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196

抑制剂 & 化合物

62

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1092 Myelin Basic Protein (MBP) (68-82), guinea pig

MBP (68-82), guinea pig,豚鼠髓磷脂碱性蛋白片段68-82

Others Others
Myelin Basic Protein (MBP) (68-82), guinea pig 是一种髓鞘碱性蛋白 (MBP) 的片段。
TP2210 VIP(Guinea pig)

VIP (guinea pig)

Others Others
Neuropeptide with many biological actions
T82518 Dynorphin B 29 (pig)

Leumorphin (pig)

Dynorphin B 29 (Leumorphin) (pig) 是一种可与大脑及孤立组织系统中的多种受体交互作用的肽,并可被用于研究免疫反应。
T80866 VIP(Guinea pig) TFA

Vasoactive Intestinal Peptide, guinea pig TFA

VIP Guinea pig TFA,作为一种胃肠激素,兼具神经递质功能,能够刺激胚胎生长,起到营养和有丝分裂因子的作用。
T76093 Peptide YY (pig)

Peptide YY (pig) 是一种由36个氨基酸组成的胃肠肽,源自猪的十二指肠。该化合物通过激活Y2 receptor来降低食欲和食物摄入量,主要在胰腺的内分泌细胞中发现,对肠动力和心血管系统具有重要影响。
T76063 Beta-defensin 1, pig

Beta-defensin 1, pig 是一种在猪舌黏膜中主要发现的抗菌肽,对包括大肠杆菌、鼠伤寒沙门氏菌、单核细胞增生性李斯特菌、金黄色葡萄球菌、百日咳博德特氏菌和白色念珠菌在内的多种细菌显示出活性。
T0930 Sulfadiazine

Sulphadiazine,磺胺嘧啶

Antibacterial; Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。
T76063L Beta-defensin 1, pig TFA

Beta-defensin 1, pig TFA 是一种在猪舌黏膜中主要发现的抗菌肽,对多种细菌如大肠杆菌、鼠伤寒沙门氏菌、单核细胞增生性李斯特菌、金黄色葡萄球菌、百日咳博德特氏菌和白色念珠菌等显示出抗菌活性。
T76064 Beta-defensin 103 isoform X1, pig

Beta-defensin 103 isoform X1, pig 是一种抗菌肽、在多种生物体内被发现,参与了先天性免疫防线。
T76064L Beta-defensin 103 isoform X1, pig TFA

Beta-defensin 103 isoform X1, pig TFA 是一种抗菌肽、在多种生物体内被发现,参与了先天性免疫防线。
T6992 Sulfadiazine sodium

Sulfadiazin-natrium,磺胺嘧啶钠,Sodium sulfadiazine

Others; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Others
Sulfadiazine sodium (Sulfadiazin-natrium) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。
T22033 ARC 239 dihydrochloride

Norepinephrine Neuroscience
ARC 239 dihydrochloride 是一种选择性 α2B 肾上腺素受体拮抗剂。
T20570 Labetalol

Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne

Adrenergic Receptor GPCR/G Protein; Neuroscience
Labetalol (Apo-Labetalol) 是一种抗高血压药物,可用于心血管疾病的研究,如妊娠期高血压。它是一种口服具有活性的选择性 α1- 和非选择性 β-肾上腺素能受体 (adrenergic receptor) 竞争性拮抗剂。
T21688L Cytochrome c - pigeon (88-104) Acetate

Cytochrome c - pigeon (88-104) Acetate (86579-06-8 Free base)

Others Others
Cytochrome c - pigeon (88-104) Acetate (Cytochrome c - pigeon ) 对 COOH 末端序列 88-1041 内的肽具有特异性。
T62560 Sirpiglenastat

DRP-104

Glutaminase Proteases/Proteasome
Sirpiglenastat (DRP-104) 是一种谷氨酰胺 (glutamine) 拮抗剂,是DON的前药,具有抗肿瘤活性,通过抑制谷氨酰胺代谢和刺激先天性和适应性免疫系统来发挥作用。
T20045 C.I. Pigment Red 172

C.I. Acid Red 51:1,Pigment Red 172,Erythrosine-aluminum lake,C.I. Food Red 14:1,Tetraiodofluorescein,Aluminum,Acid Red 51:1

C.I. Pigment Red 172 (C.I. Food Red 14:1) 是一种食品添加剂。
T34064 Pigment Blue 15

AI3-26192,EINECS 205-685-1,Blue GLA,Blue pigment,Phthalocyanine Blue BN

Pigment Blue 15, also called by many names (EINECS 205-685-1), is a bright, crystalline, synthetic blue pigment from the group of phthalocyanine dyes. Its brilliant blue is frequently used in paints and dyes. It is highly valued for its superior propertie
T126010 Epigambogellic acid

Epigambogellic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126010。
T123856 Apigenin 7,4'-di-O-alloside

Apigenin 7,4'-di-O-alloside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T123856。
T126101 Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside

Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126101。
T20059 C.I. Pigment Red 60

NSC 12455,Acid Anthracene Red G,Siloton Red 3B,NSC12455,NSC-12455,Hispacrom Red B

C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.
T126303 10alpha-Hydroxyepigambogic acid

10alpha-Hydroxyepigambogic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126303。
T39820 Dapiglutide

ZP7570

Dapiglutide (ZP7570) is a long-acting dual agonist of glucagon-like peptide-1 receptor (GLP-1R) and glucagon-like peptide-2 receptor (GLP-2R) that holds potential for short bowel syndrome (SBS) research.
T34065 Pigment Red 57

Lithol Rubine Na,Japan Red 201,Rubine Red RR 1253,Lithol rubin B

Pigment Red 57, also known as D & C Red No. 6, is a synthetic dye produced from petroleum or coal tar sources; this dye is FDA-approved for use in pharmaceuticals and cosmetics.
T126160 Apigenin 7-[rhamnosyl-(1->2)-galacturonide]

Apigenin 7-[rhamnosyl-(1->2)-galacturonide] 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126160。
T126415 9R-10alpha-Hydroxyepigambogic acid

9R-10alpha-Hydroxyepigambogic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126415。
T40742 Pigment Red 22

Pigment Red 22, a coloring agent, is a versatile compound employed in the formulation of various cosmetic products, including cleansing products, makeup, moisturizers, and night skin care products.
T124311 Apigenin 6,8-di-C-alpha-L-arabinopyranoside

Apigenin 6,8-di-C-alpha-L-arabinopyranoside 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124311,CAS号为 73140-47-3。
T20987 C.I. Pigment Yellow 74

C.I. Pigment Yellow 74 is a bioactive chemical.
T40609 Pigment Red 48:4

Pigment Red 48:4 is a manganese-complex dye suitable for applications in printing ink and paint systems.
T17301 opigolix

Others Others
Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
T82458 Epigenetic factor-IN-1

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Epigenetic factor-IN-1(40569Z)是一种针对SIRT7显示出强效结合能力的表观遗传因子抑制剂,常用于肝癌的研究领域。
T30670 C.I. Pigment Red 4

CCRIS 4907,HSDB 7720,Oralith Red,C.I. 12085

C.I. Pigment Red 4可用于印刷油墨、油漆、水彩、油漆及砚色、橡胶、天然生漆、化妆品、油漆及涂料的印刷颜色。它是黄红色粉末,颜色鲜艳。不溶于水,微溶于乙醇和苯。它在浓硝酸中呈现鲜红色,在稀氢氧化钠溶液中保持鲜红色;在乙醇-氢氧化钾溶液中呈紫色。具有良好的流动性和抗遮盖性,耐热性差。
TP2461 Lpigppal

Lysyl-prolyl-isoleucyl-glutamyl-phenylalanyl-4-nitrophenylalanyl-arginyl-leucine

Lysyl-prolyl-isoleucyl-glutamyl-phenylalanyl-4-nitrophenylalanyl-arginyl-leucine is a bioactive chemical.
T30671 C.I. Pigment Yellow 14

C.I. Pigment Yellow 14 is a yellow dye.
T124530 Apigenin-7-O-glucuronide-6'-ethyl ester

Apigenin-7-O-glucuronide-6'-ethyl ester 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124530。
T72013 Epigenetic Multiple Ligand

Epigenetic Multiple Ligand is a cell-permeable inhibitor of substrate processing by several chromatin-associated enzymes, including SIRT1/2, H3/SET7, H3/p300/CBP, H4/RmtA, PABP1/CARM1, and H4/PRMT1. It acts by inducing either apoptosis or granulocytic differentiation.
T10537 BI-749327

TRP/TRPV Channel Membrane transporter/Ion channel
BI-749327是高选择性、口服有效的TRPC6拮抗剂,对小鼠、人、豚鼠 TRPC6 作用的IC50值分别为 13 nM、19 nM 和 15 nM。BI-749327对小鼠 TRPC6 选择性比 TRPC3 高出 85 倍, 比TRPC7高出42 倍。
T38648L Cecropin P1, porcine acetate

Endogenous Metabolite Metabolism
Cecropin P1, porcine acetate 是一种在 Hyalophora cecropia 和猪肠道中发现的抗菌肽。
TP1819L Substance P 1-9 aceate

Neurotensin Receptor GPCR/G Protein
Substance P 1-9 aceate 是九肽,可减少豚鼠回肠和膀胱对 P 物质的失活。
T16026 MCI826

P-gp; LTR Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
MCI826 是一种具有有效性和选择性的 P-glycoprotein (P-gp)和肽白三烯 (p-LTs) 拮抗剂,在豚鼠晚期哮喘模型中显示出抗哮喘活性。
T19654 Guanoclor

胍氯酚,VATENSOL

Others Others
Guanoclor (VATENSOL) 也称为guanochlor,是一种交感神经药物。已知它与猪肾膜中的非肾上腺素能位点结合。
T16564 PPADS tetrasodium

P2X Receptor; Na+/Ca2+ Exchanger Membrane transporter/Ion channel; Neuroscience
PPADS tetrasodiuma 是一种有效的 P2X 受体拮抗剂,也是是豚鼠气道平滑肌 Na/Ca²⁺ 交换逆模式的抑制剂,对谷氨酸/NMDA毒性有神经保护作用。PPADS tetrasodiuma 抑制 P2X1、P2X-2、P2X-3 和 P2X-5。
T27627 Iroxanadine

BRX005,BRX-235,BRX-005,BRX235,BRX 005,BRX 235

p38 MAPK MAPK
Iroxanadine (BRX-005) 是一种新型小分子MAPK p38 抑制剂,诱导p38 SAPK 的磷酸化,在用去氧肾上腺素预先收缩的豚鼠肺动脉制剂中诱导浓度依赖性松弛,可用于治疗动脉粥样硬化、糖尿病血管病,微血管心绞痛和外周动脉疾病等血管疾病。
T12267 NSP-805

PDE Metabolism
NSP-805 是一种强心剂,是一种选择性的 phosphodiesterase 3 抑制剂,具有舒张血管的作用。
TP2026L GRP (porcine) acetate

GRP (porcine) acetate(74815-57-9 Free base)

Others Others
GRP (porcine) acetate 是从猪胰腺中提取的胃泌素释放肽。 GRP (porcine) acetate 可能在猪胰腺内分泌和外分泌的副交感神经调节中起作用。
T14941 CGP37157

7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one

Na+/Ca2+ Exchanger Membrane transporter/Ion channel
CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) 是一种 Na+/Ca2+ 交换抑制剂,抑制 Na+ 诱导的豚鼠心脏线粒体中 Ca2+ 的释放,IC50 为 0.8 μM。
T15272 Febantel

Parasite Microbiology/Virology
Febantel 是一种用于家禽和家畜的蛔虫、绦虫感染的驱虫剂。
TP1572 GR-73632

Neurokinin receptor GPCR/G Protein; Neuroscience
GR-73632 强效和选择性速激肽 NK1 受体激动剂,可通过传递瘙痒信号的 NK1 受体直接作用于初级感觉神经元的外周末端。
TP1425 Motilin (26-47), human, porcine

胃动素 (人类,猪)

Motilin Receptor GPCR/G Protein
Motilin (26-47), human, porcine 是内源性 motilin 受体的激动剂,在中国仓鼠卵巢细胞中,Ki 值和EC50值分别为 2.3 和 0.3 nM。

化合物

Myelin Basic Protein (MBP) (68-82), guinea pig
Cat.No: TP1092
Synonym: MBP (68-82), guinea pig,豚鼠髓磷脂碱性蛋白片段68-82
Target: Others
VIP(Guinea pig)
Cat.No: TP2210
Synonym: VIP (guinea pig)
Target: Others
Dynorphin B 29 (pig)
Cat.No: T82518
Synonym: Leumorphin (pig)
Target:
VIP(Guinea pig) TFA
Cat.No: T80866
Synonym: Vasoactive Intestinal Peptide, guinea pig TFA
Target:
Peptide YY (pig)
Cat.No: T76093
Synonym:
Target:
Beta-defensin 1, pig
Cat.No: T76063
Synonym:
Target:
Sulfadiazine
Cat.No: T0930
Synonym: Sulphadiazine,磺胺嘧啶
Target: Antibacterial, Antibiotic, Parasite, Autophagy
Beta-defensin 1, pig TFA
Cat.No: T76063L
Synonym:
Target:
Beta-defensin 103 isoform X1, pig
Cat.No: T76064
Synonym:
Target:
Beta-defensin 103 isoform X1, pig TFA
Cat.No: T76064L
Synonym:
Target:
Sulfadiazine sodium
Cat.No: T6992
Synonym: Sulfadiazin-natrium,磺胺嘧啶钠,Sodium sulfadiazine
Target: Others, Antibacterial, Antibiotic, Parasite
ARC 239 dihydrochloride
Cat.No: T22033
Synonym:
Target: Norepinephrine
Labetalol
Cat.No: T20570
Synonym: Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne
Target: Adrenergic Receptor
Cytochrome c - pigeon (88-104) Acetate
Cat.No: T21688L
Synonym: Cytochrome c - pigeon (88-104) Acetate (86579-06-8 Free base)
Target: Others
Sirpiglenastat
Cat.No: T62560
Synonym: DRP-104
Target: Glutaminase
C.I. Pigment Red 172
Cat.No: T20045
Synonym: C.I. Acid Red 51:1,Pigment Red 172,Erythrosine-aluminum lake,C.I. Food Red 14:1,Tetraiodofluorescein,Aluminum,Acid Red 51:1
Target:
Pigment Blue 15
Cat.No: T34064
Synonym: AI3-26192,EINECS 205-685-1,Blue GLA,Blue pigment,Phthalocyanine Blue BN
Target:
Epigambogellic acid
Cat.No: T126010
Synonym:
Target:
Apigenin 7,4'-di-O-alloside
Cat.No: T123856
Synonym:
Target:
Apigenin 6-C-(2-O-feruloyl)glucoside 8-C-glucoside
Cat.No: T126101
Synonym:
Target:
C.I. Pigment Red 60
Cat.No: T20059
Synonym: NSC 12455,Acid Anthracene Red G,Siloton Red 3B,NSC12455,NSC-12455,Hispacrom Red B
Target:
10alpha-Hydroxyepigambogic acid
Cat.No: T126303
Synonym:
Target:
Dapiglutide
Cat.No: T39820
Synonym: ZP7570
Target:
Pigment Red 57
Cat.No: T34065
Synonym: Lithol Rubine Na,Japan Red 201,Rubine Red RR 1253,Lithol rubin B
Target:
Apigenin 7-[rhamnosyl-(1->2)-galacturonide]
Cat.No: T126160
Synonym:
Target:
9R-10alpha-Hydroxyepigambogic acid
Cat.No: T126415
Synonym:
Target:
Pigment Red 22
Cat.No: T40742
Synonym:
Target:
Apigenin 6,8-di-C-alpha-L-arabinopyranoside
Cat.No: T124311
Synonym:
Target:
C.I. Pigment Yellow 74
Cat.No: T20987
Synonym:
Target:
Pigment Red 48:4
Cat.No: T40609
Synonym:
Target:
opigolix
Cat.No: T17301
Synonym:
Target: Others
Epigenetic factor-IN-1
Cat.No: T82458
Synonym:
Target: Sirtuin
C.I. Pigment Red 4
Cat.No: T30670
Synonym: CCRIS 4907,HSDB 7720,Oralith Red,C.I. 12085
Target:
Lpigppal
Cat.No: TP2461
Synonym: Lysyl-prolyl-isoleucyl-glutamyl-phenylalanyl-4-nitrophenylalanyl-arginyl-leucine
Target:
C.I. Pigment Yellow 14
Cat.No: T30671
Synonym:
Target:
Apigenin-7-O-glucuronide-6'-ethyl ester
Cat.No: T124530
Synonym:
Target:
Epigenetic Multiple Ligand
Cat.No: T72013
Synonym:
Target:
BI-749327
Cat.No: T10537
Synonym:
Target: TRP/TRPV Channel
Cecropin P1, porcine acetate
Cat.No: T38648L
Synonym:
Target: Endogenous Metabolite
Substance P 1-9 aceate
Cat.No: TP1819L
Synonym:
Target: Neurotensin Receptor
MCI826
Cat.No: T16026
Synonym:
Target: P-gp, LTR
Guanoclor
Cat.No: T19654
Synonym: 胍氯酚,VATENSOL
Target: Others
PPADS tetrasodium
Cat.No: T16564
Synonym:
Target: P2X Receptor, Na+/Ca2+ Exchanger
Iroxanadine
Cat.No: T27627
Synonym: BRX005,BRX-235,BRX-005,BRX235,BRX 005,BRX 235
Target: p38 MAPK
NSP-805
Cat.No: T12267
Synonym:
Target: PDE
GRP (porcine) acetate
Cat.No: TP2026L
Synonym: GRP (porcine) acetate(74815-57-9 Free base)
Target: Others
CGP37157
Cat.No: T14941
Synonym: 7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one
Target: Na+/Ca2+ Exchanger
Febantel
Cat.No: T15272
Synonym:
Target: Parasite
GR-73632
Cat.No: TP1572
Synonym:
Target: Neurokinin receptor
Motilin (26-47), human, porcine
Cat.No: TP1425
Synonym: 胃动素 (人类,猪)
Target: Motilin Receptor
Cat. No. Product Name Target Signaling Pathways
TN1608 (-)-Epigallocatechin-3-(3''-O-methyl) gallate

(-)-EGCG-3''-O-ME

Antioxidant; Antibacterial Microbiology/Virology; oxidation-reduction
(-)-Epigallocatechin-3-(3''-O-methyl) gallate ((-)-EGCG-3''-O-ME) 是从茶叶中分离出的一种天然产物,具有很强的抗氧化、细胞毒性和抗菌活性,可增强蚀刻漂洗粘合剂与牙本质的粘合稳定性。
T5S1026 Apigenin-7-glucuronide

Apigenin 7-O-glucuronide,芹菜素-7-葡萄糖醛酸

MMP Proteases/Proteasome
Apigenin-7-glucuronide (Apigenin 7-O-glucuronide) 能够抑制基质金属蛋白酶的活性,其对 MMP-3 (IC50:12.87 μM),MMP-8 (IC50:22.39 μM),MMP-9 (IC50:17.52 μM),MMP-13 (IC50:0.27 μM)。
T5S1526 Apigenin-7-O-(2G-rhamnosyl)gentiobioside

Apigenin 7-O-(2G-rhamnosyl)gentiobioside,芹菜素-7-0-(2G-鼠李糖)龙胆糖苷,Apigenin 7-(2-Rhamnosylgentiobioside),金银花

Others Others
Apigenin-7-O-(2G-rhamnosyl)gentiobioside 是一种黄酮类苷化合物,从Lonicera gracilipes var. glandulosa 中提取得到。
T5690 7,4'-Di-O-methylapigenin

芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE

Amylase Metabolism
7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) 可能具有抗真菌c.zeyheri 的作用,是一种潜在的抗真菌药物。它还能抑制药物流出泵(IC50 = 51.64μg /毫升)。
TN2353 8-Hydroxyapigenin

Isoscutellarein

Antioxidant; Influenza Virus Microbiology/Virology; oxidation-reduction
8-Hydroxyapigenin (Isoscutellarein) 是从植物黄芩中提取的黄铜类化合物,具有抗炎抗氧和抗流感病毒的活性。
T2988 (-)-Epigallocatechin Gallate

Epigallocatechol Gallate,(-)-表没食子儿茶素没食子酸酯,EGCG

Ferroptosis; Reactive Oxygen Species; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
(-)-Epigallocatechin Gallate (EGCG) 是茶类黄酮,具有强大的抗氧化,抗炎和抗癌作用。它可抑制EGFR 信号传导,有抗癌作用。它是谷氨酸脱氢酶 1/2 抑制剂。它通过激活细胞色素c 氧化酶来诱导氧化磷酸化。
TN7121 d-Epigalbacin

(-)-Zuonin A,表加巴辛

JNK MAPK
d-Epigalbacin ((-)-Zuonin A) 是一种天然木质素。d-Epigalbacin 是一种强效、选择性的JNKs 抑制剂,JNK1、JNK2和JNK3的IC50s 分别为1.7μM、2.9μM 和1.74μM。
T41017 Epigambogic acid

Epigambogic acid 是一种来自藤黄的小分子化合物,具有抗肿瘤、止咳、祛痰和抗炎活性。
T4S0295 Apigenin 7-glucoside

波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Apigenin 7-glucoside (Cosmosiin) 是一种 ROS 清除剂,具有抗增殖、抗氧化作用。
TN1082 Apigenin 7-O-malonylglucoside

Apigenin 7-O-(6''-O-malonylglucoside)

Apigenin 7-O-malonylglucoside (Apigenin 7-O-(6''-O-malonylglucoside)) 存在于菊花中,是一种黄酮,也是一种糖苷。
T5S0092 Epigoitrin

BA-51-090278,Goitrine,D-Goitrin,表告依春,Goitrin

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Epigoitrin (Goitrin) 是板蓝根中的一种天然生物碱,可通过线粒体抗病毒信号降低对流感病毒的易感性,具有抗病毒活性。
T2175 Apigenin

C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400

P450; Autophagy Autophagy; Metabolism
Apigenin (NSC 83244) 是从韩信草中提取的一种天然产物,是一种竞争性CYP2C9抑制剂,Ki 为 2 μM。它被用作镇静剂、温和的镇痛剂和安眠药。
T2987 (-)-Epigallocatechin

表没食子儿茶素,(-)-表没食子儿茶素,l-Epigallocatechin,Epigallocatechin,EGC

MMP; Autophagy Autophagy; Proteases/Proteasome
(-)-Epigallocatechin (Epigallocatechin) 是绿茶中含量最丰富的黄酮类天然产物,可与未折叠的天然多肽结合,阻止转化为淀粉样蛋白原纤维。
TN1609 Epigomisin O

Others Others
Epigomisin O is a natural product from Schizandra chinensis.
TN3969 Epiguajadial B

Others Others
Epiguajadial B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3969,CAS号为 1411629-26-9。
T82987 Apigenin 7-O-sophoroside

Apigenin 7-O-sophoroside, 一种黄酮苷, 可以分离自Lonicera gracilipes var. glandulosa。
TN2422 6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide

Others Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide is a natural product from Carthamus tinctorius Linn.
T10348 Apigenin-7-diglucuronide

Others Others
Apigenin-7-diglucuronide is a flavonoid glycoside that exists in an assortment of medicinal plants with anti-inflammatory or ant-oxidant activities. It protects retinas against bright light-induced photoreceptor degeneration through the inhibition of reti
T83465 10α-Hydroxyepigambogic acid

10α-Hydroxyepigambogic acid,一种从Garcinia hanburyi中提取的化合物,适用于肿瘤研究领域。
T83408 2',3'-Dihydro-2'-hydroxyprotoapigenone

2',3'-Dihydro-2'-hydroxyprotoapigenone 是一种蕨类植物中天然存在的原黄酮化合物。
TN3430 Apigenin 4'-O-rhamnoside

Others Others
Apigenin-4'-O-rhamnosylglucoside can strongly inhibit the classical pathway of the complement system.
T82985 Apigenin-6-C-β-D-xylopyranosyl-8-C-α-L-arabinopyranoside

Apigenin-6-C-β-D-xylopyranosyl-8-C-α-L-arabinopyranoside,一类黄酮化合物,具抗氧化活性,源自中药铁皮石斛。
TN5500 3',3'''-Biapigenin

3',3'''-Biapigenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5500,CAS号为 151455-26-4。
TN3213 7,4'-Di-O-methylapigenin 5-O-xylosylglucoside

Others Others
7,4'-Di-methylapigenin-5-O-xylosylglucoside shows inhibitory activity for nitric oxide(NO) production by activated RAW 264.7 cells.
TN3212 7,4-Di-O-methylapigenin 5-O-glucoside

Others Others
7,4-Di-O-methylapigenin 5-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3212,CAS号为 197018-71-6。
TN6287 Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside

Anisofolin B

Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6287,CAS号为 1448779-19-8。
T75578 Apigravin

Apigravin 是一种有效的抗菌剂。Apigravin 对 Bacillus subtilis 具有抗菌活性,MIC 值为 61 μM。
T81367 Protoapigenin

Protoapigenin是一种从Macrothelypteris torresiana地上部分分离得到的黄酮类化合物。
TN1394 Apigenin6-C-α-L-arabinopyranosyl-8-C-β-D-xylopyranoside

Apigenin 6-C-alpha-L-arabinopyranosyl-8-C-beta-D-xylopyranoside,芹菜素-6-C-Α-L-吡喃阿拉伯糖-8-C-Β-D-吡喃木糖苷,apigenin6-c-alpha-l-arabinopyranosyl-8-c-beta-d-xylopyranoside

Others Others
Apigenin 6-C-alpha-L-arabinopyranosyl-8-C-beta-D-xylopyranoside is a natural product from Viola yedoensis.
TN5356 Epiglobulol

Epiglobulol shows antibacterial activities, it can strongly inhibit the growth of foodborne microorganisms. Epiglobulol can inhibit the recombinant human UDP-glucuronosyltransferase (UGT) 2B7, it may serve as valuable lead structures for the design of pot
T82986 Apigenin triacetate

Apigenin triacetate, 作为禾谷镰刀菌的代谢产物,其含量可通过壳聚糖处理以实现下调。该化合物系由芹菜素派生。
TN2930 3-Epiglochidiol diacetate

Others Others
3-Epiglochidiol diacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2930,CAS号为 6587-37-7。
TN3432 Apigenin 5-O-neohesperidoside

Others Others
Apigenin 5-O-neohesperidoside is a natural product from Thesium chinese.
T83284 5-O-Primeverosylapigenin

5-O-Primeverosylapigenin为初级龙胆碱类化合物,源自龙胆科植物,通过分离提取获得。
TN3431 Apigenin 5-O-beta-D-glucopyranoside

Others Others
Apigenin 5-O-beta-D-glucopyranoside has inhibitory activity against the enzyme yeast a-glucosidase, withthe IC50 value of 287.12 muM.
TN6606 Apigeninidin chloride

Apigeninidin chloride 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6606,CAS号为 1151-98-0。
TN6304 Apigenin 4'-O-(2'',6''-di-O-E-p-coumaroyl)glucoside

Apigenin 4'-O-(2'',6''-di-O-E-p-coumaroyl)glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6304,CAS号为 71781-79-8。
TN3264 8,3'-Diprenylapigenin

Others Others
8,3'-Diprenylapigenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3264,CAS号为 955135-37-2。
TN2929 3-Epiglochidiol

Others Others
3-Epiglochidiol是一种天然产物,属于大戟科算盘子属,其产品编号为 TN2929,CAS号为 29028-10-2。3-Epiglochidiol可用作对照参考。
TN1241 3,8''-Biapigenin

3,8'-Biapigenin,3,8″-双芹菜素

ROS Immunology/Inflammation
3, 8''-Biapigenin can modulate intracellular ROS production.
TN5496 2'',3''-Dihydro-3',3'''-biapigenin

2,3-Dihydro-3',3'''-biapigenin

2'',3''-Dihydro-3',3'''-biapigenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5496,CAS号为 151455-25-3。
T81366 Protoapigenin 4′-O-β-D-glucoside

Protoapigenin 4'-O-β-D-glucoside是一种从Thelypteris torresiana中分离得到的黄酮苷。
T81365 Protoapigenone

Protoapigenone 是一种可从蕨类植物中分离得到的抗肿瘤剂。该化合物对 Hep G2、Hep 3B、MCF-7、A549 及 MDAMB-231 肿瘤细胞系展示了显著的抑制活性,其 IC50s 分别为 1.60、0.23、0.78、3.88 和 0.27 μg/mL。
TN5447 Apigenin 7-O-methylglucuronide

芹菜素-7-O-β-D-葡萄糖醛酸甲酯,Apigenin-7-O-β-D-glucuronide methyl ester

Apigenin 7-O-methylglucuronide did not affect GAG level or secretion, may potentially be used in osteogenesis imperfecta (OI) type I pharmacotherapy in patients with normal GAG content. Apigenin 7-O-methylglucuronide which normalized collagen synthesis in
TN2907 3,6-Dimethoxyapigenin

Others Others
3,6-Dimethoxyapigenin是一种天然产物,属于无患子科车桑子属,其产品编号为 TN2907,CAS号为 22697-65-0。3,6-Dimethoxyapigenin可用作对照参考。
TN1266 3-O-Methylquercetin

IL Receptor; cAMP; PDE GPCR/G Protein; Immunology/Inflammation; Metabolism
3-O-Methylquercetin 是分离自植物Rhamnus nakaharai 的天然产物,可抑制总 cAMP 和cGMP-phosphodiesterase (PDE)。它对PDE1、PDE5、PDE 和PDE4的IC50分别是31.9 μM、86.9 μM、18.6 μM 和1.6 μM。
T4S1422 Praeruptorin E

白花前胡素 E,白花前胡素E

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Praeruptorin E 是白花前胡中的一种主要成分,是钙拮抗剂,pD2′值为 5.2。
T6S2025 8-​O-​Acetylharpagide

8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide

Antibacterial Microbiology/Virology
8-O-Acetylharpagide 是从 Ajuga reptans 中分离得到的一种环烯醚萜,有抗肿瘤、抗病毒、抗菌和抗炎作用。它对豚鼠的离体平滑肌有生物活性。
PDK0014 3-Methylxanthine

Endogenous Metabolite Metabolism
3-Methylxanthine 是一种黄嘌呤衍生物和环磷酸鸟苷(GMP)抑制剂,在豚鼠分离的气管肌肉中测得其IC50值为 920 μM。
T6S0033 Crotonoside

巴豆苷;异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE

Others; FLT; HDAC Angiogenesis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Others; Tyrosine Kinase/Adaptors
Crotonoside (Isoguanosine) 是从中草药巴豆中分离出来的一种天然产物。 它抑制 FLT3 和 HDAC3/6,有治疗急性髓性白血病 (AML)的研究潜力。
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天然产物

(-)-Epigallocatechin-3-(3''-O-methyl) gallate
Cat.No: TN1608
Synonym: (-)-EGCG-3''-O-ME
Target: Antioxidant, Antibacterial
Apigenin-7-glucuronide
Cat.No: T5S1026
Synonym: Apigenin 7-O-glucuronide,芹菜素-7-葡萄糖醛酸
Target: MMP
Apigenin-7-O-(2G-rhamnosyl)gentiobioside
Cat.No: T5S1526
Synonym: Apigenin 7-O-(2G-rhamnosyl)gentiobioside,芹菜素-7-0-(2G-鼠李糖)龙胆糖苷,Apigenin 7-(2-Rhamnosylgentiobioside),金银花
Target: Others
7,4'-Di-O-methylapigenin
Cat.No: T5690
Synonym: 芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE
Target: Amylase
8-Hydroxyapigenin
Cat.No: TN2353
Synonym: Isoscutellarein
Target: Antioxidant, Influenza Virus
(-)-Epigallocatechin Gallate
Cat.No: T2988
Synonym: Epigallocatechol Gallate,(-)-表没食子儿茶素没食子酸酯,EGCG
Target: Ferroptosis, Reactive Oxygen Species, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite, Autophagy
d-Epigalbacin
Cat.No: TN7121
Synonym: (-)-Zuonin A,表加巴辛
Target: JNK
Epigambogic acid
Cat.No: T41017
Synonym:
Target:
Apigenin 7-glucoside
Cat.No: T4S0295
Synonym: 波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin
Target: Reactive Oxygen Species, HIV Protease
Apigenin 7-O-malonylglucoside
Cat.No: TN1082
Synonym: Apigenin 7-O-(6''-O-malonylglucoside)
Target:
Epigoitrin
Cat.No: T5S0092
Synonym: BA-51-090278,Goitrine,D-Goitrin,表告依春,Goitrin
Target: Antiviral, Influenza Virus
Apigenin
Cat.No: T2175
Synonym: C.I. Natural Yellow 1,4',5,7-Trihydroxyflavone,NSC 83244,金银花,Apigenol,芹菜素,LY 080400
Target: P450, Autophagy
(-)-Epigallocatechin
Cat.No: T2987
Synonym: 表没食子儿茶素,(-)-表没食子儿茶素,l-Epigallocatechin,Epigallocatechin,EGC
Target: MMP, Autophagy
Epigomisin O
Cat.No: TN1609
Synonym:
Target: Others
Epiguajadial B
Cat.No: TN3969
Synonym:
Target: Others
Apigenin 7-O-sophoroside
Cat.No: T82987
Synonym:
Target:
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide
Cat.No: TN2422
Synonym:
Target: Others
Apigenin-7-diglucuronide
Cat.No: T10348
Synonym:
Target: Others
10α-Hydroxyepigambogic acid
Cat.No: T83465
Synonym:
Target:
2',3'-Dihydro-2'-hydroxyprotoapigenone
Cat.No: T83408
Synonym:
Target:
Apigenin 4'-O-rhamnoside
Cat.No: TN3430
Synonym:
Target: Others
Apigenin-6-C-β-D-xylopyranosyl-8-C-α-L-arabinopyranoside
Cat.No: T82985
Synonym:
Target:
3',3'''-Biapigenin
Cat.No: TN5500
Synonym:
Target:
7,4'-Di-O-methylapigenin 5-O-xylosylglucoside
Cat.No: TN3213
Synonym:
Target: Others
7,4-Di-O-methylapigenin 5-O-glucoside
Cat.No: TN3212
Synonym:
Target: Others
Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside
Cat.No: TN6287
Synonym: Anisofolin B
Target:
Apigravin
Cat.No: T75578
Synonym:
Target:
Protoapigenin
Cat.No: T81367
Synonym:
Target:
Apigenin6-C-α-L-arabinopyranosyl-8-C-β-D-xylopyranoside
Cat.No: TN1394
Synonym: Apigenin 6-C-alpha-L-arabinopyranosyl-8-C-beta-D-xylopyranoside,芹菜素-6-C-Α-L-吡喃阿拉伯糖-8-C-Β-D-吡喃木糖苷,apigenin6-c-alpha-l-arabinopyranosyl-8-c-beta-d-xylopyranoside
Target: Others
Epiglobulol
Cat.No: TN5356
Synonym:
Target:
Apigenin triacetate
Cat.No: T82986
Synonym:
Target:
3-Epiglochidiol diacetate
Cat.No: TN2930
Synonym:
Target: Others
Apigenin 5-O-neohesperidoside
Cat.No: TN3432
Synonym:
Target: Others
5-O-Primeverosylapigenin
Cat.No: T83284
Synonym:
Target:
Apigenin 5-O-beta-D-glucopyranoside
Cat.No: TN3431
Synonym:
Target: Others
Apigeninidin chloride
Cat.No: TN6606
Synonym:
Target:
Apigenin 4'-O-(2'',6''-di-O-E-p-coumaroyl)glucoside
Cat.No: TN6304
Synonym:
Target:
8,3'-Diprenylapigenin
Cat.No: TN3264
Synonym:
Target: Others
3-Epiglochidiol
Cat.No: TN2929
Synonym:
Target: Others
3,8''-Biapigenin
Cat.No: TN1241
Synonym: 3,8'-Biapigenin,3,8″-双芹菜素
Target: ROS
2'',3''-Dihydro-3',3'''-biapigenin
Cat.No: TN5496
Synonym: 2,3-Dihydro-3',3'''-biapigenin
Target:
Protoapigenin 4′-O-β-D-glucoside
Cat.No: T81366
Synonym:
Target:
Protoapigenone
Cat.No: T81365
Synonym:
Target:
Apigenin 7-O-methylglucuronide
Cat.No: TN5447
Synonym: 芹菜素-7-O-β-D-葡萄糖醛酸甲酯,Apigenin-7-O-β-D-glucuronide methyl ester
Target:
3,6-Dimethoxyapigenin
Cat.No: TN2907
Synonym:
Target: Others
3-O-Methylquercetin
Cat.No: TN1266
Synonym:
Target: IL Receptor, cAMP, PDE
Praeruptorin E
Cat.No: T4S1422
Synonym: 白花前胡素 E,白花前胡素E
Target: Others, Calcium Channel
8-​O-​Acetylharpagide
Cat.No: T6S2025
Synonym: 8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide
Target: Antibacterial
3-Methylxanthine
Cat.No: PDK0014
Synonym:
Target: Endogenous Metabolite
Crotonoside
Cat.No: T6S0033
Synonym: 巴豆苷;异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE
Target: Others, FLT, HDAC
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