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Targets Recommended: Stearoyl-CoA Desaturase (SCD) Bradykinin Receptor

330

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP1918L Lys-[Des-Arg9]Bradykinin,TFA

Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)

Bradykinin Receptor GPCR/G Protein
Lys-[Des-Arg9]Bradykinin,TFA (71800-36-7 free base) 是内源性强效和高选择性的缓激肽 B1 受体激动剂(对人 B1 和 B2 受体的 Ki 值分别为 0.12 和 > 30000 nM)。降低体内外周血管阻力的降压药。比 [Des-Arg9]-缓激肽强 16 倍。
TP1445 [Des-Arg9]-Bradykinin acetate

[Des-Arg9]-缓激肽醋酸盐

Bradykinin Receptor GPCR/G Protein
[Des-Arg9]-Bradykinin acetate 是一种选择性缓激肽 B1 受体激动剂。
TP1918L1 Lys-[Des-Arg9]Bradykinin acetate

Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)

Bradykinin Receptor GPCR/G Protein
Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) 是一种内源性强效和高选择性的缓激肽 B1 受体激动剂(对人 B1 和 B2 受体的 Ki 值分别为 0.12 和 > 30000 nM)。降低体内外周血管阻力的降压药。比 [Des-Arg9]-缓激肽强 16 倍。
T8809 [Des-Arg9]-Bradykinin TFA

Bradykinin Receptor GPCR/G Protein
[Des-Arg9]-Bradykinin TFA 是一种缓激肽 (B1) 受体激动剂,对 B1 的选择性优于对 B2 受体的选择性。
T1883 Des(benzylpyridyl) Atazanavi

HIV Protease Microbiology/Virology; Proteases/Proteasome
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。
TP1917L1 Sar-[D-Phe8]-des-Arg9-Bradykinin acetate

Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)

Bradykinin Receptor GPCR/G Protein
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) 是一种有效的选择性缓激肽 B1 受体激动剂(兔主动脉中的 EC50 = 9.02 nM),对氨肽酶、激肽酶 I 和 II (ACE) 以及中性内肽酶切割具有抗性。在体内表现出降血压和血管生成活性。
T7645 [Des-Arg9]-Bradykinin

[Des-Arg9]-Bradykinin(2TFA),[Des-Arg9]-缓激肽

Bradykinin Receptor GPCR/G Protein
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA)) 是 Bradykinin(B1) 受体激动剂,对 B1受体选择性大于B2受体。
T1216 Diethylstilbestrol

Stilbestrol,己烯雌酚,DES

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Diethylstilbestrol (DES) 是一种非甾体雌性激素,能够用于更年期和绝经后的紊乱。
TP1181 Bradykinin (2-9)

Des-Arg1-bradykinin

Bradykinin Receptor GPCR/G Protein
Bradykinin (2-9) (Des-Arg1-bradykinin),是Bradykinin的一种氨基端截短肽类代谢物,通过Aminopeptidase P的切割作用形成。
TP2032 des-​Gln14-​Ghrelin

des-Gln14-Ghrelin (rat)

An endogenous ligand for the ghrelin receptor (GHS-R1a), produced by alternative splicing of the rat ghrelin gene. Potently induces Ca2+ release in cells expressing ghrelin receptors (EC50 = 2.4 nM) and stimulates GH release in vivo.
T36638 [Des-His1,Glu9]-Glucagon amide TFA

[Des-His1,Glu9]-Glucagon amide TFA

[Des-His1,Glu9]-Glucagon amide TFA is a potent peptide antagonist targeting the glucagon receptor, featuring a pA2 value of 7.2. It holds potential utility in diabetes pathogenesis research[1].
TP2033 [Des-His1,Glu9]-Glucagon amide

des-His1-[Glu9]-Glucagon (1-29) amide

Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes); displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitro. Blocks added glucagon-induced hy
T31634 [Des-Tyr1]-Met-Enkephalin

Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-

Enkephalin-met, des-tyr(1)- ccauses retrograde amnesia in rats.
TP2450 Argipressin, des-glynh2(9)-

9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin

Argipressin, des-glynh2(9)-, can effect on aggregation of blood platelets.
TP2241 [Des-octanoyl]-Ghrelin (human)

Others Others
[Des-octanoyl]-Ghrelin (human) is a Non-acylated, major circulating isoform of ghrelin.
TP1918 Lys-[Des-Arg9]Bradykinin

Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]
TP2242 [Des-octanoyl]-Ghrelin (rat)

Others Others
[Des-octanoyl]-Ghrelin (rat) is a Non-acylated, major circulating isoform of ghrelin.
T35602 O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine

O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine is a major metabolite of the calcium channel inhibitor amlodipine .1 1.Taguchi, R., Naito, T., Sato, H., et al.Validated LC-MS/MS method for the simultaneous determination of amlodipine and its major metabolites in human plasma of hypertensive patientsTher. Drug Monit.39(6)625-631(2017)
TP1917 Sar-[D-Phe8]-des-Arg9-Bradykinin

Potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cleavage. Exhibits hypotensive and angiogenic activity in vivo.
TP2370 Angiotensin pentapeptide

Angiotensin II (4-8),(Des-1,2,3)angiotensin II

Angiotensin pentapeptide is a peptide.
T83500 [Des-Arg10]-HOE I40

[Des-Arg10]-HOE 140 是一种有效的 B1 缓激肽受体拮抗剂,具备生物活性。
T75928 des-​Gln14-​Ghrelin TFA

des-Gln14-Ghrelin TFA为生长激素促分泌受体的第二个内源性配体。该化合物能在CHO-GHSR62细胞中诱导[Ca2+]I的提升,其EC50值为2.4 nM。
T76326 [Des-His1,Glu9] Glucagon

[Des-His1,Glu9] Glucagon 是一种有效的胰高血糖素受体系统多肽拮抗剂。[Des-His1,Glu9] Glucagon 增强胰岛细胞在葡萄糖刺激下释放胰岛素。[Des-His1,Glu9] Glucagon 可用于糖尿病的研究。
T80394 Des(8-14)brevinin-1PMa

Des(8-14)brevinin-1PMa是一种具有抗金黄色葡萄球菌和大肠杆菌活性的宿主防御肽,同时也表现出溶血性。
T80117 Lys-(Des-Arg9,Leu8)-Bradykinin

Bradykinin Receptor GPCR/G Protein
Lys-(Des-Arg9,Leu8)-Bradykinin为缓激肽B1受体的拮抗剂。
T73646 Lys-[Des-Arg9]Bradykinin TFA

Lys-[Des-Arg9]Bradykinin TFA 是一种天然存在的激肽,是一种有效且高度选择性的缓激肽 B1受体激动剂,对人,小鼠和兔子的 B1受体的 Ki 值为 0.12 nM,1.7 nM 和 0.23 nM。Lys-[Des-Arg9]Bradykinin TFA 对 B2 受体的抑制活性较低。
T80072 Des-Arg9-[Leu8]-Bradykinin acetate

Bradykinin Receptor GPCR/G Protein
Des-Arg9-[Leu8]-Bradykinin acetate 是一种B1R(缓激肽受体1)拮抗剂,主要应用于肾纤维化的研究。
T76291 Des His1, Glu8 Exendin-4

Des His1, Glu8 Exendin-4 是一种高效的GLP-1-R(胰高血糖素样肽-1 受体)拮抗剂,主要通过调控胰岛素分泌和抑制葡萄糖生成来维持葡萄糖稳态。该化合物广泛应用于2型糖尿病及胃肠道相关研究领域。
T83547 (Des-Bromo)-Neuropeptide B (1-23) (human)

'(Des-Bromo)-Neuropeptide B (1-23) (human)' 是一种作用于orphan G-protein coupled receptor的激动剂,对GPR7 (NPBW1) 的Ki值为1.2 nM,而对GPR8 (NPBW2) 的Ki值则为341 nM。
T76591 (Des-Glu5)-ACTH (1-24) (human, bovine, rat)

(Des-Glu5)-ACTH (1-24) (human, bovine, rat) 是促肾上腺皮质激素 (ACTH) 的类似物。ACTH 是一种由垂体前叶腺产生的多肽激素,调节皮质醇和雄激素的产生。
T83688 R 715 TFA

[Ac-Lys-[D-βNal7,Ile8]des-Arg9]-BK,Ac-Lys-Arg-Pro-Pro-Gly-Phe-Ser-D2Nal-Ile-OH

R 715是一种布拉迪肾上腺素B1受体拮抗剂。它抑制在表达布拉迪肾上腺素B1受体的孤立人类脐带中由布拉迪肾上腺素引发的收缩(pA2 = 8.49)。R 715(200、400及600 µg/kg)通过尾部闪烁测试减少了由链脲佐菌素(STZ)诱导的糖尿病神经病变小鼠模型中尾部撤回的潜伏期。它还在以髓磷脂少突胶质细胞糖蛋白(MOG)(35-55)(MOG35-55)抗原肽诱导的实验性自体免疫性脑炎(EAE)小鼠模型中,通过每天1 mg/kg的剂量减少了后肢无力和瘫痪的发病率,改善对称步态,并减少脊髓炎症灶点数、神经元脱髓鞘以及病灶单核细胞侵袭。R 715(0.01 nmol/动物,脑室内)能在自发性高血压大鼠中降低平均动脉血压并增加心率。
T76595 (Des-His6)-ACTH (1-24) (human, bovine, rat)

(Des-His6)-ACTH (1-24) (human, bovine, rat) 是促肾上腺皮质激素 (ACTH) 的类似物。ACTH 是一种由垂体前叶腺产生的多肽激素,调节皮质醇和雄激素的产生。
T76601 (D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)

'(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin(6-14)是一种蛙皮素(bombesin)拮抗剂,主要应用于癌症研究领域。'
T76593 (Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)

'(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)' 为一种GnRH类似物,主要用于诱导养殖鱼类排卵和/或产卵。
T76633 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin

(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin 为一种有效的加压素 V1 受体 (VP V1R) 拮抗剂,能显着降低大鼠的平均动脉压 (MAP)。
T76590 (d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin

(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin,是一种催产素受体拮抗剂,可消除 CA1 锥体神经元中催产素增强的抑制性突触后电流。
T69630 Diphenyleneiodonium (free base)

Diphenyleneiodonium (free base) is an NADPH oxidase inhibitor.
T10760 Ceramides Mixture

神经酰胺混合物,神经酰胺

Telomerase DNA Damage/DNA Repair
Ceramides Mixture 是表皮渗透屏障的主要脂质成分,参与生长抑制,细胞周期停滞和端粒酶活性的调节。它是一种内源性神经酰胺,由含羟基和非羟基脂肪酸的神经酰胺组成。
T5144 Desmopressin acetate (16679-58-6 free base)

Desmopressin acetate,醋酸去氨加压素,DDAVP

Vasopressin Receptor GPCR/G Protein
Desmopressin acetate (16679-58-6 free base) (DDAVP) 是抗利尿激素精氨酸加压素的合成类似物。
T67822L Ulodesine

BCX4208

Endogenous Metabolite Metabolism
Ulodesine (BCX4208) 是一种嘌呤核苷磷酸化酶 (PNP) 抑制剂,对 PNP 有抑制作用,IC50 值为 2.293 nM/L。Ulodesine 可用于研究高尿酸血症。
TP2323L Deslorelin acetate(57773-65-6 free base)

Deslorelin acetate

GNRH Receptor GPCR/G Protein
Deslorelin acetate(57773-65-6 free base) 是一种促性腺激素释放激素超级激动剂(GnRH agonist)
T4199 Desmethyl-VS-5584

PI3K; mTOR PI3K/Akt/mTOR signaling
Desmethyl-VS-5584 是 VS-5584 的二甲基类似物。其中VS-5584 是mTOR/PI3K 抑制剂,专门针对于吡啶 [2,3-d] 嘧啶结构。
T4572 Desoximetasone

去羟米松,Desoximetasonum,Topicort,Desoxymethasone,Desoximetasona

Others Others
Desoximetasone (Desoximetasona) 是一种可缓解皮疹等多种皮肤疾病的皮质类固醇。
T11039 Didesethyl chloroquine

Bisdesethylchloroquine

Drug Metabolite Metabolism
Didesethyl chloroquine (Bisdesethylchloroquine) 是一种有效的心肌抑制剂。Didesethyl chloroquine 是抗疟药氯喹的主要代谢产物。
T76892 Ordesekimab

AMG 714,PRV-015

IL Receptor Immunology/Inflammation
Ordesekimab (AMG 714) 是一种人 IgG1κ 抗 IL-15 (Interleukin Related) 单克隆抗体。Ordesekimab 竞争性与 IL-15 结合,会抑制 IL-15 与 IL-2Rβ 和 IL-15 受体复合物的共同 γ 链的相互作用,却不与 IL-15Rα 链发生反应。Ordesekimab 可用于研究无反应性乳糜泻 (NRCD) 。
T10138 4-Desmethoxy Omeprazole

Drug Metabolite Metabolism
4-Desmethoxy Omeprazole 是 Omeprazole 的活性代谢物。Omeprazole 是质子泵抑制剂。Omeprazole 竞争性抑制 CYP2C19 活性,Ki=2 - 6 μM。Omeprazole 还抑制革兰氏阴性菌和革兰氏阳性菌生长。
T3560 Desmethylanethol trithione

ADT-OH

VEGFR; Akt Angiogenesis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Desmethylanethol trithione (ADT-OH) 是合成硫化氢的供体。它利用上调 FADD 诱导细胞凋亡,并对体内黑色素瘤的形成具有一定的抑制作用,可用于研究癌症疾病。
T67851 rac Desmethyl Citalopram Hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
rac Desmethyl Citalopram Hydrochloride 是一种5-羟色胺摄取抑制剂,IC50值为0.013μM。
T11001L1 N-Desethyl Chloroquine Hydrochloride

(±)-Desethylchloroquine 2HCl

N-Desethyl Chloroquine Hydrochloride ((±)-Desethylchloroquine 2HCl) 是一种Desethylchloroquine 衍生物。desethylchloroquine 在体外和体内竞争性地抑制cyp2d1 /6介导的反应。
T11078 Deschloroclozapine

Serotonin Transporter Neuroscience
Deschloroclozapine 是氯氮平的代谢物,是一种高效毒蕈碱 DREADDs 激动剂。它可作为 PET 示踪剂,用于 DREADD 的影像学检查。它与 DREADD 受体亚型 hM3Dq 和 hM4Di 结合,Ki 分别为 6.3 和 4.2 nM。

化合物

Lys-[Des-Arg9]Bradykinin,TFA
Cat.No: TP1918L
Synonym: Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate
Cat.No: TP1445
Synonym: [Des-Arg9]-缓激肽醋酸盐
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate
Cat.No: TP1918L1
Synonym: Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin TFA
Cat.No: T8809
Synonym:
Target: Bradykinin Receptor
Des(benzylpyridyl) Atazanavi
Cat.No: T1883
Synonym:
Target: HIV Protease
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Cat.No: TP1917L1
Synonym: Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin
Cat.No: T7645
Synonym: [Des-Arg9]-Bradykinin(2TFA),[Des-Arg9]-缓激肽
Target: Bradykinin Receptor
Diethylstilbestrol
Cat.No: T1216
Synonym: Stilbestrol,己烯雌酚,DES
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Bradykinin (2-9)
Cat.No: TP1181
Synonym: Des-Arg1-bradykinin
Target: Bradykinin Receptor
des-​Gln14-​Ghrelin
Cat.No: TP2032
Synonym: des-Gln14-Ghrelin (rat)
Target:
[Des-His1,Glu9]-Glucagon amide TFA
Cat.No: T36638
Synonym: [Des-His1,Glu9]-Glucagon amide TFA
Target:
[Des-His1,Glu9]-Glucagon amide
Cat.No: TP2033
Synonym: des-His1-[Glu9]-Glucagon (1-29) amide
Target:
[Des-Tyr1]-Met-Enkephalin
Cat.No: T31634
Synonym: Met-enkephalin, des-tyr(1),1-De-tyr-met-enkephalin,Enkephalin-met, des-tyr(1)-
Target:
Argipressin, des-glynh2(9)-
Cat.No: TP2450
Synonym: 9-Deglycinamide-argipressin,(Arg8,de-Gly9)-vasopressin,DEAVP,DGAVP,9-Des-glynh2-argipressin
Target:
[Des-octanoyl]-Ghrelin (human)
Cat.No: TP2241
Synonym:
Target: Others
Lys-[Des-Arg9]Bradykinin
Cat.No: TP1918
Synonym:
Target:
[Des-octanoyl]-Ghrelin (rat)
Cat.No: TP2242
Synonym:
Target: Others
O-Des[2-aminoethyl]-O-carboxymethyl dehydroamlodipine
Cat.No: T35602
Synonym:
Target:
Sar-[D-Phe8]-des-Arg9-Bradykinin
Cat.No: TP1917
Synonym:
Target:
Angiotensin pentapeptide
Cat.No: TP2370
Synonym: Angiotensin II (4-8),(Des-1,2,3)angiotensin II
Target:
[Des-Arg10]-HOE I40
Cat.No: T83500
Synonym:
Target:
des-​Gln14-​Ghrelin TFA
Cat.No: T75928
Synonym:
Target:
[Des-His1,Glu9] Glucagon
Cat.No: T76326
Synonym:
Target:
Des(8-14)brevinin-1PMa
Cat.No: T80394
Synonym:
Target:
Lys-(Des-Arg9,Leu8)-Bradykinin
Cat.No: T80117
Synonym:
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin TFA
Cat.No: T73646
Synonym:
Target:
Des-Arg9-[Leu8]-Bradykinin acetate
Cat.No: T80072
Synonym:
Target: Bradykinin Receptor
Des His1, Glu8 Exendin-4
Cat.No: T76291
Synonym:
Target:
(Des-Bromo)-Neuropeptide B (1-23) (human)
Cat.No: T83547
Synonym:
Target:
(Des-Glu5)-ACTH (1-24) (human, bovine, rat)
Cat.No: T76591
Synonym:
Target:
R 715 TFA
Cat.No: T83688
Synonym: [Ac-Lys-[D-βNal7,Ile8]des-Arg9]-BK,Ac-Lys-Arg-Pro-Pro-Gly-Phe-Ser-D2Nal-Ile-OH
Target:
(Des-His6)-ACTH (1-24) (human, bovine, rat)
Cat.No: T76595
Synonym:
Target:
(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)
Cat.No: T76601
Synonym:
Target:
(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)
Cat.No: T76593
Synonym:
Target:
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
Cat.No: T76633
Synonym:
Target:
(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
Cat.No: T76590
Synonym:
Target:
Diphenyleneiodonium (free base)
Cat.No: T69630
Synonym:
Target:
Ceramides Mixture
Cat.No: T10760
Synonym: 神经酰胺混合物,神经酰胺
Target: Telomerase
Desmopressin acetate (16679-58-6 free base)
Cat.No: T5144
Synonym: Desmopressin acetate,醋酸去氨加压素,DDAVP
Target: Vasopressin Receptor
Ulodesine
Cat.No: T67822L
Synonym: BCX4208
Target: Endogenous Metabolite
Deslorelin acetate(57773-65-6 free base)
Cat.No: TP2323L
Synonym: Deslorelin acetate
Target: GNRH Receptor
Desmethyl-VS-5584
Cat.No: T4199
Synonym:
Target: PI3K, mTOR
Desoximetasone
Cat.No: T4572
Synonym: 去羟米松,Desoximetasonum,Topicort,Desoxymethasone,Desoximetasona
Target: Others
Didesethyl chloroquine
Cat.No: T11039
Synonym: Bisdesethylchloroquine
Target: Drug Metabolite
Ordesekimab
Cat.No: T76892
Synonym: AMG 714,PRV-015
Target: IL Receptor
4-Desmethoxy Omeprazole
Cat.No: T10138
Synonym:
Target: Drug Metabolite
Desmethylanethol trithione
Cat.No: T3560
Synonym: ADT-OH
Target: VEGFR, Akt
rac Desmethyl Citalopram Hydrochloride
Cat.No: T67851
Synonym:
Target: 5-HT Receptor
N-Desethyl Chloroquine Hydrochloride
Cat.No: T11001L1
Synonym: (±)-Desethylchloroquine 2HCl
Target:
Deschloroclozapine
Cat.No: T11078
Synonym:
Target: Serotonin Transporter
Cat. No. Product Name Target Signaling Pathways
T83300 5′-Des-O-methylharringtonine

5′-Des-O-methylharringtonine为Cephalotaxus harringtonia植物中提取的天然化合物。
T3S1265 Liriopesides B

山麦冬皂苷B,Nolinospiroside F

Others Others
Liriopesides B (Nolinospiroside F) 是一种甾体皂苷,分离自 Ophiopogon japonicas 中,具有抗氧化和抗衰老活性。
T1168 Desonide

Tridesilon,地索奈德,Locapred,Prednacinolone

Glucocorticoid Receptor Endocrinology/Hormones
Desonide (Prednacinolone) 是一种非氟化皮质类固醇抗炎剂,能够作用于糖皮质激素受体。
TN6786 O-Desmethyl Galanthamine

Sanguinine,O-去甲基加兰他敏

AChE Neuroscience
O-Desmethyl Galanthamine (Sanguinine) 是一种加兰他敏型生物碱,是一种乙酰胆碱酯酶 (AChE) 抑制剂,其IC50=1.83 μM。
TJS0387 Desoxyrhaponticin

去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin

Apoptosis; Fatty Acid Synthase Apoptosis; Metabolism
Desoxyrhaponticin (Deoxyrhaponticin) 是来自西藏营养食品唐古特大黄中的一种二苯乙烯苷。它是脂肪酸合成酶抑制剂,抑制细胞内 FAS 活性,下调人乳腺癌 MCF-7细胞中 FAS 的表达。它是控制糖尿病餐后高血糖的潜在药物。
T5738 7-Epi 10-desacetyl paclitaxel

10-Deacetyl-7-epipaclitaxel,7-Epi-10-deacetyltaxol,7-表-10-去乙酰基云南紫杉宁A

Others Others
7-Epi 10-desacetyl paclitaxel (10-Deacetyl-7-epipaclitaxel) 是紫杉醇衍生物,对 HeLa 细胞具有细胞毒性(IC50:85 μM)。
T2520 Desloratadine

Sch34117,地氯雷他定,NSC 675447

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Desloratadine (Sch34117) 是非镇静H1抗组胺药 Loratadine 的主要口服代谢物,可减少对支气管平滑肌、毛细血管和胃肠道平滑肌中 H1 受体的典型组胺能作用,包括血管舒张、支气管收缩、血管通透性增加、疼痛、瘙痒和胃肠道平滑肌的痉挛性收缩。它是一种选择性H1受体拮抗剂,具有抗过敏和抗炎活性。
TJS0161 Eudesmol

β-Eudesmol,桉叶醇,Β-桉叶醇

Others Others
β-Eudesmol (β-Eudesmol) 是一种倍半萜类化合物,由Streptomyces tendae 产生。
TN2755 2-Desoxy-4-epi-pulchellin

Anti-infection Microbiology/Virology
2-Desoxy-4-epi-pulchellin 是分离自 Polygonum hydropiper 的二氯甲烷可溶部分的一种化合物。
T3836 Eudesmin

MAPK; S6 Kinase MAPK; PI3K/Akt/mTOR signaling
Eudesmin 通过抑制S6K1信号通路来干扰成脂分化,具有抗肿瘤、抗炎和抗菌活性。
T8183 Deslanoside

洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C

ATPase; Drug Metabolite Membrane transporter/Ion channel; Metabolism
Deslanoside (Desacetyllanatoside C) 是一种快速作用的强心苷,可抑制Na-K-ATPase 膜泵,导致细胞内钠和钙浓度增加。它用于研究充血性心力衰竭和因折返机制引起的室上性心律失常,并在研究慢性心房颤动时控制心室率。
T3865 beta-Eudesmol

β-桉叶醇,Beta-Selinenol,beta-桉叶醇

TRP/TRPV Channel; AChR Membrane transporter/Ion channel; Neuroscience
beta-Eudesmol (Beta-Selinenol) 是天然的含氧倍半萜烯,可激活hTRPA1,EC50值为 32.5 μM。Beta-Eudesmol 有增加食欲的功效。
T2862 Desaminotyrosine

Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,对羟基苯丙酸,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid,根皮酸

Others; Influenza Virus; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
Desaminotyrosine (3-(4-Hydroxyphenyl)propionic acid) 是一种与微生物相关的代谢物,通过增强 I 型干扰素信号传导来预防流感。
T11855 Lipopolysaccharides

脂多糖,LPS

Others Others
Lipopolysaccharides (LPS) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
TN1299 Desmethylglycitein

4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone

PI3K; CDK; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) 是大豆中苷元的代谢产物,具有抗氧化性和抗癌活性。它是蛋白激酶 C(PKC)α 的直接抑制剂,抑制正常人皮肤成纤维细胞中的太阳紫外线诱导的基质金属蛋白酶1。它在体内直接结合CDK1和CDK2,抑制 CDK1 和 CDK2 活性。
TN6930 5-Desmethylsinensetin

Others Others
5-desmethylsinensetin 是分离自Stevia satureiifoliavar.satureiifolia 的天然产物,显示出抗原生动物的活性,抑制T. cruzi epimastigotes 和trypomastigotes 的IC50分别为 0.4 μg/mL 和75.1 μg/mL。
TQ0170 Desacetylcinobufagin

Deacetylcinobufagin,去乙酰华蟾蜍精

Others Others
Desacetylcinobufagin (Deacetylcinobufagin) 是一种天然化合物,可用于微生物转化。
T19711 Desmosterol

Desmesterol,24-Dehydrocholesterol

Endogenous Metabolite Metabolism
Desmosterol(24-Dehydrocholesterol) 是一种胆固醇生物合成中间体,抑制巨噬细胞炎症小体活化,防止血管炎症和动脉粥样硬化。
T5S0734 Desmethoxyyangonin

Desmethoxy yangonin,去甲氧基醉椒素,Demethoxyyangonin,5,6-Dehydrokavain

Others; Monoamine Oxidase Neuroscience; Others
Desmethoxyyangonin (5,6-Dehydrokavain) 是一种MAO-B 可逆性抑制剂。
T9358 N,N,O-Tridesmethylvenlafaxine

Tridesmethylvenlafaxine

Others; Endogenous Metabolite Metabolism; Others
N,N,O-Tridesmethylvenlafaxine (Tridesmethylvenlafaxine) 是内源性代谢产物的一种。
T22455 Vindesine sulfate

DVA,Desacetylvinblastine amide,硫酸长春地辛,DAVA,Desacetyl Vinblastine amide,VDS

Others Others
Vindesine sulfate (Desacetyl Vinblastine amide) 是一种长春花生物碱,它是长春碱的合成衍生物,与有丝分裂纺锤体的微管蛋白结合,导致微管结晶和有丝分裂停滞或细胞死亡。
T36581 Glucocerebrosides

Others Others
Glucocerebrosides 是一种天然产物。
T8270 Deserpidine

地舍平,Harmonyl

RAAS Endocrinology/Hormones
Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂,可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。
T19259 D-Desthiobiotin

Endogenous Metabolite Metabolism
D-Desthiobiotin 是一种生物素衍生物,用于蛋白质层析和亲和层析,也用于蛋白质和细胞的标记、检测和分离。
T41078 Lipopolysaccharides, Escherichiacoli

Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides, Escherichiacoli 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides, Escherichiacoli 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T75650 Rivulariapeptolides 1121

Rivulariapeptolides 1121,作为一种高效的选择性丝氨酸蛋白酶抑制剂,对胰凝蛋白酶、弹性蛋白酶和蛋白酶K展示出了显著的抑制活性,其IC50值分别为35.52 nM、13.24 nM和48.05 nM。
T75649 Rivulariapeptolides 1185

Rivulariapeptolides 1185 是一种高效的选择性丝氨酸蛋白酶抑制剂,其对胰凝蛋白酶、弹性蛋白酶和蛋白酶 K 的 IC50分别为 13.17 nM、23.59 nM 和 55.26 nM。
T80008 Stevisaliosides D

Phosphatase Metabolism
Stevisaliosides D (Compound 5) 是从甜叶菊根中提取的化合物,具有抑制PTP1B的活性(IC50:31.8 μM),应用于抗糖尿病研究。
TN4030 Eudesm-4(15)-ene-3alpha,11-diol

Eudesm-4(15)-ene-3alpha,11-diol 是一种来源于Eudesm-4(15)-ene-3alpha,11-diol 的化合物。
TN3962 epi-Eudesmol

Others Others
epi-Eudesmol is a natural product from Laggera alata var. montana C. D. Adams.
T82325 Gentiiridosides A

Gentiiridosides A为从龙胆中提取的一种化合物,采用无水乙醇作为萃取溶剂。
TN7055 N-Desmethyl Galanthamine

N-Desmethyl Galanthamine 在生命科学相关研究中具有广泛的应用。
T3841 Desrhamnosylmartynoside

Others Others
Desrhamnosylmartynoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T3841,CAS号为 136055-64-6。
TN6382 Desacetylripariochromene B

Desacetylripariochromene B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6382,CAS号为 69790-24-5。
T31728 Eudesmane

Eudesmane is a bicyclododecane terpenes.
T19782 Antidesmone

Antidesmone is one compound mainly isolated from Ajugade cumbers Thunb (Labiatae). Antidesmone prevents acute lung injury via regulating MAPK and NF-κB activities.
TN3032 4-Hydroxy-11,12,13-trinor-5-eudesmen-7-one

Others Others
4-Hydroxy-11,12,13-trinor-5-eudesmen-7-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3032,CAS号为 133369-42-3。
TN5370 1β,10β-Epoxydesacetoxymatricarin

1beta,10beta-Epoxydesacetoxymatricarin shows high anti-hypercholesterolemic potential.
T36029 Desertomycin A

Desertomycin A is fungal metabolite and the major component of the desertomycin antibiotic complex that has been found in S. flavofungini.
T82578 Desacetylxanthanol

Desacetylxanthanol (Compound 4),源自Xanthium strumarium的倍半萜类化合物,展现出抗肿瘤坏死因子相关凋亡诱导配体(TRAIL)活性。
TN5377 Nardoeudesmol A

Nardoeudesmol A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5377,CAS号为 1445952-30-6。
T11009 Destruxin B

Others Others
Destruxin B is a cyclic peptide with insecticidal and anticancer activity isolated from the insect pathogenic fungus Metarhizium isopliae. Destruxin B induces apoptosis of human non-small cell lung cancer cells through the Bcl-2 family-dependent mitochond
TN3838 Desmethylrocaglamide

Others Others
Desmethylrocaglamide is a novel inducer of cellular differentiation using HL-60 promyelocytic cells, it may be a drug for the prevention and therapy of cancer. It also has insecticidal activity.
T83386 2-Desoxypleniradin-L-α-arabinopyranoside, 2-acetate

2-Desoxypleniradin-L-α-arabinopyranoside, 2-acetate 是一种从Helenium amarum分离得到的活性化合物。
T83387 2-Desoxypleniradin-4-0-a-L-rhamnopyranoside

2-Desoxypleniradin-4-0-a-L-rhamnopyranoside为一种黄酮类化合物,可自Helenium radiatum中提取。
TN2668 1beta-Hydroxy-beta-eudesmol

Others Others
1beta-Hydroxy-beta-eudesmol is a natural product from Cymbopogon proximus STAPF.
T83431 1-Desmethylobtusin

1-Desmethylobtusin是从Cassia obtusifoliaL.分离出的蒽醌类化合物。
TN5684 5,6-Desmethylenedioxy-5-methoxyaglalactone

5,6-Desmethylenedioxy-5-methoxyaglalactone is cytotoxic to small cell lung cancer (NCI-H187) cell line. It has antimycobacterial activity against Mycobacterium tuberculosis H(37)Ra.
TN2933 3-Eudesmene-1beta,11-diol

Others Others
3-Eudesmene-1beta,11-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2933,CAS号为 658062-22-7。
TSP-41868968 alpha-Desmotroposantonin

alpha-Desmotroposantonin 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TSP-41868968。
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天然产物

5′-Des-O-methylharringtonine
Cat.No: T83300
Synonym:
Target:
Liriopesides B
Cat.No: T3S1265
Synonym: 山麦冬皂苷B,Nolinospiroside F
Target: Others
Desonide
Cat.No: T1168
Synonym: Tridesilon,地索奈德,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
O-Desmethyl Galanthamine
Cat.No: TN6786
Synonym: Sanguinine,O-去甲基加兰他敏
Target: AChE
Desoxyrhaponticin
Cat.No: TJS0387
Synonym: 去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin
Target: Apoptosis, Fatty Acid Synthase
7-Epi 10-desacetyl paclitaxel
Cat.No: T5738
Synonym: 10-Deacetyl-7-epipaclitaxel,7-Epi-10-deacetyltaxol,7-表-10-去乙酰基云南紫杉宁A
Target: Others
Desloratadine
Cat.No: T2520
Synonym: Sch34117,地氯雷他定,NSC 675447
Target: Endogenous Metabolite, Histamine Receptor
Eudesmol
Cat.No: TJS0161
Synonym: β-Eudesmol,桉叶醇,Β-桉叶醇
Target: Others
2-Desoxy-4-epi-pulchellin
Cat.No: TN2755
Synonym:
Target: Anti-infection
Eudesmin
Cat.No: T3836
Synonym:
Target: MAPK, S6 Kinase
Deslanoside
Cat.No: T8183
Synonym: 洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C
Target: ATPase, Drug Metabolite
beta-Eudesmol
Cat.No: T3865
Synonym: β-桉叶醇,Beta-Selinenol,beta-桉叶醇
Target: TRP/TRPV Channel, AChR
Desaminotyrosine
Cat.No: T2862
Synonym: Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,对羟基苯丙酸,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid,根皮酸
Target: Others, Influenza Virus, Endogenous Metabolite
Lipopolysaccharides
Cat.No: T11855
Synonym: 脂多糖,LPS
Target: Others
Desmethylglycitein
Cat.No: TN1299
Synonym: 4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone
Target: PI3K, CDK, PKC
5-Desmethylsinensetin
Cat.No: TN6930
Synonym:
Target: Others
Desacetylcinobufagin
Cat.No: TQ0170
Synonym: Deacetylcinobufagin,去乙酰华蟾蜍精
Target: Others
Desmosterol
Cat.No: T19711
Synonym: Desmesterol,24-Dehydrocholesterol
Target: Endogenous Metabolite
Desmethoxyyangonin
Cat.No: T5S0734
Synonym: Desmethoxy yangonin,去甲氧基醉椒素,Demethoxyyangonin,5,6-Dehydrokavain
Target: Others, Monoamine Oxidase
N,N,O-Tridesmethylvenlafaxine
Cat.No: T9358
Synonym: Tridesmethylvenlafaxine
Target: Others, Endogenous Metabolite
Vindesine sulfate
Cat.No: T22455
Synonym: DVA,Desacetylvinblastine amide,硫酸长春地辛,DAVA,Desacetyl Vinblastine amide,VDS
Target: Others
Glucocerebrosides
Cat.No: T36581
Synonym:
Target: Others
Deserpidine
Cat.No: T8270
Synonym: 地舍平,Harmonyl
Target: RAAS
D-Desthiobiotin
Cat.No: T19259
Synonym:
Target: Endogenous Metabolite
Lipopolysaccharides, Escherichiacoli
Cat.No: T41078
Synonym: Lipopolysaccharide, E. coli O111:B4
Target: Others
Rivulariapeptolides 1121
Cat.No: T75650
Synonym:
Target:
Rivulariapeptolides 1185
Cat.No: T75649
Synonym:
Target:
Stevisaliosides D
Cat.No: T80008
Synonym:
Target: Phosphatase
Eudesm-4(15)-ene-3alpha,11-diol
Cat.No: TN4030
Synonym:
Target:
epi-Eudesmol
Cat.No: TN3962
Synonym:
Target: Others
Gentiiridosides A
Cat.No: T82325
Synonym:
Target:
N-Desmethyl Galanthamine
Cat.No: TN7055
Synonym:
Target:
Desrhamnosylmartynoside
Cat.No: T3841
Synonym:
Target: Others
Desacetylripariochromene B
Cat.No: TN6382
Synonym:
Target:
Eudesmane
Cat.No: T31728
Synonym:
Target:
Antidesmone
Cat.No: T19782
Synonym:
Target:
4-Hydroxy-11,12,13-trinor-5-eudesmen-7-one
Cat.No: TN3032
Synonym:
Target: Others
1β,10β-Epoxydesacetoxymatricarin
Cat.No: TN5370
Synonym:
Target:
Desertomycin A
Cat.No: T36029
Synonym:
Target:
Desacetylxanthanol
Cat.No: T82578
Synonym:
Target:
Nardoeudesmol A
Cat.No: TN5377
Synonym:
Target:
Destruxin B
Cat.No: T11009
Synonym:
Target: Others
Desmethylrocaglamide
Cat.No: TN3838
Synonym:
Target: Others
2-Desoxypleniradin-L-α-arabinopyranoside, 2-acetate
Cat.No: T83386
Synonym:
Target:
2-Desoxypleniradin-4-0-a-L-rhamnopyranoside
Cat.No: T83387
Synonym:
Target:
1beta-Hydroxy-beta-eudesmol
Cat.No: TN2668
Synonym:
Target: Others
1-Desmethylobtusin
Cat.No: T83431
Synonym:
Target:
5,6-Desmethylenedioxy-5-methoxyaglalactone
Cat.No: TN5684
Synonym:
Target:
3-Eudesmene-1beta,11-diol
Cat.No: TN2933
Synonym:
Target: Others
alpha-Desmotroposantonin
Cat.No: TSP-41868968
Synonym:
Target:
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Cat. No. Product Name Species Expression System
TMPJ-00882 Desmin Protein, Human, Recombinant (His)

DES,Desmin

Human E. coli
Desmin is a cytoplasmic protein and belongs to the intermediate filament family. interacts with DST and MTM1. Desmin is only expressed in vertebrates, however homologous proteins are found in many organisms. Desmin is the main intermediate filament in mature skeletal, cardiac and smooth-muscle cells. DES founctions as homopolymers to form a stable intracytoplasmic filamentous network connecting myofibrils to each other and to the plasma membrane. .Defects in DES are cause of the myopathy myofibr...
TMPY-04960 Der p 1 Protein, Dermatophagoides pteronyssinus, Recombinant (His)

Dermatophagoides pteronyssinus HEK293 Cells
Der p 1 Protein, Dermatophagoides pteronyssinus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.7 kDa and the accession number is P08176.
TMPY-06179 IdeS Protein, Streptococcus pyogenes, Recombinant (His & GST)

Streptococcus pyogenes E. coli
IdeS (IgG-degrading enzyme of Streptococcus pyogenes) is a secreted cysteine endopeptidase from the human pathogen S. pyogenes with an extraordinarily high degree of substrate specificity, catalyzing a single proteolytic cleavage at the lower hinge of human IgG. This proteolytic degradation promotes inhibition of opsonophagocytosis and interferes with the killing of group A Streptococcus. IdeS Protein, Streptococcus pyogenes, Recombinant (His & GST) is expressed in E. coli expression system with...
TMPH-02363 TROSPA Protein, Ixodes scapularis, Recombinant (His)

Ixodes scapularis Baculovirus Insect Cells
Serves as a receptor for ospA protein of B.burgdorferi, the Lyme disease agent. Required for spirochetal colonization. Essential for pathogen adherence to the vector. TROSPA Protein, Ixodes scapularis, Recombinant (His) is expressed in Baculovirus insect cells with C-6xHis tag. The predicted molecular weight is 21.7 kDa and the accession number is Q5SDL7.
TMPH-02408 SPI Protein, Lentinula edodes, Recombinant (His)

Lentinula edodes E. coli
Serine protease inhibitor. Active against beta-trypsin and alpha-chymotrypsin with dissociation constants of 0.35 nM and 40 nM respectively. Inhibits factor XIa, but not other enzymes involved in coagulation and fibrinolysis. Does not inhibit subtilisin, lysyl endopeptidase, arginyl endopeptidase or papain.
TMPY-05078 Der f 2 Protein, Dermatophagoides farinae, Recombinant (His)

Dermatophagoides farinae E. coli
Der f 2 Protein, Dermatophagoides farinae, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 15 kDa and the accession number is Q00855.1.
TMPH-00403 Toxin A Protein, Clostridioides difficile, Recombinant (His)

Clostridioides difficile E. coli
Toxin A Protein, Clostridioides difficile, Recombinant (His) is expressed in E. coli.
TMPY-05903 Influenza A H5N1 (A/Bangladesh/207095/2008) Hemagglutinin/HA Protein (His)

Harvey rat sarcoma viral oncogene homolog

H5N1 HEK293 Cells
Influenza A H5N1 (A/Bangladesh/207095/2008) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.7 kDa.
TMPH-02407 Peroxidase Protein, Lentinula edodes, Recombinant (His & Myc)

Lentinula edodes E. coli
Peroxidase Protein, Lentinula edodes, Recombinant (His & Myc) is expressed in E. coli.
TMPY-03370 Desmocollin 2/DSC2 Protein, Rat, Recombinant (His)

desmocollin 2

Rat HEK293 Cells
Desmocollin 2/DSC2 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.1 kDa and the accession number is Q3T1K6.
TMPH-00474 Der p 6 Protein, Dermatophagoides pteronyssinus, Recombinant (GST)

DP5,Mite allergen Der p 6,DERP6,Der p 6,Allergen Der p VI

Dermatophagoides pteronyssinus E. coli
Der p 6 Protein, Dermatophagoides pteronyssinus, Recombinant (GST) is expressed in E. coli.
TMPY-04642 Desmocollin 2/DSC2 Protein, Rat, Recombinant (hFc)

desmocollin 2

Rat HEK293 Cells
Desmocollin 2/DSC2 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 101.6 kDa and the accession number is Q3T1K6.
TMPY-05518 Der p 5 Protein, Dermatophagoides pteronyssinus, Recombinant (His)

mite allergen Der p 5,DERP5 Protein, Dermatophagoides

Dermatophagoides pteronyssinus E. coli
Der p 5 Protein, Dermatophagoides pteronyssinus, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 16.6 kDa and the accession number is A0A6P6Y2A6.
TMPH-00475 DNA ligase Protein, Desulfotalea psychrophila, Recombinant (His)

Polydeoxyribonucleotide synthase [NAD(+)],ligA,DNA ligase

Desulfotalea psychrophila E. coli
DNA ligase Protein, Desulfotalea psychrophila, Recombinant (His) is expressed in E. coli.
TMPY-06023 IdeS Protein, Streptococcus pyogenes, Recombinant (His)

Streptococcus pyogenes E. coli
IdeS (IgG-degrading enzyme of Streptococcus pyogenes) is a secreted cysteine endopeptidase from the human pathogen S. pyogenes with an extraordinarily high degree of substrate specificity, catalyzing a single proteolytic cleavage at the lower hinge of human IgG. This proteolytic degradation promotes inhibition of opsonophagocytosis and interferes with the killing of group A Streptococcus. IdeS Protein, Streptococcus pyogenes, Recombinant (His) is expressed in E. coli expression system with His t...
TMPK-00967 DSG-2/Desmoglein-2 Protein, Human, Recombinant (His)

CMD1BB,Desmoglein-2,ARVC10,CDHF5,MGC117037,MGC11703...

Human HEK293 Cells
Desmoglein-2 (DSG-2) as the primary high-affinity receptor used by adenoviruses Ad3, Ad7, Ad11 and Ad14. These serotypes represent key human pathogens causing respiratory and urinary tract infections. In epithelial cells, adenovirus binding of DSG-2 triggers events reminiscent of epithelial-to-mesenchymal transition, leading to transient opening of intercellular junctions. DSG-2/Desmoglein-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted mo...
TMPH-00473 Der p 3 Protein, Dermatophagoides pteronyssinus, Recombinant (His)

Mite allergen Der p 3,Der p 3,DERP3,Allergen Der p III

Dermatophagoides pteronyssinus E. coli
Der p 3 Protein, Dermatophagoides pteronyssinus, Recombinant (His) is expressed in E. coli.
TMPY-06975 Der p 21 Protein, Dermatophagoides pteronyssinus, Recombinant

Dermatophagoides pteronyssinus E. coli
Der p 21 Protein, Dermatophagoides pteronyssinus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 15.55 kDa.
TMPH-00359 AlkB Protein, Caulobacter vibrioides, Recombinant (His & Myc)

Alpha-ketoglutarate-dependent dioxygenase AlkB homolog,DNA o...

Caulobacter vibrioides E. coli
AlkB Protein, Caulobacter vibrioides, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 31.2 kDa and the accession number is B8GWW6.
TMPH-00361 Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His)

Toxin 2,Beta-mammal toxin Cn2,Toxin II.9.2.2

Centruroides noxius P. pastoris (Yeast)
Mammal beta-toxins bind voltage-independently at site-4 of sodium channels (Nav) and shift the activation voltage to more negative potentials. This toxin is active against mammals. Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 9.6 kDa and the accession number is P01495.
TMPY-05139 Der p 10 Protein, Dermatophagoides pteronyssinus, Recombinant

Dermatophagoides pteronyssinus E. coli
Der p 10 Protein, Dermatophagoides pteronyssinus, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 32.9 kDa and the accession number is O18416.1.
TMPH-00188 BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc)

Adenosylmethionine-8-amino-7-oxononanoate aminotransferase B...

Bacteroides fragilis E. coli
Catalyzes two activities which are involved in the biotine biosynthesis: the conversion of dethiobiotin (DTB) to biotin by the insertion of a sulfur atom into dethiobiotin via a radical-based mechanism, and the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The p...
TMPY-04945 Der p 2 Protein, Dermatophagoides pteronyssinus, Recombinant (His)

Dermatophagoides pteronyssinus E. coli
Hypersensitivity to house dust mite (Dermatophagoides sp.) allergens is one of the most common allergic reactions in the world. The house dust mite allergen, Der p 2, is a major allergen and 80–90% of patients who react to mite extract, react specifically to this protein or its homologues. Although it is well characterized in terms of allergenicity, there is still some ambiguity in terms of its biological function. Three-dimensional structural analysis of Der p 2 and its close homologues indicat...
TMPH-00472 Der p 23 Protein, Dermatophagoides pteronyssinus, Recombinant (His & Myc)

Major HDM allergen Der p 23,Major mite allergen Der p 23,Der...

Dermatophagoides pteronyssinus E. coli
Der p 23 Protein, Dermatophagoides pteronyssinus, Recombinant (His & Myc) is expressed in E. coli.
TMPH-00190 Fragilysin Protein, Bacteroides fragilis, Recombinant (His)

Bacteroides fragilis E. coli
Diarrheal toxin that hydrolyzes gelatin, azocoll, actin, tropomyosin, and fibrinogen. Fragilysin Protein, Bacteroides fragilis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 46.7 kDa and the accession number is P54355.
TMPH-00362 Beta-mammal toxin Css4 Protein, Centruroides suffusus, Recombinant (His & SUMO)

Css IV,CssIV,Beta-mammal toxin Css4

Centruroides suffusus E. coli
Beta toxins bind voltage-independently at site-4 of sodium channels (Nav) and shift the voltage of activation toward more negative potentials thereby affecting sodium channel activation and promoting spontaneous and repetitive firing. This toxin is active only on mammals. Beta-mammal toxin Css4 Protein, Centruroides suffusus, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 23.6 kDa and the accession number is P60266.
TMPK-00736 DSG-2/Desmoglein-2 Protein, Mouse, Recombinant (His)

MGC117036,HDGC,Desmoglein-2,CDHF5,DSG2,MGC117037,AR...

Mouse HEK293 Cells
Desmoglein-2 (DSG-2) as the primary high-affinity receptor used by adenoviruses Ad3, Ad7, Ad11 and Ad14. These serotypes represent key human pathogens causing respiratory and urinary tract infections. In epithelial cells, adenovirus binding of DSG-2 triggers events reminiscent of epithelial-to-mesenchymal transition, leading to transient opening of intercellular junctions. DSG-2/Desmoglein-2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted mo...
TMPH-00189 HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO)

Bacteroides fragilis E. coli
Molecular chaperone. Has ATPase activity. HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 57.0 kDa and the accession number is Q5LCH4.
TMPY-05140 Der f 1 Protein, Dermatophagoides farinae, Recombinant (His)

Dermatophagoides farinae HEK293 Cells
Der f 1 Protein, Dermatophagoides farinae, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.9 kDa and the accession number is Q58A71.
TMPY-01892 Desmocollin 2/DSC2 Protein, Human, Recombinant (His)

ARVD11,desmocollin 2,DGII/III,DSC3,DG2,CDHF2

Human HEK293 Cells
Desmocollin 2/DSC2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 75 kDa and the accession number is Q02487-1.
TMPY-05710 Der p 23 Protein, Dermatophagoides pteronyssinus, Recombinant (His)

endochitinase-like,Derp 23

Dermatophagoides pteronyssinus HEK293 Cells
Der p 23 is a new major allergen of D. pteronyssinus. The house dust mite (HDM) Dermatophagoides pteronyssinus is one of most important allergen sources and a major elicitor of allergic asthma. Der p 23 may be an essential component for diagnosis and specific immunotherapy of HDM allergy.
TMPJ-00964 PRCP Protein, Human, Recombinant (His)

PCP,Proline Carboxypeptidase,PRCP,Lysosomal Pro-X Carboxypep...

Human HEK293 Cells
Lysosomal Pro-X Carboxypeptidase (PRCP) belongs to the peptidase S28 family. PRCP is detected in many tissues, with highest levels observed in placenta, lung, and liver. It is also present in the heart, brain, pancreas, and kidney. PRCP exists as a homodimer. PRCP cleaves C-terminal amino acids linked to proline in peptides such as angiotensin II, III and des-Arg9-bradykinin. This cleavage occurs at acidic pH, but enzymatic activity is retained with some substrates at neutral pH. PRCP has been s...
TMPY-02132 LYPLA2 Protein, Human, Recombinant (His)

APT-2,lysophospholipase II,DJ886K2.4,APT2

Human E. coli
Lysophospholipase II (LYPLA2, LPL-II, or LysoPLA II), also known as Acyl-protein thioesterase 2 (APT-2), belongs to the AB hydrolase 2 family. This enzyme has lysophospholipase activity and may hydrolyze fatty acids from S-acylated cysteine residues in proteins such as trimeric G alpha proteins or HRAS. Acyl-protein thioesterase 1 (APT-1) and Acyl-protein thioesterase 2 (APT-2) are cytosolic lysophospholipids hydrolyzing enzymes. The serum activity of APT-1 may play an important role in the dete...

重组蛋白

Desmin Protein, Human, Recombinant (His)
Cat.No: TMPJ-00882
Species: Human
Expression System: E. coli
Der p 1 Protein, Dermatophagoides pteronyssinus, Recombinant (His)
Cat.No: TMPY-04960
Species: Dermatophagoides pteronyssinus
Expression System: HEK293 Cells
IdeS Protein, Streptococcus pyogenes, Recombinant (His & GST)
Cat.No: TMPY-06179
Species: Streptococcus pyogenes
Expression System: E. coli
TROSPA Protein, Ixodes scapularis, Recombinant (His)
Cat.No: TMPH-02363
Species: Ixodes scapularis
Expression System: Baculovirus Insect Cells
SPI Protein, Lentinula edodes, Recombinant (His)
Cat.No: TMPH-02408
Species: Lentinula edodes
Expression System: E. coli
Der f 2 Protein, Dermatophagoides farinae, Recombinant (His)
Cat.No: TMPY-05078
Species: Dermatophagoides farinae
Expression System: E. coli
Toxin A Protein, Clostridioides difficile, Recombinant (His)
Cat.No: TMPH-00403
Species: Clostridioides difficile
Expression System: E. coli
Influenza A H5N1 (A/Bangladesh/207095/2008) Hemagglutinin/HA Protein (His)
Cat.No: TMPY-05903
Species: H5N1
Expression System: HEK293 Cells
Peroxidase Protein, Lentinula edodes, Recombinant (His & Myc)
Cat.No: TMPH-02407
Species: Lentinula edodes
Expression System: E. coli
Desmocollin 2/DSC2 Protein, Rat, Recombinant (His)
Cat.No: TMPY-03370
Species: Rat
Expression System: HEK293 Cells
Der p 6 Protein, Dermatophagoides pteronyssinus, Recombinant (GST)
Cat.No: TMPH-00474
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
Desmocollin 2/DSC2 Protein, Rat, Recombinant (hFc)
Cat.No: TMPY-04642
Species: Rat
Expression System: HEK293 Cells
Der p 5 Protein, Dermatophagoides pteronyssinus, Recombinant (His)
Cat.No: TMPY-05518
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
DNA ligase Protein, Desulfotalea psychrophila, Recombinant (His)
Cat.No: TMPH-00475
Species: Desulfotalea psychrophila
Expression System: E. coli
IdeS Protein, Streptococcus pyogenes, Recombinant (His)
Cat.No: TMPY-06023
Species: Streptococcus pyogenes
Expression System: E. coli
DSG-2/Desmoglein-2 Protein, Human, Recombinant (His)
Cat.No: TMPK-00967
Species: Human
Expression System: HEK293 Cells
Der p 3 Protein, Dermatophagoides pteronyssinus, Recombinant (His)
Cat.No: TMPH-00473
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
Der p 21 Protein, Dermatophagoides pteronyssinus, Recombinant
Cat.No: TMPY-06975
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
AlkB Protein, Caulobacter vibrioides, Recombinant (His & Myc)
Cat.No: TMPH-00359
Species: Caulobacter vibrioides
Expression System: E. coli
Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His)
Cat.No: TMPH-00361
Species: Centruroides noxius
Expression System: P. pastoris (Yeast)
Der p 10 Protein, Dermatophagoides pteronyssinus, Recombinant
Cat.No: TMPY-05139
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc)
Cat.No: TMPH-00188
Species: Bacteroides fragilis
Expression System: E. coli
Der p 2 Protein, Dermatophagoides pteronyssinus, Recombinant (His)
Cat.No: TMPY-04945
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
Der p 23 Protein, Dermatophagoides pteronyssinus, Recombinant (His & Myc)
Cat.No: TMPH-00472
Species: Dermatophagoides pteronyssinus
Expression System: E. coli
Fragilysin Protein, Bacteroides fragilis, Recombinant (His)
Cat.No: TMPH-00190
Species: Bacteroides fragilis
Expression System: E. coli
Beta-mammal toxin Css4 Protein, Centruroides suffusus, Recombinant (His & SUMO)
Cat.No: TMPH-00362
Species: Centruroides suffusus
Expression System: E. coli
DSG-2/Desmoglein-2 Protein, Mouse, Recombinant (His)
Cat.No: TMPK-00736
Species: Mouse
Expression System: HEK293 Cells
HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00189
Species: Bacteroides fragilis
Expression System: E. coli
Der f 1 Protein, Dermatophagoides farinae, Recombinant (His)
Cat.No: TMPY-05140
Species: Dermatophagoides farinae
Expression System: HEK293 Cells
Desmocollin 2/DSC2 Protein, Human, Recombinant (His)
Cat.No: TMPY-01892
Species: Human
Expression System: HEK293 Cells
Der p 23 Protein, Dermatophagoides pteronyssinus, Recombinant (His)
Cat.No: TMPY-05710
Species: Dermatophagoides pteronyssinus
Expression System: HEK293 Cells
PRCP Protein, Human, Recombinant (His)
Cat.No: TMPJ-00964
Species: Human
Expression System: HEK293 Cells
LYPLA2 Protein, Human, Recombinant (His)
Cat.No: TMPY-02132
Species: Human
Expression System: E. coli
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