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220

抑制剂 & 化合物

21

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0957 Isradipine

PN 200-110,伊拉地平

Calcium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Isradipine (PN 200-110) 是一种二氢吡啶类钙通道阻滞剂,具有抗高血压和血管扩张活性。它是一种具有口服活性的 L 型钙通道阻滞剂,也是一种潜在可行的帕金森病神经保护剂。
T12315 OR-1896

PDE Metabolism
OR-1896 is an active long-lived Levosimendan metabolite, is a highly selective inhibitor of phosphodiesterase (PDE) III isoformand a powerful vasodilator.
T67933 BAY-4931

PPAR DNA Damage/DNA Repair; Metabolism
BAY-4931 是一种有效的、共价的、选择性的 PPARγ反向激动剂,IC50为 0.17 nM。
T61214 EWP 815

Phosphatase; Hydroxylase Metabolism
EWP 815 is a disulfiram analogue that functions as a powerful inhibitor of Ins(1,4) P 2 phosphatase, Ins(1,4,5) P 3 5-phosphatase, and dopamine β-hydroxylase activity [1] [2].
T19774 Methylisothiazolinone

KB-838,MI,N-Methylisothiazolin-3-one,甲基异噻唑啉酮,Methylisothiazolinone free base

Antibacterial Microbiology/Virology
Methylisothiazolinone (MI) 是合成的杀菌剂和防腐剂,可广泛用于工业和消费产品。它作为化妆品和盥洗用品中的防腐剂。
T9879 Hydroxystilbamidine

Oxistilbamidinum,羟芪巴脒,(E)-hydroxystilbamidine,2-Hydroxy-4,4'-diguanylstilbene,Bis(8-hydroxyquinolinium) sulphate

Others Others
Hydroxystilbamidine ((E)-hydroxystilbamidine) 是一种能够结合 DNA 和 RNA 的染料, 也被发现是细胞核糖核酸酶的强效抑制剂。
T9111 8-Azaadenosine

Adenosine deaminase Metabolism
8-Azaadenosine 是 ADAR1抑制剂和是 A-to-I 编辑抑制剂。它可阻断 RNA 编辑并抑制甲状腺癌细胞的增殖、3D 生长、侵袭和迁移。
T24214 Phenamacril

JS39919,苯那普利,JS399 19

Myosin; Antifungal Cytoskeletal Signaling; Microbiology/Virology
Phenamacril (JS39919) 是一种氰基丙烯酸酯类杀菌剂,对镰刀菌,特别是禾谷镰刀菌有很强的抑制作用。它是一种特异性镰刀菌肌球蛋白 I 抑制剂。
T64347 ALDH1A3-IN-3

Dehydrogenase Metabolism
ALDH1A3-IN-3 (化合物 16) 是一种有效的 ALDH1A3 抑制剂,IC50 值为 0.26 μM。ALDH1A3-IN-3 也是 ALDH3A1 的底物。ALDH1A3-IN-3 可用于前列腺癌的研究。
T63166L (S, R)-LSN 3318839

(S, R)-LSN 3318839(Isomer-2764704-18-7)

Glucagon Receptor GPCR/G Protein
T19637 Aluminum phthalocyanine chloride

Phthalocyanine Chloroaluminum,铝酞菁,Chloroaluminum Phthalocyanine

Others Others
Aluminum phthalocyanine chloride (Phthalocyanine Chloroaluminum) 是一种强烈的蓝绿色芳香大环化合物,广泛用于染色。
T10213 A-437203

ABT-925,A37203,Lu201640

Dopamine Receptor GPCR/G Protein; Neuroscience
A-437203 (Lu201640) 是一种基于1H-pyrimidin-2-one scaffold 的、具有选择性的、新型强效的d3受体拮抗剂,对 D2, D3, 和 D4 受体,的Ki 值分别为 71, 1.6 和 6220 nM。
T35528L TD52 dihydrochloride

TD52 dihydrochloride(1798328-24-1 Free base),TD52 2HCl

Others Others
TD52 dihydrochloride (TD52 2HCl), a derivative of Erlotinib, is a potent and orally active inhibitor of protein phosphatase 2A (CIP2A). It exhibits strong anti-cancer properties by regulating the CIP2A/PP2A/p-Akt signaling pathway, resulting in the induction of apoptosis in triple-negative breast cancer (TNBC) cells. Mechanistically, TD52 dihydrochloride disrupts the binding of Elk1 to the CIP2A promoter, effectively reducing CIP2A levels. Notably, TD52 dihydrochloride demonstrates powerful anti...
T14513 BBIQ

TLR Immunology/Inflammation
BBIQ 是一种有效且选择性的 toll 样受体 7 (TLR7) 激动剂,对人 TLR7 的 EC50 为 59.1 nM。BBIQ 还是一种功能强大的疫苗佐剂,可增强机体的先天免疫应答。
T40465 SAG dihydrochloride

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
SAG dihydrochloride 是一种强效的 Smoothened(Smo)受体激动剂(EC 50 =3 nM;K d =59 nM)。SAG dihydrochloride 可激活刺猬信号通路并抵消环丙胺对 Smo 的抑制。
T67835 LKM38

LKM38是一种新型的重氮烷基胆固醇探针,是一种有前途的胆固醇模拟物。LKM38既能维持抗胆固醇细胞的生长,又能适当地调节关键的胆固醇平衡途径。LKM38可以作为研究胆固醇蛋白相互作用和贩运的有力工具。
T22574L Angiotensin 1/2 (5-7) acetate

RAAS Endocrinology/Hormones
Angiotensin 1/2 (5-7) acetate 是一种具有 H2N-Ile-His-Pro-OH 序列的肽。血管紧张素是一种寡肽,是一种激素和一种强大的双肽原。它来源于前体分子血管紧张素原,一种在肝脏中产生的血清球蛋白。它在肾素-血管紧张素系统中起重要作用。
T21610 Bradykinin (acetate)

Bradykinin Receptor GPCR/G Protein
Bradykinin (acetate) 是一种由激肽释放酶-激肽系统产生的活性肽。它是一种炎症介质,也被认为是多种血管和肾功能的神经介质和调节剂。它由血液中的 kallidin 酶促产生,是一种强大的血管扩张剂,可引起平滑肌收缩,并可能介导炎症。它具有作为人血清代谢物和血管扩张剂的作用。它是缓激肽 (2+) 的互变异构体。
T28029 Methylisothiazolinone hydrochloride

N-Methylisothiazolin-3-one,MI,2-甲基-4-异噻唑啉-3-酮盐酸盐,KB-838,Methylisothiazolinone HCl

Methylisothiazolinone is a powerful synthetic biocide and preservative.
T32436 L 1935

Compound l1935,L-1935,Histamine-liberator L 1935,L1935

L 1935 is a type of powerful histamine-liberator.
T25960 Piperic acid

NSC 129538,NSC129538,NSC-129538

Piperic acid is a powerful antioxidant and has potent antibacterial properties
T34124 Pranolium

UM-272,SC-27761,UM 272,SC 27761,SC27761

Pranolium is a quaternary dimethyl derivative of Propranolol, a well-known powerful betareceptor-blocking agent.
T71443 Amphidinolide D

Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction.
T71140 MDL-27048

MDL-27048 is a powerful and reversible microtubule inhibitor.
T33590 Nantradol HCl

MCV-4161,MCV4161,UM-1159,UM 1159,MCV 4161,UM1159

Nantradol HCl is a powerful analgesic widely used to investigate the potential therapeutic applications of cannabinoids.
T39753 Etavopivat

FT-4202

Etavopivat is a powerful, specific, orally bioavailable activator of pyruvate kinase (PKR) in red blood cells (RBCs). It exhibits potent properties against sickling.
T38822 D-threo-PPMP

D-threo-PPMP, a powerful glucosylceramide (GlcCer) synthase inhibitor, effectively impedes karyokinesis and decreases cyst formation.
T25299 Degranol

NSC 9698,NSC-9698,NSC9698

Degranol is a nitrogen mustard derivative alkylating agent utilized as antineoplastic. It causes severe bone marrow depression and is a powerful vesicant.
T30945 Cinolazepam

Gerodorm,OX-373

Cinolazepam is a benzodiazepine derivative drug.It has a powerful sedative effect, so it is mainly used as a hypnotic.
T11107 DSP-1053

Others Others
Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.
T35661 QTX125

QTX125, a powerful and highly specific HDAC6 inhibitor, demonstrates exceptional selectivity in comparison to other HDACs, resulting in robust antitumor activity[1].
T68260 Calmidazolium (cation)

Calmidazolium (cation) is a powerful inhibitor of or red blood cell Ca -ATPase & Ca transport into inside-out red blood cell vesicles; an antagonist of calmodulin.
T28464 p-SCN-Bn-TCMC HCl

p-SCN-Bn-TCMC

p-SCN-Bn-TCMC is a bifunctional chelator, it contains a powerful chelator TCMC and reactive tioisocyante linker. TCMC is a powerful chelator with capability to strongly bind radio-isotopic heavy metal ion, which are widely used for radio-diagnostic/imagin
TP2459 Lysipressin Acetate

Lysine pitressin,Lysine vasopressin,Lypressin,Lysopressin,Lysipressin Acetate. L-Lysine vasopressin,Lysine-ADH

Lysipressin Acetate is an analog of vasopressin, a powerful vasopressin used to regulate blood pressure. Endogenous vasopressin in most mammalian species.
T40943 EMD527040

EMD527040 is a powerful and highly specific αvβ6 antagonist, exhibiting notable antifibrotic properties. It is suitable for conducting research on carcinoma and liver fibrosis.
T35082 VU6010608

VU-6010608,VU 6010608

VU6010608 is an effective mGlu7 NAM with excellent CNS permeability and is powerful in electrophysiological studies in blocking long-term enhancement of high-frequency stimuli.
T38914 MPO-IN-3

MPO-IN-3, a powerful inhibitor of myeloperoxidase (MPO), is described as such in example 191 of WO2013068875A1. MPO, a heme-containing enzyme, is classified under the peroxidase superfamily.
T40841 L-2-Aminooxy-3-phenylpropanoic acid hydrobromide

L-2-Aminooxy-3-phenylpropanoic acid hydrobromide is a powerful inhibitor of L-phenylalanine ammonia-lyase, an enzyme responsible for catalyzing the conversion of L-phenylalanine to trans-cinnamic acid.
T20778 Epoprostenol

U 53217,U 53,217,U-53,217

Epoprostenol, a prostaglandin, is a powerful vasodilator. It inhibits platelet aggregation.
T61314 DC-CPin7

DC-CPin7, a powerful inhibitor of the bromodomain of CREB-binding protein (CBP), exhibits an IC50 value of 2.5 μM [1].
T11721L JDTic dihydrochloride

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
JDTic is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception.
T61310 HIV-1 inhibitor-37

HIV-1 inhibitor-37 (Compound 83) is a highly powerful HIV-1 inhibitor. It exhibits significant potential for use as an innovative latent HIV-1 reactivating agent [1].
T40642 Chlorpyrifos-oxon

Chlorpyrifos-oxon, an active metabolite of Chlorpyrifos, is a powerful phosphorylating agent with potent inhibition of AChE activity. It induces cross-linking between tubulin subunits and disrupts microtubule function[4].
T40568 Fmoc-MMAE

Fmoc-MMAE, a protective group-conjugated variant of monomethyl auristatin E (MMAE), serves as a powerful inhibitor of tubulin. It finds application in the synthesis of antibody-drug conjugates (ADC).
T36901 Pelcitoclax

Pelcitoclax (APG-1252) is a powerful inhibitor of the Bcl-2 and Bcl-xl proteins, displaying significant antineoplastic and pro-apoptotic properties[1].
T69443 Aminobutane bisphosphonate

Aminobutane bisphosphonate is a powerful inhibitor of bone resorption. It can potentially be a useful measure for controlling hypercalcemia in patients with carcinoma.
T38779 NS-102

NS-102 is a powerful and selective antagonist of the kainate receptor (GluK2), as well as a potent antagonist of the GluR6/7 receptor.
T61712 Trk-IN-8

Trk-IN-8, a powerful TRK inhibitor, demonstrates excellent potency against TRKAa, TRKA(G595R), and TRKC(G623R) with IC50 values of 0.42 nM, 0.89 nM, and 1.5 nM, respectively (WO2021115401A1, compound 3) [1].
T25316 Dexecadotril

Retorphan

Dexecadotril is a powerful and selective neprilysin inhibitor. It behaves as a prodrug of the enantiomer of thiorphan.
T75748 Indolicidin TFA

Indolicidin TFA 是一种从牛中性粒细胞的细胞质颗粒中纯化的强效抗菌肽。

化合物

Isradipine
Cat.No: T0957
Synonym: PN 200-110,伊拉地平
Target: Calcium Channel, Autophagy
OR-1896
Cat.No: T12315
Synonym:
Target: PDE
BAY-4931
Cat.No: T67933
Synonym:
Target: PPAR
EWP 815
Cat.No: T61214
Synonym:
Target: Phosphatase, Hydroxylase
Methylisothiazolinone
Cat.No: T19774
Synonym: KB-838,MI,N-Methylisothiazolin-3-one,甲基异噻唑啉酮,Methylisothiazolinone free base
Target: Antibacterial
Hydroxystilbamidine
Cat.No: T9879
Synonym: Oxistilbamidinum,羟芪巴脒,(E)-hydroxystilbamidine,2-Hydroxy-4,4'-diguanylstilbene,Bis(8-hydroxyquinolinium) sulphate
Target: Others
8-Azaadenosine
Cat.No: T9111
Synonym:
Target: Adenosine deaminase
Phenamacril
Cat.No: T24214
Synonym: JS39919,苯那普利,JS399 19
Target: Myosin, Antifungal
ALDH1A3-IN-3
Cat.No: T64347
Synonym:
Target: Dehydrogenase
(S, R)-LSN 3318839
Cat.No: T63166L
Synonym: (S, R)-LSN 3318839(Isomer-2764704-18-7)
Target: Glucagon Receptor
Aluminum phthalocyanine chloride
Cat.No: T19637
Synonym: Phthalocyanine Chloroaluminum,铝酞菁,Chloroaluminum Phthalocyanine
Target: Others
A-437203
Cat.No: T10213
Synonym: ABT-925,A37203,Lu201640
Target: Dopamine Receptor
TD52 dihydrochloride
Cat.No: T35528L
Synonym: TD52 dihydrochloride(1798328-24-1 Free base),TD52 2HCl
Target: Others
BBIQ
Cat.No: T14513
Synonym:
Target: TLR
SAG dihydrochloride
Cat.No: T40465
Synonym:
Target: Hedgehog/Smoothened
LKM38
Cat.No: T67835
Synonym:
Target:
Angiotensin 1/2 (5-7) acetate
Cat.No: T22574L
Synonym:
Target: RAAS
Bradykinin (acetate)
Cat.No: T21610
Synonym:
Target: Bradykinin Receptor
Methylisothiazolinone hydrochloride
Cat.No: T28029
Synonym: N-Methylisothiazolin-3-one,MI,2-甲基-4-异噻唑啉-3-酮盐酸盐,KB-838,Methylisothiazolinone HCl
Target:
L 1935
Cat.No: T32436
Synonym: Compound l1935,L-1935,Histamine-liberator L 1935,L1935
Target:
Piperic acid
Cat.No: T25960
Synonym: NSC 129538,NSC129538,NSC-129538
Target:
Pranolium
Cat.No: T34124
Synonym: UM-272,SC-27761,UM 272,SC 27761,SC27761
Target:
Amphidinolide D
Cat.No: T71443
Synonym:
Target:
MDL-27048
Cat.No: T71140
Synonym:
Target:
Nantradol HCl
Cat.No: T33590
Synonym: MCV-4161,MCV4161,UM-1159,UM 1159,MCV 4161,UM1159
Target:
Etavopivat
Cat.No: T39753
Synonym: FT-4202
Target:
D-threo-PPMP
Cat.No: T38822
Synonym:
Target:
Degranol
Cat.No: T25299
Synonym: NSC 9698,NSC-9698,NSC9698
Target:
Cinolazepam
Cat.No: T30945
Synonym: Gerodorm,OX-373
Target:
DSP-1053
Cat.No: T11107
Synonym:
Target: Others
QTX125
Cat.No: T35661
Synonym:
Target:
Calmidazolium (cation)
Cat.No: T68260
Synonym:
Target:
p-SCN-Bn-TCMC HCl
Cat.No: T28464
Synonym: p-SCN-Bn-TCMC
Target:
Lysipressin Acetate
Cat.No: TP2459
Synonym: Lysine pitressin,Lysine vasopressin,Lypressin,Lysopressin,Lysipressin Acetate. L-Lysine vasopressin,Lysine-ADH
Target:
EMD527040
Cat.No: T40943
Synonym:
Target:
VU6010608
Cat.No: T35082
Synonym: VU-6010608,VU 6010608
Target:
MPO-IN-3
Cat.No: T38914
Synonym:
Target:
L-2-Aminooxy-3-phenylpropanoic acid hydrobromide
Cat.No: T40841
Synonym:
Target:
Epoprostenol
Cat.No: T20778
Synonym: U 53217,U 53,217,U-53,217
Target:
DC-CPin7
Cat.No: T61314
Synonym:
Target:
JDTic dihydrochloride
Cat.No: T11721L
Synonym:
Target: JAK
HIV-1 inhibitor-37
Cat.No: T61310
Synonym:
Target:
Chlorpyrifos-oxon
Cat.No: T40642
Synonym:
Target:
Fmoc-MMAE
Cat.No: T40568
Synonym:
Target:
Pelcitoclax
Cat.No: T36901
Synonym:
Target:
Aminobutane bisphosphonate
Cat.No: T69443
Synonym:
Target:
NS-102
Cat.No: T38779
Synonym:
Target:
Trk-IN-8
Cat.No: T61712
Synonym:
Target:
Dexecadotril
Cat.No: T25316
Synonym: Retorphan
Target:
Indolicidin TFA
Cat.No: T75748
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TP1180 Dolastatin 10

尾海兔素10,NSC 376128,DLS 10

Microtubule Associated Cytoskeletal Signaling
Dolastatin 10 (DLS 10) 是一种多肽,可以抑制微管蛋白聚合,显示除抗有丝分裂的活性。
T5297 3-Indolepropionic acid

Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸

Antioxidant; Reactive Oxygen Species; Endogenous Metabolite Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
3-Indolepropionic acid (Indolepropionic acid) 是强效的抗氧化剂,具有研究阿尔兹海默症的潜能。
T3749 Pyrogallol

连苯三酚,Piral,焦榈酚,1,2,3-trihydroxybenzene

Apoptosis; Others; Endogenous Metabolite; Antifungal Apoptosis; Metabolism; Microbiology/Virology; Others
Pyrogallol (Piral) 是一种通过加热没食子酸制备的强还原剂,能产生自由基。它是一种具有抗真菌和抗牛皮癣活性的多酚。
T0965 Histamine

Ergamine,组胺

5-HT Receptor; Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine (Ergamine) 是通过组胺的酶促脱羧衍生的胺。它是一种强大的胃分泌兴奋剂、支气管平滑肌的收缩剂、血管扩张剂以及中枢作用的神经递质。
S00015 Tea polyphenol

Apoptosis; Others; Autophagy Apoptosis; Autophagy; Others
Tea polyphenol 也称为绿茶提取物,是茶中天然存在的酚类化合物,具有抗癌、抗氧化、抑制细胞增殖、诱导细胞凋亡、延缓细胞周期和调节致癌物代谢等生物活性。
T6534 Histamine dihydrochloride

组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine dihydrochloride (Ceplene) 是 Histamine 的二盐酸形式。Histamine 是一种有机氮化合物,是一种强效的胃分泌兴奋剂,支气管平滑肌收缩剂,血管舒张剂,也是一种中枢作用的神经递质。
T2S1464 Thiocolchicoside

硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl

Others; GABA Receptor Membrane transporter/Ion channel; Neuroscience; Others
Thiocolchicoside (Thiocolchicine 2-glucoside analog) 是秋水仙碱的半合成硫衍生物,是竞争性 GABAA 受体拮抗剂和甘氨酸受体拮抗剂。它是肌肉松弛剂,具有抗炎作用,可用于缓解疼痛的研究。
TC0019 Pregnenolone acetate

孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
Pregnenolone acetate 是一种强大的神经类固醇,是各种类固醇激素(包括类固醇酮)的主要前体。它作为大麻素 CB1 受体的信号特异性抑制剂,抑制由 CB1 受体介导的四氢大麻酚 (THC) 的作用。它可以保护大脑免受大麻中毒。
T10933 D-Cysteine

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-Cysteine 是一种大肠杆菌生长的有力抑制剂,是半胱氨酸的 D 型异构体。它由 D-氨基酸氧化酶介导产生 H2S,是一种对抗小脑共济失调的神经保护剂。 D-半胱氨酸可以抑制由变形链球菌和链球菌血红蛋白形成的两种生物膜的生长和致龋性。
T6S0221 Eriocitrin

eriodictyol 7-rutinoside,圣草次甙,Eriodictyol-7-O-Rutinoside,Eriodictioside,圣草次甙;圣草次苷,Eriodictyol glycoside

Apoptosis; Carbonic Anhydrase Apoptosis; Metabolism
Eriocitrin (Eriodictyol-7-O-Rutinoside) 是从柠檬中分离出来的一种黄酮类天然产物,是强效的抗氧化剂。它通过激活线粒体涉及的内在信号传导途径来触发细胞凋亡。它通过上调 p53、cyclin A、cyclin D3 和 CDK6 使 S 期细胞周期停滞,从而抑制肝癌细胞的增殖。
T40803 Isoanthricin

(Rac)-Deoxypodophyllotoxin

Isoanthricin, also known as (Rac)-Deoxypodophyllotoxin, is the racemate form of Deoxypodophyllotoxin, a powerful compound with noteworthy antitumor and anti-inflammatory properties.
T7980 Hesperidin methylchalcone

NF-κB NF-κB
Hesperidin methylchalcone 抑制氧化应激,细胞因子产生和NF-κB 活化。它能够抑制炎症和疼痛,具有血管保护作用。
TN2726 Jatrophane 5

P-gp Membrane transporter/Ion channel; Neuroscience
Jatrophane 5 demonstrates the most powerful inhibition of P-gp, higher than R(+)-verapamil and tariquidar in colorectal multi-drug resistant (MDR) cells (DLD1-TxR).
T38838 QS-21

Stimulon,QS-21

QS-21, an immunostimulatory saponin, is a powerful vaccine adjuvant that stimulates both Th2 humoral and Th1 cell-mediated immune responses by interacting with antigen presenting cells (APCs) and T cells. Additionally, QS-21 activates the NLRP3 inflammasome, leading to the release of cytokines IL-1β and IL-18, which are dependent on caspase-1.
T72731 Acremoxanthone C

Acremoxantone C 是一种有效的钙调素(CaM)抑制剂,存在于 Purpureocillium lilacinum 中。Acremoxantone C 与人钙调素 (hCaM) 生物传感器 hCaM M124C mBBr 结合,Kd 为 18.25 nM。
T37687 Cyclic ADP-ribose ammonium

Cyclic ADP-ribose ammonium (cADPR ammonium) is a powerful calcium mobilization second messenger synthesized from NAD+ by an ADP-ribosyl cyclase. It primarily raises cytosolic calcium levels through Ryanodine receptor-mediated release from the endoplasmic reticulum, while also facilitating extracellular influx through the opening of TRPM2 channels [1][2][3].
T79931 Mutanocyclin

Mutanocyclin 作为一种效能显著的抗真菌剂,能够抑制白色念珠菌 (C. albicans) 的丝状形成,并下调 HWP1、ECE1、FLO8、TEC1 基因的 mRNA 表达水平。此外,Mutanocyclin 在体外小鼠模型中亦能有效抑制酵母形态的发展。
T35895 Ingenol 3,20-dibenzoate

Ingenol 3,20-dibenzoate is a powerful activator of protein kinase C (PKC) isoforms. It effectively induces the translocation of nPKC-delta, -epsilon, and -theta as well as PKC-mu from the cytosolic fraction to the particulate fraction. Through de novo synthesis of macromolecules, it triggers apoptosis with characteristic morphology. Moreover, Ingenol 3,20-dibenzoate enhances IFN-γ production and degranulation in NK cells, particularly when stimulated by NSCLC cells[1][2].
T71750 Quinolactacin A1

Quinolactacin A1 是一种有效的乙酰胆碱酯酶 (AChE) 抑制剂,可从Penicillium citrinum 中得到。Quinolactacin A1 可用于阿尔茨海默病的研究。
T16574 Pregnenolone monosulfate sodium salt

3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt

Others Others
Pregnenolone monosulfate sodium salt is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium salt can protect the brain from cannabis intoxication. Pregnenolone monosulfate sodi
TN2727 Jatrophane 2

P-gp; Antifection Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
2,5,7,8,9,14-Hexaacetoxy-3-benzoyloxy-15-hydroxyjatropha-6(17),11E-diene (Jatrophane 2 ) exhibits significant antifeedant activity against a generalist plant-feeding insect, the cotton bollworm (Helicoverpa armigera). Jatrophane 2 also demonstrates the mo

天然产物

Dolastatin 10
Cat.No: TP1180
Synonym: 尾海兔素10,NSC 376128,DLS 10
Target: Microtubule Associated
3-Indolepropionic acid
Cat.No: T5297
Synonym: Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸
Target: Antioxidant, Reactive Oxygen Species, Endogenous Metabolite
Pyrogallol
Cat.No: T3749
Synonym: 连苯三酚,Piral,焦榈酚,1,2,3-trihydroxybenzene
Target: Apoptosis, Others, Endogenous Metabolite, Antifungal
Histamine
Cat.No: T0965
Synonym: Ergamine,组胺
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Tea polyphenol
Cat.No: S00015
Synonym:
Target: Apoptosis, Others, Autophagy
Histamine dihydrochloride
Cat.No: T6534
Synonym: 组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl
Target: Endogenous Metabolite, Histamine Receptor
Thiocolchicoside
Cat.No: T2S1464
Synonym: 硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl
Target: Others, GABA Receptor
Pregnenolone acetate
Cat.No: TC0019
Synonym: 孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate
Target: Cannabinoid Receptor, Endogenous Metabolite
D-Cysteine
Cat.No: T10933
Synonym:
Target: Endogenous Metabolite, Antibacterial
Eriocitrin
Cat.No: T6S0221
Synonym: eriodictyol 7-rutinoside,圣草次甙,Eriodictyol-7-O-Rutinoside,Eriodictioside,圣草次甙;圣草次苷,Eriodictyol glycoside
Target: Apoptosis, Carbonic Anhydrase
Isoanthricin
Cat.No: T40803
Synonym: (Rac)-Deoxypodophyllotoxin
Target:
Hesperidin methylchalcone
Cat.No: T7980
Synonym:
Target: NF-κB
Jatrophane 5
Cat.No: TN2726
Synonym:
Target: P-gp
QS-21
Cat.No: T38838
Synonym: Stimulon,QS-21
Target:
Acremoxanthone C
Cat.No: T72731
Synonym:
Target:
Cyclic ADP-ribose ammonium
Cat.No: T37687
Synonym:
Target:
Mutanocyclin
Cat.No: T79931
Synonym:
Target:
Ingenol 3,20-dibenzoate
Cat.No: T35895
Synonym:
Target:
Quinolactacin A1
Cat.No: T71750
Synonym:
Target:
Pregnenolone monosulfate sodium salt
Cat.No: T16574
Synonym: 3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt
Target: Others
Jatrophane 2
Cat.No: TN2727
Synonym:
Target: P-gp, Antifection
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