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86

抑制剂 & 化合物

58

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T67842	ERG240 EGR240	Others	Others
	ERG240 是支链氨基酸转氨酶 1 (BCAT1) 抑制剂。ERG240 有潜力用于癌症、类风湿性关节炎和骨病相关研究。
T60051	VPC-18005	Others	Others
	VPC-18005 是一种荧光素酶抑制剂。 VPC-18005 抑制 ERG 诱导的转录并直接与 ERG-ETS 结构域相互作用，从而破坏 ERG 与 DNA 的结合。
T7145	ERGi-USU 1-(2-噻唑基偶氮)-2-萘酚	Others	Others
	NSC-139021 (ERGi-USU) 是一种具有高度选择性的ERG 阳性癌细胞生长抑制剂，抑制不同细胞系的IC50值为 30-400 nM。
T11043	Dihydroergocristine mesylate 甲磺酸双氢麦角汀,DHEC (mesylate)	Beta Amyloid	Neuroscience
	Dihydroergocristine mesylate (DHEC (mesylate)) 是一种 γ-secretase (GSI) 的抑制剂，能够阿尔茨海默氏病淀粉样蛋白 β 肽 (amyloid-β) 的产生，与 γ-secretase 和 Nicastrin 结合的平衡解离常数 (Kd) 值分别为 25.7 nM 和 9.8 μM。
T28757	Sergliflozin etabonate GW-869682,GW-869682X,KGT-1251,GW869682X,GW869682,KGT1251	SGLT	GPCR/G Protein
	Sergliflozin etabonate (KGT-1251) 是一种 SGLT-2 抑制剂，可用于 2 型糖尿病和肥胖症的研究。
T9174	Icerguastat Sephin 1,lcerguastat,IFB-088	Phosphatase	Metabolism
	Icerguastat (IFB-088) 是一种缺乏 α2-肾上腺素能活性的 Guanabenz 衍生物，是一种磷酸酶调节亚单位 PPP1R15A (R15A)的选择性抑制剂。它能够抑制 eIF2α 去磷酸化，从而延长保护反应。它具有抗朊病毒作用。
T9793	Methyl Ergoline Acid	Others	Others
	Methyl Ergoline Acid 是一种麦角碱衍生物，可用作趋化因子受体配体。
T2226	Pergolide mesylate 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Pergolide mesylate salt(LY127809) 是一种有效的，具有口服活性的多巴胺 D1和 D2受体激动剂，是一种 Ergoline 衍生物，可用于帕金森氏病和高泌乳素血症的研究。
T68174	Sergliflozin A	SGLT	GPCR/G Protein
	Sergliflozin A 是一种选择型SGLT2抑制剂，以剂量依赖性方式诱导糖尿。可降低高血糖。
T1132	Nicergoline 尼麦角林,Nicergolinum,Nimergoline	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Nicergoline (Nicergolinum) 是一种有效的，选择性的、具有口服活性的α1A-肾上腺素能受体拮抗剂，是一种溴烟碱酸的麦角林衍生物。它具有血管舒张作用，可以改善阿尔茨海默症小鼠的认知功能。
T4008	Metergoline 甲麦角林,Methergoline,Liserdol	Dopamine Receptor; 5-HT Receptor; Sodium Channel	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Metergoline (Methergoline) 是多巴胺激动剂和血清素拮抗剂。它是 h5-HT7受体的高亲和力配体，Ki 为 16 nM。它还是可逆神经 Na+通道抑制剂，用于研究季节性情绪障碍、催乳激素调节。
T71707L	Romergoline 2HCl Romergoline 2HCl(107052-56-2 Free base),FCE 23884 2HCl	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Romergoline 2HCl 是一种 D1 激动剂和 D2 拮抗剂，可用于研究帕金森病。
T61062	ERGi-USU-6 mesylate
	ERGi-USU-6 (mesylate) 是一种新型选择性的 ERG 阳性前列腺癌，IC50 值为 0.089 μM，它是一种 ERGi-USU-6 盐衍生物。
T82447	Ergtoxin-1 ErgTx1
	Ergtoxin-1为钾离子通道阻断剂，源于墨西哥毒蝎Centruroides noxius的毒液。该化合物具有阻断神经、心脏及内分泌细胞ERG-K+通道的功能。
T63825	Antiallergic agent-1
	Antiallergic agent-1 是 Src 家族激酶抑制剂，是一种新的有价值的先导化合物，具有作为抗过敏剂的潜力。
T33045	Lysergine
	Lysergine is a bioactive chemical.
T82424	Experimental allergic encephalitogenic peptide (human)
	Experimental allergic encephalitogenic peptide (human) 为EAE多肽类化合物，能够诱导豚鼠发生脑脊髓炎。
T78239	Mergetpa	Carboxypeptidase	Proteases/Proteasome
	Mergetpa作为一种羧肽酶抑制剂，其功能是阻碍激肽及B2受体拮抗剂转变成无c末端精氨酸的代谢物。
T21423	Methysergide maleate Deseril, Sansert,UML 491,UML491,Methysergide,UML-491
	Methysergide is used for prophylaxis of migraine headaches/cluster headaches but is no longer recommended due to retropulmonary/retroperitoneal fibrosis. It may also be used in the treatment of serotonin syndrome. It is also used in carcinoid syndrome to
T37858	Dehydroergosterol 9,11-dehydro Ergosterol,DHE
	Dehydroergosterol is a naturally occurring, fluorescent analog of cholesterol (ex/em = 324/375 nm) that mimics the properties of cholesterol in cell membranes.[1] It is readily bound by cholesterol-binding proteins and has been used for real-time probing of the sterol environment and to elucidate intracellular sterol trafficking in living organisms.[1]
T125721	3beta-Hydroxyergost-5-en-7-one
	3beta-Hydroxyergost-5-en-7-one 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T125721。
T69337	(R)-3,4-Dimethoxydalbergione
	(R)-3,4-Dimethoxydalbergione is a novel covalent inhibitor of ca
T65361	ZWITTERGENT 3-16 Detergent
	ZWITTERGENT 3-16 Detergent 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65361，CAS号为 2281-11-0。
T68010	proterguride
	proterguride 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T68010，CAS号为 77650-95-4。
TF0004	Anzergent 3-18
	Anzergent 3-18 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 TF0004，CAS号为 13177-41-8。
T24003	Disulergine CM 29717,CH 29717,CH 29-717
	Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.
T71213	Amesergide
	Amesergide is a serotonin antagonist.
T131544	Bergenin (Vakerin; Peltophorin; Cuscutin)
	Bergenin (Vakerin; Peltophorin; Cuscutin) 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131544。
T65355	Zwittergent 3-12 Detergent
	Zwittergent 3-12 Detergent 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65355，CAS号为 14933-08-5。
T76944	Cergutuzumab amunaleukin
	Cergutuzumab amunaleukin (CEA-IL2v) 是一种靶向癌胚抗原 (CEA) 的IL-2变体，作为免疫细胞因子，展现出免疫刺激与抗肿瘤活性。
T31469	Dihydroergostin DE145,DE-145,DE 145
	Dihydroergostin is a ergot alkaloid that exhibits potential neuroprotective properties.
T69065	Tiomergine
	Tiomergine is a dopamine receptor agonist.
T68551	Cabergoline diphosphate
	Cabergoline diphosphate is a dopamine D2 receptor agonist used for prolactinoma treatment. Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.
T83611	(-)-15-Deoxyspergualin trihydrochloride
	(-)-15-Deoxyspergualin trihydrochloride，一种抗肿瘤剂，对小鼠白血病L-1210显示出显著抑制效果。
T124161	5α,8α-Epidioxyergost-6-en-3β-ol
	5α,8α-Epidioxyergost-6-en-3β-ol 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124161。
T21340	Pergolide
	Pergolide, an ergoline-based dopamine receptor agonist, is used for the treatment of Parkinson's disease, which is associated with low levels of the neurotransmitter dopamine in the brain.
T126125	8,14-Epoxyergosta-4,22-diene-3,6-dione
	8,14-Epoxyergosta-4,22-diene-3,6-dione 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T126125。
TF0052	Anzergent 3-8
	Anzergent 3-8 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 TF0052，CAS号为 15178-76-4。
T27341	Flurdihydroergotamine
	Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.
T130509	Aspergamid B
	Aspergamid B 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T130509。
T124005	Gingerglycolipid B
	Gingerglycolipid B 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T124005，CAS号为 88168-90-5。
T32655	l-Ergothionine hydrochloride l-Ergothionine HCl
	l-Ergothionine hydrochloride is a sulfur-containing amino acid, which is only produced by Actinomycetales bacteria and non-yeast-like fungi belonging to the division Basidiomycota and Ascomycota. It was originally isolated from Claviceps purpurea or rye e
T124479	Thunberginol H
	Thunberginol H 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T124479，CAS号为 64847-01-4。
T71707	Romergoline
	Romergoline 是一种新合成的麦角碱衍生物，具有独特的药理作用，在正常动物中表现出完全的多巴胺(DA)拮抗作用，而在“去神经”动物模型中表现出完全的DA 拮抗作用。
T75595	Loxosceles Bergeri Venom
	Loxosceles Bergeri Venom 是一种可以从Loxosceles Bergeri 中获得的毒液。Loxosceles 蜘蛛的毒液是一种复杂的毒素混合物，富含蛋白质、糖蛋白和低分子质量多肽。目前已鉴定出几种蛋白类，包括类虾蛋白酶金属蛋白酶、低分子杀虫肽、抑制剂半胱氨酸结肽 (ICK) 和磷脂酶 D。其中独特的酶，鞘磷脂酶 D 负责坏死的发展。
TP1108	Allergen Gal d 4 (46-61), chicken Lysozyme C (46-61) (chicken)
	Allergen Gal d 4 (46-61), chicken is a hen egg white lysozyme peptide.
T131391	3,5,25-Trihydroxyergostan-6-one
	3,5,25-Trihydroxyergostan-6-one 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131391。
T31664	Lysergamide, N-cyclopropyl-, maleate Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate
	Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate is a bioactive chemical.
T26909	Bromerguride
	Bromerguride is a dopamine antagonist with the activity of antipsychotic.
T62091	Anti-hyperglycemic agent-1
	Anti-hyperglycemic agent 1 是一种 α- 葡萄糖苷酶 (α-Glucosidase) 的有效抑制剂 (IC50: 0.53 μM)。Anti-hyperglycemic agent 1 能够用于研究糖尿病。

化合物

Cat.No: T67842

Synonym: EGR240

Target: Others

Cat.No: T60051

Target: Others

Cat.No: T7145

Synonym: 1-(2-噻唑基偶氮)-2-萘酚

Target: Others

Dihydroergocristine mesylate

Cat.No: T11043

Synonym: 甲磺酸双氢麦角汀,DHEC (mesylate)

Target: Beta Amyloid

Sergliflozin etabonate

Cat.No: T28757

Synonym: GW-869682,GW-869682X,KGT-1251,GW869682X,GW869682,KGT1251

Target: SGLT

Cat.No: T9174

Synonym: Sephin 1,lcerguastat,IFB-088

Target: Phosphatase

Methyl Ergoline Acid

Cat.No: T9793

Target: Others

Pergolide mesylate

Cat.No: T2226

Synonym: 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor

Cat.No: T68174

Target: SGLT

Cat.No: T1132

Synonym: 尼麦角林,Nicergolinum,Nimergoline

Target: Adrenergic Receptor

Cat.No: T4008

Synonym: 甲麦角林,Methergoline,Liserdol

Target: Dopamine Receptor, 5-HT Receptor, Sodium Channel

Romergoline 2HCl

Cat.No: T71707L

Synonym: Romergoline 2HCl(107052-56-2 Free base),FCE 23884 2HCl

Target: Dopamine Receptor

ERGi-USU-6 mesylate

Cat.No: T61062

Cat.No: T82447

Synonym: ErgTx1

Antiallergic agent-1

Cat.No: T63825

Cat.No: T33045

Experimental allergic encephalitogenic peptide (human)

Cat.No: T82424

Cat.No: T78239

Target: Carboxypeptidase

Methysergide maleate

Cat.No: T21423

Synonym: Deseril, Sansert,UML 491,UML491,Methysergide,UML-491

Dehydroergosterol

Cat.No: T37858

Synonym: 9,11-dehydro Ergosterol,DHE

3beta-Hydroxyergost-5-en-7-one

Cat.No: T125721

(R)-3,4-Dimethoxydalbergione

Cat.No: T69337

ZWITTERGENT 3-16 Detergent

Cat.No: T65361

Cat.No: T68010

Cat.No: TF0004

Cat.No: T24003

Synonym: CM 29717,CH 29717,CH 29-717

Cat.No: T71213

Bergenin (Vakerin; Peltophorin; Cuscutin)

Cat.No: T131544

Zwittergent 3-12 Detergent

Cat.No: T65355

Cergutuzumab amunaleukin

Cat.No: T76944

Dihydroergostin

Cat.No: T31469

Synonym: DE145,DE-145,DE 145

Cat.No: T69065

Cabergoline diphosphate

Cat.No: T68551

(-)-15-Deoxyspergualin trihydrochloride

Cat.No: T83611

5α,8α-Epidioxyergost-6-en-3β-ol

Cat.No: T124161

Cat.No: T21340

8,14-Epoxyergosta-4,22-diene-3,6-dione

Cat.No: T126125

Cat.No: TF0052

Flurdihydroergotamine

Cat.No: T27341

Cat.No: T130509

Gingerglycolipid B

Cat.No: T124005

l-Ergothionine hydrochloride

Cat.No: T32655

Synonym: l-Ergothionine HCl

Cat.No: T124479

Cat.No: T71707

Loxosceles Bergeri Venom

Cat.No: T75595

Allergen Gal d 4 (46-61), chicken

Cat.No: TP1108

Synonym: Lysozyme C (46-61) (chicken)

3,5,25-Trihydroxyergostan-6-one

Cat.No: T131391

Lysergamide, N-cyclopropyl-, maleate

Cat.No: T31664

Synonym: Ergoline-8-beta-carboxamide, N-cyclopropyl-9,10-didehydro-6-methyl-, maleate

Cat.No: T26909

Anti-hyperglycemic agent-1

Cat.No: T62091

Cat. No.	Product Name	Target	Signaling Pathways
TN7070	Ergostenol delta8(14)-Ergostenol,alpha-Ergostenol,菜油甾醇,Ergost-8(14)-en-3beta-ol	Others	Others
	Ergostenol (Ergost-8(14)-en-3beta-ol) 是一种生物前体和维生素 D2 的维生素原。
TMS0418	Dihydroergotoxine mesylate 甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Dihydroergotoxine mesylate (Ergoloid mesylates) 是系列生物碱盐混合物，对GABAA 受体高结合活性。它主要用于改善与衰老相关的精神退化的症状和身体症状。
TJS0328	Nordalbergin 6,7-dihydroxy-4-phenylcoumarin,6,7-Dihydroxy-4-Phenylchromen-2-One,6,7-二羟基-4苯基香豆素	Others	Others
	Nordalbergin 是一种香豆素，分离自Dalbergia sissoo 的木皮中。它能够显著性的诱导 HL-60 细胞的分化。
TN7127	5,6-Epoxyergosterol	Others	Others
	5,6-Epoxyergosterol 来源于内生真菌 Phyllosticta capitalensis。
T8191	Ergothioneine 麦角硫因,L-(+)-Ergothioneine	Antioxidant; Endogenous Metabolite	Metabolism; oxidation-reduction
	Ergothioneine (L-(+)-Ergothioneine) 是组氨酸甜菜碱的咪唑-2-硫酮衍生物，可以由细菌和真菌合成。Ergothioneine 是抗氧化剂。
TJS0856	Dalbergin 黄檀素,6-Hydroxy-7-Methoxy-4-Phenylcoumarin	Others	Others
	Dalbergin (6-Hydroxy-7-Methoxy-4-Phenylcoumarin) 是一种 Dalbergia Sissoo Linn. knot wood 提取物的成分。它具有强大的抗氧化活性。
T0122	Bergenin Cuscutin,Bengenin,岩白菜素	Apoptosis; IL Receptor; Virus Protease; TNF; NF-κB; Antibacterial; NOD; Autophagy; Antifungal	Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology; NF-κB
	Bergenin (Bengenin) 是一种在许多药用植物中发现的多酚，有细胞保护和抗氧化作用。它还具有广泛的保肝、抗炎、抗肿瘤、抗病毒、抗真菌以及免疫调节作用。
T2143	Bergapten 5-Methoxypsoralen,佛手柑内酯,香柑内酯	P450; Autophagy	Autophagy; Metabolism
	Bergapten (5-Methoxypsoralen) 是白芷中的一种香豆素，也是一种补骨脂素，可抑制细胞复制。
TN7071	Ergosterol Acetate Ergosta-5,7,22-trien-3-beta-yl acetate	Others	Others
	Ergosterol Acetate (Ergosta-5,7,22-trien-3-beta-yl acetate) 是来自红曲霉的 Ergosterol 的乙酸酯衍生物之一。
T5747	ISOBERGAPTEN	Others	Others
	Isobergapten 是一种化感抑制剂，分离自Hevacleum laciniatum 种子。
T2912	Ergosterol 麦角固醇,Provitamin D,Ergosterin,Provitamin D2	Others; Endogenous Metabolite	Metabolism; Others
	Ergosterol (Provitamin D2) 是真菌中的主要固醇类，具有抗炎，抗氧化和抗增殖的作用。
TN1345	8-Hydroxybergapten 8-羟基佛手柑内酯,8-羟基佛手苷内酯	Others	Others
	8-hydroxybergapten 具有优异的抗皱效果。在离散的 O-甲基转移酶介导的反应中，它被 Ruta 细胞的无细胞提取物 O-甲基化为异青霉素。
T3832	11-O-Galloylbergenin	Antioxidant; Immunology/Inflammation related	Immunology/Inflammation; oxidation-reduction
	11-O-Galloylbergenin 是从 Mallotus philippinensis 中分离出来的，具有抗氧化和抗疟原虫活性。
T15824	Lysergol	Antibacterial	Microbiology/Virology
	Lysergol 已被用作一种降血压、精神镇痛药以及刺激子宫和肠道的药物。 Lysergol 是从 Ipomoea muricata 的种子中分离出来的一种棒状生物碱，是药物和营养物质的生物增强剂，具有抗菌活性。
T5S0669	Bergamottin 5-Geranoxypsoralen,Bergamotine,Bergaptin,佛手柑素	P450	Metabolism
	Bergamottin (5-Geranoxypsoralen) 是竞争性CYP1A1抑制剂(Ki:10.703 nM)。
T14853	Cabergoline FCE-21336,卡麦角林	Dopamine Receptor; 5-HT Receptor; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Cabergoline (FCE-21336) 是一种麦角衍生的多巴胺 D2亚类受体激动剂，高亲和力作用于D2、D3和5-HT2B 受体，Ki 分别为 0.7、1.5 和 1.2。
T13686	Ergolide	NF-κB	NF-κB
	Ergolide, a sesquiterpene lactone extracted from the dried flowers of Inula Britannica, effectively hinders the expression of inducible nitric oxide synthase and cyclo-oxygenase-2 in RAW 264.7 macrophages by deactivating NF-κB.
T2S1434	Bergaptol 5-Hydroxyfuranocoumarin,4-Hydroxybergapten,5-羟基-6,7-呋喃并香豆素,5-Hydroxypsoralen	P450	Metabolism
	Bergaptol (4-Hydroxybergapten) 是CYP3A4酶脱苄基作用的抑制剂(IC50:24.92 uM)，具有抗癌、抗增殖作用。
T9057	norbergenin	IL Receptor; TNF; Reactive Oxygen Species	Apoptosis; Immunology/Inflammation; Metabolism; NF-κB
	Norbergenin 是一种 bergenin 的邻去甲基衍生物，可从白芍的根茎中分离得到，具有中等的抗氧化活性。
TN3498	Bergenin pentaacetate	Others	Others
	Bergenin pentaacetate 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3498，CAS号为 14531-47-6。
T60598	Thunbergol
	Thunbergol (Isocembrol) (Compound 17) 是TNF-α的有效抑制剂 (IC 50 = 7.2 μM)。
T75468	Asperglaucin B
	Asperglaucin B 是一种来自真菌Aspergillus chevalieriSQ-8 的烷基化水杨醛衍生物，具有抗菌活性。Asperglaucin B 对两种植物病原体Pseudomonas syringae pv actinidae(Psa)和Bacillus cereus 显示出有效的抗菌活性，MIC 值为 6.25 μM。
T72235	Antibacterial synergist 2
	Antibacterial synergist 2 是菌膜抑制剂。Antibacterial synergist 2 对肠球菌、金色葡萄球菌、铜绿假单胞菌和白色假单胞菌具有抑制效应。Antibacterial synergist 2 可用于与形成菌膜的病原体的相关研究。
TN3132	5-O-Methyldalbergiphenol	Others	Others
	5-O-Methyldalbergiphenol 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3132，CAS号为 1499946-35-8。
TN5288	Ergosterol peroxide glucoside 过氧化麦角甾醇葡萄糖苷,Ergosterol peroxide 3-O-β-D-glucopyranoside
	Ergosterol peroxide exhibits anti-cancer, amoebicidal, anticomplementary, antibacterial, antiviral, anti-oxdiant, and anti-melanogenic activities. Ergosterol peroxide could as an anti-atherosclerosis agent, it exhibits hACAT-1 and Lp-PLA2 inhibitory effec
TN3984	Ergosterol glucoside	Others	Others
	Ergosterol glucoside is a natural product from Rehmannia glutinosa.
TN3753	Dalbergioidin	Tyrosinase; ROS; Akt; PI3K; TGF-beta/Smad	Cytoskeletal Signaling; Immunology/Inflammation; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
	Dalbergioidin exhibits tyrosinase inhibitory activity with an IC50 of 20 mM. It shows a melanin biosynthesis inhibition zone in the culture plate of Streptomyces bikiniensis that has commonly been used as an indicator organism. Dalbergioidin protects MC3T3-E1 osteoblastic cells against H2O2-induced cell damage through activation of the PI3K/AKT/SMAD1 pathway, suggests that it may be useful in bone metabolism diseases, particularly osteoporosis. Dalbergioidin also ameliorates doxorubicin-induced ...
TN5299	Aspergillon A
	Aspergillon A 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5299，CAS号为 2239299-08-0。
TN3056	4-O-Galloylbergenin	Others	Others
	4-O-Galloylbergenin shows significant 2,2-diphenyl-1-picrylhydrazyl (DPPH) free-radical scavenging activity with EC50 7.8 uM, it shows more antioxidant activity than the positive control vitamin C (EC50 = 28.3 uM).
TN6432	Bergaptol O-β-D-glucopyranoside Bergaptol-beta-glucopyranoside
	Bergaptol O-β-D-glucopyranoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6432，CAS号为 131623-13-7。
T38086	Neohydroxyaspergillic Acid
	Neohydroxyaspergillic acid is a fungal metabolite produced by A. sclerotiorum that has antibiotic and antifungal activities. It inhibits the growth of P. aeruginosa, M. smegmatis, S. aureus, E. coli, K. pneumoniae, B. mycoides, and B. subtilis bacteria (MICs = 125-500 μg/ml). Neohydroxyaspergillic acid also inhibits the growth of G. convolute, S. consortiale, P. blakesleeanus, C. globosum, and T. mentagrophytes (MICs = 175-700 μg/ml) but not A. niger, P. notatum, M. verrucaria, or S. cerevisiae ...
T37810	6',7'-Epoxybergamottin
	6'7'-Epoxybergamottin is a furanocoumarin found in grapefruit. It is a potent inhibitor of the cytochrome P450 (CYP) isoform CYP3A4 with an IC50 value of 0.30 ppm in a cell-free assay, 0.33 μM in HL7 human liver cells, and 0.22 μM in S9 human intestine cells. It has been studied in the context of drug interactions with grapefruit constituents. It is found in grapefruit juice at concentrations of 0.1-7.4 μM and inhibits the transport of talinolol , a permeability glycoprotein (P-gp/ABCB1) transpo...
TN5550	Buergerinin B
	Buergerinin B是一种天然产物，属于玄参科玄参属，其产品编号为 TN5550，CAS号为 919769-83-8。Buergerinin B可用作对照参考。
T38949	Gingerglycolipid A
	Gingerglycolipid A is a monoacyldigalactosyl glycerol.
T38235	16-Keto Aspergillimide
	16-Keto Aspergillimide (SB202327) is a novel anthelmintic compound derived from the Aspergillus strain IMI 337664.
TN5798	(R)-4-Methoxydalbergione (+)-4-Methoxydalbergione,(R)-4-甲氧基黄檀醌
	(R)-4-Methoxydalbergione 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5798，CAS号为 4646-86-0。
TN3983	Ergosta-7,22-dien-3-one	NO Synthase; LTR	Immunology/Inflammation
	Ergosta-7,22-dien-3-one 是一种羊毛甾烷，能够从台湾灵芝的子实体中分离得到。Ergosta-7,22-dien-3-one 具有促炎特性，它能刺激一氧化氮的产生，诱导基因的表达，并诱导 J774A.1 细胞产生 TLRs、细胞因子、趋化因子和细胞粘附分子。
TN2893	3,5-Cycloergosta-6,8(14),22-triene	Others	Others
	3,5-Cycloergosta-6,8(14),22-triene 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN2893，CAS号为 24352-51-0。
TMA0955	Thunberginol C	Antifection	Microbiology/Virology
	Thunberginol C exhibits antimicrobial activity against oral bacteria. It shows antiallergic activity in the in vitro bioassay using the Schults-Dale reaction in sensitized guinea pig bronchial muscle.
TN3146	6',7'-Dihydroxybergamottin acetonide	Others	Others
	6',7'-Dihydroxybergamottin is a potent inhibitor of CYP3A activity, and may be primarily responsible for the effects of grapefruit juice on cytochrome P450 activity in humans.
TN5700	(+)-Dalbergiphenol (+)-黄檀酚,(R)-Dalbergiphenol
	(+)-Dalbergiphenol 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5700，CAS号为 82358-44-9。
TN3147	6',7'-Dihydroxybergamottin	P450	Metabolism
	6',7'-Dihydroxybergamottin(DHB), a well-known inhibitor of CYP3A4, the inhibition of CYP3A4 activity by DHB includes the inhibition of POR activity, DHB can inhibit nifedipine oxidation in a concentration-dependent manner.
TN5286	3β,5α,9α-Trihydroxyergosta-7,22-dien-6-one
	3β,5α,9α-Trihydroxy-ergosta-7,22-dien-6-one in the presence of NGF (20 ng/mL) exerts a significant increase in neurite-bearing cells.
T75467	Asperglaucin A
	Asperglaucin A 代表一种不寻常的类苯酞衍生物。Asperglaucin A 对两种植物病原体Pseudomonas syringae pv actinidae(Psa) 和Bacillus cereus 具有有效的抗菌活性，MIC 值为 6.25 μM。
T83462	11-O-Syringylbergenin
	11-O-Syringylbergenin为自龙骨草全草中分离出的岩白菜素类衍生物。
TN3546	Buergerinin G	Others	Others
	Buergerinin G是一种天然产物，属于玄参科地黄属，其产品编号为 TN3546，CAS号为 263764-83-6。Buergerinin G可用作对照参考。
TN3982	Ergosta-5,24(28)-diene-3,7,16-triol	Others	Others
	Ergosta-5,24(28)-diene-3,7,16-triol 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3982，CAS号为 289054-34-8。
TN1617	Ergosta-4,6,8(14),22-tetraen-3-one	BCL; Caspase; p53	Apoptosis; Proteases/Proteasome
	Ergosta-4,6,8(14),22-tetraen-3-one has cytotoxic activity against human gastric cancer cell, it can induce G2/M cell cycle arrest and apoptosis in human hepatocellular carcinoma HepG2 cells, these results would be useful for the further utilization of man
TN5314	7α-Methoxy-5α,6α-epoxyergosta-8(14),22-dien-3β-ol 5α,6α-Epoxy-7α-methoxyergosta-8(14),22-dien-3β-ol
	7α-Methoxy-5α,6α-epoxyergosta-8(14),22-dien-3β-ol 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5314，CAS号为 1207441-49-3。
TN5287	3β,5α-Dihydroxyergosta-7,22-dien-6-one
	3β,5α-Dihydroxy-(22E,24R)-ergosta-7,22-dien-6-one exhibits strong or moderate cytotoxic activities against MCF-7, A549, Hela and KB cell lines with IC50 values 4.98 (MCF-7), 1.95 (A549), 0.68(Hela), and 1.50 uM (KB), respectively.
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天然产物

Cat.No: TN7070

Synonym: delta8(14)-Ergostenol,alpha-Ergostenol,菜油甾醇,Ergost-8(14)-en-3beta-ol

Target: Others

Dihydroergotoxine mesylate

Cat.No: TMS0418

Synonym: 甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱

Target: GABA Receptor

Cat.No: TJS0328

Synonym: 6,7-dihydroxy-4-phenylcoumarin,6,7-Dihydroxy-4-Phenylchromen-2-One,6,7-二羟基-4苯基香豆素

Target: Others

5,6-Epoxyergosterol

Cat.No: TN7127

Target: Others

Ergothioneine

Cat.No: T8191

Synonym: 麦角硫因,L-(+)-Ergothioneine

Target: Antioxidant, Endogenous Metabolite

Cat.No: TJS0856

Synonym: 黄檀素,6-Hydroxy-7-Methoxy-4-Phenylcoumarin

Target: Others

Cat.No: T0122

Synonym: Cuscutin,Bengenin,岩白菜素

Target: Apoptosis, IL Receptor, Virus Protease, TNF, NF-κB, Antibacterial, NOD, Autophagy, Antifungal

Cat.No: T2143

Synonym: 5-Methoxypsoralen,佛手柑内酯,香柑内酯

Target: P450, Autophagy

Ergosterol Acetate

Cat.No: TN7071

Synonym: Ergosta-5,7,22-trien-3-beta-yl acetate

Target: Others

Cat.No: T5747

Target: Others

Cat.No: T2912

Synonym: 麦角固醇,Provitamin D,Ergosterin,Provitamin D2

Target: Others, Endogenous Metabolite

8-Hydroxybergapten

Cat.No: TN1345

Synonym: 8-羟基佛手柑内酯,8-羟基佛手苷内酯

Target: Others

11-O-Galloylbergenin

Cat.No: T3832

Target: Antioxidant, Immunology/Inflammation related

Cat.No: T15824

Target: Antibacterial

Cat.No: T5S0669

Synonym: 5-Geranoxypsoralen,Bergamotine,Bergaptin,佛手柑素

Target: P450

Cat.No: T14853

Synonym: FCE-21336,卡麦角林

Target: Dopamine Receptor, 5-HT Receptor, Autophagy

Cat.No: T13686

Target: NF-κB

Cat.No: T2S1434

Synonym: 5-Hydroxyfuranocoumarin,4-Hydroxybergapten,5-羟基-6,7-呋喃并香豆素,5-Hydroxypsoralen

Target: P450

Cat.No: T9057

Target: IL Receptor, TNF, Reactive Oxygen Species

Bergenin pentaacetate

Cat.No: TN3498

Target: Others

Cat.No: T60598

Cat.No: T75468

Antibacterial synergist 2

Cat.No: T72235

5-O-Methyldalbergiphenol

Cat.No: TN3132

Target: Others

Ergosterol peroxide glucoside

Cat.No: TN5288

Synonym: 过氧化麦角甾醇葡萄糖苷,Ergosterol peroxide 3-O-β-D-glucopyranoside

Ergosterol glucoside

Cat.No: TN3984

Target: Others

Cat.No: TN3753

Target: Tyrosinase, ROS, Akt, PI3K, TGF-beta/Smad

Cat.No: TN5299

4-O-Galloylbergenin

Cat.No: TN3056

Target: Others

Bergaptol O-β-D-glucopyranoside

Cat.No: TN6432

Synonym: Bergaptol-beta-glucopyranoside

Neohydroxyaspergillic Acid

Cat.No: T38086

6',7'-Epoxybergamottin

Cat.No: T37810

Cat.No: TN5550

Gingerglycolipid A

Cat.No: T38949

16-Keto Aspergillimide

Cat.No: T38235

(R)-4-Methoxydalbergione

Cat.No: TN5798

Synonym: (+)-4-Methoxydalbergione,(R)-4-甲氧基黄檀醌

Ergosta-7,22-dien-3-one

Cat.No: TN3983

Target: NO Synthase, LTR

3,5-Cycloergosta-6,8(14),22-triene

Cat.No: TN2893

Target: Others

Cat.No: TMA0955

Target: Antifection

6',7'-Dihydroxybergamottin acetonide

Cat.No: TN3146

Target: Others

(+)-Dalbergiphenol

Cat.No: TN5700

Synonym: (+)-黄檀酚,(R)-Dalbergiphenol

6',7'-Dihydroxybergamottin

Cat.No: TN3147

Target: P450

3β,5α,9α-Trihydroxyergosta-7,22-dien-6-one

Cat.No: TN5286

Cat.No: T75467

11-O-Syringylbergenin

Cat.No: T83462

Cat.No: TN3546

Target: Others

Ergosta-5,24(28)-diene-3,7,16-triol

Cat.No: TN3982

Target: Others

Ergosta-4,6,8(14),22-tetraen-3-one

Cat.No: TN1617

Target: BCL, Caspase, p53

7α-Methoxy-5α,6α-epoxyergosta-8(14),22-dien-3β-ol

Cat.No: TN5314

Synonym: 5α,6α-Epoxy-7α-methoxyergosta-8(14),22-dien-3β-ol

3β,5α-Dihydroxyergosta-7,22-dien-6-one

Cat.No: TN5287

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