117
8
6
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16079 |
Mirodenafil
米罗那非,SK3530 |
PDE | Metabolism |
Mirodenafil 是一种磷酸二酯酶5(PDE-5)抑制剂,可用于勃起功能紊乱的研究。 | |||
T68112 |
Nafimidone
|
||
Nafimidone 在大鼠杏仁核癫痫模型中显示出抗惊厥活性,可用于治疗慢性顽固性癫痫病。 | |||
T1543 |
Naftifine hydrochloride
Naftifungin,盐酸萘替芬,Naftifine HCl,Naftin,Exoderil |
Hedgehog/Smoothened; Antibiotic; Antifungal | GPCR/G Protein; Microbiology/Virology; Stem Cells |
Naftifine hydrochloride (Naftifine HCl) 是一种抗生素。它具有抗真菌活性,对皮肤真菌、曲霉、Sporothrix schenckii、假丝酵母属的酵母有抑制作用。 | |||
T0096 |
Vardenafil
伐地那非,Vivanza,Levitra,Vardenafil hydrochloride |
PDE | Metabolism |
Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂,IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解,从而提高 cGMP 水平。它对 PDE1 (180 nM),PDE6 (11 nM),PDE2,PDE3,PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。 | |||
T6302 |
Lonafarnib
Sarasar,氯那法尼,Sch66336 |
Raf; Transferase; Autophagy; Ras | Autophagy; GPCR/G Protein; MAPK; Metabolism |
Lonafarnib (Sch66336) 是一种可口服的 FPTase 抑制剂,作用于 H-ras、K-ras 和 N-ras,IC50分别为 1.9 nM、5.2 nM 和 2.8 nM。它具有抗肝炎三角洲病毒的活性。 | |||
T6600 |
Naftopidil dihydrochloride
KT-611,KT-611 2HCl,盐酸萘哌地尔,Naftopidil DiHCl |
5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Naftopidil dihydrochloride (KT-611 2HCl) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。 | |||
T33762 |
Fosifloxuridine nafalbenamide
NUC-3373,NUC3373,NUC 3373 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Fosifloxuridine nafalbenamide (NUC 3373) 是一种胸腺嘧啶合酶抑制剂,属于嘧啶核苷酸类似物,具有抗癌活性。它能诱发宿主免疫反应,有潜力增强免疫治疗。 | |||
T10634 |
Bunaftide
Bunaphtide,Meregon,Bunaftine |
Others | Others |
Bunaftide(Bunaphtid)具有抗心律失常作用,对乌头碱诱导的室性心动过速有抑制作用。 | |||
T15381 |
Gisadenafil
UK-369003,吉沙那非 |
PDE | Metabolism |
Gisadenafil (UK-369003) 是一种特异性磷酸二酯酶 5 (PDE5) 抑制剂,IC50 为 3.6 nM,可防止 cGMP 降解。 | |||
T6336 |
Amonafide
NSC308847,AS1413,氨萘非特,Nafidimide,AS1413,Quinamed |
Topoisomerase | DNA Damage/DNA Repair |
Amonafide (NSC-308847,AS1413) 是一种拓扑异构酶 II 的抑制剂和 DNA 的嵌入剂,通过拓扑异构酶 II 介导的反应产生蛋白质相关的 DNA 链断裂 | |||
T1312 |
Nafcillin sodium monohydrate
CL 8491,萘夫西林钠,nafcillin sodium |
Antibacterial; Antibiotic | Microbiology/Virology |
Nafcillin sodium monohydrate (CL 8491) 是一种抗生素,是可逆的β-lactamase 抑制剂。它用于治疗由耐青霉素的葡萄球菌菌株引起的感染。 | |||
T4097 |
Vardenafil hydrochloride trihydrate
Vardenafil HCl Trihydrate,BAY38-9456,盐酸瓦地那非三水合物 |
PDE | Metabolism |
Vardenafil hydrochloride trihydrate (BAY38-9456) 是一种新型 PDE 抑制剂,对 PDE5 和 PDE1 的 IC50 分别为 0.7 和 180 nM。 | |||
T10758L |
Centanafadine hydrochloride
EB-1020 hydrochloride |
Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。 | |||
T8919 |
Homo Sildenafil
蒙莫西地那非,豪莫西地那非 |
PDE | Metabolism |
Homo Sildenafil 是一种 Sildenafil 的类似物,是一种磷酸二酯酶抑制剂。 | |||
T1217 |
Butenafine hydrochloride
KP363 (Hydrochloride),Butenafine HCl,KP-363,盐酸布替萘芬 |
Antibiotic; Antifungal | Microbiology/Virology |
Butenafine hydrochloride (KP363 Hydrochloride) 通过抑制鲨烯环氧酶阻断甾醇的合成,具有抗真菌活性。 | |||
T1081 |
Naftidrofuryl oxalate
萘呋胺酯 草酸盐,Nafronyl oxalate,Nafronyl oxalate salt |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Naftidrofuryl oxalate (Nafronyl oxalate) 是一种用于治疗外周和脑血管疾病的药物,可增加细胞氧化能力,也是一种 5-HT2 受体拮抗剂。 | |||
T1497 |
Liranaftate
Piritetrate,利拉萘酯,M-732 |
Antifungal | Microbiology/Virology |
Liranaftate (Piritetrate) 是一种具有抗真菌活性的硫代氨基甲酸酯和角鲨烯环氧酶抑制剂,可研究皮肤癣菌。 | |||
T2392 |
Nafamostat mesylate
甲磺酸萘莫司他,FUT-175 |
Apoptosis; Serine/threonin kinase; SARS-CoV; Serine Protease | Apoptosis; Cell Cycle/Checkpoint; Metabolism; Microbiology/Virology; Proteases/Proteasome |
Nafamostat mesylate (FUT-175) 是一种广谱丝氨酸蛋白酶抑制剂,血管舒缓素抑制剂,能抑制血液凝固。它通过降低颗粒酶活性和 CTL 细胞溶解抑制T 细胞自身反应活性,可抑制SARS-CoV-2 的激活。它还是潜在的补体抑制剂。 | |||
T1094 |
Tolnaftate
Tonoftal,托萘酯,Sporiline,Tinactin,NP-27 |
Hedgehog/Smoothened; Antifungal | GPCR/G Protein; Microbiology/Virology; Stem Cells |
Tolnaftate (NP-27) 是一种合成的硫代氨基甲酸酯类抗真菌剂。 | |||
T8471 |
Vonafexor
EYP001,PLX007,pxl007 |
FXR; HBV | Metabolism; Microbiology/Virology |
Vonafexor (EYP001) 是一种法尼醇 X 受体激动剂,具有抗 HBV 作用。 | |||
T7346 |
Lodenafil
Hydroxyhomosildenafil,羟基豪莫西地那非 |
PDE | Metabolism |
Lodenafil (Hydroxyhomosildenafil) 是一种有效的磷酸二酯酶 5 型(PDE5)抑制剂,可用于勃起功能障碍的研究。 | |||
T33581 |
Nafetolol
K 5407,K-5407 |
Others | Others |
Nafetolol (K 5407) 是一种生化试剂,可用于合成其他化合物。 | |||
T1283 |
Clinafloxacin
克林沙星,PD 127391,CI-960,AM-1091 |
Antibacterial; Antibiotic | Microbiology/Virology |
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。 | |||
T0467 |
Sildenafil citrate
UK-92480 citrate,西地那非柠檬酸盐,枸橼酸西地那非 |
Apoptosis; PDE; Autophagy | Apoptosis; Autophagy; Metabolism |
Sildenafil citrate (UK-92480 citrate) 是一种磷酸二酯酶 5 抑制剂,IC50为 5.22 nM。 | |||
T14219 |
Aminaftone
Aminaphthone |
Endothelin Receptor | GPCR/G Protein |
Aminaftone 是 4-氨基苯甲酸的衍生物,可抑制内皮素-1 (ET-1) 的产生,可用于研究高血压和系统硬化症。 | |||
T21309 |
Nafarelin acetate(76932-56-4 free base)
RS-94991-298,醋酸萘法瑞林,Nafarelin acetate,Nafarelin acetate hydrate,Synarel |
GNRH Receptor | GPCR/G Protein |
Nafarelin acetate(76932-56-4 free base) (RS-94991-298) 是一种 GnRH 激动剂,可作为 GnRH 的类似物。 Nafarelin acetate(76932-56-4 free base) 导致促性腺激素促黄体激素 (LH) 和促卵泡激素 (FSH) 的垂体分泌减少。它可用于治疗雌激素依赖性病症。 | |||
T9220 |
Naftopidil hydrochloride
1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-,萘哌地尔盐酸盐,KT-611 hydrochloride,BM-15275 hydrochloride |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Naftopidil hydrochloride (BM-15275 hydrochloride) 是一种选择性的 alpha1-肾上腺素受体 (α1-adrenoceptor) 拮抗剂,对克隆的人类 α1a、α1b 和 α1d 亚型肾上腺素受体的亲和力 Ki 分别为 3.7 nM、20 nM、1.2 nM。它具有抗增殖活性,可用于研究前列腺增生。 | |||
T25817 |
Mitonafide
NSC-300288,米托萘胺,NSC300288,NSC 300288 |
Antibacterial | Microbiology/Virology |
Mitonafide (NSC-300288) 抑制 M. tuberculosis NAD+ 依赖性 DNA 连接酶 A 的活性。 它是一种 DNA 嵌入剂。 | |||
T36061 |
N-Desmethyl Sildenafil
Desmethylsildenafil,UK-103,320 |
Drug Metabolite | Metabolism |
N-Desmethyl Sildenafil (UK-103,320) (Desmethylsildenafil) 是Sildenafil的主要代谢物,是一种强效的磷酸二酯酶类型5(PDE5)抑制剂。 | |||
T10676 |
Carbodenafil
|
PDE | Metabolism |
Carbodenafil 是在健康食品中发现的 Sildenafil 相关化合物。其中Sildenafil 是磷酸二酯酶 5 (PDE5) 抑制剂(IC50:5.22 nM)。 | |||
T6983 |
Sildenafil Mesylate
|
PDE | Metabolism |
Sildenafil Mesylate 是 Sildenafil 的甲磺酸盐形式,Sildenafil 是磷酸二酯酶 5 的抑制剂。 | |||
T68061 |
Elinafide
|
||
Elinafide 是一种双萘酰亚胺细胞毒性剂,是 DNA 靶向抗癌剂,在体内体外实验中显示出抗肿瘤活性。 | |||
T6653 |
Salmeterol Xinafoate
Salmetedur,昔美酸沙美特罗,沙美特罗昔萘酸酯,GR 33343X xinafoate,Arial |
HIV Protease; Adrenergic Receptor | GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Salmeterol Xinafoate (GR 33343X xinafoate) 是选择性人β2肾上腺素受体激动剂。Salmeterol 有效刺激 cAMP 积累,能够作用于 CHO 细胞,对人β2,β1和β3肾上腺素受体的 pEC50分别为 9.6、6.1 和 5.9。 | |||
T2334 |
Avanafil
阿伐那非,TA1790 |
PDE | Metabolism |
Avanafil (TA1790) 是一种高活性PDE-5抑制剂,IC50=5.2 nM,对PDE1,PDE6和PDE11活性较低。 | |||
T8877 |
Bonafton
1,2-萘醌,6-溴-,Bonaphthone |
Antiviral | Immunology/Inflammation |
Bonafton (Bonaphthone) 是一种抗病毒剂。 | |||
T8405 |
Vardenafil hydrochloride
伐地那非,盐酸伐地那非 |
PDE | Metabolism |
Vardenafil hydrochloride 是口服具有活性的、高效的、选择性的磷酸二酯酶 5抑制剂。它对 PDE1 (180 nM),PDE6 (11 nM),PDE2,PDE3,PDE4 (>1000 nM) 具有选择性。它能够非竞争性地抑制环磷酸鸟苷水解,提高 cGMP 水平。它可用于勃起功能障碍的研究。 | |||
TQ0126 |
Mirodenafil dihydrochloride
SK-3530 dihydrochloride,米罗那非二盐酸盐 |
PDE | Metabolism |
Mirodenafil dihydrochloride 是一种磷酸二酯酶5(PDE-5)抑制剂,可作用于勃起功能紊乱的研究。 | |||
T21387L |
Nafoxidine
|
Estrogen Receptor/ERR | Endocrinology/Hormones |
Nafoxidine 是一种雌激素拮抗剂,已用于治疗乳腺癌。 | |||
T4992 |
Cefamandole nafate
Cephamandole nafate,头孢孟多酯钠,Cefamandole formate sodium |
Antibacterial; Antibiotic | Microbiology/Virology |
Cefamandole nafate (Cephamandole nafate) 是一种广谱头孢菌素抗生素。 | |||
T19200 | Azonafide-PEABA | Others | Others |
Azonafide-PEABA 是一种具有细胞毒性的药物。 | |||
T71658 | Indacaterol xinafoate | ||
Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist. | |||
T71519 | Chlorodenafil | ||
Chlorodenafil is a related compound of Sildenafil -- a phosphodiesterase inhibitor. | |||
T24518 |
Naftypramide
DA-992,Naftipramida,Naftypramidum,DA 992,BRN 2815141 |
||
Naftypramide is a nonsteroidal agent of anti-inflammatory. | |||
T37181 |
Avanafil metabolite M4
Avanafil metabolite M4 |
||
Avanafil metabolite M4 is a major active metabolite of the phosphodiesterase 5 (PDE5) inhibitor avanafil . Avanafil is metabolized by the cytochrome P450 (CYP450) isoforms CYP3A4 and CYP2C to the major metabolites avanafil metabolite M4 and avanafil metabolite M16 , as well as minor metabolites. Avanafil metabolite M4 inhibits PDE5 with 18% of the potency of avanafil. | |||
T36062 | N-Desmethyl Sildenafil (citrate) | ||
N-Desmethyl sildenafil is a major metabolite of sildenafil . N-Desmethyl sildenafil is formed via oxidative metabolism of sildenafil by the cytochrome (CYP) P450 isoforms CYP3A4, CYP3A5, and CYP3A7. | |||
T68665 |
Yonkenafil
Tunodafil |
||
Yonkenafil (Tunodafil) 是一种新型PDE5抑制剂,对脑梗塞、神经功能缺损、水肿及梗塞区域神经元损伤具有显著降低效果。通过调节神经发生,Yonkenafil 可改善认知功能,展现出在阿尔茨海默病研究中的潜在价值。 | |||
T40399 |
ZnAF-1
|
||
ZnAF-1, a zinc sensor compound, utilizes a fluorescein-based structure incorporating the N,N-bis(2-pyridylmethyl)ethylenediamine chelating unit. Its primary function lies in the detection of Zn2+ ions. Through its binding capability, ZnAF-1 achieves a 1:1 stoichiometry with Zn(II). | |||
T20159 |
Bilanafos
Herby,Bialaphos,Antibiotic SF 1293 |
||
Bilanafos is an agent of Anti-Bacterial. | |||
T33582 |
Nafimidone alcohol
|
||
Nafimidone alcohol is a Nafimidone metabolite. | |||
T38451 |
Clodinafop-propargyl
|
||
Clodinafop-propargyl, a prominent member of aryloxyphenoxy-propionate herbicides, is employed for postemergence management of annual grasses in cereals, such as Avena, Lolium, Setaria, Phalaris, and Alopecurus spp. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T17199 |
Udenafil
3-(6,7-二氢-1-甲基-7-氧代-3-丙基-1H-吡唑并[4,3-D]嘧啶-5-基)-N-[2-(1-甲基-2-吡咯烷基)乙基]-4-丙氧基苯磺酰胺,乌地那非 |
PDE | Metabolism |
Udenafil 是一种选择性的,有效的,具有口服活性的 5 型磷酸二酯酶 (PDE5) 抑制剂。它能够抑制 cGMP 水解,可用于研究勃起功能障碍的。 | |||
T6702 |
Terbinafine
Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067 |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Terbinafine (TDT 067) 是念珠菌属的角鲨烯环氧化酶有效的非竞争性抑制剂,Ki 值为 30 nM。它具有抗真菌感染活性。 | |||
T1411 |
Terbinafine hydrochloride
KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。 | |||
TN3880 |
Dodonaflavonol
|
Others | Others |
Dodonaflavonol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3880,CAS号为 1392213-93-2。 | |||
TN5494 |
2'',3''-Dihydroochnaflavone
|
||
2'',3''-Dihydroochnaflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5494,CAS号为 340997-02-6。 | |||
TN5501 |
Ochnaflavone
|
||
Ochnaflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5501,CAS号为 50276-96-5。 | |||
TN1283 |
4'-O-Methylochnaflavone
|
Others | Others |
4'-O-Methylochnaflavone is a natural product | |||
T5156 |
2,3,2'',3''-Tetrahydroochnaflavone
金银花 |
Others | Others |
2,3,2'',3''-Tetrahydroochnaflavone是一种天然产物,属于忍冬科忍冬属,其产品编号为 T5156,CAS号为 678138-59-5。2,3,2'',3''-Tetrahydroochnaflavone可用作对照参考。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-04726 |
IL-8/CXCL8 Protein, Human, Recombinant (His)
Interleukin-8,GCP1,MONAP,LECT,LYNAP,NAF,GCP-1,LUCT,... |
Human | P. pastoris (Yeast) |
IL-8/CXCL8 Protein, Human, Recombinant (His) is expressed in yeast with His tag. The predicted molecular weight is 9.8 kDa and the accession number is A0A024RDA5. | |||
TMPY-00472 |
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99)
NAF,GCP1,NAP1,chemokine (C-X-C motif) ligand 8,Inte... |
Human | E. coli |
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99) is expressed in E. coli expression system. The predicted molecular weight is 8.5 kDa and the accession number is A0A024RDA5. | |||
TMPY-00754 |
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99)
MONAP,MDNCF,NAP-1,白介素,NAP1,LUCT,chemokine (C-X-C motif) liga... |
Human | HEK293 Cells |
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99) is expressed in HEK293 mammalian cells. The predicted molecular weight is 8 kDa and the accession number is A0A024RDA5. | |||
TMPK-00480 |
IL-8/CXCL8 Protein, Cynomolgus, Recombinant (His)
GCP/IL-8 protein IV,MDNCF,CXCL8,GCP-1,LUCT,NAF,IL-8... |
Cynomolgus | HEK293 Cells |
Interleukin-8 (IL-8) has been revealed as a critical regulator of CNS function and development with participation in many CNS disorders including gliomas.Several promising approaches that target directly or indirectly IL-8 effects in gliomas are currently in progress while more-in-depth studies are needed to validate its biomarker role and elucidate the underlying molecular mechanisms. | |||
TMPY-00755 |
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99, hFc)
chemokine (C-X-C motif) ligand 8,Interleukin-8,LYNAP,NAP1, |
Human | HEK293 Cells |
IL-8/CXCL8 Protein, Human, Recombinant (aa 28-99, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 35 kDa and the accession number is A0A024RDA5. | |||
TMPY-00753 |
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99, hFc)
LECT,MONAP,IL-8,LYNAP,白细胞介素,chemokine (C-X-C motif) ligand 8... |
Human | HEK293 Cells |
IL-8/CXCL8 Protein, Human, Recombinant (aa 23-99, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 35.6 kDa and the accession number is A0A024RDA5. |