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Search Results for " trypsin "

70

抑制剂 & 化合物

9

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T3359	Aprotinin 抑酶肽,抑肽酶,Bovine Pancreatic Trypsin Inhibitor,Traskolan,Antilysin	Others; Serine Protease; Influenza Virus; Proteasome	Microbiology/Virology; Others; Proteases/Proteasome; Ubiquitination
	Aprotinin (Traskolan) 是分离自牛肺的一种广谱丝氨酸蛋白酶抑制剂，可抑制多种不同酯酶和蛋白酶的活性。
T76240	Urinary Trypsin Inhibitor Fragment
	Urinary Trypsin Inhibitor Fragment，一种通过蛋白水解生成的尿胰蛋白酶抑制剂片段，能通过有限蛋白水解抑制肿瘤细胞侵袭。
T8362	Benzamidine hydrochloride Benzamidine HCl,苄脒盐酸盐	Serine/threonin kinase; Serine Protease	Cell Cycle/Checkpoint; Metabolism; Proteases/Proteasome
	Benzamidine hydrochloride (Benzamidine HCl) 是可逆的胰蛋白酶样丝氨酸蛋白酶 (trypsin-like serine proteases) 竞争性抑制剂，对 uPA、类胰蛋白酶、胰蛋白酶和 Xa 因子作用的Ki 分别为 97 µM、20 µM、21 µM 和 110 µM。
T17011	TCH-165	Proteasome	Proteases/Proteasome; Ubiquitination
	TCH-165 是一种蛋白酶体组装的小分子调节剂，可增加游离 20S 水平，进而增强 IDP 蛋白水解。
T8802	2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- 2,4-Dioxaspiro[5.5]undec-8-ene, 3-(2-fur	Serine Protease	Proteases/Proteasome
	2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) 是胰蛋白酶抑制剂（人尿 urinastatin protein moiety），作为尿胰蛋白酶抑制剂（UTI），是一种从健康人尿液中分离或合成产生的糖蛋白。
T73594	Chymotrypsin Chymotrypsin A	Serine/threonin kinase	Cell Cycle/Checkpoint; Metabolism
	Chymotrypsin (Chymotrypsin A) 是胰腺产生的丝氨酸蛋白酶，可切割芳香族氨基酸羧基侧的蛋白质链。
TP2217	alpha-1 antitrypsin fragment	Others	Others
	Alpha-1 antitrypsin (A1AT) is known as a serum trypsin inhibitor and is a protease inhibitor belonging to the serpin superfamily. Alpha-1 antitrypsin is a single-chain glycoprotein consisting of 394 amino acids in the mature form and exhibits a number of
T76157	Chymotrypsinogen
	Chymotrypsinogen 是Chymotrypsin 的无活性前体。Chymotrypsinogen 是一种由胰腺产生的丝氨酸蛋白酶 (serine protease)。
TP2216	alpha-1 antitrypsin fragment 235-243 [Homo sapiens]/[Papio hamadryas]/[Cercopithecus aethiops]	Others	Others
	Protease inhibitor
T7016	VR23	Apoptosis; Proteasome; Caspase	Apoptosis; Proteases/Proteasome; Ubiquitination
	VR23 是一种蛋白酶体抑制剂，对胰蛋白酶样蛋白酶体、糜蛋白酶样蛋白酶体和半胱天冬酶样蛋白酶体的 IC50 分别是1 nM、50-100 nM 和3 μM。
T9670L	Patamostat HCl Patamostat HCl（114568-26-2 Free base）	Serine Protease; Protease	Proteases/Proteasome
	Patamostat HCl 是一种具有高效性和选择性的小分子蛋白酶 (protease) 抑制剂，对胰蛋白酶，纤溶酶和凝血酶有抑制作用，IC50 值分别为 39 nM，950 nM 和 1.9 μM。Patamostat HCl 可用于研究急性胰腺炎。
T74040	Boc-Gln-Ala-Arg-AMC hydrochloride
	Boc-Gln-Ala-Arg-AMC hydrochloride 是一种荧光化合物，可作为胰蛋白酶 (trypsin)的底物，也可用于测定 TMPRSS2 的蛋白水解活性。
T30519	BMS-363131 BMS363131,BMS 363131	Serine Protease	Proteases/Proteasome
	BMS-363131 (BMS363131) 是一种高效且具有选择性的胰蛋白酶抑制剂，IC50值 <1.7 nM。
T6370	AEBSF hydrochloride AEBSF HCl,Pefabloc SC	Thrombin; Serine Protease; Influenza Virus	Microbiology/Virology; Proteases/Proteasome
	AEBSF hydrochloride (Pefabloc SC) 是一种丝氨酸蛋白酶的不可逆抑制剂。
T6941	PI-1840 PI 1840	PARP; Proteasome	Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome; Ubiquitination
	PI-1840 是一种高效的、选择性的蛋白酶体chymotrypsin-like (CT-L)抑制剂，IC50=27nM。
T16169	N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride N-alpha-Tosyl-L-lysine_chloromethyl_ketone_hydrochloride	Others; Proteasome; COX	Immunology/Inflammation; Neuroscience; Others; Proteases/Proteasome; Ubiquitination
	N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride (N-alpha-Tosyl-L-lysine_chloromethyl_ketone_hydrochloride) 是胰蛋白酶样蛋白酶的抑制剂。 N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride 对 IFN-γ 活性具有抑制作用。
T2122	Ixazomib 艾沙佐米,MLN2238	Proteasome; Caspase; Autophagy	Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
	Ixazomib (MLN2238) 含硼肽蛋白酶体抑制剂(PI)，可抑制 20S 蛋白酶体的糜蛋白酶样蛋白水解 (β5) 位点，IC50为 3.4 nM，Ki 为 0.93 nM。它还抑制半胱天冬酶样 (β1) 和胰蛋白酶样 (β2) 蛋白水解位点，IC50值为 31和3500 nM。
T78409L	Boc-Val-Pro-Arg-MCA TFA
	Boc-Val-Pro-Arg-MCA TFA 是一种敏感性荧光底物，是凝血酶底物，可用于测定胰蛋白酶样丝氨酸蛋白酶活性。
T60248	4-Aminobenzamidine dihydrochloride p-Aminobenzamidine dihydrochloride	Serine Protease	Proteases/Proteasome
	4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) 是一种强胰蛋白酶 (trypsin)抑制剂，也是一种相对较弱的尿激酶型纤溶酶原激活剂 (uPA) 抑制剂 (Ki=82 μM)。4-Aminobenzamidine 可抑制 SCID 小鼠体内前列腺肿瘤的生长。
T2391	Camostat mesylate FOY-S980,甲磺酸卡莫司他,FOY305,Camostat mesilate	Serine/threonin kinase; SARS-CoV; Sodium Channel	Cell Cycle/Checkpoint; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
	Camostat mesylate (FOY-S980) 是口服活性合成的丝氨酸蛋白酶抑制剂，用于慢性胰腺炎。它是TMPRSS2的抑制剂，对SARS-CoV-2具有抗病毒活性。它抑制前列腺素、胰蛋白酶和苦参多糖的活性。
T63321	20S Proteasome activator 1	Proteasome	Proteases/Proteasome; Ubiquitination
	20S Proteasome activator 1 是一种 20S 蛋白酶激活剂，对胰蛋白酶样位点、胰凝乳蛋白酶样位点和半胱天冬酶位点的 IC50 分别为 0.3 μM、0.7 μM 和 1.8 μM。20S Proteasome activator 1 通过在细胞系统中翻译来防止致病性 α-synuclein A53T 突变体积累从而减少疾病发生的概率。20S Proteasome activator 1 可用于研究神经退行性疾病。
TP1832	Gluten Exorphin C	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Gluten exorphin C 是来源于谷朊粉的阿片肽。在 GPI 和 MVD 检测中，抑制 μ 阿片和 δ 阿片活性，IC50值分别为 40 和13.5 μM。
T25131	AZD8309 AZD 8309,AZD-8309	Glutathione Peroxidase; CXCR	Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism
	AZD8309 是一种强效的、可口服的趋化因子受体CXCR2的拮抗剂，能够调节中性粒细胞的转运，可显著降低胰腺和肺部的MPO，并降低胰腺内的胰蛋白酶和弹性蛋白酶活性。AZD8309 能够用于研究炎症系列疾病。
T67959	Pirodomast	Thrombin; Serine Protease	Proteases/Proteasome
	Pirodomast 是血栓素 A（TXA2）合成酶抑制剂。Pirodomast 能抑制白三烯（LT）D4、C4、E4 的形成和血栓素 B2（TXB2）的活性，但对组胺、甲氧胆碱、血清素、LTC4 或血小板活化因子诱导的豚鼠支气管痉挛的拮抗作用较弱或无效。Pirodomast 在体外对豚鼠气管只有微弱的松弛活性。Pirodomast 是一种潜在的抗过敏化合物，在体外可抑制胰蛋白酶的蛋白水解活性，在体内可阻止抗原诱发过敏绵羊的即时和晚期哮喘反应，抑制抗原诱导的过敏绵羊对组胺和卡巴胆碱的气道高反应性。
T13568L	BCX 1470 hydrochloride BCX 1470 hydrochloride(217099-43-9 Free base),BCX1470 HCl	Serine Protease; Complement System	Immunology/Inflammation; Proteases/Proteasome
	BCX 1470 hydrochloride 是一种高效的丝氨酸蛋白酶抑制剂，具有抗炎活性，能抑制 factor D 和 C1s 的酯水解和溶血活性，可用于研究水肿。
T13567	BCX 1470 methanesulfonate	Serine Protease	Proteases/Proteasome
	BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and 1.6 nM), 3.4- and 200-fold better than that of trypsin, respectively.
T13568	BCX 1470	Serine Protease	Proteases/Proteasome
	BCX 1470 inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and 1.6 nM), 3.4- and 200-fold better than that of trypsin, respectively.
T34785	TAPAP 3-Tapap
	TAPAP binds to thrombin and trypsin.
T38521	Patamostat mesylate E-3123 mesylate
	Patamostat mesylate (E-3123) is a highly potent protease inhibitor, displaying strong inhibitory activity against trypsin, plasmin, and thrombin, with IC 50 values of 39 nM, 950 nM, and 1.9 μM, respectively. This compound, Patamostat mesylate, shows promising potential in suppressing the pathogenesis and development of acute pancreatitis.
T39029	APC-6860
	APC-6860 is a trypsin-like serine proteases inhibitor with k i values of 0.21, 0.44, 1.5, 16.8, 20, 30 μM for uPA, trypsin, tryptase, tPA, thrombin and factor Xa, respectively. APC-6860 has a selectivity ratio for tPA versus uPA of 80. APC-6860 has k i values of 0.1, 0.082 μM for human and murine urokinases, respectively. APC-6860 can be used for the research of cancer.
T37053	Z-(L-Arg)-AMC (hydrochloride)
	Z-(L-Arg)-AMC is a fluorogenic substrate for trypsin, cathepsin B, and cathepsin H.1,2Upon enzymatic cleavage by trypsin, cathepsin B, or cathepsin H, 7-amino-4-methylcoumarin (AMC) is released and its fluorescence can be used to quantify trypsin, cathepsin B, and cathepsin H activity. AMC displays excitation/emission maxima of 340-360/440-460 nm, respectively. 1.Zimmerman, M., Ashe, B., Yurewicz, E.C., et al.Sensitive assays for trypsin, elastase, and chymotrypsin using new fluorogenic substrat...
T30510	BMS-262084 BMS 262084,I0IR71971G,UNII-I0IR71971G,CHEMBL71037
	BMS-262084 is a potent selective β-lactam trypsin inhibitor with therapeutic potential in the treatment of asthma.
T29969	AMG-126737 105RSZ5CNS,AMG 126737,SCHEMBL7986111
	AMG-126737 is an effective human lung mast cell trypsin inhibitor with potential therapeutic effect in lung diseases.
T78409	Boc-Val-Pro-Arg-MCA hydrochloride Boc-Val-Pro-Arg-MCA HCl
	Boc-Val-Pro-Arg-MCA hydrochloride (Boc-Val-Pro-Arg-MCA HCl) 为测定胰蛋白酶样丝氨酸蛋白酶 (trypsin-like serine proteases) 活性的敏感荧光底物。
T77221	Benzenecarboximidamide, hydrochloride, hydrate (1:1:x)
	Benzenecarboximidamide, hydrochloride, hydrate (1:1:x) (Benzamidine hydrochloride hydrate) 是一种可逆的竞争性胰蛋白酶样丝氨酸蛋白酶 (trypsin-like serine proteases) 抑制剂，对 Tryptase、Trypsin、uPA、Factor Xa、Thrombin 和 tPA 的Ki 值分别为 20、21、97、110、320 和 750 μM。
T19199	AzKTB	Others	Others
	AzKTB is a capture reagent comprising an azide module linked to TAMRA/PEG-biotin labels through a short trypsin-cleavable peptide sequence.
T62464	Bz-D-Arg-pNA hydrochloride
	Bz-D-Arg-pNA hydrochloride 是一种竞争性胰蛋白酶抑制剂。
T19218	Bz-Lys-OMe	Others	Others
	Bz-Lys-Ome is a methyl ester substrate of trypsin.
T19580	Thrombin (MW 37kDa) 凝血酶,Thrombin	Thrombin	Proteases/Proteasome
	Thrombin (MW 37kDa) 是一种 Na+激活的胰蛋白酶样别构丝氨酸蛋白酶。它能够利用凝血酶识别序列对融合蛋白进行位点特异性切割，并可用于消化 GST 标记的蛋白。
T36686	Ac-Arg-Gly-Lys(Ac)-AMC
	Ac-RGK(Ac)-AMC, fluorogenic substrate for assaying histone deacetylase (HDAC) activity in a two-step enzymatic reaction. The assay consists of the initial lysine deacetylation by HDAC followed by the release of the fluorescent group by trypsin.
T37011	Boc-LRR-AMC
	Boc-LRR-AMC is a fluorogenic substrate for the trypsin-like activity of the 26S proteasome or 20S proteolytic core. Upon enzymatic cleavage by the 26S proteasome or 20S proteolytic core, amino-4-methylcoumarin (AMC) is released and its fluorescence can be used to quantify 26S proteasome or 20S proteolytic core trypsin-like activity. AMC displays excitation/emission maxima of 340-360/440-460 nm, respectively.
T6564L	Leupeptin Leupeptin Ac-LL,NK-381
	Leupeptin is a competitive protease inhibitor produced by actinomycetes. Leupeptin can inhibit cysteine, serine and threonine peptidases. Leupeptin inhibits serine proteinases (trypsin (Ki=3.5 nM), plasmin (Ki= 3.4 nM), porcine kallikrein), and cysteine p
T78402	Boc-Gln-Ala-Arg-AMC acetate
	Boc-Gln-Ala-Arg-AMC醋酸盐是trypsin的一种荧光底物，主要用于检测TMPRSS2的蛋白水解活性。
T37019	p-APMSF (hydrochloride)
	p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 μM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively. It is selective for these proteases over bovine chymotrypsin and acetylcholinesterase.
T80211	Ac-KQL-AMC
	Ac-KQL-AMC是量化蛋白酶体样活性的荧光底物，其被裂解时释放可检测的荧光信号。
T72736	Aeruginosin 98-B
	Aeruginosin 98-B为一种蛋白酶抑制剂，能够抑制胰蛋白酶、纤溶酶和凝血酶，其IC50值依次为0.6、7.0和10.0 μg/mL。
T41085	UK122 UK122
	UK122 is a highly effective and specific inhibitor of urokinase-type plasminogen activator (uPA) with an IC50 value of 0.2 μM. It displays negligible to minimal inhibition towards tissue-type plasminogen activator (tPA), plasmin, thrombin, and trypsin (all IC50 >100 μM). Functioning as a 4-oxazolidinone analogue, UK122 is an anticancer agent that effectively inhibits cancer cell migration and invasion.
T78625	Z-Ala-Arg-Arg-AMC Z-ARR-AMC,Fluorogenic Proteasome Substrate	Proteasome	Proteases/Proteasome; Ubiquitination
	Z-Ala-Arg-Arg-AMC (FluorogenicProteasomeSubstrate) 作为荧光底物，专用于检测蛋白酶体中的胰蛋白酶样活性。
T76619	Methoxycarbonyl-D-Nle-Gly-Arg-pNA
	Methoxycarbonyl-D-Nle-Gly-Arg-pNA，这是一种底物，主要用于FIXa (Factors IXa) 和 FXa (Factors Xa)的合成蛋白酶。
T35887	MBD
	MBD, a novel fluorescent probe (7-(p-Methoxybenzylamino)-4-nitrobenz-2,1,3-oxadiazole), is utilized to study the conformation of protein and nucleoprotein. Its application is extended to bacterial ribosomes, as well as bovine trypsinogen and trypsin. MBD exhibits significant fluorescence when it binds to the hydrophobic region of macromolecules [1][2].

化合物

Cat.No: T3359

Synonym: 抑酶肽,抑肽酶,Bovine Pancreatic Trypsin Inhibitor,Traskolan,Antilysin

Target: Others, Serine Protease, Influenza Virus, Proteasome

Urinary Trypsin Inhibitor Fragment

Cat.No: T76240

Benzamidine hydrochloride

Cat.No: T8362

Synonym: Benzamidine HCl,苄脒盐酸盐

Target: Serine/threonin kinase, Serine Protease

Cat.No: T17011

Target: Proteasome

2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-

Cat.No: T8802

Synonym: 2,4-Dioxaspiro[5.5]undec-8-ene, 3-(2-fur

Target: Serine Protease

Cat.No: T73594

Synonym: Chymotrypsin A

Target: Serine/threonin kinase

alpha-1 antitrypsin fragment

Cat.No: TP2217

Target: Others

Chymotrypsinogen

Cat.No: T76157

alpha-1 antitrypsin fragment 235-243 [Homo sapiens]/[Papio hamadryas]/[Cercopithecus aethiops]

Cat.No: TP2216

Target: Others

Cat.No: T7016

Target: Apoptosis, Proteasome, Caspase

Cat.No: T9670L

Synonym: Patamostat HCl（114568-26-2 Free base）

Target: Serine Protease, Protease

Boc-Gln-Ala-Arg-AMC hydrochloride

Cat.No: T74040

Cat.No: T30519

Synonym: BMS363131,BMS 363131

Target: Serine Protease

AEBSF hydrochloride

Cat.No: T6370

Synonym: AEBSF HCl,Pefabloc SC

Target: Thrombin, Serine Protease, Influenza Virus

Cat.No: T6941

Synonym: PI 1840

Target: PARP, Proteasome

N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride

Cat.No: T16169

Synonym: N-alpha-Tosyl-L-lysine_chloromethyl_ketone_hydrochloride

Target: Others, Proteasome, COX

Cat.No: T2122

Synonym: 艾沙佐米,MLN2238

Target: Proteasome, Caspase, Autophagy

Boc-Val-Pro-Arg-MCA TFA

Cat.No: T78409L

4-Aminobenzamidine dihydrochloride

Cat.No: T60248

Synonym: p-Aminobenzamidine dihydrochloride

Target: Serine Protease

Camostat mesylate

Cat.No: T2391

Synonym: FOY-S980,甲磺酸卡莫司他,FOY305,Camostat mesilate

Target: Serine/threonin kinase, SARS-CoV, Sodium Channel

20S Proteasome activator 1

Cat.No: T63321

Target: Proteasome

Gluten Exorphin C

Cat.No: TP1832

Target: Opioid Receptor

Cat.No: T25131

Synonym: AZD 8309,AZD-8309

Target: Glutathione Peroxidase, CXCR

Cat.No: T67959

Target: Thrombin, Serine Protease

BCX 1470 hydrochloride

Cat.No: T13568L

Synonym: BCX 1470 hydrochloride(217099-43-9 Free base),BCX1470 HCl

Target: Serine Protease, Complement System

BCX 1470 methanesulfonate

Cat.No: T13567

Target: Serine Protease

Cat.No: T13568

Target: Serine Protease

Cat.No: T34785

Synonym: 3-Tapap

Patamostat mesylate

Cat.No: T38521

Synonym: E-3123 mesylate

Cat.No: T39029

Z-(L-Arg)-AMC (hydrochloride)

Cat.No: T37053

Cat.No: T30510

Synonym: BMS 262084,I0IR71971G,UNII-I0IR71971G,CHEMBL71037

Cat.No: T29969

Synonym: 105RSZ5CNS,AMG 126737,SCHEMBL7986111

Boc-Val-Pro-Arg-MCA hydrochloride

Cat.No: T78409

Synonym: Boc-Val-Pro-Arg-MCA HCl

Benzenecarboximidamide, hydrochloride, hydrate (1:1:x)

Cat.No: T77221

Cat.No: T19199

Target: Others

Bz-D-Arg-pNA hydrochloride

Cat.No: T62464

Cat.No: T19218

Target: Others

Thrombin (MW 37kDa)

Cat.No: T19580

Synonym: 凝血酶,Thrombin

Target: Thrombin

Ac-Arg-Gly-Lys(Ac)-AMC

Cat.No: T36686

Cat.No: T37011

Cat.No: T6564L

Synonym: Leupeptin Ac-LL,NK-381

Boc-Gln-Ala-Arg-AMC acetate

Cat.No: T78402

p-APMSF (hydrochloride)

Cat.No: T37019

Cat.No: T80211

Aeruginosin 98-B

Cat.No: T72736

Cat.No: T41085

Synonym: UK122

Z-Ala-Arg-Arg-AMC

Cat.No: T78625

Synonym: Z-ARR-AMC,Fluorogenic Proteasome Substrate

Target: Proteasome

Methoxycarbonyl-D-Nle-Gly-Arg-pNA

Cat.No: T76619

Cat.No: T35887

Cat. No.	Product Name	Target	Signaling Pathways
TN6872	Trypsin	Protease-activated Receptor	GPCR/G Protein
	Trypsin 是一种可从鱼类分离出的丝氨酸蛋白酶，可水解赖氨酸或精氨酸羧基侧蛋白质。Trypsin 具有抗炎活性，可通过 PDCoV 的 S 糖蛋白与 pAPN 的相互作用诱导 PDCoV 感染的细胞膜融合，可激活 PAR2 和 PAR4，促进细胞增殖和分化。Trypsin 可用于促进伤口愈合和研究神经源性炎症。
T5S0689	Demethylwedelolactone 去甲蟛蜞菊内酯,去甲基蟛蜞内酯	Serine Protease	Proteases/Proteasome
	Demethylwedelolactone 是一种分离自 Eclipta alba 中的 coumestan 天然产物。它能抑制乳腺癌细胞的移动和侵袭，是一种有效的trypsin 抑制剂(IC50:3.0 μM)。
T16012	Marizomib NPI-0052,Salinosporamide A,ML858	Proteasome	Proteases/Proteasome; Ubiquitination
	Marizomib (ML858) 是一种新型不可逆的脑渗透性泛蛋白酶体 (proteasome) 抑制剂，对 20S 蛋白酶体的 CT-L (β5)、CT-T-laspase 样 (C-L, β1) 和胰蛋白酶样 (T-L, β2) 具有抑制作用， IC50 分别为 3.5, 28, 430 nM。
TN1372	Alpha-Amyrin alpha-Amyrenol,α-Amyrin,alpha-Amyrine,Viminalol,α-香树脂醇	P450; Serine Protease; ROS	Immunology/Inflammation; Metabolism; Proteases/Proteasome
	Alpha-Amyrin (alpha-Amyrine) 是一种具有抗肿瘤作用的胰蛋白酶和糜蛋白酶抑制剂。 alpha-Amyrin 可用于作为肝调节剂的研究。
T2O2730	L-Serine (S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid	Endogenous Metabolite	Metabolism
	L-Serine (serine) 是一种人体非必需氨基酸，它存在于许多蛋白质中，并且在功能上很重要。L-Serine 也存在于丝氨酸蛋白酶类的活性位点，包括胰蛋白酶和凝乳胰蛋白酶。
T6S0071	Fraxinellone	HIF/HIF Prolyl-Hydroxylase; STAT; PD-1/PD-L1	Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Metabolism; Stem Cells
	Fraxinellone 是从白鲜的根皮中分离出来的一种天然产物，是PD-L1抑制剂，可抑制HIF-1α蛋白质合成。它通过靶向 PD-L1，有用于癌症免疫的潜力。
T39367	Suomilide
	Suomilide effectively inhibits human trypsin-2 and trypsin-3, displaying IC50 values of 4.7 nM and 11.5 nM, respectively. Additionally, it exhibits inhibition of trypsin-1 with an IC50 value of 104 nM.
T41033	Fetuin, Fetal Bovine Serum
	Fetuin, Fetal Bovine Serum is a glycoprotein weighing 64 kDa that is secreted by the liver and obtained from fetal bovine serum. It acts as an inhibitor of trypsin activity and facilitates cellular attachment, growth, and differentiation.
T75647	Nostosin G
	Nostosin G 是一种独特的线性肽，含有 3 个亚基，4-羟基苯乳酸 (Hpla)，高酪氨酸 (Hty) 和精氨酸。Nostosin G 具有有效的胰蛋白酶抑制特性，其 IC50值为 0.1 μM。

天然产物

Cat.No: TN6872

Target: Protease-activated Receptor

Demethylwedelolactone

Cat.No: T5S0689

Synonym: 去甲蟛蜞菊内酯,去甲基蟛蜞内酯

Target: Serine Protease

Cat.No: T16012

Synonym: NPI-0052,Salinosporamide A,ML858

Target: Proteasome

Cat.No: TN1372

Synonym: alpha-Amyrenol,α-Amyrin,alpha-Amyrine,Viminalol,α-香树脂醇

Target: P450, Serine Protease, ROS

Cat.No: T2O2730

Synonym: (S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid

Target: Endogenous Metabolite

Cat.No: T6S0071

Target: HIF/HIF Prolyl-Hydroxylase, STAT, PD-1/PD-L1

Cat.No: T39367

Fetuin, Fetal Bovine Serum

Cat.No: T41033

Cat.No: T75647

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