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105

抑制剂 & 化合物

28

天然产物

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Cat. No. Product Name Target Signaling Pathways
T41303 Isoflupredone

Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone

Others Others
Isoflupredone (Isoflupredonum) 是一种合成的皮质类固醇,通过与动物 (如马) 的糖皮质激素和矿皮质激素受体结合抑制炎症细胞和抑制炎症介质的表达在生物体内发挥作用。Isoflupredone 具有抗炎和免疫抑制作用, 可应用于治疗各种肌肉骨骼、过敏性和全身炎症性疾病。
T7107 δ-Sleep Inducing Peptide

DSIP,Delta-Sleep Inducing Peptide,依米地肽

Antioxidant oxidation-reduction
δ-Sleep Inducing Peptide (DSIP) 是一种具有抗氧化和抗焦虑活性的神经肽。
T41328 Delta-12-Prostaglandin J2

Delta-12-Prostaglandin J2 在生命科学相关研究中具有广泛的应用。
T124900 Delta-9-Tetrahydrocannabivarinic acid

Delta-9-Tetrahydrocannabivarinic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124900。
T82587 Delta (Phospho) Sleep Inducing Peptide

DSIP-P

Delta (Phospho) Sleep Inducing Peptide (DSIP-P) 是促进睡眠效应持久的多肽,能诱导大鼠昼夜运动行为的改变。
T78005 δ-Sleep Inducing Peptide acetate

Delta-Sleep Inducing Peptide acetate

δ-Sleep Inducing Peptide acetate为具备抗氧化及抗焦虑功能的神经肽。
T125797 Longilactone, delta-4(18)-Isomer, 2alpha-alcoho

Longilactone, delta-4(18)-Isomer, 2alpha-alcoho 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125797,CAS号为 149155-28-2。
T32266 Jasmine lactone

Jasmolactone, delta-,EINECS 247-074-2,FEMA No. 3745

Jasmine lactone is a lactone and aroma compound. Its chemical formula is C10H16O2. It exists in some natural product in jasmine oil, tuberose, gardenia, mimosa, honeysuckle, lily, tea, peach, and ginger. It can be mainly used for the preparation of apri
T78271 Anti-Mouse TCR gamma/delta Antibody (UC7-13D5)

Anti-Mouse TCR gamma/delta Antibody为针对小鼠TCR gamma/delta的IgG类免疫抑制抗体,其宿主为亚美尼亚仓鼠。
T66182 2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone

2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66182,CAS号为 32384-65-9。
T35321 Zymostenol

delta(8)-Cholestenol,5a-Cholest-8-en-3b-ol,Δ8-Cholesterol

Endogenous Metabolite; ROR Metabolism
Zymostenol (5a-Cholest-8-en-3b-ol) 是一种 RORγ 激动剂 ,EC50为1 μM。Zymostenol 是胆固醇生物合成的后期前体。
T39516 Bocidelpar

PPAR DNA Damage/DNA Repair; Metabolism
Bocidelpar 是一种有效的过氧化物酶体增殖物激活受体 delta 调节剂,可改善杜兴肌营养不良肌肉细胞中的线粒体生物合成和功能。
T38862 Nandrolone acetate

19-Nortestosterone 17β-acetate

Others Others
Nandrolone acetate (19-Nortestosterone 17β-acetate) 是一种甾体酮,是异构酶的竞争性抑制剂,对Δ5-3-酮甾体异构酶的 Ki 为 7 μM。
T70289 Terpendole E

Terpendole E is an atypical L5 site inhibitor.
T9713 δ-secretase inhibitor 11

Beta Amyloid; Caspase Apoptosis; Neuroscience; Proteases/Proteasome
δ-secretase inhibitor 11是一种分泌酶抑制剂,可用作 阿尔茨海默病(AD) 治疗转化开发的先导化合物。
T26370 (25S)-delta7-Dafachronic acid

(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.
TP2145 JTP10-△-R9 TFA

JNK MAPK
JTP10-△-R9 TFA is a selective inhibitor of JNK2 peptide (IC50: 89 nM), exhibiting 10-fold selectivity for JNK2 over JNK1 and JNK3.
TP2146 JTP10-△-TATi TFA

JNK MAPK
JTP10-△-TATi TFA is a selective inhibitor of JNK2 peptide (IC50: 92 nM), exhibiting 10-fold selectivity for JNK2 over JNK1 and JNK3.
T5002 Methyl Aminolevulinate Hydrochloride

5-Aminolevulinic acid methyl ester,Methyl δ-aminolevulinate hydrochloride,5-氨基酮戊酸甲酯盐酸盐,Methyl 5-aminolevulinate Hydrochloride,Aminolevulinic acid methyl ester Hydrochloride

Others Others
Methyl Aminolevulinate Hydrochloride (5-Aminolevulinic acid methyl ester) 是增敏剂,可用于光动力疗法。Methyl aminolevulinate 是一种前药,可代谢为原卟啉 IX。
T6462 Deltarasin

PDE; Ras GPCR/G Protein; MAPK; Metabolism
Deltarasin 是一种 KRAS-PDEδ 相互作用的小分子抑制剂,与纯化的 PDEδ 结合,Kd 值为 38 nM。
T25302 Deltakephalin

DTLET,Enkephalin leu, thr(2)-thr(6)-

Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.
T23976 Deltasonamide 1

Deltasonamide

Deltasonamide is a potent and selective inhibitor of PDE6δ‐KRas.
T10994L2 Deltasonamide 2 (TFA)

PDE Metabolism
Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.
T12461 PI3Kdelta inhibitor 1

PI3K PI3K/Akt/mTOR signaling
PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an IC50 of 1.3 nM.
T25303 Deltamycin A1

Deltamycin A1 is a novel macrolide antibiotic.
T73864 Deltasonamide 1 TFA

Deltasonamide 1 TFA 是一种PDE6δ-KRas 抑制剂。Deltasonamide 1 可以抑制 PDE6δ-KRas,KD 为 203 pM。Deltasonamide 1 可用于肿瘤的研究。
T10994L Deltasonamide 2 hydrochloride

Deltasonamide 2 hydrochloride (2088485-34-9 free base)

PDE Metabolism
Deltasonamide 2 hydrochloride is a competitive high-affinity PDEδ inhibitor with a Kd of approximately 385 pM.
T10994 Deltasonamide 2

PDE Metabolism
Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.
T23977 Deltazinone

Deltazinone is a selective PDEδ inhibitor. Deltazinone exhibits less unspecific cytotoxicity and demonstrates a high correlation with the phenotypic effect of PDEδ knockdown in a set of human pancreatic cancer cell lines.
T70646 Deltarasin HCl

Deltarasin is a high affinity PDEδ-KRAS interaction inhibitor. Deltarasin can inhibit KRAS-PDEδ interactions by binding to a hydrophobic pocket on PDEδ, resulting in the impairment of cell growth, KRAS activity, and RAS/RAF signaling in human pancreatic ductal adenocarcinoma cell lines. The anti-cancer cell activity of deltarasin can be enhanced by simultaneously blocking tumor protective" autophagy
T22752L (D-Ser2)-Leu-Enkephalin-Thr

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
(D-Ser2)-Leu-Enkephalin-Thr 是阿片受体的 delta 选择性药物,具有镇痛作用。
TP1367 [D-Ala2]leucine-enkephalin

(D-ALA2)-亮氨酸脑啡肽

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
[D-Ala2]leucine-enkephalin 是 δ 阿片类激动剂,是能长效抗降解的亮氨酸脑非肽,可用于研究 δ 阿片受体的信号通路。
T15575 Indeglitazar

PPM 204

PPAR DNA Damage/DNA Repair; Metabolism
Indeglitazar (PPM 204) 是 PPAR 的泛激动剂,包括亚型 alpha (α)、delta (δ) 和 gamma (γ)。
T0102 Naloxone hydrochloride

盐酸纳洛酮,Naloxone HCl

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Naloxone hydrochloride (Naloxone HCl) 是一种特异性、没有激动剂活性的opiate 拮抗剂。它是 mu、delta 和 kappa 阿片受体的竞争性拮抗剂。
T27667 JNJ-20788560

JNJ 20788560

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
JNJ-20788560 是一种δ阿片受体(DOR)激动剂,具有镇痛活性。它对 DOR 的选择性高于μ阿片受体(MOR)。
T8992 BMS986188

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
BMS986188 是一种新型的强效选择性正向变构调节剂,用于 δ-阿片受体。
T29663 ADL-5747

ADL-5747 (free base),ADL5747,ADL-5747 free base

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
ADL-5747 (ADL-5747 (free base)) (free base)是一种δ opioid 受体激动剂,可用于治疗神经系统疾病、皮肤和肌肉骨骼疾病,可用于研究疱疹后神经痛、膝关节炎和疼痛。
T28903 T-3364366

T 3364366,T3364366

Others Others
T-3364366 是一种噻吩并嘧啶酮 delta-5 去饱和酶 (Δ5D) 抑制剂,在 HepG2 和 RLN-10 细胞中的 IC50 分别为 1.9 nM 和 2.1 nM。
T67888L Samidorphan HCl

Samidorphan HCl(852626-89-2 free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Samidorphan HCl 是一种具有口服活性和高效性的 opioid 系统调节剂,可与 μ‐opioid、 κ‐opioid 和 δ‐opioid 受体结合。Samidorphan HCl 是一种新型 μ‐opioid 受体拮抗剂,是 k-opioid 受体和 δ‐opioid 受体的部分激动剂。Samidorphan HCl 可用于预防和治疗精神分裂。
T30188L1 (Iso)-Atagabalin HCl

(Iso)-Atagabalin HCl((Iso)-223445-75-8)

Others Others
(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) 是一种可用于治疗非恢复性睡眠的α -2- δ配体。
T76698 Rovalpituzumab

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Rovalpituzumab 是一种靶向 delta 样蛋白 3 (DLL3) 的人源化单克隆抗体。Rovalpituzumab 可用于合成抗体-活性分子偶联物 (ADC)。Rovalpituzumab 具有抗癌活性,可用于治疗小细胞肺癌 (SCLC)。
T32804 LJ-001

LJ 001,LJ001

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
LJ-001 显示出对几乎所有包膜 RNA 和 DNA 病毒的广谱活性。 LJ001 抑制传染性胃肠炎病毒 (TGEV) 和猪 delta 冠状病毒 (PDCoV) 的感染。
T64350 Casein kinase 1δ-IN-3

Casein Kinase Metabolism; Stem Cells
Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) 是一种酪蛋白激酶 1δ (CK1d) 抑制剂,pIC50 为 6.5376。
T1473 Trilostane

曲洛斯坦,Win 24540,曲洛司坦

Dehydrogenase Metabolism
Trilostane (Win 24540) 是一种3 β-羟化类固醇脱氢酶抑制剂,能够作用于库兴氏综合征。
T13140 Umbralisib R-enantiomer

TGR-1202 R-enantiomer,RP5264 R-enantiomer

PI3K PI3K/Akt/mTOR signaling
Umbralisib R-enantiomer (RP5264 R-enantiomer) 是 PI3K 的δ型抑制剂,是 TGR-1202 活性较低的对映体。Umbralisib R-enantiomer 对δ型 pi3激酶的 IC50,至少比抑制剂对其他 PI3K 亚型(A, β和γ)的 IC50低20倍。
T8991 BMS986187

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
BMS986187 是一种有效的δ-阿片受体选择性正变构调节剂 (PAM),其 EC50= 0.03 μM,pKB= 6.02 (~1 μM)。BMS986187 对 μ 受体无明显 PAM 活性 (EC50=3 μM)。
T1988 Duvelisib

INK1197,IPI-145,度维利塞

PI3K PI3K/Akt/mTOR signaling
Duvelisib (INK1197) 是 p100δ的选择性抑制剂,能够作用于 p110δ (IC50:2.5 nM)、p110γ (IC50:27.4 nM)、p110β (IC50:85 nM) 和 p110α (IC50:1602 nM)。
T1197 Trimebutine maleate

Debridat,Polibutin,马来酸曲美布汀

Calcium Channel; Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Trimebutine maleate (Polibutin) 是一种外周 μ、δ 和 kappa 阿片受体激动剂,用作治疗慢性和急性腹痛的解痉药物。
T64387 2-Nitrobenzoic acid

o-Nitrobenzoic acid

Others Others
2-Nitrobenzoic acid (o-Nitrobenzoic acid) 是一种抗增殖化合物,对表达 T 型钙通道α1H 或其剪接变体δ25的 jurkat 细胞系显示出8.3μM 的 IC50。
T20435L Leuphasyl TFA

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Leuphasyl TFA 是一种酰胺肽,一种 δ-阿片受体激动剂,是一种抗降解的长效 Leu-脑啡肽类似物,用于研究 δ 阿片受体的信号通路。 它 是一种有效的长效 Leu-脑啡肽类似物,可抵抗酶促降解。

化合物

Isoflupredone
Cat.No: T41303
Synonym: Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone
Target: Others
δ-Sleep Inducing Peptide
Cat.No: T7107
Synonym: DSIP,Delta-Sleep Inducing Peptide,依米地肽
Target: Antioxidant
Delta-12-Prostaglandin J2
Cat.No: T41328
Synonym:
Target:
Delta-9-Tetrahydrocannabivarinic acid
Cat.No: T124900
Synonym:
Target:
Delta (Phospho) Sleep Inducing Peptide
Cat.No: T82587
Synonym: DSIP-P
Target:
δ-Sleep Inducing Peptide acetate
Cat.No: T78005
Synonym: Delta-Sleep Inducing Peptide acetate
Target:
Longilactone, delta-4(18)-Isomer, 2alpha-alcoho
Cat.No: T125797
Synonym:
Target:
Jasmine lactone
Cat.No: T32266
Synonym: Jasmolactone, delta-,EINECS 247-074-2,FEMA No. 3745
Target:
Anti-Mouse TCR gamma/delta Antibody (UC7-13D5)
Cat.No: T78271
Synonym:
Target:
2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone
Cat.No: T66182
Synonym:
Target:
Zymostenol
Cat.No: T35321
Synonym: delta(8)-Cholestenol,5a-Cholest-8-en-3b-ol,Δ8-Cholesterol
Target: Endogenous Metabolite, ROR
Bocidelpar
Cat.No: T39516
Synonym:
Target: PPAR
Nandrolone acetate
Cat.No: T38862
Synonym: 19-Nortestosterone 17β-acetate
Target: Others
Terpendole E
Cat.No: T70289
Synonym:
Target:
δ-secretase inhibitor 11
Cat.No: T9713
Synonym:
Target: Beta Amyloid, Caspase
(25S)-delta7-Dafachronic acid
Cat.No: T26370
Synonym:
Target:
JTP10-△-R9 TFA
Cat.No: TP2145
Synonym:
Target: JNK
JTP10-△-TATi TFA
Cat.No: TP2146
Synonym:
Target: JNK
Methyl Aminolevulinate Hydrochloride
Cat.No: T5002
Synonym: 5-Aminolevulinic acid methyl ester,Methyl δ-aminolevulinate hydrochloride,5-氨基酮戊酸甲酯盐酸盐,Methyl 5-aminolevulinate Hydrochloride,Aminolevulinic acid methyl ester Hydrochloride
Target: Others
Deltarasin
Cat.No: T6462
Synonym:
Target: PDE, Ras
Deltakephalin
Cat.No: T25302
Synonym: DTLET,Enkephalin leu, thr(2)-thr(6)-
Target:
Deltasonamide 1
Cat.No: T23976
Synonym: Deltasonamide
Target:
Deltasonamide 2 (TFA)
Cat.No: T10994L2
Synonym:
Target: PDE
PI3Kdelta inhibitor 1
Cat.No: T12461
Synonym:
Target: PI3K
Deltamycin A1
Cat.No: T25303
Synonym:
Target:
Deltasonamide 1 TFA
Cat.No: T73864
Synonym:
Target:
Deltasonamide 2 hydrochloride
Cat.No: T10994L
Synonym: Deltasonamide 2 hydrochloride (2088485-34-9 free base)
Target: PDE
Deltasonamide 2
Cat.No: T10994
Synonym:
Target: PDE
Deltazinone
Cat.No: T23977
Synonym:
Target:
Deltarasin HCl
Cat.No: T70646
Synonym:
Target:
(D-Ser2)-Leu-Enkephalin-Thr
Cat.No: T22752L
Synonym:
Target: Opioid Receptor
[D-Ala2]leucine-enkephalin
Cat.No: TP1367
Synonym: (D-ALA2)-亮氨酸脑啡肽
Target: Opioid Receptor
Indeglitazar
Cat.No: T15575
Synonym: PPM 204
Target: PPAR
Naloxone hydrochloride
Cat.No: T0102
Synonym: 盐酸纳洛酮,Naloxone HCl
Target: Opioid Receptor
JNJ-20788560
Cat.No: T27667
Synonym: JNJ 20788560
Target: Opioid Receptor
BMS986188
Cat.No: T8992
Synonym:
Target: Opioid Receptor
ADL-5747
Cat.No: T29663
Synonym: ADL-5747 (free base),ADL5747,ADL-5747 free base
Target: Opioid Receptor
T-3364366
Cat.No: T28903
Synonym: T 3364366,T3364366
Target: Others
Samidorphan HCl
Cat.No: T67888L
Synonym: Samidorphan HCl(852626-89-2 free base)
Target: Opioid Receptor
(Iso)-Atagabalin HCl
Cat.No: T30188L1
Synonym: (Iso)-Atagabalin HCl((Iso)-223445-75-8)
Target: Others
Rovalpituzumab
Cat.No: T76698
Synonym:
Target: Gamma-secretase
LJ-001
Cat.No: T32804
Synonym: LJ 001,LJ001
Target: Antiviral, HIV Protease
Casein kinase 1δ-IN-3
Cat.No: T64350
Synonym:
Target: Casein Kinase
Trilostane
Cat.No: T1473
Synonym: 曲洛斯坦,Win 24540,曲洛司坦
Target: Dehydrogenase
Umbralisib R-enantiomer
Cat.No: T13140
Synonym: TGR-1202 R-enantiomer,RP5264 R-enantiomer
Target: PI3K
BMS986187
Cat.No: T8991
Synonym:
Target: Opioid Receptor
Duvelisib
Cat.No: T1988
Synonym: INK1197,IPI-145,度维利塞
Target: PI3K
Trimebutine maleate
Cat.No: T1197
Synonym: Debridat,Polibutin,马来酸曲美布汀
Target: Calcium Channel, Opioid Receptor
2-Nitrobenzoic acid
Cat.No: T64387
Synonym: o-Nitrobenzoic acid
Target: Others
Leuphasyl TFA
Cat.No: T20435L
Synonym:
Target: Opioid Receptor
Cat. No. Product Name Target Signaling Pathways
T6000 Delta-Tocopherol

(+)-DELTA-生育酚,D-DELTA-TOCOPHEROL

Endogenous Metabolite Metabolism
Delta-Tocopherol 是维生素 E 的异构体,具有抗氧化活性。
T4821 Tetrahydro-2H-pyran-2-one

δ-Valerolactone,δ-Valeryllactone,delta-戊内酯,2-Oxotetrahydropyran

Others; Endogenous Metabolite Metabolism; Others
Tetrahydro-2H-pyran-2-one (δ-Valerolactone) 是内源性代谢产物的一种。
T10109 3-Carene

Delta-3-Carene

COX; Antifungal Immunology/Inflammation; Microbiology/Virology; Neuroscience
3-Carene(Delta-3-Carene) 是西部落叶松和花旗松中提取的双环单萜烯,可做为植物杀菌剂。3-Carene 对痛觉刺激引起的炎症浸润和 COX-2 过表达有抑制作用。3-Carene 具有抗伤害作用,能促进成骨细胞分化的早期标志物碱性磷酸酶的活性和表达。
T10993 δ-Amyrenone

Delta-Amyrone,Α-香树脂酮

Others Others
δ-Amyrenone (Delta-Amyrone) 分离自 S. lineare,具有抗炎作用。
TN3817 Delta-Caesalpin

Others Others
Delta-Caesalpin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3817,CAS号为 7716-14-5。
T19274 delta-Valerobetaine

Others Others
delta-Valerobetaine is a precursor of trimethylamine N-oxide (TMAO).
T8044 Ajmalicine

阿吗里新,Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin

Adrenergic Receptor GPCR/G Protein; Neuroscience
Ajmalicine (Raubasine) 是一种有效的抗肾上腺素 (adrenolytic) 剂,优先阻断 α1-肾上腺素受体 (α1-adrenoceptor)。Ajmalicine 是一种可逆性但非竞争性尼古丁受体 (nicotine receptor) 完全抑制剂,IC50 为 72.3 μM。Ajmalicine 还可用于降压、蛇毒,具有镇静活性。
TN3816 delta-Amyrin acetate

Others Others
β-Amyrin acetate and β-Amyrin acetate have antidyslipidemic activity.
TN6697 Delta-Nonalactone

Delta-Nonalactone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6697,CAS号为 3301-94-8。
TMA2474 δ-Tocotrienol

Delta-Tocotrienol,δ-生育三烯酚

ERK; BCL; VEGFR; Akt; PI3K; PDK; p53 Angiogenesis; Apoptosis; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
δ-Tocotrienol (Delta-Tocotrienol) 是一种维生素 E,存在于蔬菜,水果,种子,坚果,谷物和油等。维生素 E 是抗氧化剂、神经保护剂和抗癌剂,可以降低胆固醇和其他脂质,保护心血管疾病。
TN3815 Delta 7-avenasterol

Delta 7-avenasterol has antioxidant activity.
TN3814 Delta 5-avenasterol

Others Others
Delta 5-avenasterol has antioxidant activity.
T0933 D-(+)-Glucono-1,5-lactone

Gluconic acid lactone,Delta-Gluconolactone,Gluconolactone,葡萄糖酸内酯

Others; Reactive Oxygen Species; Endogenous Metabolite Immunology/Inflammation; Metabolism; NF-κB; Others
D-(+)-Glucono-1,5-lactone (Gluconolactone) 是聚羟基酸,可螯合金属离子,具有保湿、抗氧化特性。
T31993 Grayanotoxin II

G-II,Deacetylanhydroandromedotoxin,delta(sup 10 (18))-Andromedenol

Grayanotoxins are a group of closely related neurotoxins named after Leucothoe grayana. Extract from leaves of Ericaceae.
T40815 δ-Decalactone

Others Others
δ-Decalactone 存在于脱脂奶粉和水果中,具有甜味。
T2919 Sesamin

Fagarol,Fsesamin,芝麻素

Others Others
Sesamin (Fsesamin) 是多不饱和脂肪酸生物合成中的选择性delta 5 去饱和酶抑制剂,是在芝麻油中存在丰富的木脂素。它对脑缺血具有有效的神经保护作用。
T4034 Solamargine

Solamargin,δ-Solanigrine,澳洲茄边碱

Apoptosis; p38 MAPK; P-gp; STAT Apoptosis; JAK/STAT signaling; MAPK; Membrane transporter/Ion channel; Neuroscience; Stem Cells
Solamargine (δ-Solanigrine) 是一种来源于茄属植物的类固醇 Solasodine 的衍生物,诱导非选择性细胞毒性和 P-gp 抑制作用。它通过下调 MMP-2 和 MMP-9 的表达和活性来显著抑制 HepG2 细胞的迁移和侵袭,在多种癌症中均表现出抗癌活性。
T35409 (+)-δ-Cadinene

Apoptosis; Antibacterial Apoptosis; Microbiology/Virology
(+)-δ-Cadinene 是一种从G. hirsutum 中发现的倍半萜,具有抗菌、杀虫、抗癌和抗增殖活性。 它对肺炎双球菌的MIC 值为31.25 μg/ml,对 A. stephensi、A. aegypti 和 C. quinquefasciatust 三龄幼虫的LC50s 值分别8.23、9. 2和3。(+)-δ-Cadinene(10、50 和 100 μM)可诱导 OVCAR-3 人类卵巢癌细胞凋亡并抑制其增殖。
TN2409 6-Deoxy-3-O-methyl-β-allopyranosyl (1→4)-β-cymaronic acid δ-lactone

Others Others
6-Deoxy-3-O-methyl-β-allopyranosyl (1→4)-β-cymaronic acid δ-lactone is a natural product from Marsdenia tenacissima
T20754 Deltamethrin

Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974

Others Others
Deltamethrin (RU 22974) 是一种具有神经毒性的拟除虫菊酯杀虫剂,在大鼠中能够产生一系列可逆的运动症状(如包括后肢僵硬、舞蹈性关节炎)。
T3S1888 Deltaline

德尔塔林,Deltamine 6-acetate,Eldelin

Others Others
Deltaline (Eldelin) 是一种从滇川翠雀花属植物中分离出来的二萜类生物碱。它可用于缓解疼痛的研究,滇川翠雀花属植物也被用于风湿痛、中风引起的麻痹、类风湿性关节炎的研究。
TN6070 Deltatsine

Deltatsine是一种天然产物,属于毛茛科翠雀属,其产品编号为 TN6070,CAS号为 92631-66-8。Deltatsine可用作对照参考。
T4868 gamma-Linolenic acid

gamolenic acid,γ-Linolenic acid,γ-亚麻酸

Endogenous Metabolite Metabolism
gamma-Linolenic acid (gamolenic acid) 是一种 omega-6 (n-6),18 碳 (18C-) 多不饱和脂肪酸 (PUFA),可以从人乳和植物种子油中提取。
T3417 Amentoflavone

Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin

Apoptosis; P450; Phospholipase; Reactive Oxygen Species; Opioid Receptor; COX; Antibacterial; RSV; Antifungal Apoptosis; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
Amentoflavone (3',8''-Biapigenin) 是一种具有很多生物活性的双黄酮类天然产物,有抗炎、抗氧化和神经保护等作用。
T41253 Sterculic acid

Sterculic acid 是一种硬脂酰辅酶 A 去饱和酶 1 (SCD1) 抑制剂。Sterculic acid 剂量依赖性抑制 delta-9 去饱和酶 (Δ9D) 活性,IC50值为 0.9 μM。
TN3367 Akuammidine

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively.
T35895 Ingenol 3,20-dibenzoate

Ingenol 3,20-dibenzoate is a powerful activator of protein kinase C (PKC) isoforms. It effectively induces the translocation of nPKC-delta, -epsilon, and -theta as well as PKC-mu from the cytosolic fraction to the particulate fraction. Through de novo synthesis of macromolecules, it triggers apoptosis with characteristic morphology. Moreover, Ingenol 3,20-dibenzoate enhances IFN-γ production and degranulation in NK cells, particularly when stimulated by NSCLC cells[1][2].
TN3368 Akuammigine

Opioid Receptor; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki val

天然产物

Delta-Tocopherol
Cat.No: T6000
Synonym: (+)-DELTA-生育酚,D-DELTA-TOCOPHEROL
Target: Endogenous Metabolite
Tetrahydro-2H-pyran-2-one
Cat.No: T4821
Synonym: δ-Valerolactone,δ-Valeryllactone,delta-戊内酯,2-Oxotetrahydropyran
Target: Others, Endogenous Metabolite
3-Carene
Cat.No: T10109
Synonym: Delta-3-Carene
Target: COX, Antifungal
δ-Amyrenone
Cat.No: T10993
Synonym: Delta-Amyrone,Α-香树脂酮
Target: Others
Delta-Caesalpin
Cat.No: TN3817
Synonym:
Target: Others
delta-Valerobetaine
Cat.No: T19274
Synonym:
Target: Others
Ajmalicine
Cat.No: T8044
Synonym: 阿吗里新,Lamuran,Delta-Yohimbine,Raubasine,Ajmalicin
Target: Adrenergic Receptor
delta-Amyrin acetate
Cat.No: TN3816
Synonym:
Target: Others
Delta-Nonalactone
Cat.No: TN6697
Synonym:
Target:
δ-Tocotrienol
Cat.No: TMA2474
Synonym: Delta-Tocotrienol,δ-生育三烯酚
Target: ERK, BCL, VEGFR, Akt, PI3K, PDK, p53
Delta 7-avenasterol
Cat.No: TN3815
Synonym:
Target:
Delta 5-avenasterol
Cat.No: TN3814
Synonym:
Target: Others
D-(+)-Glucono-1,5-lactone
Cat.No: T0933
Synonym: Gluconic acid lactone,Delta-Gluconolactone,Gluconolactone,葡萄糖酸内酯
Target: Others, Reactive Oxygen Species, Endogenous Metabolite
Grayanotoxin II
Cat.No: T31993
Synonym: G-II,Deacetylanhydroandromedotoxin,delta(sup 10 (18))-Andromedenol
Target:
δ-Decalactone
Cat.No: T40815
Synonym:
Target: Others
Sesamin
Cat.No: T2919
Synonym: Fagarol,Fsesamin,芝麻素
Target: Others
Solamargine
Cat.No: T4034
Synonym: Solamargin,δ-Solanigrine,澳洲茄边碱
Target: Apoptosis, p38 MAPK, P-gp, STAT
(+)-δ-Cadinene
Cat.No: T35409
Synonym:
Target: Apoptosis, Antibacterial
6-Deoxy-3-O-methyl-β-allopyranosyl (1→4)-β-cymaronic acid δ-lactone
Cat.No: TN2409
Synonym:
Target: Others
Deltamethrin
Cat.No: T20754
Synonym: Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974
Target: Others
Deltaline
Cat.No: T3S1888
Synonym: 德尔塔林,Deltamine 6-acetate,Eldelin
Target: Others
Deltatsine
Cat.No: TN6070
Synonym:
Target:
gamma-Linolenic acid
Cat.No: T4868
Synonym: gamolenic acid,γ-Linolenic acid,γ-亚麻酸
Target: Endogenous Metabolite
Amentoflavone
Cat.No: T3417
Synonym: Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin
Target: Apoptosis, P450, Phospholipase, Reactive Oxygen Species, Opioid Receptor, COX, Antibacterial, RSV, Antifungal
Sterculic acid
Cat.No: T41253
Synonym:
Target:
Akuammidine
Cat.No: TN3367
Synonym:
Target: Opioid Receptor
Ingenol 3,20-dibenzoate
Cat.No: T35895
Synonym:
Target:
Akuammigine
Cat.No: TN3368
Synonym:
Target: Opioid Receptor, Adrenergic Receptor
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