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139

抑制剂 & 化合物

65

天然产物

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Cat. No. Product Name Target Signaling Pathways
T9073 SRS16-86

Ferroptosis Apoptosis
SRS16-86 是一种铁死亡抑制剂,可研究肾缺血再灌注损伤和脊髓损伤。它在体内比 Ferrostatin-1 对代谢和血浆更稳定。
T4612 NS309

EGFR; Potassium Channel; HER Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
NS309 是选择性钙依赖性钾离子通道 SK/IK 的激活剂,在 BK 通道上没有激活作用。
T68139 Scio-323

p38 MAPK MAPK
Scio-323是一种可口服的 p38丝裂原活化蛋白(MAPK)激酶抑制剂。
T20657 Muscimol HBr

Agarin hydrobromide,Muscimol Hydrobromide,Agarin HBr

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Muscimol HBr (Agarin HBr) 是GABAA 受体的激动剂
T9422 Fosciclopirox

CPX-POM

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Fosciclopirox (CPX-POM) 利用靶向γ-分泌酶,抑制尿路上皮癌的生长。静脉给药后,它选择性地将活性代谢物 Ciclopirox 递送至整个尿路。Ciclopirox 在许多实体和血液恶性肿瘤中显示出抗癌活性。
T5177 Asciminib

ABL001

Bcr-Abl Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Asciminib (ABL001) 是一种有效的、选择性的变构BCR-ABL1抑制剂,能够抑制 Ba/F3 细胞生长 (IC50:0.25 nM)。
T6493 Escitalopram Oxalate

草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Escitalopram Oxalate ((S)-(+)Citalopram oxalate) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T22304 Desciclovir

BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV

Antifection Microbiology/Virology
Desciclovir (DCV) 是抗疱疹药物阿昔洛韦的前药,口服有活性,在体内被黄嘌呤氧化酶转化成为阿昔洛韦。
T77046 Ivonescimab

Ivonescimab (AK112) 是一种PD-1/VEGF 双特异性抗体。Ivonescimab 可用于癌症研究。
T74219 Maximiscin

Maximiscin 是一种真菌代谢产物,可诱导DNA damage 损伤,并对一种三阴性乳腺癌亚型显示出选择性的细胞毒活性。
T34291 Rescinnamidine

Reserpic acid

Rescinnamidine is an alkaloid.
T125173 Fasciculic acid D

Fasciculic acid D 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125173,CAS号为 261638-74-8。
T126320 Anthriscifoldine B

Anthriscifoldine B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126320。
T25404 Fasciculic acid A

Fasciculic acid A is a calmodulin antagonist isolated from mushroom Naematoloma fasciculare.
T34290 Rescimetol

WHO-4939,WHO4939,WHO 4939

Rescimetol is a biochemical.
T34585 Scillicyanoside

Scillicyanosid

Scillicyanoside is a cardiac glycoside.
T124831 Scillarenin

Scillarenin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124831,CAS号为 465-22-5。
T34265 Raunescine monohydrate

Raunescine monohydrate is a biochemical.
T33889 Passitrifasciatin

Passitrifasciatin is a cyclopentanoid cyanohydrin glycoside isolated from Passiflora trifasciata.
T34581 Scicinib

Scicinib is a biologically active chemical that may be used to treat cancers of the blood and solid tumors.
T82415 Fasciculin-I

FAS-I

Fasciculin-I 是从曼巴蛇的毒液中分离出的化合物。该物质通过抑制乙酰胆碱酯酶(AChE)来发挥其毒性,同时阻碍烟碱乙酰胆碱受体与α-神经毒素以及心脏毒素与细胞膜的相互作用。
T25406 Fasciculic acid C

Fasciculic acid C is a calmodulin antagonist isolated from mushroom Naematoloma fasciculare.
T34587 Scirpusin A

Scirpusin-A

Scirpusin A is a hydroxystilbene dimer from the rhizome of Scirpus fluviatilis and Xinjiang wine grape.
T80378 Tilapia piscidin 3

Tilapia piscidin 3 是具抗菌谱广的肽类化合物,有效对抗多种革兰氏阳性菌与阴性菌,其对 V. vulnificus 204、V. alginolyticus、S. agalactiae 819、E. faecalis BCRC 10066、S. agalactiae BCRC 10787 的最小抑菌浓度 (MIC) 分别为 2.44、2.44、9.78、19.55、0.61 μg/mL。同時,Tilapia piscidin 3 对鱼红细胞显示出溶血性。
TP2283 parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]

Others Others
parathyroid hormone (7-34) [Homo sapiens] [Macaca fascicularis] is a peptide with the sequence H2N-LMHNLGKHLNSMERVEWLRKKLQDVHNF-OH, MW= 3474.03. Parathyroid hormone (PTH) is secreted by the chief cells of the parathyroid glands as a polypeptide containing
T80286 TP4 (Nile tilapia piscidin)

Necroptosis Apoptosis
TP4(Nile tilapia piscidin)是一种piscidin样的抗菌肽,其口服活性被证实。此化合物对多种革兰氏阳性及阴性菌株均有效(MIC: 0.03-10 μg/mL),并展现了溶血性。TP4还能增强免疫响应、提升抗氧化能力和改善肠道健康,助于防御细菌感染。除此之外,TP4显示抗肿瘤效果,并可通过激发癌细胞线粒体功能障碍导致坏死(necrosis)。
T28965 Thiomuscimol hydrobromide

Thiomuscimol hydrobromide is an agonist of GABAA receptor.
T34583 Scillabiose

Glucosidorhamnose

Scillabiose is a Glycone of both hellebrin and transvaalin.
T25405 Fasciculic acid B

Fasciculic acid B is the ester of fasciculol B and 3-hydroxy-3-methylglutaric acid. Fasciculic acid B is calmodulin antagonist from mushroom Naematoloma fasciculare.
T125410 Polyscioside D

Polyscioside D 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125410,CAS号为 202585-62-4。
T126360 Abscisic alcohol

Abscisic alcohol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126360,CAS号为 113472-20-1。
T31250 Deacetylscilliroside

6-Desacetyl-scilliroside,Desacetylscilliroside

Deacetylscilliroside is a biochemical.
T40755 Glabrescione B

Glabrescione B is a novel compound that specifically binds to Gli1, an important modulator of the Hedgehog (Hh) signaling pathway. By disrupting the Gli1-DNA interaction, Glabrescione B effectively impairs the activity of Gli1. Moreover, Glabrescione B demonstrates potent inhibitory effects on the growth of tumor cells that rely on Hedgehog signaling, as well as on the self-renewal capacity and clonogenicity of tumor-derived stem cells.
T126411 Glucoscillaren A

Glucoscillaren A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126411,CAS号为 11003-96-6。
T33291 Meproscillarin

KY-18,Rambufaside,Clift,KY 18,KY18

Meproscillarin is a glycoside with high bioavailability (about 70%) and an elimination independent of renal function.
TP1521 Piscidin-1 (22-42) (TFA)

Piscidin-1 (22-42) (TFA) is a highly potent, multi-functional Antimicrobial Peptide (AMP) produced by Orange-spotted grouper (Epinephelus coioides).
T31946 Glutamylputrescine

NGGP

Glutamylputrescine catalyzes the gamma-glutamylation of putrescine.
T37581 SCIO 469 hydrochloride

Selective, ATP-competitive p38 inhibitor (IC50 = 9 nM for p38α in vitro). Displays approximately 10-fold selectivity for p38α over p38β and 2000-fold selectivity for p38α over 20 other kinases. Reduces p38α phosphorylation in multiple myeloma cells in vitro and in vivo; activity results in decreased tumor burden and angiogenesis in murine models of multiple myeloma. Also enhances bortezomib-induced cytotoxicity against multiple myeloma cells. Hideshima et al (2004) p38 MAPK inhibition enhances P...
T33670 Nigrescigenin

Canescegenine,Canescegenin,Sarmentosigenin A

Nigrescigenin is a cardenolide from Parquetina nigrescens.
TP1475 Piscidin-1 (22-42)

Piscidin-1 (22-42) is a highly potent, multi-functional Antimicrobial Peptide (AMP) produced by Orange-spotted grouper (Epinephelus coioides).
T131538 Reserpinine (Raubasinine, Pubescine)

Reserpinine (Raubasinine, Pubescine) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131538。
T33352 Methylepoxyproscillaridin

Methylepoxyproscillaridin is a semisynthetic cardiac glycoside.
T73608 Muscimol hydrochloride

Muscimol (Agarin; Agarine) hydrochloride 是一种具有精神活性的异恶唑。Muscimol hydrochloride 也是抑制性神经递质 GABA 离子型受体的选择性激动剂。Muscimol hydrochloride 可以从毒蝇伞和相关蘑菇中分离出来。总之,Muscimol 是一种有效的 GABAA 受体激动剂 (EC50=0.2 μM),部分 GABAC 受体激动剂和无活性的 GABAB 受体激动剂。Muscimol hydrochloride 具有镇静、抗焦虑和致幻作用。
T126541 Viscic acid

Viscic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126541,CAS号为 100664-47-9。
T30152 Ascididemin

Leptoclinidinone,CRL 8274,NSC-675670,NSC 675670,NSC675670

Ascididemin can be regarded as a fused phenanthroline with quinoline.
T124458 Fasciculol C

Fasciculol C 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124458,CAS号为 65694-19-1。
T75381 Bodipy TMR-X muscimol

Bodipy TMR-X muscimol为标记有Bodipy的Muscimol(Ex=543 nm, Em=572 nm),是GABAA受体的激动剂。该化合物适用于可视化可逆脑失活的扩散研究。
T31746 Fasciculol A

Fasciculol A is a terpenoid.
T63226 Asciminib hydrochloride

Asciminib (ABL001) hydrochloride 是选择性的、有效的变构 BCR-ABL1 抑制剂,能够抑制 Ba/F3 细胞生长(IC50: 0.25 nM)。
T34265L Raunescine monoacetate monohydrate

Raunescine monoacetate monohydrate is a biochemical.

化合物

SRS16-86
Cat.No: T9073
Synonym:
Target: Ferroptosis
NS309
Cat.No: T4612
Synonym:
Target: EGFR, Potassium Channel, HER
Scio-323
Cat.No: T68139
Synonym:
Target: p38 MAPK
Muscimol HBr
Cat.No: T20657
Synonym: Agarin hydrobromide,Muscimol Hydrobromide,Agarin HBr
Target: GABA Receptor
Fosciclopirox
Cat.No: T9422
Synonym: CPX-POM
Target: Gamma-secretase
Asciminib
Cat.No: T5177
Synonym: ABL001
Target: Bcr-Abl
Escitalopram Oxalate
Cat.No: T6493
Synonym: 草酸右旋西酞普兰,依他普仑草酸盐,Cipralex,(S)-(+)Citalopram oxalate
Target: Others, 5-HT Receptor, Serotonin Transporter
Desciclovir
Cat.No: T22304
Synonym: BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV
Target: Antifection
Ivonescimab
Cat.No: T77046
Synonym:
Target:
Maximiscin
Cat.No: T74219
Synonym:
Target:
Rescinnamidine
Cat.No: T34291
Synonym: Reserpic acid
Target:
Fasciculic acid D
Cat.No: T125173
Synonym:
Target:
Anthriscifoldine B
Cat.No: T126320
Synonym:
Target:
Fasciculic acid A
Cat.No: T25404
Synonym:
Target:
Rescimetol
Cat.No: T34290
Synonym: WHO-4939,WHO4939,WHO 4939
Target:
Scillicyanoside
Cat.No: T34585
Synonym: Scillicyanosid
Target:
Scillarenin
Cat.No: T124831
Synonym:
Target:
Raunescine monohydrate
Cat.No: T34265
Synonym:
Target:
Passitrifasciatin
Cat.No: T33889
Synonym:
Target:
Scicinib
Cat.No: T34581
Synonym:
Target:
Fasciculin-I
Cat.No: T82415
Synonym: FAS-I
Target:
Fasciculic acid C
Cat.No: T25406
Synonym:
Target:
Scirpusin A
Cat.No: T34587
Synonym: Scirpusin-A
Target:
Tilapia piscidin 3
Cat.No: T80378
Synonym:
Target:
parathyroid hormone (7-34) [Homo sapiens]/[Macaca fascicularis]
Cat.No: TP2283
Synonym:
Target: Others
TP4 (Nile tilapia piscidin)
Cat.No: T80286
Synonym:
Target: Necroptosis
Thiomuscimol hydrobromide
Cat.No: T28965
Synonym:
Target:
Scillabiose
Cat.No: T34583
Synonym: Glucosidorhamnose
Target:
Fasciculic acid B
Cat.No: T25405
Synonym:
Target:
Polyscioside D
Cat.No: T125410
Synonym:
Target:
Abscisic alcohol
Cat.No: T126360
Synonym:
Target:
Deacetylscilliroside
Cat.No: T31250
Synonym: 6-Desacetyl-scilliroside,Desacetylscilliroside
Target:
Glabrescione B
Cat.No: T40755
Synonym:
Target:
Glucoscillaren A
Cat.No: T126411
Synonym:
Target:
Meproscillarin
Cat.No: T33291
Synonym: KY-18,Rambufaside,Clift,KY 18,KY18
Target:
Piscidin-1 (22-42) (TFA)
Cat.No: TP1521
Synonym:
Target:
Glutamylputrescine
Cat.No: T31946
Synonym: NGGP
Target:
SCIO 469 hydrochloride
Cat.No: T37581
Synonym:
Target:
Nigrescigenin
Cat.No: T33670
Synonym: Canescegenine,Canescegenin,Sarmentosigenin A
Target:
Piscidin-1 (22-42)
Cat.No: TP1475
Synonym:
Target:
Reserpinine (Raubasinine, Pubescine)
Cat.No: T131538
Synonym:
Target:
Methylepoxyproscillaridin
Cat.No: T33352
Synonym:
Target:
Muscimol hydrochloride
Cat.No: T73608
Synonym:
Target:
Viscic acid
Cat.No: T126541
Synonym:
Target:
Ascididemin
Cat.No: T30152
Synonym: Leptoclinidinone,CRL 8274,NSC-675670,NSC 675670,NSC675670
Target:
Fasciculol C
Cat.No: T124458
Synonym:
Target:
Bodipy TMR-X muscimol
Cat.No: T75381
Synonym:
Target:
Fasciculol A
Cat.No: T31746
Synonym:
Target:
Asciminib hydrochloride
Cat.No: T63226
Synonym:
Target:
Raunescine monoacetate monohydrate
Cat.No: T34265L
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2064 Physcion 8-O-β-D-glucopyranoside

大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside

TNF Apoptosis
Physcion 8-O-β-D-glucopyranoside (Physcion 8-O-beta-D-monoglucoside) 具有抗炎和抗癌活性。Physcion 8-O-β-D-glucopyranoside 可用于常见恶性肿瘤的研究。
T3771 Methyl protodioscin

山药,Smilax saponin B,NSC-698790

Apoptosis Apoptosis
Methyl protodioscin (Smilax saponin B) 是一种甾二糖苷,能诱导细胞周期阻滞,具有抗肿瘤活性。
T5S2129 Sciadopitysin

TNF; NF-κB Apoptosis; NF-κB
Sciadopitysin 是一种双黄酮类化合物,来自银杏叶片中。它通过抑制NF-κB 活化并降低c-Fos 和NFATc1的表达来抑制 RANKL 诱导的破骨细胞生成和骨丢失。
T3019 Physcion

大黄素甲醚,Physcione,Parietin,Rheochrysidin

Dehydrogenase; Antibacterial Metabolism; Microbiology/Virology
Physcion (Physcione) 是一种从中药大黄中分离的蒽醌,作为 6-磷酸葡萄糖酸脱氢酶的抑制剂,IC50和 Kd 值分别为 38.5 μM 和 26.0 μM。它具有通便、保肝、抗炎、抗菌、抗增殖、抗肿瘤作用。
T5S0246 Pseudoprotodioscin

山药

Others; Fatty Acid Synthase Metabolism; Others
Pseudoprotodioscin 是一种呋喃葡糖苷,抑制SREBP1/2和microRNA 33a/b 水平,降低胆固醇和甘油三酯合成相关的基因表达。
T8846 beta-Escin

B-escin,AESCINE,beta-七叶素

Immunology/Inflammation related Immunology/Inflammation
beta-Escin 是七叶树种子的主要活性成分。它可抑制碱性成纤维细胞生长因子所诱导的增殖、迁移、管形成以及体内 CAM 血管生成。它具有研究抗血管生成作用的分子机制的潜力。
T7508 N-Acetylputrescine hydrochloride

Endogenous Metabolite Metabolism
N-Acetylputrescine hydrochloride 是腐胺衍生物。
T3932 Viscidulin I

Others Others
Viscidulin I 存在于黄芩中,是一种天然产物。
T3014 (±)-Abscisic acid

Abscisic acid,Dormin,脱落酸,Abscisinsaeure

Others Others
(±)-Abscisic acid (Dormin) 是一种口服具有活性的植物激素,也存在与动物中。它可以调节哺乳动物的血糖。
T0278 Escin

七叶皂苷,七叶皂素,Aescin

Apoptosis; Others Apoptosis; Others
Escin (Aescin) 是从七叶树种子中分离得到的一种三萜皂苷,有血管保护、抗炎、抗水肿和抗伤害作用。
T4429 Rauwolscine hydrochloride

Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。
T2321 Protodioscin

Furostanol I,原薯蓣皂苷

Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Protodioscin (Furostanol I) 是一种山药根茎中的主要甾体皂苷,具有抗高血脂、抗癌活性。
T5S1389 Escin IB

七叶皂苷B,七叶皂苷 IB

5-HT Receptor; NO Synthase GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escin IB 是一种皂苷,分离自马栗子种子的皮和胚乳中,能够抑制 pancreatic lipase 的活性。
TN2107 Protoescigenin

Others Others
Protoescigenin 来自七叶树皂甙混合物,可用作用于选择性保护的探索性化学的底物。
T4S1387 Isoescin IA

七叶皂苷C,异七叶皂苷 IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Isoescin IA 是一种从七叶树种子中分离出来的三萜皂苷。它具有抗HIV-1蛋白酶活性。
T8918 Feruloylputrescine

Others Others
Feruloylputrescine 是一种天然产物。
T3027 Sodium Aescinate

Escin sodium salt,七叶皂苷钠

HIF Angiogenesis; Chromatin/Epigenetic
Sodium Aescinate (Escin sodium salt) 是一种三萜皂苷,来源于Aesculus hippocastanum 的种子,具有抗炎、抗氧化作用。它可以通过靶向 CARMA3/NF-κB 途径,抑制抑制肝癌生长。
T6473 Dioscin

山药,CCRIS 4123,Collettiside III,Saponin

Apoptosis; Autophagy Apoptosis; Autophagy
Dioscin (Collettiside III) 是一种来源植物的天然甾体皂苷,针对多种癌细胞有较好的抗癌活性。
T6368 Abscisic Acid

Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)

Others; Proton pump; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Abscisic Acid (Dormin) 是具有口服活性的植物激素,存在于蔬菜和水果中,也是内源性的哺乳动物激素。它是生长抑制剂,可以调节植物生长发育。他抑制质子泵,并导致 Ca2+依赖性的质膜去极化。它是 LANCL2 的天然配体,属于胰岛素敏感化合物,在糖尿病前期,2 型糖尿病和代谢综合征的研究中具有价值。
TN1777 Isoescin IB

Others Others
Isoescin IB 是 Escin IB 的异构体,两者是 Escin 中的主要活性成分。
T4S1383 Escin IA

Aescin IA,Escin IA;Aescin IA,Escin IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Escin IA (Escin IA;Aescin IA);Aescin IA 是从马蹄中七叶树分离出的一种三萜皂苷,抑制HIV-1蛋白酶,IC50值为 35 μM。它具有抗 TNBC 转移活性,其作用机制涉及通过下调 LOXL2 表达抑制上皮-间质转化过程。
TN2302 Viscidulin III

Ganhuangenin

Glucosidase Metabolism
Viscidulin III (Ganhuangenin) 存在于黄芩中,可作为α-葡萄糖苷酶抑制剂。
TN4963 Scillascillin

Others Others
Scillascillin has anticancer activity, it is significantly active against human cancer cell lines MCF-7 (breast cancer) and DU-145 (prostate cancer) with inhibitory concentration (IC)50 values 9.59 and 11.32 ug/ml respectively.
TN1967 N-​Caffeoylputrescine,​(E)​-

咖啡酰丁二胺,(E)-N-Caffeoylputrescine

Others Others
N-Caffeoylputrescine has antioxidant activity.
TN7009 CANNABISCITRIN

CANNABISCITRIN is a natural product.
T81768 Molluscicidal agent-1

Molluscicidal agent-1 (Compound 3)为从S. vesicaria分离得到的皂苷类化合物。
T79996 N,N′-Diferuloylputrescine

Melanocortin Receptor GPCR/G Protein; Neuroscience
N,N′-Diferuloylputrescine 作为pigmentation的抑制剂,有效减少了57%的色素沉着,并显著降低了MITF蛋白水平。同时,该化合物对活性氧表现出强大的抗氧化活性。
TN1358 Escin IIa

七叶皂苷C,Aescin IIA

Others Others
Aescin IIA is a natural product
TN4965 Scillascillone

Others Others
Scillascillone is a natural product from Scilla scilloides.
T34584 Scillaren A

Transvaalin,Scillaglykosid A

Scillaren A is a a crystalline steroidal glycoside from Scilla maritima.
TN2765 2-Hydroxy-7-O-methylscillascillin

Others Others
2-Hydroxy-7-O-methylscillascillin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2765,CAS号为 52096-50-1。
TN3882 Dodoviscin A

cAMP; Tyrosinase; transporter GPCR/G Protein; Metabolism; Proteases/Proteasome
Dodoviscin A may be a new promising pigmentation-altering agent for cosmetic and therapeutic applications, it can inhibit melanin biosynthesis induced by 3-isobutyl-1-methylxanthine and PD98059.Dodoviscin A can promote adipocyte differentiation as charact
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T39605 β-D-Glucopyranosyl abscisate

ABA-GE,β-D-Glucopyranosyl abscisate,(S)-cis,trans-Abscisicacidglucosylester

β-D-Glucopyranosyl abscisate (ABA-GE) is a hydrolyzable conjugate of abscisic acid (ABA), which predominantly accumulates in the vacuole and likely in the endoplasmic reticulum. The deconjugation of β-D-Glucopyranosyl abscisate enables a swift release of free ABA in response to abiotic stress factors like dehydration and salt stress. β-D-Glucopyranosyl abscisate plays a crucial role in maintaining ABA homeostasis.
TN4801 Piscidinol A

Others Others
Piscidinol A is toxic against the 4T1 and HEp2 cancer cell lines, the IC50 of 8.0 ± 0.03 and 8.4 ± 0.01 uM, respectively. It can inhibit NO production in mouse peritoneal macrophages with inhibitory ratios ranging from 39.8±7.7 to 68.2±4.5%.
TN4781 Physcion 8-O-rutinoside

Others Others
Physcion 8-O-rutinoside is a natural product from Rhamnus libanoticus.
T12093 Monascin

Others Others
Monascin is a kind of azaphilonoid pigments extracted from Monascus pilosus-fermented rice (red-mold rice),exhibits anti-tumor-initiating activity and anti-inflammatory activity .
TN4964 Scillascillol

Others Others
Scillascillol is a natural product from Scilla scilloides.
T32575 Lascivol

Lascivol is a bitter substance derived from Tricholoma lascivum.
TN5239 Viscidulin III tetraacetate

Others Others
Viscidulin III tetraacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5239,CAS号为 96684-81-0。
TN3885 Dodoviscin J

transporter Metabolism
Dodoviscin J can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
TN1623 Escin IIB

Others; NOS Immunology/Inflammation; Others
Escin IIB has positive effects on acute inflammation in animals, it can inhibit the induced by serotonin in rats, the hind paw edema induced by carrageenin, and the scratching behavior induced by compound 48/80 in mice.
T82036 Isoescin Ie

Isoescin Ie,一种Aescine的衍生物,系由Aesculi Semen提取物中分离得到。
T15111 Diacetoxyscirpenol

Others Others
Diacetoxyscirpenol, a trichothecene mycotoxin, is a secondary metabolite product of fungi. Diacetoxyscirpenol consumption induces hematological disorders in humans and animals.
TN6024 N-p-Coumaroyl-N'-caffeoylputrescine

N-p-Coumaroyl-N'-caffeoylputrescine是一种天然产物,属于蔷薇科白鹃梅属,其产品编号为 TN6024,CAS号为 1138156-77-0。N-p-Coumaroyl-N'-caffeoylputrescine可用作对照参考。
T39080 Escin Ie

Escin Ie is a derivative of Aescine in Aesculi Semen extract.
TN5364 Boscialin

Boscialin can inhibit signal transducer and activator of transcription 1 translocation at a concentration of 10 uM.
TN5238 Viscidulin II

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Viscidulin II can be potential therapeutic agents against P. acnes-induced skin inflammation, it can significantly suppress P. acnes-induced IL-8 and IL-1β production in THP-1 cells, concomitant intradermal injection of viscidulin II with P. acnes can effectively attenuate P. acnes-induced ear swelling, and decrease the production of IL-6 and tumor necrosis factor-α in ear homogenates.
TN3772 Datiscin

Others Others
Datiscin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3772,CAS号为 16310-92-2。
TN4966 Scillascilloside B-1

Others Others
Scillascilloside B-1 is a natural product from Scilla scilloides.
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天然产物

Physcion 8-O-β-D-glucopyranoside
Cat.No: TN2064
Synonym: 大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside
Target: TNF
Methyl protodioscin
Cat.No: T3771
Synonym: 山药,Smilax saponin B,NSC-698790
Target: Apoptosis
Sciadopitysin
Cat.No: T5S2129
Synonym:
Target: TNF, NF-κB
Physcion
Cat.No: T3019
Synonym: 大黄素甲醚,Physcione,Parietin,Rheochrysidin
Target: Dehydrogenase, Antibacterial
Pseudoprotodioscin
Cat.No: T5S0246
Synonym: 山药
Target: Others, Fatty Acid Synthase
beta-Escin
Cat.No: T8846
Synonym: B-escin,AESCINE,beta-七叶素
Target: Immunology/Inflammation related
N-Acetylputrescine hydrochloride
Cat.No: T7508
Synonym:
Target: Endogenous Metabolite
Viscidulin I
Cat.No: T3932
Synonym:
Target: Others
(±)-Abscisic acid
Cat.No: T3014
Synonym: Abscisic acid,Dormin,脱落酸,Abscisinsaeure
Target: Others
Escin
Cat.No: T0278
Synonym: 七叶皂苷,七叶皂素,Aescin
Target: Apoptosis, Others
Rauwolscine hydrochloride
Cat.No: T4429
Synonym: Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
Protodioscin
Cat.No: T2321
Synonym: Furostanol I,原薯蓣皂苷
Target: Androgen Receptor, Endogenous Metabolite
Escin IB
Cat.No: T5S1389
Synonym: 七叶皂苷B,七叶皂苷 IB
Target: 5-HT Receptor, NO Synthase
Protoescigenin
Cat.No: TN2107
Synonym:
Target: Others
Isoescin IA
Cat.No: T4S1387
Synonym: 七叶皂苷C,异七叶皂苷 IA
Target: HIV Protease
Feruloylputrescine
Cat.No: T8918
Synonym:
Target: Others
Sodium Aescinate
Cat.No: T3027
Synonym: Escin sodium salt,七叶皂苷钠
Target: HIF
Dioscin
Cat.No: T6473
Synonym: 山药,CCRIS 4123,Collettiside III,Saponin
Target: Apoptosis, Autophagy
Abscisic Acid
Cat.No: T6368
Synonym: Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)
Target: Others, Proton pump, Endogenous Metabolite
Isoescin IB
Cat.No: TN1777
Synonym:
Target: Others
Escin IA
Cat.No: T4S1383
Synonym: Aescin IA,Escin IA;Aescin IA,Escin IA
Target: HIV Protease
Viscidulin III
Cat.No: TN2302
Synonym: Ganhuangenin
Target: Glucosidase
Scillascillin
Cat.No: TN4963
Synonym:
Target: Others
N-​Caffeoylputrescine,​(E)​-
Cat.No: TN1967
Synonym: 咖啡酰丁二胺,(E)-N-Caffeoylputrescine
Target: Others
CANNABISCITRIN
Cat.No: TN7009
Synonym:
Target:
Molluscicidal agent-1
Cat.No: T81768
Synonym:
Target:
N,N′-Diferuloylputrescine
Cat.No: T79996
Synonym:
Target: Melanocortin Receptor
Escin IIa
Cat.No: TN1358
Synonym: 七叶皂苷C,Aescin IIA
Target: Others
Scillascillone
Cat.No: TN4965
Synonym:
Target: Others
Scillaren A
Cat.No: T34584
Synonym: Transvaalin,Scillaglykosid A
Target:
2-Hydroxy-7-O-methylscillascillin
Cat.No: TN2765
Synonym:
Target: Others
Dodoviscin A
Cat.No: TN3882
Synonym:
Target: cAMP, Tyrosinase, transporter
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
β-D-Glucopyranosyl abscisate
Cat.No: T39605
Synonym: ABA-GE,β-D-Glucopyranosyl abscisate,(S)-cis,trans-Abscisicacidglucosylester
Target:
Piscidinol A
Cat.No: TN4801
Synonym:
Target: Others
Physcion 8-O-rutinoside
Cat.No: TN4781
Synonym:
Target: Others
Monascin
Cat.No: T12093
Synonym:
Target: Others
Scillascillol
Cat.No: TN4964
Synonym:
Target: Others
Lascivol
Cat.No: T32575
Synonym:
Target:
Viscidulin III tetraacetate
Cat.No: TN5239
Synonym:
Target: Others
Dodoviscin J
Cat.No: TN3885
Synonym:
Target: transporter
Escin IIB
Cat.No: TN1623
Synonym:
Target: Others, NOS
Isoescin Ie
Cat.No: T82036
Synonym:
Target:
Diacetoxyscirpenol
Cat.No: T15111
Synonym:
Target: Others
N-p-Coumaroyl-N'-caffeoylputrescine
Cat.No: TN6024
Synonym:
Target:
Escin Ie
Cat.No: T39080
Synonym:
Target:
Boscialin
Cat.No: TN5364
Synonym:
Target:
Viscidulin II
Cat.No: TN5238
Synonym:
Target: IL Receptor, TNF
Datiscin
Cat.No: TN3772
Synonym:
Target: Others
Scillascilloside B-1
Cat.No: TN4966
Synonym:
Target: Others
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