Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Lodenafil (Hydroxyhomosildenafil) 是一种有效的磷酸二酯酶 5 型(PDE5)抑制剂,可用于勃起功能障碍的研究。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 397 | 现货 | ||
2 mg | ¥ 595 | 现货 | ||
5 mg | ¥ 996 | 现货 | ||
10 mg | ¥ 1,580 | 现货 | ||
25 mg | ¥ 2,690 | 现货 | ||
50 mg | ¥ 3,960 | 现货 | ||
100 mg | ¥ 5,650 | 现货 | ||
1 mL * 10 mM (in DMSO) | ¥ 1,150 | 现货 |
产品描述 | Lodenafil (Hydroxyhomosildenafil) is a potent PDE5 inhibitor, with treatment of erectile dysfunction (ED) |
体内活性 | Investigated right ventricular hypertrophy (RVH) and IL-1 levels in lung fragments. The number of cases of RVH was significantly higher in the monocrotaline group than in the lodenafil and control groups, as were mPAP and IL-1 levels. Lodenafil can prevent monocrotaline-induced PH, RVH, and inflammation[1]. |
动物实验 | Thirty male Sprague-Dawley rats were randomly divided into three groups: control; monocrotaline (experimental model); and lodenafil (experimental model followed by lodenafil treatment, 5 mg/kg daily for 28 days) Mean pulmonary artery pressure (mPAP) was obtained by right heart catheterization[1]. |
别名 | Hydroxyhomosildenafil, 羟基豪莫西地那非 |
分子量 | 504.6 |
分子式 | C23H32N6O5S |
CAS No. | 139755-85-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (495.44 mM)
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 1.9818 mL | 9.9088 mL | 19.8177 mL | 49.5442 mL |
5 mM | 0.3964 mL | 1.9818 mL | 3.9635 mL | 9.9088 mL | |
10 mM | 0.1982 mL | 0.9909 mL | 1.9818 mL | 4.9544 mL | |
20 mM | 0.0991 mL | 0.4954 mL | 0.9909 mL | 2.4772 mL | |
50 mM | 0.0396 mL | 0.1982 mL | 0.3964 mL | 0.9909 mL | |
100 mM | 0.0198 mL | 0.0991 mL | 0.1982 mL | 0.4954 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Lodenafil 139755-85-4 Metabolism PDE inhibit Hydroxyhomosildenafil Phosphodiesterase (PDE) 羟基豪莫西地那非 Inhibitor inhibitor