137
57
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T81403 |
Priliximab
cM-T412,CEN 000029 |
||
Priliximab (CEN 000029) 是一种针对CD4的人源化单克隆抗体。其与T细胞表面CD4的结合作用可引起循环中CD4+T细胞的显著并持久的减少,适用于类风湿性关节炎 (RA) 研究。 | |||
T14495 |
Baloxavir
Baloxavir acid,S-033447 |
Influenza Virus | Microbiology/Virology |
Baloxavir (S-033447) 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。 | |||
TNU1173 |
2'-Fluoro-2'-deoxy-ara-U-3'-phosphoramidite
|
||
2'-Fluoro-2'-deoxy-ara-U-3'-phosphoramidite is a Nucleoside Phosphoramidite; Nucleoside Derivative - Fluoro-modified nucleoside. | |||
T14927 |
Centrinone
LCR-263 |
PLK; Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
Centrinone (LCR-263) 是 polo 样激酶 4 的可逆抑制剂,对PLK4的Ki 值为0.16 nM。 | |||
T69691 |
Pocenbrodib
FT-7051,P-300 |
Epigenetic Reader Domain | Chromatin/Epigenetic |
Pocenbrodib (FT-7051) 是一种有效的 CBP/p300 家族的溴结构域抑制剂,具有潜在的抗肿瘤活性,可口用于研究癌症。 | |||
T68127 |
Picenadol
LY-150720,LY150720,LY 150720 |
Others | Others |
Picenadol (LY 150720) 是N-甲基-4-苯基哌啶衍生物的外消旋混合物,具有激动剂 - 拮抗剂阿片性质。Picenadol 具有中枢镇痛活性。 | |||
TP1104L |
Melanin Concentrating Hormone, salmon acetate
MCH (salmon),Melanin Concentrating Hormone, salmon acetate(87218-84-6 free base) |
Others; Melanin-concentrating Hormone Receptor (MCHR) | GPCR/G Protein; Others |
Melanin Concentrating Hormone, salmon acetate (MCH (salmon))(87218-84-6 free base) 是一种 19 个氨基酸的环状肽,主要在下丘脑中表达。 | |||
T19589 |
trans-2-Undecenoic acid
(E)-2-Undecenoic acid,反-2-十一烯酸,(E)-Undec-2-enoic acid |
Others | Others |
trans-2-Undecenoic acid ((E)-Undec-2-enoic acid) 是一种 α,β-不饱和羧酸,其特征在于酸二聚体,相应的二聚体通过羧基 C=O···H-O 的分子间氢键连接。 | |||
T10758L |
Centanafadine hydrochloride
EB-1020 hydrochloride |
Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。 | |||
T12832 |
Amcenestrant
SAR439859 |
Estrogen Receptor/ERR; Estrogen/progestogen Receptor | Endocrinology/Hormones |
Amcenestrant (SAR439859) 是一种有效的 ER 拮抗剂,具有 ER 降解活性,EC50为 0.2 nM。它是一种具有口服活性,非甾体和选择性雌激素受体降解剂 (SERD)。它可在 ER+乳腺癌中表现出强大的抗肿瘤功效和有限的交叉耐药性。 | |||
T9499 |
Icenticaftor
QBW251 |
CFTR | Membrane transporter/Ion channel |
Icenticaftor (QBW251) 是一种具有口服活性CFTR 通道增强剂,可用于慢性阻塞性肺疾病 (COPD) 和囊性纤维化研究,对F508del 和G551D CFTR 的EC50分别为 79 和 497 nM。 | |||
TP2338L |
Cenupatide acetate
Cenupatide acetate(1006388-38-0 Free base) |
Others | Others |
Cenupatide acetate 是一种尿激酶纤溶酶原激活物受体 (uPAR) 抑制剂,用于治疗与细胞迁移改变相关的疾病,例如癌症。 | |||
T22216 |
10-Undecen-1-ol
|
Others | Others |
10-Undecen-1-ol 是由蓖麻油酸转化得到,是一种能够引入官能团的共聚单体。 | |||
T6269 |
Bemcentinib
R428,BGB324 |
TAM Receptor | Tyrosine Kinase/Adaptors |
Bemcentinib (R428) 是具有选择性的、高效的 Axl 抑制剂,其 IC50=14 nM。 | |||
T31425 |
Dibenz[a,h]anthracene
CCRIS 208,二苯葸,NSC 22433,AI3-18996,DB(a,h)A |
DNA | DNA Damage/DNA Repair |
Dibenz[a,h]anthracene (CCRIS 208) 诱导细菌DNA 损伤和基因突变,并在几种哺乳动物细胞培养物中诱导基因突变和转化。 | |||
T10038 |
11-cis-Vaccenyl acetate
(Z)-Octadec-11-enyl acetate |
Endogenous Metabolite | Metabolism |
11-cis-Vaccenyl acetate ((Z)-Octadec-11-enyl acetate) 激活位于触角 T1 感受器的嗅觉神经元,并介导雄性和雌性果蝇的聚集行为。 | |||
TQ0297 |
Cenicriviroc
TAK-652,TBR-652 |
HIV Protease; CCR | Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Cenicriviroc (TAK-652) 是一种可口服的CCR2/CCR5拮抗剂,可抑制 HIV-1 和 HIV-2,具有抗炎、抗感染作用。 | |||
T14924 |
Cenerimod
ACT-334441 |
S1P Receptor | GPCR/G Protein |
Cenerimod (ACT-334441) 是一种具有口服活性、选择性和高效性的磷酸鞘氨醇 1 受体(S1P1)激动剂(EC50:1 nM)。Cenerimod 对多种 S1P 的亚型具有抑制作用,可用于研究鼠类实验性自身免疫性脑脊髓炎 (EAE)和鼠类硬皮病。 | |||
T8157 |
Centhaquin
PMZ-2010,Centhaquine |
Others | Others |
Centhaquin (Centhaquine)e 是一种具有研究出血性休克的潜力的试剂。在出血模型中,它能够减少全身血管阻力。 | |||
T7332 |
(E)-2-Decenoic acid
trans-2-Decenoic acid,反式-2-癸烯酸 |
Others | Others |
(E)-2-Decenoic acid (trans-2-Decenoic acid) 是一种存在于蜂王浆中的脂肪酸。 | |||
T4274 |
Melitracen hydrochloride
盐酸美利曲辛,盐酸美力他欣,Thymeol hydrochloride,Melixeran |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Melitracen hydrochloride (Thymeol hydrochloride) 是一种可口服的双相抗抑郁药和抗焦虑药。它可以通过突触前膜抑制去甲肾上腺素和5-羟色胺(5-HT)的吸收,从而诱导突触空间中单胺递质的增加。 | |||
T7193 |
Encenicline
EVP-6124 |
AChR | Neuroscience |
Encenicline (EVP-6124) 是一种新型α7神经元烟碱乙酰胆碱受体 (nAChRs)激动剂,用于治疗精神分裂症和阿尔茨海默病的认知障碍。 | |||
T2285 |
Encenicline hydrochloride
(R)-7-氯-N-(奎宁环-3-基)苯并[b]噻吩-2-甲酰胺盐酸盐,EVP-6124 (hydrochloride),EVP-6124 hydrochloride |
AChR | Neuroscience |
Encenicline hydrochloride (EVP-6124 hydrochloride) 是一种新型的α7神经元烟碱乙酰胆碱受体激动剂。 | |||
T71384 | Cenisertib benzoate | ||
Cenisertib benzoate is an orally bioavailable, synthetic, small-molecule multi-Aurora kinase inhibitor with potential antineoplastic activity. | |||
T67235 | (S)-1-[(S)-tert-Butylphosphinoyl]-2-[(S)-1-(diphenylphosphino)ethyl]ferrocene | ||
(S)-1-[(S)-tert-Butylphosphinoyl]-2-[(S)-1-(diphenylphosphino)ethyl]ferrocene 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67235。 | |||
T124174 | 2-Pentadecenedioic acid | ||
2-Pentadecenedioic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124174。 | |||
T32659 | Lettucenin A | ||
Lettucenin A is a sesquiterpenoid lactone phytoalexin. | |||
T36431 | 7,10-dihydroxy-8(E)-Octadecenoic Acid | ||
7,10-dihydroxy-8(E)-Octadecenoic acid is a hydroxy fatty acid and metabolite of oleic acid that is produced byP. aeruginosafrom vegetable oils.1It is active against the food-borne pathogenic bacteriaS. aureus,S. typhimurium,L. monocytogenes,B. subtilis, andE. coli(MIC50s = 31.3, 125, 125, 62.5, and 250 μg/ml, respectively), as well as the plant pathogenic bacteriaErwinia,R. solanacearum,C. glutamicum, andP. syringae(MIC90s = 125, 125, 250, and 500 μg/ml, respectively).2,1 1.Sohn, H.-R., Bae, J.-... | |||
T125821 | 2E-Decenoylpiperidide | ||
2E-Decenoylpiperidide 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125821。 | |||
T31299 | Decamethylrhenocene | ||
Decamethylrhenocene is a biochemical. | |||
T76490 |
Fluorescent HIV Substrate
|
||
FluorescentHIVSubstrate 是 HIV 底物。 | |||
T40400 |
Enhanced Green Fluorescent Protein (EGFP) (200-208)
|
||
Enhanced Green Fluorescent Protein (EGFP) (200-208) is a reporter protein obtained from Aequorea Victoria jellyfish. EGFP is widely used as a marker gene product due to its strong fluorescence properties, making it easily detectable. | |||
T82023 |
Ivicentamab
GEN-3009 |
||
Ivicentamab (GEN-3009),一种人源化IgG1κ亚型的单克隆抗体,靶向CD37,主要应用于癌症相关研究。 | |||
T78347 |
Serratia marcescens nuclease
|
||
Serratia marcescens nuclease,为一种非特异性核酸酶,因具备强大消化DNA与RNA活性,应用范围广泛。 | |||
T74029 |
cis-11-Methyl-2-dodecenoic acid
|
||
cis-11-Methyl-2-dodecenoic acid 是群体感应 (QS) 信号分子,在微生物及真菌的细胞外通讯系统中扮演扩散信号因子(DSF)的角色。它参与调控多种细菌病原体的毒性及生物膜的生成。 | |||
T125104 |
Lucenin II
|
||
T10757 |
Cenobamate S-Enantiomer
|
Others | Others |
Cenobamate S-Enantiomer is a Cenobamate's S-enantiomer. | |||
T123819 |
4'-O-Methyllucenin II (Diosmetin 6,8-di-C-glucoside)
|
||
4'-O-Methyllucenin II (Diosmetin 6,8-di-C-glucoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T123819。 | |||
T124811 |
Lushanrubescensin H
|
||
Lushanrubescensin H 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124811。 | |||
T29255 |
(E)-4-Undecenal
|
||
(E)-4-Undecenal is a bioactive chemical. | |||
T124378 |
(2S,3R,4E)-2-Amino-4-heptadecene-1,3-diol
|
||
(2S,3R,4E)-2-Amino-4-heptadecene-1,3-diol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124378。 | |||
T60227 |
[1,1'-Bis(diphenylphosphino)ferrocene]dichloropalladium(II)
PDCL2(DPPF) |
Others | Others |
[1,1'-Bis(diphenylphosphino)ferrocene]dichloropalladium(II) (PDCL2(DPPF))是一种催化剂。 | |||
T124254 |
(E/Z)-10-Hydroxy-2-decenoic acid
|
||
(E/Z)-10-Hydroxy-2-decenoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124254,CAS号为 765-01-5。 | |||
T32115 |
Hydrogenated didecene
1-Decene,dimers,Dec-1-ene,hydrogenated,dimer |
||
Hydrogenated didecene as skin-softening agent derived from didecene, which is a hydrocarbon. Hydrocarbons are organic compounds that contain only carbon and hydrogen. Examples of common hydrocarbons include mineral oil, petroleum, and paraffin wax. | |||
T31353 |
Decenyl cyclopentanone
AI 3-34972,AI3-34972 |
||
Decenyl cyclopentanone is a biochemical. | |||
TD0003L |
CelGreen nucleic acid gel stain *10,000× concentrate in DMSO*
|
||
CelGreen nucleic acid gel stain *10,000× concentrate in DMSO* is a fluorescent dye with a unique involvement that binds to all dsDNA double helix sulcus regions.In the free state, the side strand and CelGreen emit weak fluorescence, but the fluorescence is greatly enhanced once they are combined with the double-stranded DNA. Therefore, the fluorescence signal strength of CelGreen is related to the amount of double-stranded DNA, and the amount of double-stranded DNA in the PCR system can be detec... | |||
T9296 |
Methyl Undecenate
10-十一烯酸甲酯,Methyl undec-10-enoate,Methyl 10-undecenoate |
Others | Others |
Methyl Undecenate (Methyl undec-10-enoate) 是 10-十一碳烯酸的脂肪酸甲酯。它具有作为代谢物的作用。它衍生自 10-十一碳烯酸。 | |||
T125431 | 9,10-Anthracenedione | ||
9,10-Anthracenedione 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125431。 | |||
T129791 | 5,5'-(4-Tetradecene-1,4-diyl)bis[1,3-benzenediol] | ||
5,5'-(4-Tetradecene-1,4-diyl)bis[1,3-benzenediol] 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T129791。 | |||
T123995 | Hebeirubescensin L | ||
Hebeirubescensin L 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123995,CAS号为 887333-34-8。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0251 |
(Z)-2-decenoic acid
(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid |
Others | Others |
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。 | |||
T3851 |
Vicenin 2
Vicenin -2,维采宁 2,新西兰牡荆苷 |
RAAS | Endocrinology/Hormones |
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。 | |||
T2P2870 |
Damascenone
trans-damascenone,Beta-Damascenone,大马烯酮,大马酮 |
Others; NF-κB; Endogenous Metabolite | Metabolism; NF-κB; Others |
Damascenone (trans-damascenone) 是一种 E-和 Z-异构体大马士革酮的混合物,源于 Epipremnum pinnatum 的具有抗炎特性的特性化合物。 | |||
TWS1563 |
Incensole
|
Others | Others |
Incensole 是一种 14-membered 二萜类化合物,分离自烯属植物的香精油和乳香树脂中。它能够激活脑中离子通道,并可以缓解焦虑或抑郁,从而显示出抗炎和抗抑郁的特性。 | |||
TN2182 |
Sarracenin
脱水莫诺苷元,金银花 |
Others | Others |
Sarracenin 是一种的环烯醚萜,分离自鸢尾草的根和根茎中。它对肿瘤细胞显示出细胞毒作用。 | |||
T0306 |
10-Undecenoic acid
Undecylenic acid,Undecenoic acid,10-十一烯酸 |
Endogenous Metabolite; Antibiotic; Antifungal | Metabolism; Microbiology/Virology |
10-Undecenoic acid (Undecylenic acid) 是一种天然或合成的抑菌脂肪酸,具有抗真菌活性。 | |||
TQ0194 |
trans-Vaccenic acid
TVA,(11E)-octadec-11-enoic acid,11E)-octadec-11-enoic acid |
Endogenous Metabolite | Metabolism |
Trans-Vaccenic acid(TVA)是一种天然存在的反式脂肪酸,存在于反刍动物的脂肪和乳制品中,可通过 GPCR-CREB 通路调控 CD8+ T 细胞增殖,具有抗肿瘤活性。Trans-Vaccenic acid 可在瘤胃中合成饱和脂肪酸,在组织水平合成共轭亚油酸。 | |||
T8240 |
Cis-5-Dodecenoic Acid
|
Others | Others |
Cis-5-Dodecenoic Acid 是一种单不饱和脂肪酸,具有 C12 链作为主链,C5 位具有顺式双键。 | |||
T5834 |
Myrcene
|
Others | Others |
Myrcene 是具有可挥发性的芳香族化合物,对 TNFα 诱导的 NF-κB 具有抑制作用,且具有抗侵袭的能力。 | |||
T13299 |
Vicenin 3
维采宁-3,维采宁 3 |
RAAS | Endocrinology/Hormones |
Vicenin 3来源于广金钱草的地上部分。Vicenin 3是血管紧张素转换酶抑制剂,IC50=46.91 μM。 | |||
T7914 |
Acenaphthylene
|
Others | Others |
Acenaphthylene 是多环芳烃。其中多环芳烃是自然衍生于煤和焦油沉积物中,并由有机质的不完全燃烧得到。 | |||
TQ0197 |
Acenocoumarol
醋硝香豆素,新抗凝 |
||
Acenocoumarol 是一种抗凝血剂,与 Vitamin K 拮抗剂的功能相似。 | |||
T20225 |
Dicentrine, (-)-
L-Dicentrine,荷包牡丹碱,NSC 251699,NSC251699,NSC-251699 |
Others | Others |
Dicentrine, (-)- (NSC-251699) 是一种在几种植物物种中发现的非卟啉生物碱,在小鼠内脏痛的急性模型中显示出显著的镇痛活性。 | |||
T21130 |
Precocene II
早熟素Ⅱ,AI3-36847,Ageratochromene,BRN 0160683 |
Others | Others |
Precocene II (Ageratochromene) 是一种抗异体激素化合物,可抑制保幼激素的生物合成。 Precocene II 具有杀虫、抗真菌、抗菌和抗氧化活性。 | |||
T8241 |
cis-10-Heptadecenoic acid
|
Others | Others |
cis-10-Heptadecenoic acid 是反刍动物脂肪的次要成分。 | |||
T41335 |
cis-Vaccenic acid
cis-11-Octadecenoic acid,Asclepic acid,(Z)-octadec-11-enoic acid |
Antiviral | Immunology/Inflammation |
cis-Vaccenic acid (Asclepic acid) 是来自 Rhodopseudomonas capsulate 的抗病毒提取物,是 Rhodopseudomonas capsulate 的主要活性成分,cis-Vaccenic acid 可用作潜在的胎儿血红蛋白诱导剂。 | |||
T0744 |
10-Undecenoic acid zinc salt
Zinc diundec-10-enoate,Zinc 10-undecenoate,Zinc undecylenate,十一烯酸锌 |
Antibiotic; Antifungal | Microbiology/Virology |
10-Undecenoic acid zinc salt (Zinc undecylenate) 是一种天然的或合成的抗真菌脂肪酸, 在乳膏中可局部用于治疗湿疹、真菌感染、癣和其他皮肤病。 锌具有收敛作用。 | |||
T8271 |
10Z-Nonadecenoic acid
|
Endogenous Metabolite | Metabolism |
10Z-Nonadecenoic acid 是一种长链脂肪酸,具有抗肿瘤特性。 | |||
TN2295 |
Vicenin-1
Vicenin -1 |
Antioxidant; Angiotensin-converting Enzyme (ACE) | Metabolism; oxidation-reduction |
Vicenin-1 (Vicenin -1) 是一种来自豆科植物胡卢巴种子中分离出来的类黄酮糖苷,具有强大的抗炎和抗氧化活性,抑制血管紧张素转换酶 (ACE) 。 | |||
T17214 |
Valencene
NSC 148969,NSC-148969,NSC148969 |
Others; Antioxidant; NF-κB | NF-κB; Others; oxidation-reduction |
Valencene (NSC-148969) 是一种从 Cyperus rotundus 中分离出来的倍半萜类化合物,是柑橘类水果和柑橘类衍生气味的香气成分。ValenceneValencene 具有抗过敏、抗炎、抗黑色素生成、和抗氧化活性。通过阻断 NF-κB 通路,Valencene 通过阻断 NF-κB 通路抑制 Th2 趋化因子和促炎性趋化因子的过度表达。 | |||
TN2981 | 3-Phenyl-1,2-dihydroacenaphthylene-1,2-diol | Others | Others |
3-Phenyl-1,2-dihydroacenaphthylene-1,2-diol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2981,CAS号为 193892-33-0。 | |||
T38658 | 3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione | ||
3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione, also known as an anthraquinone, has been specifically extracted from Rubia cordifolia. | |||
T81504 |
Peucenin 7-O-methyl ether
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"Peucenin 7-O-methyl ether"是从Rosa rugosa的花中提取的一种天然产物。 | |||
TN2992 |
(3S,7S)-5,6-Dehydro-4''-de-O-methylcentrolobine
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Others | Others |
(3S,7S)-5,6-Dehydro-4''-de-O-methylcentrolobine is a natural product from Alpinia blepharocalyx. | |||
TN1577 |
Dicentrine
荷苞牡丹碱,荷包牡丹碱 |
Others | Others |
Dicentrine, a selective α±(1)-adrenoceptor antagonist with potent antiarrhythmic and antihypertensive activities, it also has antinociception in different models of chemical pain. | |||
T75560 | 4(1H)-Quinolinone, 1-methyl-2-(5Z)-5-undecen-1-yl- | ||
4(1H)-Quinolinone, 1-methyl-2-(5Z)-5-undecen-1-yl- (化合物2) 是一种从蛇床子提取的喹诺酮类生物碱。该化合物对耐甲氧西林金黄色葡萄球菌(MRSA)表现出活性,其最小抑制浓度(MIC)值对ATCC 33591和ATCC 25923株分别为32 μg/mL和16 μM/mL。 | |||
T75507 | 1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone | ||
1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone 对幽门螺杆菌菌株 51 表现出有效的抗菌活性,MIC50 值和 MIC90 值分别为 22 µM 和 50 µM。该化合物展现了在研究胃及十二指肠溃疡方面的潜力。 | |||
TN6309 |
Heteropeucenin 7-methyl ether
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Heteropeucenin 7-methyl ether 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6309,CAS号为 26213-95-6。 | |||
T83134 |
Alterbrassicene B
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Alterbrassicene B,一种从甘蓝链格孢菌(Alternaria brassicicola)分离得到的抗癌化合物。 | |||
TN1559 |
Dehydrodicentrine
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AChR | Neuroscience |
Dehydrodicentrine showed strong acetylcholinesterase (AChE) inhibitory effects with the IC50 value of 2.98 μM. | |||
TN2793 | 2-Picenecarboxylic acid | Others | Others |
2-Picenecarboxylic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2793,CAS号为 118172-80-8。 | |||
TN6899 | 1-Octadecene | ||
1-Octadecene is a natural product. | |||
TN2217 |
Sophoflavescenol
槐苦参醇,槐黄醇 |
Others; Beta-Secretase; BACE; PDE; AChR; AChE | Metabolism; Neuroscience; Others |
Sophoflavescenol 是异戊烯基黄酮类化合物,能够抑制PDE5的活性,IC50=0.013 μM。它也抑制 RLAR,HRAR,BACE1,AChE 和 BChE,IC50值分别为 0.30 µM,0.17 µM,10.98 µM,8.37 µM 和 8.21 µM。 | |||
T79977 |
Maceneolignan A
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Maceneolignan A,一种可从肉豆蔻(肉豆蔻科)假种皮分离的天然产品,有能力抑制RBL-2H3细胞内β-己糖胺酶释放,其IC50值为48.4 μM。同样,Maceneolignan A对抗原激活的RBL-2H3细胞中TNF-α释放的抑制作用,其IC50为63.7 μM。 | |||
T82747 |
Centellasaponin A
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Centellasaponin A (compound 10)为五环三萜皂苷类化合物,可通过积雪草甲醇提取物进行分离提取。 | |||
TN6057 |
1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone
(Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one |
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(Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one shows strong inhibitory activity on leukotriene biosynthesis in human polymorphonuclear granulocytes, and it is very effective against mycobacteria. | |||
TN3837 |
Desmethoxycentaureidin
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Others | Others |
Desmethoxycentaureidin shows high inhibitory activity against HeLa cell growth (GI50 9 microM). | |||
TN4058 |
Filicenol B
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Others | Others |
Filicenol B is a natural product from Adiantum lunulatum. | |||
TN4010 |
Erythrocentaurin
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Antifection | Microbiology/Virology |
Erythrocentaurin has antibacterial activity; it also exhibits a concentration-dependent α-amylase inhibition (IC(50) 1.67 ± 0.28 mg/mL). | |||
TN3621 |
Centrolobol
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Caspase | Apoptosis; Proteases/Proteasome |
(-)-Centrolobol has antifibrotic activity, it can significantly inhibit the proliferation of HSC-T6 cells in a dose-dependent manner. Centrolobol exhibits strong cytotoxic activity against KB cell line. | |||
T81908 |
Lucenin 1
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Lucenin-1为一种黄酮类化合物,可从Erucaria microcarpa Boiss (小叶芥菜) 地上部分提取。 | |||
TN6168 | Teuvincenone B | ||
Teuvincenone B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6168,CAS号为 127419-64-1。 | |||
T78467 |
trans-10-Heptadecenoic acid
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trans-10-Heptadecenoic acid 是一种能在特定酶作用下参与生物合成与代谢过程的反式脂肪酸。在 2,4-二烯酰基-CoA 还原酶与 Delta3,Delta2-烯酰基-CoA 异构酶催化下,trans-10-Heptadecenoic acid 可合成聚羟基链烷酸酯。当缺乏 2,4-二烯酰基-CoA 还原酶时,该化合物则经由多功能酶 (MFE) 中的烯酰辅酶 A 水合酶 II 进行降解。此外,trans-10-Heptadecenoic acid 能通过还原酶依赖性与直接 MFE 依赖性途径引起细胞内的碳外流。 | |||
TN1764 |
Incensole acetate
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TNF; NF-κB | Apoptosis; NF-κB |
Incensole acetate is a novel anti-inflammatory compound that inhibits NF-κB activation. | |||
TN6843 |
1-Hexadecene
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1-Hexadecene is a natural product. | |||
TN6906 |
1-Pentadecene [Standard Material for GC]
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1-Pentadecene [Standard Material for GC] is a natural product. | |||
T34931 |
Trichodecenin II
Trichodecenin-II,4-Decenoyl-gly-gly-leu-aib-gly-leu-lol |
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Trichodecenin II is a peptaibol isolated from Trichoderma viride. | |||
T81907 | Lucenin 3 | ||
Lucenin 3,一种生物活性类黄酮,具备生物医学领域内的功能性特性。 | |||
T32979 | Lushanrubescensin E | ||
Lushanrubescensin E is a bioactive chemical. | |||
T75499 | Maceneolignan H | ||
Maceneolignan H (Compound 8)是一种新的木脂素化合物,从肉豆蔻假种皮中分离而来。它表现为选择性CCR3拮抗剂(EC50=1.4 μM),具有研究过敏性疾病潜力。 | |||
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