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80

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T24805 SMA-12b

SMA 12b,SMA12b

SMA-12b is an IL-1 inhibitor.
T4283 SRI-011381

TGF-beta/Smad Stem Cells
SRI011381 是口服具有活力的 TGF-β信号通路的激活剂,具有神经保护活性。
T14080 AA147

ATF6-activator-147

Others Others
AA147 (ATF6-activator-147) 是小分子内质网蛋白稳态调节剂,能够选择性激活未折叠蛋白反应的 ATF6臂。
T16886 Sinefungin

Adenosyl-Ornithine,西奈芬净,A-9145,Antibiotic 32232RP

Others; Histone Methyltransferase; Antibiotic; Antifungal Chromatin/Epigenetic; Microbiology/Virology; Others
Sinefungin (Adenosyl-Ornithine) 是病毒粒子mRNA (鸟嘌呤-7-)-甲基转移酶、 mRNA (核苷-2'-)-甲基转移酶和病毒增殖的有效抑制剂。它还抑制SET7/9,通过抑制H3K4甲基化来改善肾纤维化。
T4641 Branaplam

LMI 070,NVS-SM1

Others; Potassium Channel; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Others
Branaplam (LMI 070) 是一种高效、选择性和口服活性的小分子 SMN2 剪接调节剂,对 SMN 的 EC50为 20 nM。它可提高全长 SMN 蛋白并延长其生存期,也抑制 hERG,IC50为 6.3 μM。
T81149 SMA4

SMA4是一款选择性的PKG1α激活剂,其对PKG1α的EC50为29 μM。该化合物能够在细胞内促进PKG1底物——血管扩张刺激磷蛋白(VASP)的磷酸化,同时能够抑制人肺动脉平滑肌细胞(hPASMC)的增殖,适用于心血管疾病研究。
T5129 SRI-011381 hydrochloride

SRI-011381 hydrochloride [1629138-41-5(free base)]

TGF-beta/Smad Stem Cells
SRI-011381 hydrochloride 是口服具有活力的TGF-β信号通路的激活剂,具有神经保护活性。
T1606 Fasudil

HA-1077,AT877,法舒地尔

ROCK; Serine/threonin kinase; Calcium Channel; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil (HA-1077) 是一种非特异性 RhoA/ROCK 抑制剂,也是 Ca2+通道拮抗剂和血管扩张剂。它对蛋白激酶有抑制作用,ROCK1 的 Ki 值为 0.33 μM,ROCK2 和 PKA、PKC、PKG 的 IC50值分别 0.158 μM 和 4.58 μM、12.30 μM、1.650 μM。
T3060 Fasudil hydrochloride

Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877

ROCK; Serine/threonin kinase; Calcium Channel; HIV Protease; PKA; PKC; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
Fasudil hydrochloride (HA-1077) 是一种非特异性RhoA/ROCK 抑制剂,也抑制蛋白激酶,对 ROCK1、PKA、PKC 和 MLCK 的 Ki 值分别为 0.33 μM、1.0 μM、9.3 μM 和 55 μM。
T28466 PSMA-11

HBED-CC-PSMA,Psma-hbed-CC,PSMA11

PSMA-11 (HBED-CC-PSMA)通过与前列腺特异性膜抗原(PSMA)的细胞外结构域结合来检测前列腺癌的复发和转移。PSMA-11常被用作正电子发射断层扫描(PET)中用作表达PSMA 的肿瘤的示踪剂,通过静脉注射镓Ga 68标记的PSMA-11,Glu-urea-Lys(Ahx)分子靶向并结合表达PSMA 的肿瘤细胞。内化后,PSMA 表达的肿瘤细胞可在PET 成像中被检测到。
T2277 Losmapimod

GSK-AHAB,GW856553X,6-[5-(环丙基氨基甲酰基)-3-氟-2-甲基苯基]-N-(2,2-二甲基丙基)吡啶-3-甲酰胺,GW856553,洛批莫德,SB856553

p38 MAPK; Autophagy Autophagy; MAPK
Losmapimod (GSK-AHAB) 是一种可口服的特异性 p38 MAPK 抑制剂,抑制 p38α 和 p38β 的 pKi 值分别为 8.1 和 7.6。
T23370 SMANT hydrochloride

N-(4-Bromophenyl)-3,5-dimethyl-1-piperidinepropanamide hydrochloride,hydrochloride,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide;hydrochloride,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide,SMANT HCl,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) 是一种 Smoothened 积聚的拮抗剂。
T13890 SMARCA-BD ligand 1 for Protac dihydrochloride

Epigenetic Reader Domain Chromatin/Epigenetic
SMARCA-BD ligand 1 for Protac dihydrochloride 是一种能够与 BAF ATPase 亚基 SMARCA2 结合的化合物,基于 PROTAC 技术,使 SMARCA2 降解。
T9568 SGC-SMARCA-BRDVIII

Epigenetic Reader Domain Chromatin/Epigenetic
SGC-SMARCA-BRDVIII 是SMARCA2/4和PB1(5)选择性抑制剂,其Kd 值分别为 35 nM,36 nM 和 13 nM。它还抑制PB1(2)和PB1(3),Kd 值分别为 3.7 和 2.0 μM。它可阻断 3T3-L1 鼠成纤维细胞的脂肪生成。
T19957 Bismaleimide

XU 292A,XU-292A,XU292A

Others Others
Bismaleimide (XU 292A) 具有抗热性、抗氧化性、抗辐射性,可用于制备电器绝缘材料、耐磨材料、增强塑料添加剂、砂轮粘结剂等。
T77019 Garetosmab

REGN 2477

TGF-beta/Smad Stem Cells
Garetosmab (REGN 2477) 是一种全人 IgG4 单克隆抗体,可选择性抑制激活素 A (activin A),可作用于 COVID-44。Garetosmab 具有潜在的抗癌活性,可用于研究骨化性纤维发育不良 (FOP) 和癌症。
T13848 SMARCA-BD ligand 1 for Protac

Epigenetic Reader Domain Chromatin/Epigenetic
SMARCA-BD ligand 1 for Protac 能够与 BAF ATPase 亚基 SMARCA2 结合,可用于 PROTAC 技术,用于降解 SMARCA2。
TP1844L Small Cardioactive Peptide B SCPB acetate

Small Cardioactive Peptide B SCPB acetate(84746-43-0 free base)

Others Others
Small Cardioactive Peptide B SCPB acetate (Small Cardioactive Peptide B SCPB acetate (84746-43-0 free base)) 是一种神经活性肽,可刺激心脏和鳃组织颗粒部分的腺苷酸环化酶活性,EC50 分别为 0.1 和 1.0 μM。
T77750 Rosmantuzumab

OMP-131R10

Others Others
Rosmantuzumab (OMP-131R10) 是一种 人源化抗 R-spondin 3 (RSPO3)单克隆抗体。Rosmantuzumab 具有潜在的抗肿瘤活性,可用于研究晚期复发难治性实体瘤。
T69924 PSMA-1007

PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.
T11314 Fosmanogepix

APX001,E1211

Others Others
Fosmanogepix (APX001) is a first-in-class, orally available broad-spectrum antifungal agent. It acts as an N-phosphonooxymethyl prodrug that undergoes rapid and complete metabolism by systemic alkaline phosphatases. This metabolism leads to the formation of the active moiety, APX001A. Fosmanogepix (APX001), with its ability to target the highly conserved Gwt1 fungal enzyme, holds great potential for the development of treatments against invasive fungal infections.
T34660 SMART-F

SMART-F is a biochemical.
T83738 SMAP 29 (ovine) TFA

Sheep Myeloid Antimicrobial Peptide 29

SMAP 29是一种抗微生物肽,同时也是绵羊防御素前体肽的C末端切割产物。在低盐和高盐条件下,对P. aeruginosa菌株PAO1具有杀菌作用,该作用在能量依赖的发光测定中表现出来(EC50s分别为0.05和0.06 µM)。它还能够以浓度依赖的方式引起绵羊红细胞的溶血。
T12934 SMAP-2

DT-1154

Phosphatase Metabolism
SMAP-2 is an orally bioavailable activator of phosphatase 2A (PP2A) which binds to the PP2A Aα scaffold subunit to drive conformational changes in PP2A. It inhibits the growth of KRAS-mutant lung cancers .
T78412 Biotin-NH-PSMA-617

Biotin-NH-PSMA-617为标记有生物素的PSMA-617小分子,专门针对前列腺特异性膜抗原(PSMA),后者为肿瘤细胞所特有表达。
TP2407 Small cardioactive peptide A

SCPA

Small cardioactive peptide A, as a neuropeptide that modulates neuromuscular synapsis in Aplysia, can also function as a neural cotransmitter in molluscs and exert a role in both the central and peripheral modulation of the control of feeding behavior.
T79321 nSMase2-IN-1

Phospholipase Metabolism
nSMase2-IN-1是一款口服活性的nSMase2抑制剂,具有0.13 ± 0.06 μM的IC50。该化合物在肝脏微粒体内具有良好的代谢稳定性,口服给药后获得较高的脑血浆比值,适用于神经系统疾病研究。
T20053 Jasmacyclen

EC 226-501-6,NSC-6598,Verdyl acetate,Greenyl acetate,NS 6598,NSC 6598

Jasmacyclen is a compound in which has an aroma.
T80262 SMAP-18

SMAP-18是一种具有高生物活性的18氨基酸残基肽酰胺,为SMAP-29 (羊髓系抗菌肽-29) 的缩短版本。SMAP-29对假单胞菌菌株、其他革兰氏阴性菌及多重耐药病原体有很强的抗菌作用。SMAP-18相较于母体SMAP-29,表现出更高的细胞选择性,因其降低了溶血活性同时保留了抗菌能力。
TP1844 Small Cardioactive Peptide B (SCPB)

Small Cardioactive Peptide B SCPB

Small Cardioactive Peptide B (SCPB), a neurally active peptide, stimulates adenylate cyclase activity in particulate fractions of both heart and gill tissues with EC50s of 0.1 and 1.0 μM, respectively.
TF0097 BisMalt-20

BisMalt-20 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0097,CAS号为 1423237-53-9。
T61403 Plasma kallikrein-IN-3

Plasma kallikrein-IN-3, a potent inhibitor ( IC 50 : 0.15 μM) of plasma kallikrein, finds application in research related to hereditary angioedema, diabetic macular edema, and diabetic retinopathy [1].
T125437 14-Hydroxy-7-O-methylrosmanol

14-Hydroxy-7-O-methylrosmanol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125437,CAS号为 197649-67-5。
T35205 Xylosmacin

Xylosmacin is a biochemical.
T126198 Rosmaquinone

Rosmaquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126198。
T124419 Clausmarin A

Clausmarin A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124419。
T40312 Plasma kallikrein-IN-1

Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.
T30474 Bismark Brown Y

AI3 52758,AI352758,AI3-52758

Bismark Brown Y is a brown dye.
T39172 SMAP-29

SMAP-29 is a broad spectrum antibacterial and antifungal α-helical cathelicidin-derived peptide with strong potential as an antiinfective agent. It effectively permeabilizes bacterial membranes and induces significant alterations in the surface morphology of susceptible microorganisms.
T78927 PSMA-IN-3

PSMA-IN-3(compound 17)是一种高亲和力的新型PSMA抑制剂,IC50为13 nM。该化合物可作为开发18F标记的放射性配体的基础,用于前列腺癌PSMA的PET成像。
T40326 PSMA–DA1

PSMA–DA1

PSMA–DA1 may be a useful PSMA-targeting radiotheranostic agent.
TF0006 BisMalt-22

BisMalt-22 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0006,CAS号为 1198081-47-8。
T28818 SMAPP1

SMAPP1 is an activator of protein phosphatase 1 (PP1). SMAPP1 induces PP1 activity in vitro and activates latent HIV-1 provirus in cultured and primary T cells.
T35217 Xysmalorin

Xysmalorin is a biochemical.
T34391 Rosmarinine

Rosmarinine is a non-toxic pyrrolizidine alkaloid.
T81361 PSMA-Val-Cit-PAB-MMAE

PSMA-Val-Cit-PAB-MMAE是一种靶向前列腺特异性膜抗原(PSMA)的小分子化合物,用MMAE作为药效基团进行前列腺癌治疗。
T81376 PROTAC SMARCA2 degrader-2

PROTACs PROTAC
PROTACSMARCA2 degrader-2,作为一种高效的SMARCA2/4PROTAC降解剂,在HeLa HiBiT检测中显示出极低的IC50值(<0.1 μΜ)。该化合物对于SMARCA4相关或缺陷癌症研究具有潜在应用价值。
T71742 SMases D inhibitor-1

SMases D inhibitor-1 is a novel inhibitor of loxosceles sphingomyelinases d (smases d)
TF0053 BisMalt-28

BisMalt-28 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0053,CAS号为 1198081-49-0。
T125796 Osmanthuside H

Osmanthuside H 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125796,CAS号为 149155-70-4。

化合物

SMA-12b
Cat.No: T24805
Synonym: SMA 12b,SMA12b
Target:
SRI-011381
Cat.No: T4283
Synonym:
Target: TGF-beta/Smad
AA147
Cat.No: T14080
Synonym: ATF6-activator-147
Target: Others
Sinefungin
Cat.No: T16886
Synonym: Adenosyl-Ornithine,西奈芬净,A-9145,Antibiotic 32232RP
Target: Others, Histone Methyltransferase, Antibiotic, Antifungal
Branaplam
Cat.No: T4641
Synonym: LMI 070,NVS-SM1
Target: Others, Potassium Channel, DNA/RNA Synthesis
SMA4
Cat.No: T81149
Synonym:
Target:
SRI-011381 hydrochloride
Cat.No: T5129
Synonym: SRI-011381 hydrochloride [1629138-41-5(free base)]
Target: TGF-beta/Smad
Fasudil
Cat.No: T1606
Synonym: HA-1077,AT877,法舒地尔
Target: ROCK, Serine/threonin kinase, Calcium Channel, PKA, PKC, Autophagy
Fasudil hydrochloride
Cat.No: T3060
Synonym: Fasudil (HA-1077) HCl,盐酸法舒地尔,HA-1077,Fasudil HCl,HA-1077 hydrochloride,AT-877
Target: ROCK, Serine/threonin kinase, Calcium Channel, HIV Protease, PKA, PKC, Autophagy
PSMA-11
Cat.No: T28466
Synonym: HBED-CC-PSMA,Psma-hbed-CC,PSMA11
Target:
Losmapimod
Cat.No: T2277
Synonym: GSK-AHAB,GW856553X,6-[5-(环丙基氨基甲酰基)-3-氟-2-甲基苯基]-N-(2,2-二甲基丙基)吡啶-3-甲酰胺,GW856553,洛批莫德,SB856553
Target: p38 MAPK, Autophagy
SMANT hydrochloride
Cat.No: T23370
Synonym: N-(4-Bromophenyl)-3,5-dimethyl-1-piperidinepropanamide hydrochloride,hydrochloride,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide;hydrochloride,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide,SMANT HCl,N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride
Target: Hedgehog/Smoothened
SMARCA-BD ligand 1 for Protac dihydrochloride
Cat.No: T13890
Synonym:
Target: Epigenetic Reader Domain
SGC-SMARCA-BRDVIII
Cat.No: T9568
Synonym:
Target: Epigenetic Reader Domain
Bismaleimide
Cat.No: T19957
Synonym: XU 292A,XU-292A,XU292A
Target: Others
Garetosmab
Cat.No: T77019
Synonym: REGN 2477
Target: TGF-beta/Smad
SMARCA-BD ligand 1 for Protac
Cat.No: T13848
Synonym:
Target: Epigenetic Reader Domain
Small Cardioactive Peptide B SCPB acetate
Cat.No: TP1844L
Synonym: Small Cardioactive Peptide B SCPB acetate(84746-43-0 free base)
Target: Others
Rosmantuzumab
Cat.No: T77750
Synonym: OMP-131R10
Target: Others
PSMA-1007
Cat.No: T69924
Synonym:
Target:
Fosmanogepix
Cat.No: T11314
Synonym: APX001,E1211
Target: Others
SMART-F
Cat.No: T34660
Synonym:
Target:
SMAP 29 (ovine) TFA
Cat.No: T83738
Synonym: Sheep Myeloid Antimicrobial Peptide 29
Target:
SMAP-2
Cat.No: T12934
Synonym: DT-1154
Target: Phosphatase
Biotin-NH-PSMA-617
Cat.No: T78412
Synonym:
Target:
Small cardioactive peptide A
Cat.No: TP2407
Synonym: SCPA
Target:
nSMase2-IN-1
Cat.No: T79321
Synonym:
Target: Phospholipase
Jasmacyclen
Cat.No: T20053
Synonym: EC 226-501-6,NSC-6598,Verdyl acetate,Greenyl acetate,NS 6598,NSC 6598
Target:
SMAP-18
Cat.No: T80262
Synonym:
Target:
Small Cardioactive Peptide B (SCPB)
Cat.No: TP1844
Synonym: Small Cardioactive Peptide B SCPB
Target:
BisMalt-20
Cat.No: TF0097
Synonym:
Target:
Plasma kallikrein-IN-3
Cat.No: T61403
Synonym:
Target:
14-Hydroxy-7-O-methylrosmanol
Cat.No: T125437
Synonym:
Target:
Xylosmacin
Cat.No: T35205
Synonym:
Target:
Rosmaquinone
Cat.No: T126198
Synonym:
Target:
Clausmarin A
Cat.No: T124419
Synonym:
Target:
Plasma kallikrein-IN-1
Cat.No: T40312
Synonym:
Target:
Bismark Brown Y
Cat.No: T30474
Synonym: AI3 52758,AI352758,AI3-52758
Target:
SMAP-29
Cat.No: T39172
Synonym:
Target:
PSMA-IN-3
Cat.No: T78927
Synonym:
Target:
PSMA–DA1
Cat.No: T40326
Synonym: PSMA–DA1
Target:
BisMalt-22
Cat.No: TF0006
Synonym:
Target:
SMAPP1
Cat.No: T28818
Synonym:
Target:
Xysmalorin
Cat.No: T35217
Synonym:
Target:
Rosmarinine
Cat.No: T34391
Synonym:
Target:
PSMA-Val-Cit-PAB-MMAE
Cat.No: T81361
Synonym:
Target:
PROTAC SMARCA2 degrader-2
Cat.No: T81376
Synonym:
Target: PROTACs
SMases D inhibitor-1
Cat.No: T71742
Synonym:
Target:
BisMalt-28
Cat.No: TF0053
Synonym:
Target:
Osmanthuside H
Cat.No: T125796
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN7057 rosmarinate acid

(R)-rosmarinic acid,rosmarinic acid,迷迭香素,Rosemary acid

MAO; Endogenous Metabolite; Transferase Metabolism; Neuroscience
Rosmarinate acid(Rosemary acid) 抑制 MAO-A、MAO-B 和 COMT 酶,IC50 分别为 50.1、184.6 和 26.7 μM。
TN1334 7-Methoxyrosmanol

7ALPHA-甲氧基迷迭香酚,7-O-Methylrosmanol

cAMP GPCR/G Protein
7-Methoxyrosmanol (7-O-Methylrosmanol) 是一种酚类二萜,从迷迭香中分离得到,可抑制 PEPCK 和 G6Pase 启动子的 cAMP 反应。
T7033 Rosmanol

Antioxidant; COX Immunology/Inflammation; Neuroscience; oxidation-reduction
Rosmanol 能够显著抑制脂多糖诱导的 INOS、COX-2 的表达,抑制低密度脂蛋白的氧化,并具有抗炎作用。
TN6784 ethyl rosmarinate

迷迭香酸乙酯

MMP; Tyrosinase; Glucosidase Metabolism; Proteases/Proteasome
ethyl rosmarinate 抑制酪氨酸酶、α-葡萄糖苷酶和基质金属蛋白酶-1 (MMP-1) 的活性。
T9135 Epirosmanol

Others Others
Epirosmanol 是含有内酯部分的二萜类化合物。 Epirosmanol 是一种极弱碱性(基本中性)的化合物(基于其 pKa)。
TN1928 Methyl rosmarinate

MMP; Anti-infection; Tyrosinase Microbiology/Virology; Proteases/Proteasome
Methyl rosmarinate 是一种非竞争性 tyrosinase 抑制剂,从 Rabdosia serra 中分离得到的,对蘑菇酪氨酸酶作用的 IC50值为 0.28 mM,也能抑制a-glucosidase。
T2765 Rosmarinic acid

Labiatenic acid,迷迭香酸,Rosemary acid

Apoptosis; IκB/IKK; MAO; Endogenous Metabolite; Transferase; Monoamine Oxidase Apoptosis; Metabolism; Neuroscience; NF-κB
Rosmarinic acid (Labiatenic acid) 广泛存在植物中,具有抗氧化、抗炎和抗菌活性。它抑制 MAO-A,MAO-B 和 COMT,IC50分别为 50.1,184.6 和 26.7 μM。
T31728 Eudesmane

Eudesmane is a bicyclododecane terpenes.
T4S0818 Chasmanine

Chasmanine, hypaconitine, and deoxyaconitine are anti-inflammatory pharmacodynamic components in Heishunpian (HSP) with positive relations with HSP efficacy. Chasmanine has insecticidal activities against larvae of Bradysia odoriphaga Yan et Zhang.
TN4285 Isodorsmanin A

Others Others
Isodorsmanin A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4285,CAS号为 118266-99-2。
T75538 Alismanol M

Alismanol M,一种法尼酯 X 受体 (FXR) 激动剂,具有 50.25 μM 的 EC50 值。作为一种源自东方红根茎的原丹类三萜化合物,Alismanol M 主要应用于胆汁淤积与非酒精性脂肪性肝炎的研究。
TN3257 7beta-Methoxyrosmanol

Transferase Metabolism
7beta-Methoxyrosmanol inhibited acyl CoA:diacylglycerol acyltransferase (DGAT)1 activity, with the IC50 values ranging from 39.5 ± 0.6 to 144.2 ± 3.1 μM.
T35216 Xysmalogenin

BRN0051836,,BRN-0051836,BRN 0051836

Xysmalogenin is a biochemical.
TN1798 Isorosmanol

异迷迭香酚

Beta Amyloid; AChR Neuroscience
Isorosmanol 具有抗氧化、神经保护和神经营养作用,可能用于老年性疾病,如认知功能下降和色素沉着。
TN3149 6,8-Cyclo-1,4-eudesmanediol

Others Others
6,8-Cyclo-1,4-eudesmanediol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3149,CAS号为 213769-80-3。
TN6523 Rosmarinyl glucoside

Rosmarinyl glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6523,CAS号为 910028-78-3。
TN3888 Dorsmanin A

Others Others
Dorsmanin A is a natural product from Psoralea corylifolia.
TN4031 Eudesma-3,11-dien-2-one

Others Others
Eudesma-3,11-dien-2-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4031,CAS号为 86917-79-5。
T80009 Osmanthuside B

Osmanthuside B,从Pseuderanthemum carruthersii (Seem.) Guill. var.atropurpureum (Bull.) Fosb 中分离得到,展现出较弱的乙酰胆碱酯酶抑制活性。
TN6351 Dorsmanin I

Dorsmanin I 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6351,CAS号为 329703-46-0。
TN2495 1,4,7-Eudesmanetriol

Antifection Microbiology/Virology
1α,4β,7β-Eudesmanetriol and 1β,4β,7β-Eudesmanetriol can inhibit growth of Pseudomonas stutzeri with a MIC value of 117 uM, they also show remarkable activities against acetylcholinesterase enzyme with IC50 values ranging between 25 and 26 uM.
TN1329 7-Ethoxyrosmanol

Antifection Microbiology/Virology
7-Ethoxyrosmanol has cytotoxic and antimicrobial activities.
T5S0896 Loureirin A

龙血素 A,龙血素A

Akt; PI3K Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Loureirin A 是一种黄酮类物质,从龙血树中分离得到,能够降低Akt 的磷酸化,具有抗血小板聚集作用。

天然产物

rosmarinate acid
Cat.No: TN7057
Synonym: (R)-rosmarinic acid,rosmarinic acid,迷迭香素,Rosemary acid
Target: MAO, Endogenous Metabolite, Transferase
7-Methoxyrosmanol
Cat.No: TN1334
Synonym: 7ALPHA-甲氧基迷迭香酚,7-O-Methylrosmanol
Target: cAMP
Rosmanol
Cat.No: T7033
Synonym:
Target: Antioxidant, COX
ethyl rosmarinate
Cat.No: TN6784
Synonym: 迷迭香酸乙酯
Target: MMP, Tyrosinase, Glucosidase
Epirosmanol
Cat.No: T9135
Synonym:
Target: Others
Methyl rosmarinate
Cat.No: TN1928
Synonym:
Target: MMP, Anti-infection, Tyrosinase
Rosmarinic acid
Cat.No: T2765
Synonym: Labiatenic acid,迷迭香酸,Rosemary acid
Target: Apoptosis, IκB/IKK, MAO, Endogenous Metabolite, Transferase, Monoamine Oxidase
Eudesmane
Cat.No: T31728
Synonym:
Target:
Chasmanine
Cat.No: T4S0818
Synonym:
Target:
Isodorsmanin A
Cat.No: TN4285
Synonym:
Target: Others
Alismanol M
Cat.No: T75538
Synonym:
Target:
7beta-Methoxyrosmanol
Cat.No: TN3257
Synonym:
Target: Transferase
Xysmalogenin
Cat.No: T35216
Synonym: BRN0051836,,BRN-0051836,BRN 0051836
Target:
Isorosmanol
Cat.No: TN1798
Synonym: 异迷迭香酚
Target: Beta Amyloid, AChR
6,8-Cyclo-1,4-eudesmanediol
Cat.No: TN3149
Synonym:
Target: Others
Rosmarinyl glucoside
Cat.No: TN6523
Synonym:
Target:
Dorsmanin A
Cat.No: TN3888
Synonym:
Target: Others
Eudesma-3,11-dien-2-one
Cat.No: TN4031
Synonym:
Target: Others
Osmanthuside B
Cat.No: T80009
Synonym:
Target:
Dorsmanin I
Cat.No: TN6351
Synonym:
Target:
1,4,7-Eudesmanetriol
Cat.No: TN2495
Synonym:
Target: Antifection
7-Ethoxyrosmanol
Cat.No: TN1329
Synonym:
Target: Antifection
Loureirin A
Cat.No: T5S0896
Synonym: 龙血素 A,龙血素A
Target: Akt, PI3K
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