1068
333
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10242 |
ACT-389949
|
Others | Others |
ACT-389949 是一种高效的甲酰肽受体 2/脂蛋白 A4 受体(FPR2)/(ALX)选择性激动剂,对 FPR2/ALX 进行内化入单核细胞的EC50值为 3 nM。它对炎性疾病具有潜在的研究价值。 | |||
T26559 |
ACT-462206
|
OX Receptor | GPCR/G Protein; Neuroscience |
ACT-462206 是一种可口服且可穿过血脑屏障的Orexin 1/Orexin 2 受体拮抗剂。ACT-462206 具有高效性,可用于研究睡眠和焦虑。 | |||
T14119 |
ACT-678689
Compound Example 1.53.4 |
Hydroxylase | Metabolism |
ACT-678689 (Compound Example 1.53.4) 是一种色氨酸羟化酶 (TPH) 抑制剂,IC50=8 nM。 | |||
T9149 |
2BAct
2B-Act,2B Act |
PERK | Apoptosis |
2BAct 是一种具有口服活性的高选择性真核起始因子eIF2B 活化剂,EC50为 33 nM。它可防止由慢性综合应激反应引起的神经系统缺陷。 | |||
T14924 |
Cenerimod
ACT-334441 |
S1P Receptor | GPCR/G Protein |
Cenerimod (ACT-334441) 是一种具有口服活性、选择性和高效性的磷酸鞘氨醇 1 受体(S1P1)激动剂(EC50:1 nM)。Cenerimod 对多种 S1P 的亚型具有抑制作用,可用于研究鼠类实验性自身免疫性脑脊髓炎 (EAE)和鼠类硬皮病。 | |||
T2058 |
Palosuran
ACT-058362 |
GPR | Endocrinology/Hormones; GPCR/G Protein |
Palosuran (ACT-058362) 是人类 UT 受体的新型强效特异性拮抗剂,对表达人重组受体的 CHO 细胞膜的IC50值为 3.6 nM。它可改善糖尿病大鼠的胰腺和肾脏功能。 | |||
T40542 |
Sinbaglustat
ACT-519276,Sinbaglustat,OGT2378 |
Transferase | Metabolism |
Sinbaglustat (OGT2378) (OGT2378) 是葡萄糖神经酰胺合成酶 (GCS) 和非溶酶体葡萄糖神经酰胺酶 (GBA2) 的双重抑制剂。Sinbaglustat 是一种可透过血脑屏障的的口服N-烷基亚氨基糖。Sinbaglustat 可用于治疗溶酶体贮积症和研究溶酶体功能障碍相关的中枢神经退行性疾病。 | |||
T3258 |
Ponesimod
ACT-128800 |
S1P Receptor; LPL Receptor | GPCR/G Protein |
Ponesimod (ACT-128800) 是一种选择性 S1P1可口服激动剂,在放射性配体结合试验中的 IC50值为 6 nM。它可高效激活 S1P1介导的信号转导,EC50为5.7 nM。它可预防淋巴细胞介导的组织炎症,具有潜在的免疫调节活性。 | |||
T4689 |
Palosuran hydrochloride 540769-28-6(free base)
ACT-058362 hydrochloride |
GPR | Endocrinology/Hormones; GPCR/G Protein |
Palosuran hydrochloride 540769-28-6(free base) (ACT-058362 hydrochloride) 是一种新型强效特异性人 UT 受体拮抗剂,IC50 为 3.6±0.2 nM。 | |||
T26557 |
ACT-209905
ACT 209905,ACT209905 |
||
ACT-209905 is an agonist of S1P1 receptor. | |||
T4020 |
Cadazolid
ACT-179811,卡达唑利德 |
Antibacterial; Antibiotic | Microbiology/Virology |
Cadazolid (ACT-179811) 是一种新型恶唑烷酮类抗生素,对Clostridium difficile 有活性。 | |||
T2561 |
Macitentan
马西替坦,ACT-064992 |
Apoptosis; Endothelin Receptor | Apoptosis; GPCR/G Protein |
Macitentan (ACT-064992) 是一种内皮素受体拮抗剂,用于治疗肺动脉高压。 | |||
T35623 |
ACT-373898
|
||
ACT-373898 is a metabolite of the endothelin (ET) receptor type A (ETA) and ETBdual antagonist macitentan .1 1.Dingemanse, J., Sidharta, P.N., Maddrey, W.C., et al.Efficacy, safety and clinical pharmacology of macitentan in comparison to other endothelin receptor antagonists in the treatment of pulmonary arterial hypertensionExpert Opin. Drug Saf.13(3)391-405(2013) | |||
T2613 |
Almorexant
阿莫伦特,ACT 078573 |
OX Receptor | GPCR/G Protein; Neuroscience |
Almorexant (ACT 078573) 是一种有效的竞争性食欲素 1 受体 (OX1)/食欲素 2 受体 (OX2) 双重拮抗剂,OX1 和 OX2 的 Ki 值分别为 1.3 和 0.17 nM。 | |||
T3520 |
Setipiprant
KYTH-105,塞替匹仑,ACT-129968 |
GPR; Prostaglandin Receptor | Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation |
Setipiprant (ACT-129968) 是一种口服的选择性 CRTH2 拮抗剂,IC50为6.0 nM。 | |||
T70616 |
ACT-672125
|
||
ACT-672125 is a Potent CXCR3 Antagonist with Therapeutic Potential in Autoimmune Diseases. ACT-672125 showed good physicochemical properties and safety profile. In a proof-of-mechanism model of lung inflammation, ACT-672125 inhibited the recruitment of CXCR3 expressing T cells into the inflamed lung in a dose-dependent manner. | |||
T3216 |
Selexipag
NS-304,ACT-293987,赛乐西帕,Uptravi |
Others; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Others |
Selexipag (ACT-293987) 是前列环素受体激动剂,可引起肺血管舒张,用于治疗肺动脉高压。 | |||
T70475 | ACT-280778 | ||
ACT-280778 is a potent L/T calcium channel blocker. | |||
T14123 |
ACT 178882
|
RAAS | Endocrinology/Hormones |
ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM). | |||
T21850 |
ACT 335827
|
||
ACT-335827 是一种可口服的、脑渗透性 orexin 1 型 (orexin type 1) 受体选择性拮抗剂。ACT-33582 作用于 OXR1 和 OXR2 的 IC50值分别是 6 nM 和 417 nM。ACT-33582 可用于神经系统疾病的相关研究。 | |||
T14120 |
ACT-709478
|
Others | Others |
ACT-709478 is a potent, selective T-type calcium channel blocker that is orally active and capable of penetrating the brain. It is currently utilized in research focusing on generalized epilepsies[1]. | |||
T39665 |
ACT-1004-1239
|
||
ACT-1004-1239 is a highly potent and selective antagonist of CXCR7, which can be administered orally. It exhibits an impressive inhibitory concentration (IC50) value of 3.2 nM. | |||
T71363 | ACT-281959 | ||
ACT-281959, a prodrug of ACT-246475, is a novel potent and selective P2Y12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel. ACT-281959 showed antithrombotic efficacy after oral administration in the rat ferric chloride model. ACT-281959 entered clinical studies in healthy volunteers. | |||
T26558 |
ACT-387042
ACT387042 |
||
ACT-387042 is a Bacterial Topoisomerase Inhibitor, it has broad-spectrum activity against Gram-positive and Gram-negative bacteria. | |||
T23625 |
ACT-451840
ACT451840 |
||
ACT-451840 is a drug of antimalarial activity. It has effective activity against sensitive and resistant Plasmodium falciparum strains. | |||
T7817 |
Aprocitentan
ACT-132577,N-[5-(4-溴苯基)-6-[2-[(5-溴-2-嘧啶基)氧基]乙氧基]-4-嘧啶基]氨基磺酰胺 |
Endothelin Receptor | GPCR/G Protein |
Aprocitentan (ACT-132577) 是一种 Macitentan 的主要活性代谢物。它是 ETA/ETB 的双重拮抗剂,其 pA2值分别为 6.7 和 5.5,IC50分别为 3.4 nM 和 987 nM。 | |||
T73148 |
ACT-777991
|
||
ACT-777991为一种选择性、口服生效的CXCR3拮抗剂,于动物模型中展现出微粒体及肝细胞稳定性,能抑制活化T细胞向CXCL11迁移。 | |||
T63761 | ACT-660602 | ||
ACT-660602 是口服具有活力的趋化因子受体 CXCR3 拮抗剂 (IC50: 204 nM)。ACT-660602 能够抑制 T 细胞迁移,并在体内急性肺损伤模型中显示出显著作用。ACT-660602 能够用于研究自身免疫性疾病。 | |||
T73100 |
ACT-606559
|
||
ACT-606559,ACT451840的一种代谢物,为新型抗疟活性化合物,可用于研究疟疾。 | |||
T77442 |
Glenzocimab
ACT017 |
Others | Others |
Glenzocimab (ACT017) 是人源化抗 GPVI 单克隆抗体的 Fab 片段。Glenzocimab 在缺血性卒中模型对胶原诱导的血小板聚集显示出抑制作用。Glenzocimab 具有研究急性缺血性脑卒中和脑血栓。 | |||
T24478 |
MK-8141
MK 8141,ACT 077825,ACT077825,ACT-077825 |
||
MK-8141 is a renin inhibitor. It displays some antihypertensive efficacy in hypertensive patients. | |||
T10351 |
Aprocitentan D4
ACT-132577 D4 |
Others | Others |
Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5). | |||
T11934 |
Macitentan-d4
Macitentan D4,ACT-064992 D4 |
Endothelin Receptor | GPCR/G Protein |
Macitentan-d4 (ACT-064992 D4) 是一种 Macitentan 氘代物,可被当作非多肽 ETA 和 ETB (内皮素受体)双拮抗剂。Macitentan-d4 比 Macitentan 毒性更低,半衰期更长,可用于研究由内皮素受体介导介导的疾病。 | |||
T6155 |
Almorexant hydrochloride
ACT-078573 hydrochloride,Almorexant HCl |
OX Receptor | GPCR/G Protein; Neuroscience |
Almorexant hydrochloride (ACT-078573 hydrochloride) 是一种有效的竞争性食欲素 1 受体(OX1)/食欲素 2 受体 (OX2) 双重拮抗剂,OX1 和 OX2 的 Ki 值分别为 1.3 和 0.17 nM。 | |||
T70474 |
Gallamine
|
||
Gallamine is an allosteric antagonist at muscarinic M2 acetylcholine receptors and an inhibitor of acetylcholinesterase. | |||
T70614 |
SLR080811 HCl
|
||
SLR080811 is a SphK inhibitor. Sphingosine-1-phosphate (S1P) is a ubiquitous, endogenous small molecule that is synthesized by two isoforms of sphingosine kinase (SphK1 and 2). Intervention of the S1P signaling pathway has attracted significant attention because alteration of S1P levels is linked to several disease states including cancer, fibrosis, and sickle cell disease. | |||
T71361 | CHS-828 nicotinate | ||
CHS-828 nicotinate is a CHS-828 salt with Nicotinic acid.. CHS-828 also known as GMX-1778, is a potent and selective NAMPT inhibitor. CHS-828 inhibits cellular synthesis of NAD. CHS 828 kill tumour cells by inhibiting the nuclear factor-kappaB translocation but unlikely through down-regulation of proteasome. CHS 828 has shown promising anticancer activity in experimental tumor models and primary cultures of cancer cells from patients. CHS 828 showed a synergistic effect with melphalan in 67%, ... | |||
T7744 |
Piperaquine tetraphosphate tetrahydrate
4,4'-(1,3-丙烷双-4,1-哌嗪基)双(7-氯喹啉)磷酸盐水合物,四磷酸哌喹四水合物 |
Parasite | Microbiology/Virology |
Piperaquine tetraphosphate tetrahydrate 是一种双喹啉抗寄生虫剂,可与青蒿素联用研究抗疟。 | |||
T71362 |
GCC-4401C free base
|
||
GCC-4401C free base is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE). | |||
T7532 |
Piperaquine
|
Parasite | Microbiology/Virology |
Piperaquine 是一种双喹啉化合物,可抑制来自疟疾感染患者的恶性疟原虫分离株的离体生长,IC50 范围为 11.8-217.3 nM。 | |||
T6179 |
Moxalactam sodium salt
Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy |
Antibacterial; Antibiotic | Microbiology/Virology |
Moxalactam sodium salt (LY-127935) 是一种抗生素, 对大肠杆菌和绿脓杆菌有作用。 | |||
T0299 |
Lactitol monohydrate
D-Lactitol monohydrate,单水合乳糖醇 |
Others | Others |
Lactitol monohydrate (D-Lactitol monohydrate) 是一种乳果糖的糖类似物,是一种糖醇,用作替代甜味剂。有用于便秘和肝性脑病的研究潜力。。 | |||
TP1106L |
α-Factor Mating Pheromone, yeast acetate
Mating Factor α acetate,α-Factor Mating Pheromone, yeast acetate(59401-28-4 free base) |
Others | Others |
α-Factor Mating Pheromone, yeast acetate (Mating Factor α acetate)(59401-28-4 free base) 是由酿酒酵母α细胞分泌的13个氨基酸的肽。 | |||
T3189 |
B7/CD28 interaction inhibitor 1
CTLA-4 inhibitor |
Others | Others |
B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。 | |||
T10674 |
Potassium Channel Activator 1
钾离子通道激活剂1,ZINC34634569 |
Potassium Channel | Membrane transporter/Ion channel |
Potassium Channel Activator 1 可用于治疗多巴胺能系统被破坏的疾病或病症的研究,例如情绪障碍 ADHD、精神分裂症和其他精神病状态。 | |||
T37192 |
4-Methylumbelliferyl-α-D-Galactopyranoside
4MU-α-Gal |
Others | Others |
4-Methylumbelliferyl-α-D-Galactopyranoside (4MU-α-Gal) (4-MU-α-Gal)是α-半乳糖苷酶的荧光底物。除了用于表征新的α-半乳糖苷酶外,4-MU-α-Gal 还用于评估与法布里病相关的α-半乳糖糖苷酶活性的缺乏。 | |||
T60000 | STING (WT/R232) activity regulator 126 | STING | Immunology/Inflammation |
STING (WT/R232) activity regulator 126 是一种具有抗菌和抗病毒作用的 STING 调节剂。 | |||
T9501 |
Enterobactin
Enterochelin |
Others | Others |
Enterobactin (Enterochelin) 是一种高亲和力铁载体,可为微生物系统获取铁。 | |||
T7627L |
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA(4037-01-8(free base)),Acth (4-10) |
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) 是一种有效的黑皮质素 (MC4R) 受体激动剂。 | |||
TP1245L |
ACTH 4-11 acetate
ACTH 4-11 acetate (67224-41-3 Free base) |
Others | Others |
ACTH 4-11 acetate 是一种促肾上腺皮质激素片段,具有与 α-黑素细胞刺激素 (MSH) 相同的氨基酸序列。 ACTH 4-11 acetate 仅在高剂量时表现出微弱的 MSH 效力。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3S2007 |
MRE-269
3-氧代-12-烯-28-乌苏酸,MRE 269,ACT-333679,MRE269 |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
MRE-269 (ACT-333679) 是一种口服的长效前列环素受体激动剂前药,是 Selexipag 的活性代谢物,用于治疗肺动脉高压。 | |||
T10943 |
D-(-)-Lactic acid
(R)-2-Hydroxypropionic acid,D-乳酸 |
Others; Endogenous Metabolite | Metabolism; Others |
D-(-)-Lactic acid 是糖发酵(氧化、代谢)中的一种正常中间体。它被鉴定为植物中 ProDH(脯氨酸脱氢酶)的竞争性抑制剂。 | |||
T2833 |
Dehydrocostus Lactone
Epiligulyl oxide,去氢木香内酯,(-)-Dehydrocostus lactone,去氢木香烃内酯 |
IκB/IKK | NF-κB |
Dehydrocostus Lactone ((-)-Dehydrocostus lactone) 是一种倍半萜内酯,从云木香中分离得到。 | |||
T6520 |
Grape Seed Extract
Grape Seed P.E.,葡萄籽提取物 |
Apoptosis; Others | Apoptosis; Others |
Grape Seed Extract (Grape Seed P.E.) 是葡萄植物 Vitis vinifera 的种子分泌物,能诱导人类结肠直肠癌细胞凋亡,具有抗炎和抗增殖作用。它对脂肪代谢酶、胰脂肪酶和脂蛋白脂肪酶有抑制作用。 | |||
T5S0167 |
Atractylenolide I
白术内酯 I,白术内酯I;苍术内酯I |
IL Receptor; TNF; TLR; JAK; STAT | Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells |
Atractylenolide I 是从白术根中得到的一种倍半萜烯,具有神经保护、抗过敏、抗炎和抗癌等多种生物活性。它是一种TLR4拮抗剂,在 A375 细胞中,能够降低JAK2和STAT3的磷酸化水平。 | |||
T35709 |
N-acetyl-D-Lactosamine
N-Acetyllactosamine |
Endogenous Metabolite | Metabolism |
N-acetyl-D-Lactosamine (N-Acetyllactosamine) 是一种由半乳糖和N-乙酰葡萄糖组成的二糖,是各种寡糖的重要组成部分,可作为合成各种寡糖的起始材料。N-acetyl-D-Lactosamine 可能被都当作一种结构元素自然出现在各种糖结合物中,也可用于表征凝集素,具有益生元的作用。 | |||
T8085 |
(-)-Corey lactone diol
科立内脂二醇,Corey Lactone Diol |
Others | Others |
(-)-Corey lactone diol 是 corey aldehyde 的还原形式,也是化学合成中的砌块。 | |||
T20255 |
L-Galactose
Galactose, L- |
Endogenous Metabolite | Metabolism |
L-Galactose (Galactose, L-) 是一种天然产物,广泛存在动植物体内。L-Galactose 在Pistia stratiotes 中被证明是D-葡萄糖转化为草酸的分子途径中的关键中间体。 | |||
T3999 |
D(+)-Galactosamine hydrochloride
D-半乳糖胺盐酸盐,D-氨基半乳糖盐酸盐,D-Galactosamine HCl |
Others | Others |
D(+)-Galactosamine hydrochloride (D-Galactosamine HCl) 是一种被证实的实验毒素,它能够产生自由基及UTP 核苷酸的消耗导致肝损伤,中毒剂量会造成肾功能不全,而肾功能衰竭通常和终末期肝损伤有关。脂多糖/D-Galactosamine 诱导的急性肝损伤是一种已知的暴发性肝衰竭动物模型。 | |||
TN7021 |
Ent-toddalolactone
|
Others | Others |
Ent-toddalolactone 是一种天然化合物,属于香豆素类,来源于两面针,具有抗炎、抗癌活性。 | |||
T1353 |
DL-Mevalonolactone
甲瓦龙酸内酯,Mevalonolactone |
Others; Endogenous Metabolite | Metabolism; Others |
DL-Mevalonolactone (Mevalonolactone),一种人内源性代谢物,是甲羟戊酸的 δ-lactone 形式,甲羟戊酸途径的一个前体。它能够降低大脑中线粒体膜电位(∆Ψm),Ca2+的保留能力和 NAD (P) H 的含量 , 而且还诱导线粒体肿胀。 | |||
T4845 |
L-Lactic acid
2-HYDROXYPROPIONIC ACID,L-乳酸,L-(+)-Lactic acid,(S)-2-Hydroxypropanoic acid |
Endogenous Metabolite; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology |
L-Lactic acid ((S)-2-Hydroxypropanoic acid) 属于天然产物,由丙酮酸的无氧糖酵解产生。L-Lactic acid 是组织缺氧的敏感指标,可作为危重病人的血流动力学指标。 | |||
TJO2795 |
D-Galacturonic acid hydrate
D-(+)-Galacturonic acid,D-半乳糖醛酸 |
Others; Endogenous Metabolite | Metabolism; Others |
D-Galacturonic acid hydrate 是内源性代谢产物的一种。 | |||
T0591 |
D-Galactose
D-(+)-Galactose,alpha-D-半乳糖,D-半乳糖,D-Galactopyranose,Alpha-D-galactose |
Endogenous Metabolite | Metabolism |
D-Galactose (Alpha-D-galactose) 是一种天然的己糖,是葡萄糖的C-4差向异构体。 | |||
T13827 |
Pronase E (Activity ≥ 7000 U/g)
Pronase,Pronase E |
Others | Others |
Pronase E 是一种蛋白水解酶混合物,从灰色链霉菌 (Streptomyces griseus) 中获得,能够将蛋白质消化成单个氨基酸。 | |||
TN6700 |
gamma-Nonanolactone
|
Others | Others |
gamma-Nonanolactone 是蒸小麦的香气成分。 | |||
T6102 |
2'-acetylacteoside
|
Antioxidant; Reductase | Endocrinology/Hormones; Metabolism; oxidation-reduction |
2'-Acetylacteoside 是一种苯乙醇苷类化合物,分离自来江藤中,可抑制自由基诱导的红细胞溶血,具有清除自由基的作用。 | |||
T6528 |
Gynostemma Extract
Gypenoside IX,七叶胆皂甙,Gypenoside,Gynostemma Pentaphyllum,绞股蓝提取物,Notoginsenoside Fd,Ginsenoside C-Mx1,Gynosaponin I |
Others; Endogenous Metabolite | Metabolism; Others |
Gynostemma Extract (Gypenoside IX) 是一种天然产物。 | |||
T1262 |
Tazobactam
Tazobactamum,Tazobactam acid,他唑巴坦酸,YTR-830H,CL-298741,他唑巴坦 |
Antibacterial; Antibiotic | Microbiology/Virology |
Tazobactam (YTR-830H) acid 是一种具有抗菌活性的β-内酰胺酶抑制剂。 | |||
T8078 |
Gamma-decalactone
Decan-4-olide,γ-Decalactone,丙位癸内酯 |
Others | Others |
Gamma-decalactone (Decan-4-olide) 是一种具有果味桃子味的食品添加剂。蓖麻油酸 (12-羟基-十八烷基-9-烯酸) 常作为 γ-Decalactone 的生产过程中的底物。 | |||
T125211 |
Deoxy euphorbia factor L1
|
Others | Others |
Deoxy euphorbia factor L1是一种天然产物,存在于植物续随子 Euphorbia lathyris L 的种子中。 | |||
T4S0592 |
Toddalolactone
(+)-Toddalolactone,飞龙掌血内酯,毛两面针素 |
PAI-1 | Metabolism |
Toddalolactone ((+)-Toddalolactone) 是一种Toddalia asiatica 的主要成分,能够抑制重组人纤溶酶原激活物抑制物-1(PAI-1)的活性, IC50=37.31 μM。 | |||
T5663 |
α-Lactose
D-乳糖单水合物,Lactose |
Others | Others |
α-Lactose 是牛奶中的主要的糖。它一般以 α 和 β 两个异构体的形式存在,其中α 形式通常以一水合物的形式结晶。 | |||
TN6744 |
Undecanoic gamma-lactone
|
Others | Others |
Undecanoic gamma-lactone 是一种天然产物。 | |||
T3384 |
Wedelolactone
蟛蜞菊内酯,IKK Inhibitor II |
Apoptosis; NF-κB; Lipoxygenase; Caspase | Apoptosis; Metabolism; NF-κB; Proteases/Proteasome |
Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物,通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录,具有抗癌,抗炎和抗氧化活性。 | |||
T5798 |
Euphorbia Factor L2
千金子素L2,euphorbiafactor L2,大戟因子L2 |
Apoptosis; NF-κB | Apoptosis; NF-κB |
Euphorbia Factor L2 是从大戟种子中分离得到的一种赤藓烷二萜,显示强烈的细胞毒性并通过线粒体途径诱导细胞凋亡,具有抗癌活性。 | |||
T2S0410 |
Euphorbia factor L1
Euphorbiasteroid,大戟因子L1,大戟因子 L1 |
Apoptosis; P-gp | Apoptosis; Membrane transporter/Ion channel; Neuroscience |
Euphorbia factor L1 (Euphorbiasteroid) 可降低 Bcl-2,PI3K,AKT 和 mTOR 蛋白和 mRNA 水平,上调 caspase-9 and caspase-3 蛋白水平。它可诱导自噬,具有抗癌、抗脂肪生成、抗破骨细胞生成和多重耐药调节作用。 | |||
T7933 |
D(+)-LACTIDE
|
Others | Others |
D(+)-LACTIDE 是丙酮的环状二聚体,用于合成各种药物和其他化合物,也可用于生物化学和生理学研究。 | |||
TN1106 |
Cyanidin-3-O-galactoside chloride
Ideain chloride |
Antioxidant | oxidation-reduction |
Cyanidin-3-O-galactoside chloride (Ideain chloride)是从山楂果皮 (EPHF)中提取的小分子化合物,具有抗氧化和抗肿瘤作用,可用于研究肥胖。 | |||
T8064 |
Lactobionic acid
|
Others; Antibacterial | Microbiology/Virology; Others |
Lactobionic acid 是在里海酸奶中的一种仿生酸,化学上由与半乳糖键合的葡萄糖酸组成。它是具有抗氧化、抗菌和保湿特性的乳糖酸。 | |||
T0799 |
Lactulose
Duphalac,4-O-β-D-Galactopyranosyl-D-fructose,D-Lactulose,Lactulosum,乳果糖 |
Others | Others |
Lactulose (Lactulosum) 是一种不易吸收的糖,一般给药 8 到 12 小时后开始发挥药效,但可能需要两天时间改善便秘。它可用于便秘和肝性脑病的研究。 | |||
T0933 |
D-(+)-Glucono-1,5-lactone
Gluconic acid lactone,Delta-Gluconolactone,Gluconolactone,葡萄糖酸内酯 |
Others; Reactive Oxygen Species; Endogenous Metabolite | Immunology/Inflammation; Metabolism; NF-κB; Others |
D-(+)-Glucono-1,5-lactone (Gluconolactone) 是聚羟基酸,可螯合金属离子,具有保湿、抗氧化特性。 | |||
T5742 |
Isodemethylwedelolactone
异去甲蟛蜞菊内酯,Isodemethylwedelolacton |
Others | Others |
Isodemethylwedelolactone (Isodemethylwedelolacton) 是一种促凝剂,也是溶血性成分,分离自 Eclipta alba。 | |||
T4708 |
D-N-Acetylgalactosamine
D-GalNAc,N-Acetyl-D-galactosamine,N-乙酰-D-半乳糖胺 |
Others; Endogenous Metabolite | Metabolism; Others |
D-N-Acetylgalactosamine (N-Acetyl-D-galactosamine) 是脑杂多糖(糖蛋白)的重要组成部分。 | |||
T8098 |
γ-Hexalactone
γ-caprolactone,gamma-己内酯,γ-己内酯 |
Others | Others |
γ-Hexalactone (γ-caprolactone) 是一种存在成熟水果中的 gamma 内酯。它会导致 DNA 损伤,可用作对氧磷酶 1 的底物 (PON1)。 | |||
T3234 |
Dihydroactinidiolide
R-(-)Dihydro actinidiolide,二氢猕猴桃内酯 |
Others | Others |
Dihydroactinidiolide (R-(-)Dihydro actinidiolide) 是一种植物生长抑制剂,也是基因表达的调节剂,存在于植物叶片和果实中,能够负责拟南芥中的光适应。它具有抗氧化活性,抗菌活性,抗癌活性和神经保护作用。 | |||
TN1634 |
Euphorbia factor L7b
千金子素L7B |
Others | Others |
Euphorbia factor L7b 是从大戟属植物大戟中提取的天然产物。 | |||
T3S1227 |
Aristolactam I
Aristolactam,Aristololactam I,马兜铃内酰胺I,Aristololactum |
Apoptosis; Caspase | Apoptosis; Proteases/Proteasome |
Aristolactam I (Aristololactum) 是马兜铃酸 I (AA-I) 的主要代谢产物,参与导致肾损伤的过程。它具有细胞毒性,通过诱导半胱天冬酶 3 依赖性途径中的细胞凋亡介导。 | |||
T1683 |
Actriol
异雌三醇,Epiestriol |
Glucocorticoid Receptor | Endocrinology/Hormones |
Actriol (Epiestriol) 是内源性雌激素雌酮的代谢物,拥有抗炎及抗菌活性。 | |||
TN6796 |
2'-FUCOSYLLACTOSE
2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖 |
Others | Others |
2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) 是一种含岩藻糖的寡糖。 | |||
TN2539 |
1beta-Hydroxyalantolactone
|
IL Receptor; TNF | Apoptosis; Immunology/Inflammation |
1beta-Hydroxyalantolactone 是从药用植物大英花的花头中分离出的小分子化合物,可抑制细胞中TNF-α、IL-17、IFN-γ的表达,促进TNF-α、IFN-γ、IL-17的分泌,可防治类风湿性关节炎。 | |||
T20576 |
Lactitol
NSC 231323,Lactit,D-Lactitol,NSC231323,乳糖醇,NSC-231323,Lactosit Miruhen |
Others | Others |
Lactitol (Lactit) 是一种乳果糖的糖类似物, 是一种糖醇,可用作甜味剂的替代品。有用于便秘和肝性脑病研究的潜力。 | |||
T5578 |
L-Gulono-1,4-lactone
|
Others; Endogenous Metabolite | Metabolism; Others |
L-Gulono-1,4-lactone 是一种 L-古洛糖酸-γ-内酯氧化还原酶的作用底物,该酶能促进维生素 C 合成的末步。它是动物、植物和一些原生生物中维生素 C 的直接前体。 | |||
TN6718 |
Dehydrocostuslactone
|
Others | Others |
Dehydrocostuslactone 是一种从奥克兰提取的天然产物。它具有广泛的生物作用,包括抗炎、抗癌、抗病毒、抗菌、抗真菌、抗氧化、抗糖尿病、抗溃疡和驱虫活性。 | |||
T4455 |
DL-3-Phenyllactic acid
DL-3-苯乳酸,3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid |
Others; Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology; Others |
DL-3-Phenyllactic acid (3-Phenyllactic acid) 是广谱抗菌化合物,对细菌和真菌具有活性。 | |||
T3902 |
Atractylenolide III
白术内酯 III,ICodonolactone,8β-Hydroxyasterolide |
Apoptosis | Apoptosis |
Atractylenolide III (ICodonolactone) 是白术根茎主要成分,通过诱导细胞色素 c 的释放、上调 Bax 的表达和易位凋亡诱导因子,是治疗人肺癌的潜力。 | |||
T3791 |
Atractyloside A
|
AChR | Neuroscience |
Atractyloside A 是存在于一些植物中的贝壳杉类二萜糖苷,具有降血压、降血糖、抗肿瘤等活性。 | |||
T0434 |
D-Glucuronic acid lactone
Glucuronolactone,D-Glucurone,Dicurone,葡醛内酯 |
Others; Endogenous Metabolite | Metabolism; Others |
D-Glucuronic acid lactone (Dicurone) 是内源性代谢产物的一种。 | |||
TN1823 |
Kaempferol 3-O-β-D-galactopyranoside
Kaempferol 3-O-beta-D-galactoside,Kaempferol-3-O-galactoside,三叶豆苷 |
Immunology/Inflammation related | Immunology/Inflammation |
Kaempferol 3-O-β-D-galactopyranoside 是黄酮类化合物的衍生物,分离自木樨状菌 (Consolida oliverana) 的地上部分。 | |||
T0586 |
Lactose
|
Others; Endogenous Metabolite | Metabolism; Others |
Lactose 是半乳糖和葡萄糖衍生的二糖,是大多数物种乳汁中的主要糖分,能够调节人类肠道的微生物菌群。 | |||
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