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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6393 ARQ 621

Kinesin Cytoskeletal Signaling
ARQ 621 是一种变构和选择性 Eg5 有丝分裂运动蛋白抑制剂,具有抗肿瘤活性。
T11689 ITI-214

ITI214

PDE Metabolism
ITI-214 是一种中枢神经系统活性抑制剂,具有口服生物活性的PDE1抑制剂 (Kiof 58 pM),对其他 PDE 家族成员和一系列酶、受体、转运体和离子通道具有良好的选择性,在各种运动和认知功能的动物模型中显示出有效性。
T22103 ML-193

CID 1261822

Cannabinoid Receptor GPCR/G Protein
ML-193 (CID 1261822) 是一种有效的选择性GPR55拮抗剂,IC50值为 221 nM,对 GPR55 的选择性比 GPR35、CB1 和 CB2 高 27 倍以上,可改善帕金森病 (PD) 大鼠的运动和感觉运动缺陷。
T13554 Arimoclomol maleate

BRX-220

HSP Cytoskeletal Signaling; Metabolism
Arimoclomol maleate (BRX-220) 是一种热休克蛋白 (HSP) 的共诱导剂。它通过增强 Hsp 表达来保护运动神经元,进而通过蛋白酶体-泛素系统直接影响蛋白质聚集和错误折叠装配体的清除
T1030 Triprolidine hydrochloride monohydrate

盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Triprolidine hydrochloride monohydrate 是一种组胺 H1 拮抗剂,用于过敏性鼻炎、哮喘。
T4641 Branaplam

LMI 070,NVS-SM1

Others; Potassium Channel; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Others
Branaplam (LMI 070) 是一种高效、选择性和口服活性的小分子 SMN2 剪接调节剂,对 SMN 的 EC50为 20 nM。它可提高全长 SMN 蛋白并延长其生存期,也抑制 hERG,IC50为 6.3 μM。
T13553 Arimoclomol

阿瑞洛莫,BRX-220 free base

HSP Cytoskeletal Signaling; Metabolism
Arimoclomol (BRX-220 free base) 是热休克蛋白 (HSP) 的共诱导剂,可用于治疗肌萎缩侧索硬化症的研究。
T24047 Etilevodopa hydrochloride

Levodopa ethyl ester,Etilevodopa HCl, L-DOPA ethyl ester

Others; Dopamine Receptor; Drug Metabolite GPCR/G Protein; Metabolism; Neuroscience; Others
Etilevodopa hydrochloride (L-DOPA ethyl ester) 是 Levodopa 的前药,在胃肠道中被非特异性酯酶快速水解产生 Levodopa 和乙醇。Levodopa 是多巴胺的前体,有助于中枢神经系统的渗透和传递多巴胺。Etilevodopa HCl 可用于帕金森病 (PD)的相关研究。
T3336 Rg3039

PF-06687859

Others Others
Rg3039 (PF-06687859) 是一种具有口服活性、能够透过血脑屏障的DcpS 抑制剂,其IC50=0.069 nM。
T27084 Crisdesalazine

AAD2004,AAD 2004,AAD-2004

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Crisdesalazine (AAD 2004) 是微粒体前列腺素 E2 合酶 1 (mPGES-1) 的抑制剂。 Crisdesalazine 可减少自噬体形成、轴索病变和运动神经元变性,改善运动功能并延长寿命。
T6209 CW-069

CW069

Kinesin; Microtubule Associated Cytoskeletal Signaling
CW-069 是一种微管运动蛋白 HSET 的变构选择性抑制剂,IC50值为 75 μM,对 KSP 具有显着的特异性。
T16757 Risdiplam

RO7034067,RG7916

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Risdiplam (RO7034067) 是一种中枢和外周分布的 SMN2 前 mRNA 剪接修饰剂,可增加运动神经元存活 (SMN) 蛋白水平。
T8631 pyridostigmine

Regonol,Mestinon-SR,UNII-19QM69HH21,PyridostigmineBromine,Pyridostigminum

Others Others
Pyridostigmine(Regonol) 是一种乙酰胆碱酯酶抑制剂,可通过增加突触后运动终板的乙酰胆碱来治疗重症肌无力。
T4029 BTB-1

BTB 1,NSC156750

Microtubule Associated Cytoskeletal Signaling
BTB-1 (NSC156750) 是一种新型的有丝分裂运动蛋白 Kif18A 的小分子抑制剂,IC50值为1.69 μM。
T3525 PD150606

Cysteine Protease Proteases/Proteasome
PD150606 是一种具有选择性的非肽 calpain 抑制剂,具有神经保护活性,抑制 μ-calpains 和 m-calpains ,抑制红藻氨酸诱导的 Ca2+ 内流,干扰兴奋性毒性依赖性运动神经元死亡。
T2039 GSK-923295

Apoptosis; Kinesin Apoptosis; Cytoskeletal Signaling
GSK923295 是一种特异性的变构着丝粒相关蛋白-E 驱动蛋白 ATPase 活性抑制剂,作用于人类和犬类此酶,Ki 分别为 3.2±0.2 nM 和 1.6±0.1 nM。
T23331 SC 51089

SC 51089 free base

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
SC 51089 是一种选择性的前列腺素受体 PGE2 拮抗剂,对前列腺素受体亚型具有选择性,具有抗伤害活性,可改善亨廷顿病 R6/1 小鼠模型中的运动缺陷并挽救记忆力下降。
T34399 Rovatirelin

KPS-0373,S0373,S-0373,S 0373

AChE Neuroscience
Rovatirelin (S-0373) 是一种新合成的促甲状腺激素释放激素(TRH)类似物,通过乙酰胆碱和多巴胺神经传递改善胞嘧啶阿拉伯糖苷诱导的脊髓小脑变性大鼠模型的运动功能障碍。
TP1852L Myomodulin acetate(110570-93-9 free base)

Potassium Channel; Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Myomodulin acetate(110570-93-9 free base) 存在于两个已识别的海兔神经元中,它们包含肌调节蛋白 A、ARC 运动神经元 B16 和腹部神经元 L10。
T77586 Eg5-IN-1

Kinesin Cytoskeletal Signaling
Eg5-IN-1 是一种有效的驱动蛋白家族运动蛋白 (Eg5) 抑制剂,对 Eg5 的 IC50 值为 1.97 µM。Eg5-IN-1 可用于研究癌症。
T10659 Ca2+ channel agonist 1

Calcium Channel; CDK Cell Cycle/Checkpoint; Membrane transporter/Ion channel; Metabolism
Ca2+channel agonist 1 是 N-型钙离子通道激动剂和Cdk2的抑制剂,EC50分别为 14.23 μM 和 3.34 μM,可用作运动神经末梢功能障碍的潜在治疗方法。
T7352 Pridopidine

ACR16,ASP2314,FR310826,4-[3-(甲磺酰基)苯基]-1-丙基哌啶

Dopamine Receptor GPCR/G Protein; Neuroscience
Pridopidine (FR310826) 是多巴胺稳定剂,是一种低亲和力的多巴胺 D2 受体拮抗剂。它高亲和力作用于 sigma 1受体,Ki=70-80 nM,比其对 D2R 的亲和力高约 100 倍。
T8741 MitoBloCK-10

3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m

Others Others
MitoBloCK-10 (3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m) 是第一个能够减弱PAM 复合体活性的小分子调节剂,对 C 末端结构域的Tim44与前体和 Hsp70 结合具有抑制作用。
T14965 Ciliobrevin D

ATPase; Hedgehog/Smoothened GPCR/G Protein; Membrane transporter/Ion channel; Stem Cells
Ciliobrevin D 是细胞渗透性,可逆和特异性的 AAA + ATPase 运动细胞质动力蛋白抑制剂。它在体外抑制依赖于动力蛋白的微管滑动和 ATPase 活性。它抑制Hedgehog 信号和初级纤毛形成。
TP2047L CRF (6-33) acetate(120066-38-8 free base)

CRFR GPCR/G Protein
CRF (6-33) acetate(120066-38-8 free base) 是促肾上腺皮质激素释放因子结合蛋白 (CRFBP) 抑制肽;从 CRFBP 中替换 CRF。在体内抑制肥胖大鼠的体重增加并增加运动活动。
T16398 Opicapone

BIA 9-1067

Transferase Metabolism
Opicapone (BIA 9-1067) 是第三代儿茶酚-O-甲基转移酶 (COMT)抑制剂,能够降低细胞 ATP 含量,IC50=98 μM。它有用于帕金森病和运动波动的研究潜力。
T13248 UK-240455

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
UK-240455是一种有效的且具有选择性的 N-甲基 D-天冬氨酸 (NMDA) 甘氨酸受体拮抗剂,具有神经保护作用和改善帕金森病模型的运动的功能,是治疗帕金森病的潜在候选化合物。
T0166 Pancuronium dibromide

Pancuronium bromide,Pavulon,泮库溴铵

AChR Neuroscience
Pancuronium dibromide (Pavulon) 是一种双季基类固醇,是一种神经肌肉松弛剂。它通过与乙酰胆碱竞争 nACh 受体上的结合位点来抑制神经肌肉传递。它还可抑制心脏毒蕈碱受体并具有拟交感神经作用。
T24754 Hh-Ag1.5

SAG-1.5,SAG1.5,SAG 1.5

Hedgehog/Smoothened GPCR/G Protein; Stem Cells
Hh-Ag1.5 (SAG-1.5) 是一种高效的 Hedgehog (Hh) 激动剂(EC50: 1 nM)和Smoothened (Smo)受体激动剂,对Smo的 EC50 为 1 nM、 Ki值在 0.5 和 2.3 nM 之间。Hh-Ag1.5 介导的重编程打破了非损伤肝脏干细胞的静止状态,从而挽救了肝衰竭。Hh-Ag1.5 诱导 hiPSCs 分化为皮肤前体细胞、脊髓运动神经元和脊髓感觉神经元。
TP1325L Gastrin-Releasing Peptide, human(TFA)

Others Others
Gastrin-Releasing Peptide, human(TFA) (93755-85-2 free base) 是一种调节性人类肽,可引发胃泌素释放并调节胃酸分泌和肠道运动功能。支配胃G 细胞的迷走神经节后纤维释放GRP,刺激G 细胞释放胃泌素。
T2546 Pimozide

R6238,匹莫奇特,匹莫齐特

Potassium Channel; Dopamine Receptor; Adrenergic Receptor; STAT GPCR/G Protein; JAK/STAT signaling; Membrane transporter/Ion channel; Neuroscience; Stem Cells
Pimozide (R6238) 是多巴胺受体拮抗剂,对多巴胺 D1、D2 和 D3 受体的 Ki 值分别为 588、1.4 和 2.5 nM。它也是STAT3和STAT5的抑制剂,对 α1 肾上腺素受体也有较高亲和性,Ki 值为 39 nM。
T67729 UCM-1306

Dopamine Receptor GPCR/G Protein; Neuroscience
UCM-1306 是具有口服活性的人多巴胺 D1 受体变构调节剂 (PAM)。UCM-1306 增加结合在人和小鼠 D1 受体的内源性多巴胺 (DA) 效应。UCM-1306可以改善运动症状,解决与长期帕金森病(PD) 相关的关键共病认知障碍。
T0939 Phenytoin

苯妥英,Diphenylhydantoin,5,5-Diphenylhydantoin

Virus Protease; Sodium Channel Membrane transporter/Ion channel; Microbiology/Virology
Phenytoin (5,5-Diphenylhydantoin) 是一种有效的电压门控钠离子通道阻滞剂,可减少小鼠乳腺肿瘤的生长和转移,具有抗癫痫活性。
T37816 SB 243213

SB 243213 is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 has improved anxiolytic profile and has the potential for schizophrenia and motor disorders[1]. SB 243213 shows little affinity (pKi<6) for cloned human 5-HT1A, 5-HT1B, 5-HT1E, 5- HT1F and 5-HT7 receptors. It shows...
T28866 Stemazole

Apoptosis Apoptosis
Stemazole 是一种新型小分子人类干/祖细胞增殖激活剂 ,可促进人类胚胎干细胞的存活并保持干性 ,促进少突胶质细胞前体细胞在体外的存活。Stemazole 能显著提高细胞存活率和克隆形成数,并呈剂量依赖性,降低细胞凋亡率,促进运动功能障碍的恢复和髓鞘的修复。Stemazole 可作为脱髓鞘疾病的治疗剂,促进OPC 体外存活和体内再生。
T35689 MTP 131 acetate

Others Others
MTP 131 acetate 是一种小的线粒体靶向四肽。
T30167 ASP-5854

UNII-BJS8Y4IC5V,ASP 5854,C524699

ASP-5854 is an adenosine A(2A) receptor antagonist with the potential to improve motor deficits in Parkinson's disease.
T71828 Syntelin

Syntelin is a selectively CENP-E inhibitor. Syntelin inhibited CENP-E motility in a dose-dependent manner with an IC50 value of 160 nM. Among an extensive list of mitotic kinesins examined, syntelin was found to be highly selective for CENP-E. Syntelin binds to different sites from those of GSK923295, a recently identified CENP-E ATPase inhibitor, as syntelin inhibits CENP-E mutants resistant to GSK923295 in a manner indistinguishable from that of wild type motor. Syntelin represents a novel cla...
T21466 MK-212

MK 212,MK212

MK-212 is a 5HT2C-receptor agonist. Intraperitoneal injection of MK-212 in 0.5 and 1.0 mg/kg increased the blood level of corticosterone in mice and reduced their motor activity. In 0.1 and 0.2 mg/kg, the agonist reduced anxiety with no effect on motor ac
T38828 Mesdopetam

IRL790

Mesdopetam (IRL790) is a dopamine D3 receptor antagonist with a Ki of 90 nM and an IC50 of 9.8 μM for the human recombinant D3 receptor. It exhibits psychomotor stabilizing properties and is utilized in the study of motor and psychiatric complications associated with Parkinson's disease.
T63612 ATX inhibitor 8

ATX inhibitor 8 是自分泌运动因子 Autotaxin (ATX) 抑制剂。
T34664 SMN2-Stablizer-27

SMN2-Stablizer 27,SMN2 Stablizer-27

SMN2-Stablizer-27 is a stablizer of survival of motor neuron 2 (SMN2), and a post-translationally stablizing SMN protein for the treatment of spinal muscular atrophy (SMA).
T68881 OL-135

OL-135 is a CNS penetrant, highly potent and selective reversible inhibitor of FAAH. OL-135 exhibits analgesic pharmacology in various animal models without the motor impairment associated with direct CB1 agonism.
T21393 Ethopropazine Hydrochloride

Lysivane,Parphezein,Dibutil,Parfezin,Profenamine HCl,Pardisol

Ethoproprazine hydrochloride is an butyrylcholinesterase inhibitor. It reduces extrapyramidal motor effects and used as an antidyskinetic, characteristic of Parkinson′s disease. It also alleviates thermal hyperalgesia in rats.
T28680 SB-215505

SB215505 is a potent 5-HT2B/2C receptor antagonist (pKi values are 8.3, 7.66 and 6.77 for 5-HT2B, 5-HT2C and 5-HT2A respectively). It Increases wakefulness and motor activity in rats.
TP2047 CRF(6-33)(human)

CRF (6-33)

CRF(6-33)(human) is a Corticotropin-releasing factor binding protein (CRFBP) inhibitor peptide; displaces CRF from CRFBP. Suppresses body weight gain and increases motor activity in obese rats in vivo.
T30576 Brasofensine

BMS-204756,CID9554198,BMS204756,UNII-1YP2S94RVH,BMS 204756

Brasofensine is a monoamine reuptake blocker, which is a benztoalkane. In animal models of Parkinson's disease, Brasofensine is effective in stimulating LMA and reversing motor inactivity. Brasofensine is being developed to treat Parkinson's disease and A
T35594 Cuspin-1

The Survival of Motor Neurons (SMN) protein participates in RNA splicing. Decreases in SMN, typically a consequence of defects in the smn1 gene, result in the death of motor neurons and lead to the neurodegenerative disease, spinal muscular atrophy (SMA). Cuspin-1 is a small molecule upregulator of SMN that has been shown in vitro to increase levels of SMN in SMA patient fibroblasts by 50% at 18 μM. Its mechanism of action is thought to involve increased phosphorylation of ERK to initiate Ras-Ra...
T69152 Bromopride hydrochloride

Bromopride hydrochloride is the salt form of Bromopride, a dopamine D2 receptor blocker. Bromopride exerts is a gastrointestinal prokinetic exploited clinically for the management of motor disorders of the upper gastrointestinal tract, including functional dyspepsia, gastric stasis of various origins and emesis.
T12859 SB 243213 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It has improved anxiolytic profile and has the potential for schizophrenia and motor disorders.

化合物

ARQ 621
Cat.No: T6393
Synonym:
Target: Kinesin
ITI-214
Cat.No: T11689
Synonym: ITI214
Target: PDE
ML-193
Cat.No: T22103
Synonym: CID 1261822
Target: Cannabinoid Receptor
Arimoclomol maleate
Cat.No: T13554
Synonym: BRX-220
Target: HSP
Triprolidine hydrochloride monohydrate
Cat.No: T1030
Synonym: 盐酸曲普利啶,盐酸曲普利啶一水合物,Triprolidine hydrochloride
Target: Histamine Receptor
Branaplam
Cat.No: T4641
Synonym: LMI 070,NVS-SM1
Target: Others, Potassium Channel, DNA/RNA Synthesis
Arimoclomol
Cat.No: T13553
Synonym: 阿瑞洛莫,BRX-220 free base
Target: HSP
Etilevodopa hydrochloride
Cat.No: T24047
Synonym: Levodopa ethyl ester,Etilevodopa HCl, L-DOPA ethyl ester
Target: Others, Dopamine Receptor, Drug Metabolite
Rg3039
Cat.No: T3336
Synonym: PF-06687859
Target: Others
Crisdesalazine
Cat.No: T27084
Synonym: AAD2004,AAD 2004,AAD-2004
Target: Prostaglandin Receptor
CW-069
Cat.No: T6209
Synonym: CW069
Target: Kinesin, Microtubule Associated
Risdiplam
Cat.No: T16757
Synonym: RO7034067,RG7916
Target: DNA/RNA Synthesis
pyridostigmine
Cat.No: T8631
Synonym: Regonol,Mestinon-SR,UNII-19QM69HH21,PyridostigmineBromine,Pyridostigminum
Target: Others
BTB-1
Cat.No: T4029
Synonym: BTB 1,NSC156750
Target: Microtubule Associated
PD150606
Cat.No: T3525
Synonym:
Target: Cysteine Protease
GSK-923295
Cat.No: T2039
Synonym:
Target: Apoptosis, Kinesin
SC 51089
Cat.No: T23331
Synonym: SC 51089 free base
Target: Prostaglandin Receptor
Rovatirelin
Cat.No: T34399
Synonym: KPS-0373,S0373,S-0373,S 0373
Target: AChE
Myomodulin acetate(110570-93-9 free base)
Cat.No: TP1852L
Synonym:
Target: Potassium Channel, Calcium Channel, Sodium Channel
Eg5-IN-1
Cat.No: T77586
Synonym:
Target: Kinesin
Ca2+ channel agonist 1
Cat.No: T10659
Synonym:
Target: Calcium Channel, CDK
Pridopidine
Cat.No: T7352
Synonym: ACR16,ASP2314,FR310826,4-[3-(甲磺酰基)苯基]-1-丙基哌啶
Target: Dopamine Receptor
MitoBloCK-10
Cat.No: T8741
Synonym: 3-fluoro-N'-[(E)-(5-nitrothiophen-2-yl)m
Target: Others
Ciliobrevin D
Cat.No: T14965
Synonym:
Target: ATPase, Hedgehog/Smoothened
CRF (6-33) acetate(120066-38-8 free base)
Cat.No: TP2047L
Synonym:
Target: CRFR
Opicapone
Cat.No: T16398
Synonym: BIA 9-1067
Target: Transferase
UK-240455
Cat.No: T13248
Synonym:
Target: NMDAR, iGluR
Pancuronium dibromide
Cat.No: T0166
Synonym: Pancuronium bromide,Pavulon,泮库溴铵
Target: AChR
Hh-Ag1.5
Cat.No: T24754
Synonym: SAG-1.5,SAG1.5,SAG 1.5
Target: Hedgehog/Smoothened
Gastrin-Releasing Peptide, human(TFA)
Cat.No: TP1325L
Synonym:
Target: Others
Pimozide
Cat.No: T2546
Synonym: R6238,匹莫奇特,匹莫齐特
Target: Potassium Channel, Dopamine Receptor, Adrenergic Receptor, STAT
UCM-1306
Cat.No: T67729
Synonym:
Target: Dopamine Receptor
Phenytoin
Cat.No: T0939
Synonym: 苯妥英,Diphenylhydantoin,5,5-Diphenylhydantoin
Target: Virus Protease, Sodium Channel
SB 243213
Cat.No: T37816
Synonym:
Target:
Stemazole
Cat.No: T28866
Synonym:
Target: Apoptosis
MTP 131 acetate
Cat.No: T35689
Synonym:
Target: Others
ASP-5854
Cat.No: T30167
Synonym: UNII-BJS8Y4IC5V,ASP 5854,C524699
Target:
Syntelin
Cat.No: T71828
Synonym:
Target:
MK-212
Cat.No: T21466
Synonym: MK 212,MK212
Target:
Mesdopetam
Cat.No: T38828
Synonym: IRL790
Target:
ATX inhibitor 8
Cat.No: T63612
Synonym:
Target:
SMN2-Stablizer-27
Cat.No: T34664
Synonym: SMN2-Stablizer 27,SMN2 Stablizer-27
Target:
OL-135
Cat.No: T68881
Synonym:
Target:
Ethopropazine Hydrochloride
Cat.No: T21393
Synonym: Lysivane,Parphezein,Dibutil,Parfezin,Profenamine HCl,Pardisol
Target:
SB-215505
Cat.No: T28680
Synonym:
Target:
CRF(6-33)(human)
Cat.No: TP2047
Synonym: CRF (6-33)
Target:
Brasofensine
Cat.No: T30576
Synonym: BMS-204756,CID9554198,BMS204756,UNII-1YP2S94RVH,BMS 204756
Target:
Cuspin-1
Cat.No: T35594
Synonym:
Target:
Bromopride hydrochloride
Cat.No: T69152
Synonym:
Target:
SB 243213 hydrochloride
Cat.No: T12859
Synonym:
Target: 5-HT Receptor
Cat. No. Product Name Target Signaling Pathways
T20754 Deltamethrin

Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974

Others Others
Deltamethrin (RU 22974) 是一种具有神经毒性的拟除虫菊酯杀虫剂,在大鼠中能够产生一系列可逆的运动症状(如包括后肢僵硬、舞蹈性关节炎)。
TN1913 Marmin

Calcium Channel; Antifection; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and secondarily due to the prevention of the effects of endogenous acetylcholine and histamine.
TN4519 Mesuaxanthone A

胡桐,海棠木

Others Others
Mesuaxanthone A and mesuaxanthone B are two yellow pigments.They produce varying degrees of C.N.S. depression characterised by ptosis, sedation, decreased spontaneous motor activity, loss of muscle tone, potentiation of pentobarbitone sleeping time and et
T13123 Tentoxin

Endogenous Metabolite Metabolism
Tentoxin 是一种由植物致病真菌产生的环状肽,在敏感植物中,当其浓度在纳摩尔到微摩尔之间时,会使 F1马达失活,而更高的浓度会超过该酶的天然活性
T75576 Solidagonic acid

Solidagonic acid 通过促进异常单极纺锤体向双极纺锤体的转变来抑制 HSET 运动活动。Solidagonic acid 抑制裂殖酵母细胞死亡,并使有丝分裂纺锤体从单极形态逆转为双极形态。Solidagonic acid 对 Lactuca sativaL. 和 Lolium multiflorumLam 的幼苗具有生长抑制活性。

天然产物

Deltamethrin
Cat.No: T20754
Synonym: Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974
Target: Others
Marmin
Cat.No: TN1913
Synonym:
Target: Calcium Channel, Antifection, Histamine Receptor
Mesuaxanthone A
Cat.No: TN4519
Synonym: 胡桐,海棠木
Target: Others
Tentoxin
Cat.No: T13123
Synonym:
Target: Endogenous Metabolite
Solidagonic acid
Cat.No: T75576
Synonym:
Target:
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