成no-carrier-added 6-[18F]fluoro-L-DOPA (6-FDOPA)。它可用于研究多巴胺能系统的PET。
T0239 Lonidamine

AF1890,氯尼达明,DICA,Diclondazolic Acid

Apoptosis; Hexokinase; Mitochondrial Metabolism Apoptosis; Metabolism
Lonidamine (Diclondazolic Acid) 是一种抗肿瘤药物,是己糖激酶、线粒体丙酮酸载体和质膜单羧酸转运蛋白抑制剂,同时也抑制线粒体复合物 II。
T30680 Cabiotraxetan

Cabiotraxetan is a therapeutic carrier.
T32255 Jam 2-263

Jam 2 263l,Jam-2-263,Jam2263

Jam 2-263 is a spermidine-based catechol ferric carrier - carbocephalosporin.
T28732 SCH-538415

SCH-538415 is an inhibitor of acyl carrier protein synthase from a microorganism. SCH-538415 exhibited inhibitory activity in the acyl carrier protein synthase (AcpS) assay with an IC(50) value of 4.19 microM and showed antibacterial activity against Stap
T26184 Seproxetine HCl

(S)-Norfluoxetine hydrochloride,Seproxetine hydrochloride,(S)-Desmethylfluoxetine Hydrochloride

Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.
T33929 Perflubrodec

AF0144,AF-0144,AF 0144

Perflubrodec is a component of an intravascular temporary oxygen carrier to enhance oxygen transport.
T32619 Lead phthalocyanine

Lead phthalocyanine, a selective carrier, can be used for the preparation of a cysteine-selective electrode.
T24841 Sulfo-MBS Crosslinker

Sulfo-MBS Cross linker,Sulfo-MBS Cross-linker

Sulfo-MBS Crosslinker is a non-cleavable, water-soluble, heterobifunctional protein crosslinking reagent. It is commonly used to crosslink haptens to carrier proteins and enzymes to antibodies.
T32598 Lauroyl-coenzyme A

Dodecanoyl-coa,Coenzyme A, lauroyl-,Lauroyl-coa

Lauroyl-coenzyme A can function as an acyl group carrier, acetyl-CoA. It can be used as an intermediate in lipid metabolism and is involved in lipid biosynthesis and fatty acid transport.
T12635L Plevitrexed

BGC9331,ZD 9331

Others Others
Plevitrexed is taken up via the α-folate receptor as well as the reduced folate carrier. Plevitrexed is an orally active and effective thymidylate synthase (TS) inhibitor (Ki: 0.44 nM). Plevitrexed is used for gastric cancer in clinical.
T26635 Antifolate C1

AGF 94,AGF94,AGF-94

Antifolate C1 is an inhibitor of de novo purine biosynthesis. Antifolate C1 has selectivity for cellular uptake by high affinity folate receptors and the proton-coupled folate transporter (PCFT) over the reduced folate carrier (RFC).
T60313 Sucistil

Sucistil 是一种活性生化物质。hemoglobin sucistil (bovine) 是一种氧载体。
T25980 Pralatrexate, (R)-

Pralatrexate, (R)- is a folate analog dihydrofolate reductase (DHFR) inhibitor exhibiting high affinity for reduced folate carrier-1 (RFC-1) with antineoplastic and immunosuppressive activities. Pralatrexate selectively enters cells expressing RFC-1; intr
T73990 Lipid M

Lipid M (pKa: 6.75) 可用于递送 mRNA 疫苗,引发强大的免疫反应并提高耐受性。
T34316 Rhizoferrin

Others Others
Rhizoferrin 是一种来自真菌Rhizopus microsporus var.rhizopodiformis 的新型铁载体,可用于研究植物缺铁引起的萎黄病。
T70499 Afabicin diolamine

Afabicin (formerly Debio 1450, AFN-1720) is a prodrug of afabicin desphosphono, an enoyl-acyl carrier protein reductase (FabI) inhibitor, and is a first-in-class antibiotic with a novel mode of action to specifically target fatty acid synthesis in Staphylococcus spp.
T5137 Corn oil

玉米油

Others Others
Corn oil 是一种药物分子的载体,是一种从玉米胚芽中提取出来的油。
T25981 Pralatrexate, (S)-

Pralatrexate, (S)- is a folate analog dihydrofolate reductase (DHFR) inhibitor exhibiting high affinity for reduced folate carrier-1 (RFC-1) with antineoplastic and immunosuppressive activities. Pralatrexate selectively enters cells expressing RFC-1; intr
T76568 Aminopeptidase N Ligand (CD13) NGR peptide

AminopeptidaseN Ligand (CD13) NGR peptide 是靶向CD13的多肽,常见于癌症研究中,用作细胞内传递的载体介质。
T37070 Pyridomycin

Pyridomycin is a structurally unusual antimycobacterial cyclodepsipeptide whose composition includes two rare moieties: 3-(3-pyridyl)-L-alanine and 2-hydroxy-3-methylpent-2-enoic acid. It inhibits NADH-dependent enoyl (Acyl-Carrier-Protein) reductase InhA, preventing mycolic acid synthesis in M. tuberculosis, including isoniazid-resistant strains (MICs = 0.31-0.63 μg/ml).
T74304 C16 PEG-Ceramide

C16 PEG-Ceramide为一种聚乙二醇化神经酰胺,具备脂质载体传递功能,并能诱导自噬(autophagy),在癌症研究中有应用。
T73085 Talotrexin

PT523

Talotrexin (PT523) 是一种 Aminopterin 的类似物,是一种非聚谷氨酸化的经典抗叶酸剂 (antifolate)。 Talotrexin 是一种 RFC(还原型叶酸载体)的特异性抑制剂,可选择性地抑制 RFC 转运。Talotrexin 通过靶向 DHFR 抑制肿瘤生长显示出抗肿瘤活性。
T74859 SLC7A11-IN-1

SLC7A11-IN-1 是一种有效的 SLC7A11抑制剂。SLC7A11-IN-1 显示出抗增殖活性。SLC7A11-IN-1 抑制细胞侵袭和转移。SLC7A11-IN-1 诱导细胞凋亡 (Apoptosis) 和细胞周期停滞在 S 期。SLC7A11-IN-1 具有抗肿瘤活性。
T35957 PBD-BODIPY

PBD-BODIPY is a probe for the spectrophotometric measurement of autoxidation reactions. Co-autoxidation of the PBD-BODIPY signal carrier and a hydrocarbon co-substrate can be quantified by monitoring loss of absorbance at 591 nm. PBD-BODIPY has been used to measure the activity of radical-trapping antioxidants in cell-free assays. It has also been used as a fluorescent probe for the detection of epoxidation activity.
T73032 MtInhA-IN-1

MtInhA-IN-1是一种口服活性的选择性结核分枝杆菌NADH依赖性烯酰基载体蛋白还原酶(MtInhA)抑制剂,IC50值为0.23 μM。对结核分枝杆菌H37Rv菌株,其MIC为0.4 μM。

化合物

Acyl Carrier Protein (ACP) (65-74)
Cat.No: TP1837
Synonym: Acyl Carrier Protein (ACP) 65-74
Target:
CTPI-2
Cat.No: T8732
Synonym:
Target: Others, Mitochondrial Metabolism
MSDC 0160
Cat.No: T2607
Synonym: CAY10415,Mitoglitazone,MSDC0160,MSDC-0160
Target: Others, IGF-1R, Mitochondrial Metabolism
Perfluamine
Cat.No: T19507
Synonym: FTPA,Tris(perfluoropropyl)amine,Perfluorotripropylamine
Target: Others
DLIN-MC4-DMA
Cat.No: T83656
Synonym:
Target: Others
Nilofabicin
Cat.No: T19642
Synonym: CG 0549,CG-0549,CG-400549,CG 400549,CG0549,CG400549
Target: Antibacterial
DLIN-MC2-DMA
Cat.No: T83655
Synonym: DLin-M-C2-DMA
Target: Others
Pep-1 (uncapped)
Cat.No: TP1798
Synonym: Pep-1 uncapped
Target: Others
Dlin-MeOH
Cat.No: T74233
Synonym:
Target: Others
Dilinoleyl Ketone
Cat.No: T83654
Synonym: Bis(linoleyl) ketone
Target: Others
FCCP
Cat.No: T6834
Synonym: Carbonyl cyanide 4-(trifluoromethoxy)phenylhydrazone,Trifluoromethoxy carbonylcyanide phenylhydrazone
Target: ATPase, Mitochondrial Metabolism
Macropa-NH2
Cat.No: T11938L
Synonym:
Target: Others
L319
Cat.No: T41324
Synonym: Di((Z)-Non-2-en-1-yl) 9-((4-(dimethylamino)butanoyl)oxy)heptadecanedioate
Target: Others
CPDS
Cat.No: T9807
Synonym:
Target: Others
AFN-1252
Cat.No: T4105
Synonym: Debio 1452,API-1252
Target: Others, Antibacterial, Antibiotic
MSDC-0602K
Cat.No: T38715
Synonym: MSDC-0602K,Azemiglitazone potassium
Target: PPAR
CCCP
Cat.No: T7081
Synonym: Carbonyl Cyanide m-Chlorophenylhydrazone,Carbonyl cyanide 3-chlorophenylhydrazone,羰基氰化氯苯腙
Target: Apoptosis, IκB/IKK, COX, Mitochondrial Metabolism, STING, IFNAR, Antibacterial
UK-5099
Cat.No: T4441
Synonym: UK 5099,PF-1005023,UK5099
Target: Others, Mitochondrial Metabolism
ZINC00640089
Cat.No: T72968
Synonym:
Target: Akt
1,4-Dipierazino-2,3,5,6-tetrafluorobenzene
Cat.No: T9405
Synonym:
Target: Others
Elesclomol
Cat.No: T6170
Synonym: 伊利司莫,STA-4783
Target: Apoptosis, HSP, Reactive Oxygen Species
Pralatrexate
Cat.No: T6120
Synonym: Folotyn,10-炔丙基-10-去氮杂氨基蝶呤,10-Propargyl-10-deazaaminopterin,普拉曲沙
Target: Apoptosis, DHFR, Antifolate, TAM Receptor
MCT1-IN-3
Cat.No: T67727
Synonym:
Target: Monocarboxylate transporter
SLC26A3-IN-1
Cat.No: T72054
Synonym:
Target: transporter
DMNB
Cat.No: T8637
Synonym: 6-Nitroveratraldehyde,6-硝基藜芦醛
Target: DNA-PK
Lonidamine
Cat.No: T0239
Synonym: AF1890,氯尼达明,DICA,Diclondazolic Acid
Target: Apoptosis, Hexokinase, Mitochondrial Metabolism
Cabiotraxetan
Cat.No: T30680
Synonym:
Target:
Jam 2-263
Cat.No: T32255
Synonym: Jam 2 263l,Jam-2-263,Jam2263
Target:
SCH-538415
Cat.No: T28732
Synonym:
Target:
Seproxetine HCl
Cat.No: T26184
Synonym: (S)-Norfluoxetine hydrochloride,Seproxetine hydrochloride,(S)-Desmethylfluoxetine Hydrochloride
Target:
Perflubrodec
Cat.No: T33929
Synonym: AF0144,AF-0144,AF 0144
Target:
Lead phthalocyanine
Cat.No: T32619
Synonym:
Target:
Sulfo-MBS Crosslinker
Cat.No: T24841
Synonym: Sulfo-MBS Cross linker,Sulfo-MBS Cross-linker
Target:
Lauroyl-coenzyme A
Cat.No: T32598
Synonym: Dodecanoyl-coa,Coenzyme A, lauroyl-,Lauroyl-coa
Target:
Plevitrexed
Cat.No: T12635L
Synonym: BGC9331,ZD 9331
Target: Others
Antifolate C1
Cat.No: T26635
Synonym: AGF 94,AGF94,AGF-94
Target:
Sucistil
Cat.No: T60313
Synonym:
Target:
Pralatrexate, (R)-
Cat.No: T25980
Synonym:
Target:
Lipid M
Cat.No: T73990
Synonym:
Target:
Rhizoferrin
Cat.No: T34316
Synonym:
Target: Others
Afabicin diolamine
Cat.No: T70499
Synonym:
Target:
Corn oil
Cat.No: T5137
Synonym: 玉米油
Target: Others
Pralatrexate, (S)-
Cat.No: T25981
Synonym:
Target:
Aminopeptidase N Ligand (CD13) NGR peptide
Cat.No: T76568
Synonym:
Target:
Pyridomycin
Cat.No: T37070
Synonym:
Target:
C16 PEG-Ceramide
Cat.No: T74304
Synonym:
Target:
Talotrexin
Cat.No: T73085
Synonym: PT523
Target:
SLC7A11-IN-1
Cat.No: T74859
Synonym:
Target:
PBD-BODIPY
Cat.No: T35957
Synonym:
Target:
MtInhA-IN-1
Cat.No: T73032
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T10857 Coenzyme A

Endogenous Metabolite Metabolism
Coenzyme A 是所有活细胞中必需的辅助因子,由泛酸,三磷酸腺苷和半胱氨酸合成的。Coenzyme A 与过氧化物酶 5 共价结合导致其过氧化物酶活性完全抑制,通过 DTT 还原能够逆转。Coenzyme A 及其硫酯衍生物是主要分解代谢,合成代谢途径和基因表达调控的关键参与者。
T15717 Lasalocid

Lasalocid-A,Antibiotic X-537A,Ionophore X-537A

Antibacterial Microbiology/Virology
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。
T8170 Carboxyatractyloside

羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt

Others Others
Carboxyatractyloside (Carboxyatractyloside tripotassium salt) tripotassium salt 是一种 ADP/ATP 载体蛋白 (ADP/ATP carrier) 抑制剂,抑制线粒体 ADP/ATP 的转运。它是一种具有毒性的天然产物,
T2796 Coenzyme Q10

Ubiquinone-10,辅酶Q10,CoQ10

Ferroptosis; Reactive Oxygen Species; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Metabolism; NF-κB
Coenzyme Q10 (CoQ10)是来自藤仓赤霉菌的一种天然产物,在线粒体呼吸链中充当电子载体。
T1609 NAD+

烟酰胺腺嘌呤二核苷酸,Cozymase,煙酸胺,β-DPN,DPN,β-Nicotinamide Adenine Dinucleotide,β-NAD

NADPH; Endogenous Metabolite Metabolism
NAD+ (β-Nicotinamide Adenine Dinucleotide) 即烟酰胺腺嘌呤二核苷酸,是转递氢离子的辅酶。
T22446 NADP disodium salt

Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐

Others Others
NADP disodium salt (Disodium NADP) 是一种氧化还原辅助因子,是一种烟酰胺腺嘌呤二核苷酸。它是代谢中电子转移的关键辅因子,可以被交替氧化 (NADP+) 和还原 (NADPH)。
T3092 Nigericin sodium salt

尼日利亚菌素,尼日利亚菌素钠盐

Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。
TWA2417 Sodium taurocholate

牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium

Others Others
Sodium taurocholate (Taurocholate Sodium) hydrate 具有显著的生物学效应,例如通过上调 VEGF-A 的表达抑制肝动脉结扎所致的胆道损伤。对免疫系统具有一定的调节作用。
T0326 DL-Glutamine

Glutamin,DL-Gl,(±)-Glutamine,DL-谷氨酰胺,2-amino-4-carbamoylbutanoic acid

Ferroptosis; Amino Acids and Derivatives; Endogenous Metabolite Apoptosis; Metabolism
DL-Glutamine (2-amino-4-carbamoylbutanoic acid) 是一种非必需氨基酸,大量存在于全身并参与许多代谢过程。 它由谷氨酸和氨合成,是体内氮的主要载体,是许多细胞的重要能量来源,用于制药和供生物化学研究。
T38499 κ-Carrageenan

κ-Carrageenan, a natural polymer found predominantly in red seaweeds, can serve as an effective drug carrier for delivering curcumin to cancer cells and inducing apoptosis. Additionally, κ-Carrageenan holds promise as a potential inflammatory agent, amplifying existing intestinal inflammation.
T38069 Aquastatin A

Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC50= 3.2 μM) andS. aureusfatty acid synthesis (IC50= 3.5 μM).2Aquastatin A also inhibits the Na+/K+-ATPase and H+/K+-ATPase (IC50s = 7.1 and 6.2 μM, respectively), as well as protein tyrosine phosphatase 1B (PTP1B; IC50= 0.19 μM).1,3 1.Hamano, K., Kinoshita-Okami, M., Minagawa, K....
T78465 H-γ-Glu-Gln-OH

γ-Glutamylglutamine,γ-Glu-Gln

H-γ-Glu-Gln-OH 是一种水溶性肽类化合物,用于药物结合。该载体特征为高溶解度、药物负载效能、优良生物相容性、低毒性,并能增强抗癌药物对肿瘤的靶向作用及疗效。
T36439 Gramicidin A

Antibacterial; HIF; Parasite Angiogenesis; Chromatin/Epigenetic; Microbiology/Virology
Gramicidin A 是一种从从 B. brevis 分离出来的多肽类抗生素。Gramicidin A 是一种高度疏水的通道形成离子载体,在人工膜中形成一价阳离子可渗透的通道。Gramicidin A 诱导缺氧诱导因子 1α (HIF-1α) 的降解,并能降低人肾细胞癌小鼠异种移植模型的生长。Gramicidin A 具有抗菌、抗疟活性以及溶血活性。

天然产物

Coenzyme A
Cat.No: T10857
Synonym:
Target: Endogenous Metabolite
Lasalocid
Cat.No: T15717
Synonym: Lasalocid-A,Antibiotic X-537A,Ionophore X-537A
Target: Antibacterial
Carboxyatractyloside
Cat.No: T8170
Synonym: 羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt
Target: Others
Coenzyme Q10
Cat.No: T2796
Synonym: Ubiquinone-10,辅酶Q10,CoQ10
Target: Ferroptosis, Reactive Oxygen Species, Endogenous Metabolite
NAD+
Cat.No: T1609
Synonym: 烟酰胺腺嘌呤二核苷酸,Cozymase,煙酸胺,β-DPN,DPN,β-Nicotinamide Adenine Dinucleotide,β-NAD
Target: NADPH, Endogenous Metabolite
NADP disodium salt
Cat.No: T22446
Synonym: Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐
Target: Others
Nigericin sodium salt
Cat.No: T3092
Synonym: 尼日利亚菌素,尼日利亚菌素钠盐
Target: Potassium Channel, NOD-like Receptor (NLR), Antibacterial, Antibiotic, NOD
Sodium taurocholate
Cat.No: TWA2417
Synonym: 牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium
Target: Others
DL-Glutamine
Cat.No: T0326
Synonym: Glutamin,DL-Gl,(±)-Glutamine,DL-谷氨酰胺,2-amino-4-carbamoylbutanoic acid
Target: Ferroptosis, Amino Acids and Derivatives, Endogenous Metabolite
κ-Carrageenan
Cat.No: T38499
Synonym:
Target:
Aquastatin A
Cat.No: T38069
Synonym:
Target:
H-γ-Glu-Gln-OH
Cat.No: T78465
Synonym: γ-Glutamylglutamine,γ-Glu-Gln
Target:
Gramicidin A
Cat.No: T36439
Synonym:
Target: Antibacterial, HIF, Parasite
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