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117

抑制剂 & 化合物

14

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Cat. No. Product Name Target Signaling Pathways
T19840 GSK-F1

PI4KA inhibitor-F1

PI4K PI3K/Akt/mTOR signaling
GSK-F1 (PI4KA inhibitor-F1) 是一种新型强效 PI4KA 抑制剂。
T67837 (3S)-GSK-F1

PI4KA inhibitor-F1

PI4K PI3K/Akt/mTOR signaling
(3S)-GSK-F1是一种选择性PI4KIIIα抑制剂,pIC50=8.3。
T83670 F1 TFA

Tat-IKIP (46-60),Tat-Inhibitor of NF-κB Kinase-interacting Peptide

F1是一种抗炎肽,由HIV-1 Tat蛋白质转导域与对应于抑制因子NF-κB激酶-相互作用肽(IKIP)46-60残基的15氨基酸肽链接而成。在5 µM浓度下,F1抑制了小鼠腹腔巨噬细胞中LPS诱导的IκB激酶α(IKKα)和IKKβ的磷酸化以及NF-κB(p65)的核内转移。在体内,F1(5 mg/kg)降低了LPS诱导的脓毒症小鼠模型中IL-6、TNF-α和IL-1β的血清水平,并增加了生存率。
T126048 Coreanoside F1

Coreanoside F1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126048,CAS号为 132282-69-0。
T125155 Schidigerasaponin F1

Schidigerasaponin F1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125155,CAS号为 266998-42-9。
TP2476 Tnrnflrfamide

Thr-asn-arg-asn-phe-leu-arg-phe-NH2,Peptide F(1), lobster,F1 Peptide, lobster,Lobster peptide F1

Tnrnflrfamide is a SCP (small cardioactive peptide)-like peptide found in lobster neurons; exhibits FMRFamide-like immunoreactivity.
T11254 F-1

ROS; ALK; ROS Kinase Angiogenesis; Immunology/Inflammation; Tyrosine Kinase/Adaptors
F-1 是 ALK 和 ROS1 的双重抑制剂,抑制 ALK 的磷酸化及下游通路,可作用于对 ALKWT (IC50:2.1 nM),ROS1WT (IC50:2.3 nM),ALKL1196M (IC50:1.3 nM) 和 ALKG1202R (IC50:3.9 nM)。
T37919 Prostaglandin F1α

PGF1α,Prostaglandin F1α

Prostaglandin F1α (PGF1α) is the putative metabolite of dihomo-γ-linolenic acid (DGLA) via the cyclooxygenase (COX) pathway. Both PGF1α and PGF2α have been shown to act as priming pheromones for male Atlantic salmon with a threshold concentration of 10-11 M. [1] PGF1α binds to the ovine corpus luteum FP receptor at only 8% of the relative potency of PGF2α. [2] It is only half as active as PGF2α in inducing human respiratory smooth muscle contractions in vitro. [3]
T36162 8-iso Prostaglandin F1α

8-iso Prostaglandin F1α

8-iso PGF1α is an isoprostane that was first identified in human semen. It is a member of the isoprostane family, which are eicosanoids of non-cyclooxygenase origin. 8-iso PGF1α is present along with its 19-hydroxy congener at 5-10 μg/ml of seminal plasma.
T36163 8-iso Prostaglandin F1β

8-iso Prostaglandin F1β

8-iso PGF1β is a potential autoxidation product of DGLA. There are no published reports on its isolation from any biological source or on its biological activity.
T36772 11-deoxy Prostaglandin F1β

11-deoxy Prostaglandin F1β

11-deoxy PGF1β is a synthetic analog of PGF1β. In contrast to PGF2α and PGF1α, 11-deoxy PGF1β exhibits vasodepressor and bronchodilator activities in guinea pigs at a dose of 500 μg/kg.
T37990 15-keto Prostaglandin F1α

15-keto Prostaglandin F1α

15-keto PGF1α is the initial metabolite of PGF1α via 15-hydroxy PGDH. In mammals, oxidation of C-15 markedly attenuates receptor binding and activity. In fish, the 15-keto compounds serve as post-ovulatory pheromones and are more active than the parent prostaglandins.
T36771 11-deoxy Prostaglandin F1α

11-deoxy Prostaglandin F1α

11-deoxy PGF1α is a synthetic analog of PGF1α. In whole animal studies, a dose of 32 mg/kg inhibited gastric acid secretion by 35%. 11-deoxy PGF1α is also known to cause rat uterine contractions at a dose 0.3 times that of PGF1α. It also exhibits vasopressor and bronchoconstrictor activities at about half the potency of PGF2α in guinea pigs.
T36148 13,14-dihydro-15-keto Prostaglandin F1α

13,14-dihydro-15-keto Prostaglandin F1α

13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach. The measurement of 13,14-dihydro-15-keto PGF1α can be used as a marker of the in vivo production of PGF1α.
T36724 6,15-diketo-13,14-dihydro Prostaglandin F1α

6,15-diketo-13,14-dihydro Prostaglandin F1α

6,15-diketo-13,14-dihydro PGF1α is a metabolite of PGI2. It was shown to enhance intracellular cAMP and cholesterol catabolism in bovine arterial smooth muscle cells.
T83662 2,3-dinor-8-iso Prostaglandin F1α

2,3-dinor-8-iso PGF1α,2,3-dinor-iPF1α-III,2,3-dinor-5,6-dihydro-15-F2t-Isoprostane,2,3-dinor-5,6-dihydro-15-F2t-IsoP

2,3-dinor-8-iso Prostaglandin F1α(2,3-dinor-8-iso PGF1α)是一种异前列腺素和花生四烯酸的活性代谢物,也是血小板聚集抑制剂8-iso PGF2α的产物。它通过花生四烯酸的非酶促自由基过氧化作用形成。2,3-dinor-8-iso PGF1α在孤立的猪视网膜和大脑微血管中引起血管收缩(EC50s分别为12.8和18.5 nM),但在31 µM的浓度下使用时不会引起孤立的大鼠主动脉环的收缩。在1 µM的浓度下使用时,它能增加孤立的猪大脑切片中的血栓素B2(TXB2)水平,这一效应可以通过血栓素A合成酶抑制剂CGS 12970、电压门控钙通道抑制剂SKF 96365或烟碱型乙酰胆碱受体(nAChR)拮抗剂α-conotoxin来逆转。
T13194 CSF1R-IN-2

c-Fms; c-Met/HGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
CSF1R-IN-2 是一种口服具有活力的、有效的 SRC,MET 和 c-FMS 抑制剂,它们的 IC50 值分别为 0.12 nM,0.14 nM 和 0.76 nM。
T77745 N6F11

GPX oxidation-reduction
N6F11是一种新型且具有选择性和有效性的铁死亡诱导剂,具有抗癌抗肿瘤活性,通过与癌细胞中的TRIM25结合从而促进GPX4降解。N6F11 可用于研究胰腺癌。
T10894 CSF1R-IN-1

c-Fms Tyrosine Kinase/Adaptors
CSF1R-IN-1 是一种 CSF1R 抑制剂 (IC50:0.5 nM)。
T64066 CSF1R-IN-3

c-Fms; CSF-1R Tyrosine Kinase/Adaptors
CSF1R-IN-3是一种口服有效的 CSF-1R 抑制剂,IC50值为2.1nM。CSF1R-IN-3对结直肠癌细胞具有抗增殖活性。CSF1R-IN-3 通过抑制巨噬细胞的迁移,诱导 M2 型巨噬细胞重新编程为 M1 型巨噬细胞,从而表现出抗肿瘤作用和提高免疫力的作用,展现对结直肠癌细胞的活性。
T13324 VUF11207 fumarate

CXCR; Arrestin Autophagy; GPCR/G Protein; Immunology/Inflammation
VUF11207 fumarate 是一种 CXCR7激动剂和高效CXCR7配体,pKi 为 8.1。它可诱导CXCR7的β-arrestin2募集和随后的内在化,pEC50分别为 8.8 和 7.9。
T77767L1 GLF16 HCl

Others Others
GLF16 HCl 是一种荧光团偶联的苏丹黑 B 类似物,可通过通过荧光显微镜和流式细胞术快速检测、分离和实时跟踪衰老细胞。
T61112 SLF1081851

LPL Receptor GPCR/G Protein
SLF1081851 是一种 Spns2 抑制剂,抑制 S1P 释放 (IC50=1.93 μM)。SLF1081851 在发育和免疫系统中起关键作用。
T6667 SF1670

PTP CD45 Inhibitor,PTPase CD45 Inhibitor

Phosphatase; PTEN; Autophagy Autophagy; Metabolism; PI3K/Akt/mTOR signaling
SF1670 (PTPase CD45 Inhibitor) 是一种特异性 PTEN 抑制剂,IC50 为 2 μM。
T15266 F16

(E)-4-(3-indolylvinyl)-N-methylpyridinium iodide

Others Others
F16 ((E)-4-(3-indolylvinyl)-N-methylpyridinium iodide)抑制neu-overeigning 细胞的生长和乳腺上皮的增殖。
T60026 KIF18A-IN-2

Microtubule Associated Cytoskeletal Signaling
KIF18A-IN-2 是有丝分裂驱动蛋白 Kif18A 的抑制剂,IC50 为 28 nM,可用于染色体不稳定性相关漏洞的研究。
T4308 F1063-0967

Phosphatase Metabolism
F1063-0967 是双特异性磷酸酶 26 抑制剂,其IC50=11.62 μM。
T16904 Smurf1-IN-A01

A01

Others Others
Smurf1-IN-A01 (A01) 是泛素连接酶 Smad 泛素化调节因子-1(Smurf1)抑制剂,其kd=3.664 nM。它能够抑制 Smurf1 介导的 Smad1/5 降解,并提高 BMP-2 的反应性。
T22774L eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA)

Others Others
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA) 是延伸因子 1 亚基。真核翻译延伸因子 1 alpha 1 (EEF1A1) 编码延伸因子 alpha 亚基的同种型- 1 复合物,负责将氨酰 tRNA 酶促递送至核糖体。这种亚型(α 1)在脑、胎盘、肺、肝、肾和胰腺中表达,另一种亚型(α 2)在脑、心脏和骨骼肌中表达。这种亚型在 66% 的 Felty 综合征患者中被鉴定为自身抗原。已发现该基因在许多染色体上具有多个拷贝,其中一些(如果不是全部)代表不同的假基因。
T12125 MuRF1-IN-1

Others Others
MuRF1-IN-1 是MuRF1抑制剂,能减少心脏恶病质中的骨骼肌萎缩和功能障碍。
T15409 GNF179

Parasite Microbiology/Virology
GNF179 是8,8-二甲基 IP 类似物。 它表现出对多药耐药菌株 W2 的效力,具有良好的体外代谢稳定性和体内口服生物相容性。
T9890 HIF1-IN-3 

Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-

HIF Angiogenesis; Chromatin/Epigenetic
HIF1-IN-3 (Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-) 是HIF-1的有效抑制剂(EC50 = 0.9 μM),可用于抗癌的研究。
T4125 HSF1A

HSP Cytoskeletal Signaling; Metabolism
HSF1A 是一种可渗透细胞的 HSF1 激活剂,可保护哺乳动物细胞免受应激诱导的细胞凋亡。它还是 TRiC/CCT 的特异性抑制剂。
T3963 VUF10460

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
VUF10460 是一种非咪唑组胺 H4 受体激动剂,与大鼠H4受体结合的pKi 值为7.46。
T24949 VUF10132

VUF-10132,VUF 10132

VUF10132 is a full inverse CXCR3 N3.35A agonist.
T40232 KIF18A-IN-1

KIF18A-IN-1

KIF18A-IN-1 is a potent inhibitor of the mitotic kinesin KIF18A. This compound demonstrates significant anti-tumor properties.
T26785 BFF122

BFF 122,BF5,BFF-122

BFF122 is an inhibitor of kynurenine aminotransferase II (KAT II).
T70872 Smurf1 inhibitor 1

Smurf1 inhibitor 1 is a inhibitor that promotes bone formation.
T62318 CSF1R-IN-9

CSF1R-IN-9 (Compound 46) 是一种 CSF-1R 抑制剂 (IC50: 0.028 μM)。
T74271 TRIM24/BRPF1-IN-2

TRIM24/BRPF1-IN-2 (compound 20l) 是一种有效的 TRIM24/BRPF1双重抑制剂,IC50值分别为 0.98 和 1.16 μM。 TRIM24/BRPF1-IN-2 显示出 TRIM24/BRPF1 溴结构域结合亲和力。 TRIM24/BRPF1-IN-2 可用于前列腺癌研究。
TP1268 CEF19, Epstein-Barr Virus latent NA-3A (458-466)

CEF19,Epstein-Barr Virus latent NA-3A 458-466

CEF19, Epstein-Barr Virus latent NA-3A (458-466) is a single peptide epitope, YPLHEQHGM, representing residues 458-466 of the type 1 Epstein-Barr Virus (EBV) nuclear antigen 3A protein (B95.8 strain).
T15661 Kif15-IN-1

Others Others
Kif15-IN-1, a mitotic Kinesin family member 15 (Kif15) inhibitor, is utilized in the study of cellular proliferative diseases.
TP2402 Peptide VF13N

Epitope VF13N

Peptide VF13N is a synthetic rabies virus glycoprotein T helper cell epitope.
T77932 PF15 TFA

PROTACs PROTAC
PF15 TFA是一种连接FLT3 kinase配体和CRBN配体的PROTAC,作为FLT3-ITD的高选择性降解剂,DC50值为76.7 nM。该化合物可显著抑制FLT3-ITD阳性细胞增殖,并降低FLT3和STAT5磷酸化水平。PF15 TFA亦能抑制小鼠模型的肿瘤生长,并可用于白血病研究。
T70403 VUF14480

VUF14480 is a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor. VUF14480 was shown to be a partial agonist of hH4 receptor-mediated G protein signalling and β-arrestin2 recruitment. VUF14480 bound covalently to the hH₄ receptor with submicromolar affinity. Serine substitution of C98(3.36) prevented this covalent interaction.
T62364 CSF1R-IN-5

CSF1R-IN-5 是一种 CSF1R 的有效抑制剂。其中 CSF-1R 表达于巨噬细胞中,巨噬细胞的存活和分化依赖于 CSF-1/CSF-1R 信号通路。CSF1R-IN-5 可以影响 TAM 和胶质瘤细胞之间炎症因子的交换。CSF1R-IN-5 具有潜力进行癌症疾病的研究。
T74336 YF135

YF135为一种效能高的KRASG12CPROTAC,能可逆地促使共价结合。该化合物采用KRAS G12C inhibitor 48(compound 6d)作为配体,并以MRTX849搭配VHL配体作为框架进行设计与合成。通过E3连接酶VHL介导的蛋白酶体途径,YF135显著诱导KRASG12C的降解并可逆地降低ERK磷酸化水平。
T28790 SKF1

SKF1 is a suppressor of the ability of FK506. SKF1 inhibits cell growth in the presence of high levels of NaCl, induces cell death in low salt conditions, interacts directly with yeast mitochodria.
T76245L CKLF1-C27 TFA

CKLF1-C27 是 CKLF1 的 C 末端肽,与 CCR4受体结合并激活 ERK1/2通路。CKLF1-C27 可以通过竞争 CCR4受体来消除 CKLF1 对细胞的影响。CKLF1-C27对促进 HUVECs 增殖有很大的作用。CKLF1-C27 具有用于银屑病研究的潜力。
T61554 CSF1R-IN-13

CSF1R-IN-13 is a powerful CSF1R inhibitor with potential applications in researching cancer diseases [1]. CSF1R, also known as colony stimulating factor 1 receptor, is a critical growth factor that regulates various cell types, including bone marrow progenitor cells, monocytes, macrophages, and giants [1]. CSF1R-IN-13 shows promise in furthering our understanding of cancer-related disorders (WO2019134661A1, compound 32) [1].

化合物

GSK-F1
Cat.No: T19840
Synonym: PI4KA inhibitor-F1
Target: PI4K
(3S)-GSK-F1
Cat.No: T67837
Synonym: PI4KA inhibitor-F1
Target: PI4K
F1 TFA
Cat.No: T83670
Synonym: Tat-IKIP (46-60),Tat-Inhibitor of NF-κB Kinase-interacting Peptide
Target:
Coreanoside F1
Cat.No: T126048
Synonym:
Target:
Schidigerasaponin F1
Cat.No: T125155
Synonym:
Target:
Tnrnflrfamide
Cat.No: TP2476
Synonym: Thr-asn-arg-asn-phe-leu-arg-phe-NH2,Peptide F(1), lobster,F1 Peptide, lobster,Lobster peptide F1
Target:
F-1
Cat.No: T11254
Synonym:
Target: ROS, ALK, ROS Kinase
Prostaglandin F1α
Cat.No: T37919
Synonym: PGF1α,Prostaglandin F1α
Target:
8-iso Prostaglandin F1α
Cat.No: T36162
Synonym: 8-iso Prostaglandin F1α
Target:
8-iso Prostaglandin F1β
Cat.No: T36163
Synonym: 8-iso Prostaglandin F1β
Target:
11-deoxy Prostaglandin F1β
Cat.No: T36772
Synonym: 11-deoxy Prostaglandin F1β
Target:
15-keto Prostaglandin F1α
Cat.No: T37990
Synonym: 15-keto Prostaglandin F1α
Target:
11-deoxy Prostaglandin F1α
Cat.No: T36771
Synonym: 11-deoxy Prostaglandin F1α
Target:
13,14-dihydro-15-keto Prostaglandin F1α
Cat.No: T36148
Synonym: 13,14-dihydro-15-keto Prostaglandin F1α
Target:
6,15-diketo-13,14-dihydro Prostaglandin F1α
Cat.No: T36724
Synonym: 6,15-diketo-13,14-dihydro Prostaglandin F1α
Target:
2,3-dinor-8-iso Prostaglandin F1α
Cat.No: T83662
Synonym: 2,3-dinor-8-iso PGF1α,2,3-dinor-iPF1α-III,2,3-dinor-5,6-dihydro-15-F2t-Isoprostane,2,3-dinor-5,6-dihydro-15-F2t-IsoP
Target:
CSF1R-IN-2
Cat.No: T13194
Synonym:
Target: c-Fms, c-Met/HGFR, Src
N6F11
Cat.No: T77745
Synonym:
Target: GPX
CSF1R-IN-1
Cat.No: T10894
Synonym:
Target: c-Fms
CSF1R-IN-3
Cat.No: T64066
Synonym:
Target: c-Fms, CSF-1R
VUF11207 fumarate
Cat.No: T13324
Synonym:
Target: CXCR, Arrestin
GLF16 HCl
Cat.No: T77767L1
Synonym:
Target: Others
SLF1081851
Cat.No: T61112
Synonym:
Target: LPL Receptor
SF1670
Cat.No: T6667
Synonym: PTP CD45 Inhibitor,PTPase CD45 Inhibitor
Target: Phosphatase, PTEN, Autophagy
F16
Cat.No: T15266
Synonym: (E)-4-(3-indolylvinyl)-N-methylpyridinium iodide
Target: Others
KIF18A-IN-2
Cat.No: T60026
Synonym:
Target: Microtubule Associated
F1063-0967
Cat.No: T4308
Synonym:
Target: Phosphatase
Smurf1-IN-A01
Cat.No: T16904
Synonym: A01
Target: Others
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA)
Cat.No: T22774L
Synonym:
Target: Others
MuRF1-IN-1
Cat.No: T12125
Synonym:
Target: Others
GNF179
Cat.No: T15409
Synonym:
Target: Parasite
HIF1-IN-3 
Cat.No: T9890
Synonym: Benzenepropanamide, N-[(8-hydroxy-7-quinolinyl)(4-methoxyphenyl)methyl]-
Target: HIF
HSF1A
Cat.No: T4125
Synonym:
Target: HSP
VUF10460
Cat.No: T3963
Synonym:
Target: Histamine Receptor
VUF10132
Cat.No: T24949
Synonym: VUF-10132,VUF 10132
Target:
KIF18A-IN-1
Cat.No: T40232
Synonym: KIF18A-IN-1
Target:
BFF122
Cat.No: T26785
Synonym: BFF 122,BF5,BFF-122
Target:
Smurf1 inhibitor 1
Cat.No: T70872
Synonym:
Target:
CSF1R-IN-9
Cat.No: T62318
Synonym:
Target:
TRIM24/BRPF1-IN-2
Cat.No: T74271
Synonym:
Target:
CEF19, Epstein-Barr Virus latent NA-3A (458-466)
Cat.No: TP1268
Synonym: CEF19,Epstein-Barr Virus latent NA-3A 458-466
Target:
Kif15-IN-1
Cat.No: T15661
Synonym:
Target: Others
Peptide VF13N
Cat.No: TP2402
Synonym: Epitope VF13N
Target:
PF15 TFA
Cat.No: T77932
Synonym:
Target: PROTACs
VUF14480
Cat.No: T70403
Synonym:
Target:
CSF1R-IN-5
Cat.No: T62364
Synonym:
Target:
YF135
Cat.No: T74336
Synonym:
Target:
SKF1
Cat.No: T28790
Synonym:
Target:
CKLF1-C27 TFA
Cat.No: T76245L
Synonym:
Target:
CSF1R-IN-13
Cat.No: T61554
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3401 Ginsenoside F1

人参皂苷 F1,20(S)-Ginsenoside F1

P450; Endogenous Metabolite Metabolism
Ginsenoside F1 (20(S)-Ginsenoside F1) 是一种 Ginsenoside Rg1 的酶促修饰衍生物,它竞争性抑制CYP3A4,对 CYP2D6 具有较弱的抑制作用。
TN1942 Momordicoside F1

苦瓜皂苷 F1

Others Others
Momordicoside F1 may have antiproliferative activities against MCF-7, WiDr, HEp-2, and Doay human tumor cell lines.
TN1989 Niga-ichigoside F1

苦莓苷F1

Others; Nrf2 Immunology/Inflammation; Others
Niga-ichigoside F1(NI) has anti-inflammatory, gastroprotective ,antinociceptive, and cytotoxic effects.
TN4161 Goshonoside F1

Goshonoside F1是半糯米品种水稻的脂质代谢产物,可被当作培育优良水稻的一个指标。
TN1080 Kaji-ichigoside F1

蔷薇苷

Kaji-ichigoside F1 shows antiinflammatory/antinociceptive action in acetic acid-induced writhing and hot plate testing and in a carrageenan-induced paw edema model in mice and rats. Kaji-ichigoside F1 exhibits in vivo hepatoprotective effects, it inhibite
TN6448 3-Acetyl-ginsenoside F1

3-Acetyl-ginsenoside F1 可用于生命科学领域的相关研究,其产品编号为 TN6448。
T81853 Marstenacisside F1

Marstenacisside F1(化合物1)为从通关藤(Marsdenia tenacissima)分离的抗炎聚氧孕烷苷,能抑制脂多糖激活的RAW 264.7细胞产生一氧化氮(NO),属Tenacigenin B衍生物。
TN2242 Suavissimoside R1

甜叶苷R1,Suavissimoside F1

Others Others
Suavissimoside F1 is a natural product
T3920 Pseudoginsenoside F11

Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11

Others; Endogenous Metabolite Metabolism; Others
Pseudoginsenoside F11 (Ginsenoside A1) 从人参根和叶中分离得到。PF11在一系列心血管和中枢神经系统疾病中具有广泛的保护作用。
TN4049 F1839-I

Others Others
F1839-I is a natural product from Stachybotrys sp.
T19328 Fructo-oligosaccharide DP11/GF10

Others Others
Fructo-oligosaccharide DP11/GF10 is a fructooligosaccharide (FOS) compound with a degree of polymerization (DP) equal to 11. FOS consists of 10 fructose units connected by (2→1)-β-glycosidic bonds, with a single D-glucosyl unit present at the non-reducing end.
T19329 Fructo-oligosaccharide DP12/GF11

蔗果十二糖

Others Others
Fructo-oligosaccharide DP12/GF11 is a member of fructooligosaccharides (FOS) characterized by a degree of polymerization (DP) of 12. FOS compounds consist of 11 fructose units connected by (2→1)-β-glycosidic bonds, with a lone D-glucosyl unit located at the non-reducing end.
T3S0153 Xanthatin

苍耳亭,叶黄制菌素

Apoptosis; VEGFR; Lipoxygenase; Wnt/beta-catenin; Antibacterial Angiogenesis; Apoptosis; Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Stem Cells; Tyrosine Kinase/Adaptors
Xanthatin 是一种从Xanthium strumarium 叶子中提取的天然产物,可诱导细胞凋亡。它抑制布鲁氏菌的IC50值为 2.63 μg/ mL,对寄生虫特异性锥虫硫磷还原酶具有不可逆的弱抑制作用。它通过抑制PGE2的合成和 5-脂氧合酶的活性而显示出抗炎活性。
T13123 Tentoxin

Endogenous Metabolite Metabolism
Tentoxin 是一种由植物致病真菌产生的环状肽,在敏感植物中,当其浓度在纳摩尔到微摩尔之间时,会使 F1马达失活,而更高的浓度会超过该酶的天然活性

天然产物

Ginsenoside F1
Cat.No: T3401
Synonym: 人参皂苷 F1,20(S)-Ginsenoside F1
Target: P450, Endogenous Metabolite
Momordicoside F1
Cat.No: TN1942
Synonym: 苦瓜皂苷 F1
Target: Others
Niga-ichigoside F1
Cat.No: TN1989
Synonym: 苦莓苷F1
Target: Others, Nrf2
Goshonoside F1
Cat.No: TN4161
Synonym:
Target:
Kaji-ichigoside F1
Cat.No: TN1080
Synonym: 蔷薇苷
Target:
3-Acetyl-ginsenoside F1
Cat.No: TN6448
Synonym:
Target:
Marstenacisside F1
Cat.No: T81853
Synonym:
Target:
Suavissimoside R1
Cat.No: TN2242
Synonym: 甜叶苷R1,Suavissimoside F1
Target: Others
Pseudoginsenoside F11
Cat.No: T3920
Synonym: Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11
Target: Others, Endogenous Metabolite
F1839-I
Cat.No: TN4049
Synonym:
Target: Others
Fructo-oligosaccharide DP11/GF10
Cat.No: T19328
Synonym:
Target: Others
Fructo-oligosaccharide DP12/GF11
Cat.No: T19329
Synonym: 蔗果十二糖
Target: Others
Xanthatin
Cat.No: T3S0153
Synonym: 苍耳亭,叶黄制菌素
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
Tentoxin
Cat.No: T13123
Synonym:
Target: Endogenous Metabolite
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